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Journal articles on the topic '–Aminobenzenesulfonamide'

Author: Grafiati

Published: 2 June 2025

Last updated: 31 July 2025

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1

Benmebarek, Sabrina, Mhamed Boudraa, Sofiane Bouacida, Hocine Merazig та George Dénès. "Bis(4-aminobenzenesulfonamide-κN4)dichloridozinc". Acta Crystallographica Section E Structure Reports Online 70, № 1 (2013): m28—m29. http://dx.doi.org/10.1107/s160053681303417x.

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2

Kaneda, Kyosuke. "Synthesis of Cyclic Compounds Containing Aminobenzenesulfonamide." YAKUGAKU ZASSHI 140, no. 9 (2020): 1087–94. http://dx.doi.org/10.1248/yakushi.20-00139.

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3

Kravchenya, N. A. "Selective N-acylation of 4-aminobenzenesulfonamide." Pharmaceutical Chemistry Journal 23, no. 4 (1989): 332–34. http://dx.doi.org/10.1007/bf00758426.

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4

Güzel-Akdemir, Özlen, Atilla Akdemir, Nilgün Karalı, and Claudiu T. Supuran. "Discovery of novel isatin-based sulfonamides with potent and selective inhibition of the tumor-associated carbonic anhydrase isoforms IX and XII." Organic & Biomolecular Chemistry 13, no. 23 (2015): 6493–99. http://dx.doi.org/10.1039/c5ob00688k.

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A series of 2/3/4-[(2-oxo-1,2-dihydro-3H-indol-3-ylidene)amino]benzenesulfonamides, obtained from substituted isatins and 2-, 3- or 4-aminobenzenesulfonamide, showed low nanomolar inhibitory activity against the tumor associated carbonic anhydrases IX and XII.

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5

H. Naser, Noor, Monther F. Mahdi, Tagreed N-A Omar, and Amar A. Fadhil. "Synthesis and Preliminary Pharmacological Evaluation of New Analogues of Diclofenac as Potential Anti-inflammatory Agents." Iraqi Journal of Pharmaceutical Sciences ( P-ISSN: 1683 - 3597 , E-ISSN : 2521 - 3512) 20, no. 1 (2017): 25–32. http://dx.doi.org/10.31351/vol20iss1pp25-32.

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A group of amine derivatives [4-aminobenzenesulfonamide derivatives, 2-aminopyridine and 2-aminothiazole] incorporated to Î±-carbon of diclofenac a well known non-steroidal anti-inflammatory drug (NSAID) to increase bulkiness were designed and synthesized for evaluation as a potential anti-inflammatory agents with expected COX-2 selectivity. In vivo acute anti-inflammatory activity of the selected final compounds (9, 12 and 13) was evaluated in rats using egg-white induced edema model of inflammation in a dose equivalent to (3 mg/Kg) of diclofenac sodium. All tested compounds produced a signif

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6

F. Mahdi, Monther. "Synthesis and Preliminary Pharmacological Evaluation of Aminobenzensulfonamides Derivatives of Mefenamic Acid as a Potential Anti-inflammatory Agents." Iraqi Journal of Pharmaceutical Sciences ( P-ISSN: 1683 - 3597 , E-ISSN : 2521 - 3512) 17, no. 1 (2017): 7–15. http://dx.doi.org/10.31351/vol17iss1pp7-15.

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A group of amino derivatives [4-aminobenzenesulfonamide,4-amino-NÂ¹ methylbenzenesulfonamide, or NÂ¹-(4-aminophenylsulfonyl)acetamide] bound to carboxyl group of mefenamic acid a well known nonsteroidal anti-inflammatory drugs (NSAIDs) were designed and synthesized for evaluation as a potential anti-inflammatory agent. In vivo acute anti-inflammatory activity of the final compounds (9, 10 and 11) was evaluated in rat using egg-white induced edema model of inflammation in a dose equivalent to (7.5mg/Kg) of mefenamic acid. All tested compounds produced a significant reduction in paw edema with r

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7

Gein, V. L., O. V. Nazarets, A. V. Romanova, et al. "Synthesis and biological activity of 4-aryl-2-hydroxy-4-oxo-<i>N</i>-(2-sulfamoylphenyl)but-2-enamides." Журнал общей химии 93, no. 5 (2023): 664–69. http://dx.doi.org/10.31857/s0044460x23050025.

