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Dissertations / Theses on the topic 'Isoxazolino'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Knight, Julian Gary. "Diphenylphosphinoylalkyk isoxazoles and isoxazolines." Thesis, University of Cambridge, 1989. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.306451.

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2

Lager, Markku. "Isoxazoline Synthese, Eigenschaften und N-O-Bindungsspaltungen /." [S.l.] : [s.n.], 2005. http://deposit.ddb.de/cgi-bin/dokserv?idn=974370304.

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3

Young, Anne A. "Nitrile oxide/isoxazoline approach to higher sugars." Thesis, University of Edinburgh, 1990. http://hdl.handle.net/1842/11655.

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The application of nitrile oxide/isoxazoline chemistry towards the synthesis of higher sugars (monosaccharides containing seven or more contiguous carbon atoms) has been investigated. This convergent approach, involving the cycloaddition of sugar derived alkene and nitrile oxide fragments and subsequent manipulation of the resulting isoxazoline, has much of the product stereochemistry preselected. Three ω-unsaturated monosaccharides were chosen for study: the D-glucose-derived six carbon unit (<i>94</i>), its C-3 epimer (<i>102</i>) and a seven carbon alkene, (<i>97</i>), prepared from D-galac

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4

Boyd, Ewan Campbell. "Synthetic applications of nitrile oxide/isoxazoline chemistry." Thesis, University of Edinburgh, 1992. http://hdl.handle.net/1842/12525.

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Three alkenes, (<i>R/S</i>)-2-phenyl-4-vinyl-4,5-dihydro-oxazole (<i>11</i>), (4<i>R</i>)-3-<i>N-t</i>-butoxycarbonyl-2,2-dimethyl-4-vinyloxazolidine (<i>12</i>) and (2<i>R</i>)-2-(<i>N-t</i>-butoxycarbonyl)aminobut-3-en-1-ol (<i>13</i>), have been prepared from (<i>S</i>)-serine and used in cycloaddition reactions with some common nitrile oxides, to investigate the effect of an allylic nitrogen at an α-chiral centre on π-facial selectivity. Alkene (<i>11</i>) was prepared in racemic form after an unexpected racemisation during its synthesis. Cycloaddition reactions with three nitrile oxides (

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5

Penman, Kenneth J. "The nitrile oxide/isoxazoline route to carbon-linked disaccharides." Thesis, University of Edinburgh, 1993. http://hdl.handle.net/1842/11249.

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A route to carbon-linked disaccharides (two monosaccharide units linked by a carbon bridge rather than a glycosidic oxygen) employing nitrile oxide/isoxazoline chemistry has been investigated. This convergent approach is based on cycloaddition of sugar-derived alkene and nitrile oxide fragments, followed by ring cleavage and functional group manipulation of the resulting 2-isoxazoline. Careful selection of the nitrile oxide and alkene fragments defines much of the stereochemistry of the products. Two ω-unsaturated hexofuranoses were chosen for study: 3-<i>O</i>-benzyl-5,6-dideoxy-1,2-<i>O</i>-

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6

Tavares, Aline. "Isoxazolinas: uma classe de materiais avançados revisitada." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2010. http://hdl.handle.net/10183/32776.

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Este trabalho descreve a síntese e caracterização de séries inéditas de materiais líquidocristalinos contendo o N-heterociclo isoxazolina. Este anel foi obtido a partir da reação de cicloadição [3+2] 1,3-dipolar de óxidos de nitrila a diferentes dipolarófilos. As propriedades térmicas foram analisadas por MOLP, DSC e TGA, e as propriedades ópticas através de espectros de absorção. O presente trabalho apresenta três publicações, um artigo submetido e dois em fase final de redação, todos relacionados à Tese. Na primeira publicação (Eur. J. Org. Chem. 2009, 889-897) foi obtida uma coleção de isox

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7

March, Andrew Ronald. "Application of nitrile oxide/isoxazoline chemistry in C-glycoside synthesis." Thesis, University of Edinburgh, 2000. http://hdl.handle.net/1842/12565.