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The reaction of methyl esters of 4-aryl-2-hydroxy-4-oxobut-2-enoic (aroylpyruvic) acids with 2-aminobenzenesulfonamide in glacial acetic acid in the presence of anhydrous sodium acetate, 4-aryl-2-hydroxy-4-oxo N -(2-sulfamoylphenyl)but-2-enamides were obtained. The analgesic and antimicrobial activity of the obtained compounds was studied.

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8

S. Salem, Bader, Monther F. Mahdi, and Mohammed H. Mohammed. "Synthesis and Preliminary Pharmacological Study of Sulfonamide Conjugates with Ibuprofen and Indomethacin as New Anti-Inflammatory Agents." Iraqi Journal of Pharmaceutical Sciences ( P-ISSN: 1683 - 3597 , E-ISSN : 2521 - 3512) 18, no. 2 (2017): 39–45. http://dx.doi.org/10.31351/vol18iss2pp39-45.

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4-aminobenzenesulfonamide conjugates of ibuprofen (compound 10) and indomethacin (compound 11) have been designed and synthesized by the reaction of sulfanilamide (compound 7) with 2-(4-isobutylphenyl) propanoic acid (ibuprofen) and 2-(1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid (indomethacin) for the evaluation as potential anti-inflammatory agents with expected selectivity against COX-2 enzyme. In vivo acute anti-inflammatory activity of the synthesized final compounds (10 and 11) was evaluated in rats using egg-white induced edema model of inflammation in a dose equival

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9

Nasser, Noor H., Nethal H. Hammud, Samer A. Hasan, Abbas Hamid Abdalsadh, and Ahmed kareem Hussein. "Design and Synthesis of new Naproxen Analogues as Potential Anti-inflammatory Agents." Al Mustansiriyah Journal of Pharmaceutical Sciences 17, no. 1 (2018): 9. http://dx.doi.org/10.32947/ajps.v17i1.61.

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4-aminobenzenesulfonamide derivatives were linked to α-carbon of naproxen a non-selective non-steroidal anti-inflammatory drug (NSAID) to increase its size, so; increase its selectivity toward COX-2 enzyme, rather than COX-1 enzyme, that lead to reduce gastrointestinal side effects of this drug.The chemical structures of the synthesized compounds and their intermediates were confirmed and characterized using elemental microanalysis (CHN), FTIR, and other physicochemical properties like melting points, Rf values.

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10

González, Myriam, María Ovejero-Sánchez, Alba Vicente-Blázquez, et al. "Microtubule Destabilizing Sulfonamides as an Alternative to Taxane-Based Chemotherapy." International Journal of Molecular Sciences 22, no. 4 (2021): 1907. http://dx.doi.org/10.3390/ijms22041907.

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Pan-Gyn cancers entail 1 in 5 cancer cases worldwide, breast cancer being the most commonly diagnosed and responsible for most cancer deaths in women. The high incidence and mortality of these malignancies, together with the handicaps of taxanes—first-line treatments—turn the development of alternative therapeutics into an urgency. Taxanes exhibit low water solubility that require formulations that involve side effects. These drugs are often associated with dose-limiting toxicities and with the appearance of multi-drug resistance (MDR). Here, we propose targeting tubulin with compounds directe

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11

Jin, Jun-su, Xue-mei Pei, Jia-lin Li, and Ze-ting Zhang. "Solubility ofp-Aminobenzenesulfonamide in Supercritical Carbon Dioxide with Acetone Cosolvent." Journal of Chemical & Engineering Data 54, no. 1 (2009): 157–59. http://dx.doi.org/10.1021/je800700r.

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12

Gein, V. L., O. V. Nazarets, A. V. Romanova, O. V. Bobrovskaya, and M. V. Dmitriev. "Reactions of Anthranilamide and 2-Aminobenzenesulfonamide with Pyruvic Acid Esters." Russian Journal of Organic Chemistry 61, no. 1 (2025): 180–83. https://doi.org/10.1134/s1070428024604758.