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A route to <i>C</i>-glycosides and <i>C</i>-disaccharides with functionalised linkages has been investigated. This convergent strategy involves cycloaddition of selected alkenes and sugar derived nitrile oxide moieties. The resultant 2-isoxazolines can be modified and subsequently ring opened to afford compounds with carbonyl or amino containing linkages. The alkenes selected for study were two w-unsaturated monosaccharide derivatives: 5,6-dideoxy-1,2-<i>O</i>-isopropylidene-a-D-<i>xylo</i>-hex-5-enofuranose and methyl 5,6-dideoxy-2,3-<i>O</i>-isopropylidene-a-D-<i>lyxo</i>-hex-5-enofuranoside

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8

Leandro, Gonçalves Bonfim Reis Silvio. "Síntese e avaliação preliminar da atividade antinoceptiva e toxicidade de novas isoxazolil-aril-hidrazonas." Universidade Federal de Pernambuco, 2008. https://repositorio.ufpe.br/handle/123456789/3215.

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Made available in DSpace on 2014-06-12T16:28:59Z (GMT). No. of bitstreams: 2 arquivo2102_1.pdf: 2203105 bytes, checksum: 355011545cb1b9f8b811ca232623d364 (MD5) license.txt: 1748 bytes, checksum: 8a4605be74aa9ea9d79846c1fba20a33 (MD5) Previous issue date: 2008<br>Fundação de Amparo à Ciência e Tecnologia do Estado de Pernambuco<br>A Química Medicinal, através de estratégias específicas, vem para estudar as razões moleculares da ação dos fármacos, descrevendo a relação entre a estrutura química e a atividade farmacológica, com objetivo de planejar, sintetizar e produzir moléculas com potenc

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9

Correia, de Almeida Gleybson. "Síntese e avaliação preliminar da atividade antimicrobiana e antichagásica de novas isoxazolil-aril-semicarbazonas, e tiossemicarbazonas e isoxazolil-nitrofurfuril-hidrazonas." Universidade Federal de Pernambuco, 2010. https://repositorio.ufpe.br/handle/123456789/2969.

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Made available in DSpace on 2014-06-12T16:25:37Z (GMT). No. of bitstreams: 2 arquivo1125_1.pdf: 3490678 bytes, checksum: 347a62790e8d9bfb7abcdf2e63109656 (MD5) license.txt: 1748 bytes, checksum: 8a4605be74aa9ea9d79846c1fba20a33 (MD5) Previous issue date: 2010<br>Coordenação de Aperfeiçoamento de Pessoal de Nível Superior<br>Na literatura, há um grande número de trabalhos que buscam obter derivados de semicarbazonas e tiossemicarbazonas, contendo heterociclos, com aplicações farmacológicas, como antimicrobiana, antichagásica, antifúngica, antineoplásica e anticonvulsivante. Pesquisas vêm obte

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10

Wierschem, Frank Georg. "Darstellung und Modifizierung von 2-Oxo-piperazin-basierenden Isoxazolinen und Isoxazolidinen in Lösung und an fester Phase." [S.l.] : [s.n.], 2004. http://deposit.ddb.de/cgi-bin/dokserv?idn=971626812.

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11

Leilane, Souza Santana Maria. "Síntese e avaliação da atividade antitumoral de novos aminoácidos isoxazolínicos de conformação restringida." Universidade Federal de Pernambuco, 2011. https://repositorio.ufpe.br/handle/123456789/3665.

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Made available in DSpace on 2014-06-12T16:32:58Z (GMT). No. of bitstreams: 2 arquivo9012_1.pdf: 1156402 bytes, checksum: 455074848a3e717cd6059d914fcaae0b (MD5) license.txt: 1748 bytes, checksum: 8a4605be74aa9ea9d79846c1fba20a33 (MD5) Previous issue date: 2011<br>De acordo com a literatura, há uma grande quantidade de trabalhos com a intenção de obter derivados do ácido glutâmico com aplicações farmacológicas, como a neurotransmissora, antitumoral, anti-inflamatória. Também se deve salientar a variedade de trabalhos contendo o núcleo 2-isoxazolina explorando as mais diversas atividades biológ

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12

Ferguson, William James. "The nitrile oxide/isoxazoline route to novel C-glycosides and C-disaccharides." Thesis, University of Edinburgh, 1996. http://hdl.handle.net/1842/13815.