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13

Aboud, Wasfi, Harith Y. Mahmood, Rasha M. Othman, and Wasan M. Shaker. "The NMR Study and Antimicrobial Activity of Some Schiff Bases Derived From Sulphonamide Drug." JOURNAL OF ADVANCES IN CHEMISTRY 12, no. 2 (2016): 4009–17. http://dx.doi.org/10.24297/jac.v12i2.2157.

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Some Schiff base compounds derived from sulfonamide drug were synthesized by reaction of 4-aminobenzenesulfonamide with aromatic aldehydes (2-hydroxy-1-naphthaldehyde, 3,4-dihydroxybenzaldehyde and 2-hydroxy benzaldehyde) in good yields. Characterization of synthesized compound was carried by elemental analysis, IR, 1H,13C, HSQC and HMBC- NMR spectroscopy. The synthesized compounds were screened for their antibacterial activity against Staphylococcus aureus, Streptococcus sp., Bacillus subtillus, Escherichia coli and Klebsiella pneumonia. Additionally, the compounds were tested for antifungici

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14

Jiang, Pingping, and Zhanzhong Wang. "Solubility ofp-Aminobenzenesulfonamide in Different Solvents from (283.15 to 323.15) K." Journal of Chemical & Engineering Data 54, no. 6 (2009): 1945–46. http://dx.doi.org/10.1021/je900038m.

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15

Hiremath, Kavita B., and Murugesh Shivashankar. "Efficient detection of Sn2+ by 4-aminobenzenesulfonamide based Schiff base chemosensor." Journal of Photochemistry and Photobiology A: Chemistry 450 (May 2024): 115437. http://dx.doi.org/10.1016/j.jphotochem.2023.115437.

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16

Novotný, Ladislav, Hubert Hřebabecký, and Jiří Beránek. "Synthesis of the sulfonamido derivatives of arabinonucleosides." Collection of Czechoslovak Chemical Communications 50, no. 2 (1985): 383–92. http://dx.doi.org/10.1135/cccc19850383.

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Reaction of the sodium salt of 4-aminobenzenesulfonamide with cyclocytidine I and cyclouridine II led to the 2-sulfonamido derivatives V and VI while the reaction with the 5'-chloro derivatives of anhydronucleosides III and IV afforded compounds VIII and IX containing nitrogen bridge between the carbon atoms in position 2 and 5'. Kinetics of the model cyclization reaction of 5'-chloroarabinosylisocytosine (XI) was followed and the structure of prepared compounds was confirmed. Inhibition activity against L 1210 leukemia cells in the experiments in vitro was exhibited by compounds V (1.4 . 10-5

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17

Chern, Ji-Wang, Ching-Po Ho, Ying-Hwa Wu, et al. "1,2,4-benzothiadiazine 1,1-dioxides 3. Reactions of 2-aminobenzenesulfonamide with chloroalkyl isocyanates." Journal of Heterocyclic Chemistry 27, no. 7 (1990): 1909–15. http://dx.doi.org/10.1002/jhet.5570270712.

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18

Zaib, Sumera, Aamer Saeed, Karin Stolte, Ulrich Flörke, Mohammad Shahid, and Jamshed Iqbal. "New aminobenzenesulfonamide–thiourea conjugates: Synthesis and carbonic anhydrase inhibition and docking studies." European Journal of Medicinal Chemistry 78 (May 2014): 140–50. http://dx.doi.org/10.1016/j.ejmech.2014.03.023.

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19

Kallmayer, H. J., and R. Bender. "ChemInform Abstract: Reaction of 2-/4-Aminobenzenesulfonamide Structures with Thymol/Sodium Hypochlorite." ChemInform 32, no. 30 (2010): no. http://dx.doi.org/10.1002/chin.200130074.

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20

Chern, Ji-Wang, Ying-Hwa Wu, and Kang-Chien Liu. "2H-1,2,4-benzothiadiazine 1,1-dioxides2. A condensation of 2-aminobenzenesulfonamide with chloroalkyl isothiocyanates." Journal of Heterocyclic Chemistry 27, no. 5 (1990): 1485–88. http://dx.doi.org/10.1002/jhet.5570270556.

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21

Maloshitskaya, Olga A., Jari Sinkkonen, Valery V. Alekseyev, Kirill N. Zelenin, and Kalevi Pihlaja. "A comparison of ring-chain tautomerism in heterocycles derived from 2-aminobenzenesulfonamide and anthranilamide." Tetrahedron 61, no. 30 (2005): 7294–303. http://dx.doi.org/10.1016/j.tet.2005.04.074.

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22

Kaneda, Kyosuke, Risa Naruse, and Syota Yamamoto. "2-Aminobenzenesulfonamide-Containing Cyclononyne as Adjustable Click Reagent for Strain-Promoted Azide–Alkyne Cycloaddition." Organic Letters 19, no. 5 (2017): 1096–99. http://dx.doi.org/10.1021/acs.orglett.7b00123.

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23

Alafeefy, Ahmed M., Rehan Ahmad, Maha Abdulla, et al. "Development of certain new 2-substituted-quinazolin-4-yl-aminobenzenesulfonamide as potential antitumor agents." European Journal of Medicinal Chemistry 109 (February 2016): 247–53. http://dx.doi.org/10.1016/j.ejmech.2016.01.001.

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24

Kaneda, Kyosuke, Risa Naruse, Syota Yamamoto, and Teppei Satoh. "Reactivity of the Sultam and Strained Alkyne Groups in 2-Aminobenzenesulfonamide-Containing Cyclononyne (ABSACN)." Asian Journal of Organic Chemistry 7, no. 4 (2018): 793–801. http://dx.doi.org/10.1002/ajoc.201700687.

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25

Zheng, Jun, Yan Mei Jin, Xi Nan Yang, et al. "Self-Assembly Mode and Supramolecular Framework of Cyclopentanocucurbit[6]uril and Aromatic Amines." Current Organic Chemistry 25, no. 23 (2021): 2902–8. http://dx.doi.org/10.2174/1385272825666211117153451.

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Single-crystal X-ray diffraction analysis, nuclear magnetic resonance (NMR), and other characterization methods are used to characterize the complexes formed by cyclopentano- cucurbit[6]uril (abbreviated as CyP<sub>6</sub>Q[6]) as a host interacting with p-aminobenzenesulfonamide (G1), 4,4&#039;-diaminobiphenyl (G2), and (E)-4,4&#039;-diamino-1,2-diphenylethene (G3) as guests, respectively. The experimental results show that these three aromatic amine molecules have the same interaction mode with CyP<sub>6</sub>Q[6], interacting with its negatively electric pote

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26

Anandakumaran, J., M. Sundararajan, T. Jeyakumar, and Mohammad Uddin. "Transition Metal Complexes of 4-aminobenzenesulfonamide 1,3-benzodioxole-5-carbaldehyde: Synthesis, Characterization and Biological Activities." American Chemical Science Journal 11, no. 3 (2016): 1–14. http://dx.doi.org/10.9734/acsj/2016/22807.

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27

CHERN, J. W., C. P. HO, Y. H. WU, et al. "ChemInform Abstract: 1,2,4-Benzothiadiazine 1,1-Dioxides. Part 3. Reactions of 2- Aminobenzenesulfonamide with Chloroalkyl Isocyanates." ChemInform 22, no. 18 (2010): no. http://dx.doi.org/10.1002/chin.199118197.

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28

Gelmboldt, V. O., A. A. Ennan, Ed V. Ganin, Yu A. Simonov, M. S. Fonari, and M. M. Botoshansky. "Synthesis and structure of fluorosilicic acid compounds with 4-aminobenzoic acid and with 4-aminobenzenesulfonamide." Journal of Fluorine Chemistry 125, no. 12 (2004): 1951–57. http://dx.doi.org/10.1016/j.jfluchem.2004.08.003.

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29

Starshinova, N. V., and M. N. Filimonova. "Nuclease Biosynthesis and Growth of Serratia marcescens in the Presence of 2-(p-Aminobenzenesulfonamide)-thiazole." Microbiology 74, no. 3 (2005): 310–13. http://dx.doi.org/10.1007/s11021-005-0068-x.

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30

Maloshitskaya, O. A., V. V. Alekseev, and K. Pihlaja. "Tautomeric equilibria in solutions of the products of reaction between 2-aminobenzenesulfonamide and 3-oxo aldehydes." Chemistry of Heterocyclic Compounds 42, no. 2 (2006): 280–81. http://dx.doi.org/10.1007/s10593-006-0085-3.

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31

Gideon, A.Shallangwa, Musa Haliru, and Ogbe Elizabeth. "Design and Synthesis of New Series of One Pot Schiff Bases of 4-AminobenzenesulfonAmideas Potent Antibacterial and Anti-Fungal Agents." Journal of Progressive Research in Chemistry 1, no. 1 (2015): 14–21. https://doi.org/10.5281/zenodo.3970062.

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Schiff bases are imines formed by the condensation of a primary amine and a carbonyl compound. These classes of compounds are very important due to their wide range of biological activities and industrial applications. In this study, some Schiff bases (coded GAS1-5) were synthesized by condensation of 4–Aminobenzenesulfonamide and some selected carbonyl molecules via MW irradiation for 1 minute at 385 watt power; and were characterized by FT-IR and elemental analyses. These Schiff bases were then evaluated for their bactericidal effects against two Gram positive and two Gram negative bac

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32

Lin, Zhaoliang, Zhaohua Huang, Lianjun Shi, and Junlian Huang. "Synthesis of a new monomerN?-(?-methacryloyloxyethyl)-2-pyrimidyl-(p-benzyloxycarbonyl)aminobenzenesulfonamide and its copolymerization withN-phenyl maleimide." Journal of Polymer Science Part A: Polymer Chemistry 38, no. 14 (2000): 2548–54. http://dx.doi.org/10.1002/1099-0518(20000715)38:14<2548::aid-pola50>3.0.co;2-s.

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33

CHERN, J. W., Y. H. WU, and K. C. LIU. "ChemInform Abstract: 2H-1,2,4-Benzothiadiazine 1,1-Dioxides. Part 2. A Condensation of 2- Aminobenzenesulfonamide with Chloroalkyl Isothiocyanates." ChemInform 22, no. 1 (2010): no. http://dx.doi.org/10.1002/chin.199101250.

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34

Havránková, Eva, Nikola Čalkovská, Tereza Padrtová, Jozef Csöllei, Radka Opatřilová, and Pavel Pazdera. "New 1,3,5-Triazine Derivatives Incorporating Aminobenzenesulfonamide, Aminoalcohol, Piperazine, Chalcone or Stilbene Structural Motifs and Evaluation of Their Antioxidative Activity." Proceedings 41, no. 1 (2019): 17. http://dx.doi.org/10.3390/ecsoc-23-06598.

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A series of 1,3,5-triazine derivatives, incorporating aminobenzenesulfonamide, aminoalcohol/phenol, piperazine, chalcone, or stilbene structural motifs, were evaluated as potential antioxidants. The compounds were prepared by using step by step nucleophilic substitution of chlorine atoms in starting 2,4,6-trichloro-1,3,5-triazine. Reactions were catalyzed by Cu(I)-supported on a weakly acidic resin. The radical scavenging activity was determined in terms of %inhibition activity and IC50, using the ABTS method. Trolox and ascorbic acid (ASA) were used as standards. In the lowest used concentrat

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35

Sharif, Muhammad, Julita Opalach, Peter Langer, Matthias Beller, and Xiao-Feng Wu. "Oxidative synthesis of quinazolinones and benzothiadiazine 1,1-dioxides from 2-aminobenzamide and 2-aminobenzenesulfonamide with benzyl alcohols and aldehydes." RSC Adv. 4, no. 1 (2014): 8–17. http://dx.doi.org/10.1039/c3ra45765f.

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36

Hajiaghababaei, Leila, Babak Ghasemi, Alireza Badiei, Hassan Goldooz, Mohammad Reza Ganjali, and Ghodsi Mohammadi Ziarani. "Aminobenzenesulfonamide functionalized SBA-15 nanoporous molecular sieve: A new and promising adsorbent for preconcentration of lead and copper ions." Journal of Environmental Sciences 24, no. 7 (2012): 1347–54. http://dx.doi.org/10.1016/s1001-0742(11)60892-9.

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37

Mikulová, Mária Bodnár, Dáša Kružlicová, Daniel Pecher, Andrea Petreni, Claudiu T. Supuran, and Peter Mikuš. "Synthesis and Inhibition Activity Study of Triazinyl-Substituted Amino(alkyl)-benzenesulfonamide Conjugates with Polar and Hydrophobic Amino Acids as Inhibitors of Human Carbonic Anhydrases I, II, IV, IX, and XII." International Journal of Molecular Sciences 22, no. 20 (2021): 11283. http://dx.doi.org/10.3390/ijms222011283.

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Primary sulfonamide derivatives with various heterocycles represent the most widespread group of potential human carbonic anhydrase (hCA) inhibitors with high affinity and selectivity towards specific isozymes from the hCA family. In this work, new 4-aminomethyl- and aminoethyl-benzenesulfonamide derivatives with 1,3,5-triazine disubstituted with a pair of identical amino acids, possessing a polar (Ser, Thr, Asn, Gln) and non-polar (Ala, Tyr, Trp) side chain, have been synthesized. The optimized synthetic, purification, and isolation procedures provided several pronounced benefits such as a sh

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38

Danilkina, Natalia A., Ekaterina A. Khmelevskaya, Anna G. Lyapunova, et al. "Functionalized 10-Membered Aza- and Oxaenediynes through the Nicholas Reaction." Molecules 27, no. 18 (2022): 6071. http://dx.doi.org/10.3390/molecules27186071.

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The scope and limitations of the Nicholas-type cyclization for the synthesis of 10-membered benzothiophene-fused heterocyclic enediynes with different functionalities were investigated. Although the Nicholas cyclization through oxygen could be carried out in the presence of an ester group, the final oxaenediyne was unstable under storage. Among the N-type Nicholas reactions, cyclization via an arenesulfonamide functional group followed by mild Co-deprotection was found to be the most promising, yielding 10-membered azaendiynes in high overall yields. By contrast, the Nicholas cyclization throu

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39

Alibeg, Ammar Abdul Aziz, and Tuqa Salim Hussein. "In Silico Study of New Isatin- Sulfonamide Derivatives as Carbonic Anhydrase Inhibitors." Wiadomości Lekarskie 77, no. 10 (2024): 2027–32. https://doi.org/10.36740/wlek/193997.

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AimBackground: This study uses molecular docking to describes the potential binding affinity of new sulfonamides derivatives by incorporating substituted Isatin moiety as tail groups linked to 4-amino benzene sulfonamide as zinc binding group through a 4-amino ethyl benzoate linker, that targeted carbonic anhydrase XII enzyme in some firm tumors like breast and colon cancer by using CA XII (PDB: 1JCZ /chain A). Aims: to evaluate compound I, II, III, and IV's anticancer properties that have just been produced. These substances were created with the specific purpose of targeting solid tumors' ca

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40

Mikulová, Mária Bodnár, Dáša Kružlicová, Daniel Pecher, Claudiu T. Supuran, and Peter Mikuš. "Synthetic Strategies and Computational Inhibition Activity Study for Triazinyl-Substituted Benzenesulfonamide Conjugates with Polar and Hydrophobic Amino Acids as Inhibitors of Carbonic Anhydrases." International Journal of Molecular Sciences 21, no. 10 (2020): 3661. http://dx.doi.org/10.3390/ijms21103661.

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Various sulfonamide derivatives are intensively studied as anticancer agents owing to their inhibitory activity against human tumor-associated carbonic anhydrase isoforms. In this work, different synthetic procedures for the series of 1,3,5-triazinyl-aminobenzenesulfonamide conjugates with amino acids, possessing polar uncharged, negatively charged, and hydrophobic side chain, were studied and optimized with respect to the yield/purity of the synthesis/product as well as the time of synthetic reaction. These procedures were compared to each other via characteristic HPLC-ESI-DAD/QTOF/MS analyti

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41

Akocak, Suleyman, Özlen Güzel-Akdemir, Rajesh Kishore Kumar Sanku, et al. "Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII." Bioorganic Chemistry 103 (October 2020): 104204. http://dx.doi.org/10.1016/j.bioorg.2020.104204.

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42

Sbîrnă, Liana Simona, and Clementina Moldovan. "Research on three complex compounds of divalent first-row transition metal ions having the Schiff base derived from sulfanilamide and N-acetylisatin as bidentate ligand." Annals of the University of Craiova Series Chemistry 28, no. 2 (2022): 5–13. http://dx.doi.org/10.52846/aucchem.2022.2.01.

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The present paper aims to describe the research performed on three complex compounds formed by divalent first-row transition metal ions – namely M = Co(II), Ni(II) and Zn(II) (representing the complex kernels) with the Schiff base derived from the condensation of sulfanilamide with N-acetylisatin (which proved itself to be able to act as a bidentate ligand in all these cases). This Schiff base is N-(1-acetyl-2-oxoindolin-3-ylidene)-4-aminobenzenesulfonamide, which appears twice in each complex, but is not the only ligand in the structure, as two water molecules are also part of the coordinatio

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43

Asadi, Prashanth, Kalyani Kodide, Mounika Kota, and Jyothi Thati. "Determination and correlation of solubility and solution thermodynamics of 4-aminobenzenesulfonamide in five binary solvent mixtures from 278.15 to 318.15 K." Journal of Molecular Liquids 303 (April 2020): 112670. http://dx.doi.org/10.1016/j.molliq.2020.112670.

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44

Sharif, Muhammad, Julita Opalach, Peter Langer, Matthias Beller, and Xiao-Feng Wu. "ChemInform Abstract: Oxidative Synthesis of Quinazolinones and Benzothiadiazine 1,1-Dioxides from 2-Aminobenzamide and 2-Aminobenzenesulfonamide with Benzyl Alcohols and Aldehydes." ChemInform 45, no. 28 (2014): no. http://dx.doi.org/10.1002/chin.201428181.

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Dvorkin, A. A., M. S. Fonar', S. T. Malinovskii, et al. "Crystal and molecular structure of the 1:2 complex of cis-anti-cis diastereomer of dicyclohexano-18-crown-6 with 4-aminobenzenesulfonamide." Journal of Structural Chemistry 30, no. 3 (1989): 440–44. http://dx.doi.org/10.1007/bf00751906.

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Kovalenko, S. N., V. P. Chernykh, A. E. Shkarlat, I. V. Ukrainets, V. I. Gridasov, and S. A. Rudnev. "Recyclization of 2-imino-2H-1-benzopyrans under the influence of nucleophilic reagents. 2. Reaction of 2-iminocoumarin-3-carboxamides witho-aminobenzenesulfonamide." Chemistry of Heterocyclic Compounds 34, no. 7 (1998): 791–95. http://dx.doi.org/10.1007/bf02251684.

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Popova, Angelina D., Miglena K. Georgieva, Ognyan I. Petrov, Katya V. Petrova, and Evelina A. Velcheva. "IR spectral and structural studies of 4-aminobenzenesulfonamide (sulfanilamide)-d0, -d4, and -15N, as well as their azanions: Combined DFT B3LYP/experimental approach." International Journal of Quantum Chemistry 107, no. 8 (2007): 1752–64. http://dx.doi.org/10.1002/qua.21242.

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Hen, Naama, Meir Bialer, Boris Yagen, et al. "Anticonvulsant 4-Aminobenzenesulfonamide Derivatives with Branched-Alkylamide Moieties: X-ray Crystallography and Inhibition Studies of Human Carbonic Anhydrase Isoforms I, II, VII, and XIV." Journal of Medicinal Chemistry 54, no. 11 (2011): 3977–81. http://dx.doi.org/10.1021/jm200209n.

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Sun, Jinwei, Tao Tao, Dan Xu, et al. "Metal-free oxidative cyclization of 2-amino-benzamides, 2-aminobenzenesulfonamide or 2-(aminomethyl)anilines with primary alcohols for the synthesis of quinazolinones and their analogues." Tetrahedron Letters 59, no. 21 (2018): 2099–102. http://dx.doi.org/10.1016/j.tetlet.2018.04.054.

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Xi, Long-Yi, Ruo-Yi Zhang, Lei Shi, Shan-Yong Chen, and Xiao-Qi Yu. "Iodine-mediated synthesis of 3-acylbenzothiadiazine 1,1-dioxides." Beilstein Journal of Organic Chemistry 12 (May 24, 2016): 1072–78. http://dx.doi.org/10.3762/bjoc.12.101.

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Abstract:

An iodine-mediated synthesis of 3-acylbenzothiadizine 1,1-dioxides is described. A range of electronically diverse acetophenones reacted well with several 2-aminobenzenesulfonamides, affording 3-acylbenzothiadiazine 1,1-dioxides in good yields.

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