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A convergent route, based on nitrile oxide/isoxazoline chemistry to carbon-linked disaccharides (<I>C</I>-disaccharides) and <I>C</I>-glycosides with functionalised linkages has been investigated. The sequence involves three steps. Firstly, the cycloaddition of a sugar-derived nitrile oxide to a terminal alkene provides a 3,5-disubstituted 2-isoxazoline. Next, the substituents attached to the isoxazoline may be modified, and finally the heterocycle subjected to either hydrogenolysis or reductive cleavage to afford a <I>C</I>-glycoside with a carbonyl or an amino functionalised linkage. Four te

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13

Huang, Sheng-Lin Kevin. "Cycloaddition reactions in the construction of isoxazoline, azacyanine, and imidazopyridinium/pyridopyrimidium heterocycles /." For electronic version search Digital dissertations database. Restricted to UC campuses. Access is free to UC campus dissertations, 2002. http://uclibs.org/PID/11984.

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14

Tout, Jaki. "The synthesis and reactions of alkenyl isoxazoles and isoxazolines." Thesis, University of Edinburgh, 1993. http://hdl.handle.net/1842/14563.

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Four vinyl-isoxazoles and -2-isoxazolines have been synthesised as potential monomers for polymerisation studies. 5-Phenyl-3-vinylisoxazole was prepared in 38% overall yield by a sequence involving cycloaddition of ethoxycarbonyl-formonitrile oxide to phenylacetylene and then reduction of the resulting 3-carbethoxyisoxazole to the aldehyde using di-isobutylaluminium hydride. In the final stage Wittig olefination of the formyl-isoxazole afforded the target compound. 5-Phenyl-3-vinylisoxazole (17%) and 5-phenyl-3-vinyl-2-isoxazoline (26%) were synthesised similarily from ethyl propiolate & benzo

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15

Chhetri, Manjit Singh. "N-cyclohenyl, N-phenyl nitrones and their potentiality in isoxazolidine and isoxazoline syntheses." Thesis, University of North Bengal, 2010. http://hdl.handle.net/123456789/1364.

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16

Vilela, Guilherme Drechsler. "Síntese de polimetacrilatos, triarilaminase perilenos derivados de isoxazóis e isoxazolinas." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2014. http://hdl.handle.net/10183/109702.

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Este trabalho descreve a síntese e caracterização de diferentes séries inéditas de isoxazolinas e isoxazóis dirigida para a área de materiais orgânicos eletrônicos e a sua derivatização em polimetacrilatos líquido-cristalinos, em aminas terciárias e em derivados do perileno. As isoxazolinas foram sintetizadas por meio de reação de cicloadição [3+2] 1,3-dipolar de óxidos de nitrila com alcenos escolhidos, com posterior oxidação do anel para isoxazol via MnO2, gerando os isoxazóis 5a-c. Isoxazóis 3-aril-5-hidroximetil substituídos 37a-c foram obtidos através da reação de cicloadição [3+2] entre

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17

Todd, Christine Joy. "Application of nitrile oxide-isoxazoline chemistry for the synthesis of 2-ulosonic acid analogues." Thesis, University of Edinburgh, 1995. http://hdl.handle.net/1842/13143.

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Nitrile oxide-isoxazoline methodology has been employed in a novel convergent approach towards 2-ulosonic acid analogues, in particular those of 3-deoxy-D-<I>arabino</I>-2-heptulosonic acid (DAH) and 3-deoxy-D-<I>manno</I>-octulosonic acid (KDO). It involves regio- and diastereoselective [3+2] cycloaddition of a nitrile oxide to carbohydrate alk-1-enes containing four, five or six carbons, yielding 2-isoxazolines. Subsequent deprotection followed by reductive hydrolytic cleavage affords the 2-ulosonic acid analogues. The four carbon alkene 1,2-dideoxy-3,4-<I>0</I>-cyclohexylidene-D-<I>glycero<

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18

McGhie, Karen E. "Application of nitrile oxide-isoxazoline chemistry for the synthesis of higher monosaccharides and azasugars." Thesis, University of Edinburgh, 1994. http://hdl.handle.net/1842/15332.

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Nitrile oxide-isoxazoline chemistry has been utilised in a convergent approach towards the synthesis of a series of undecose monosaccharides. The sequence involves three stages. The cycloaddition of a five-carbon nitrile oxide to a hex-5-enofuranose derivative provides an eleven carbon framework incorporating a 2-isoxazoline. Reductive hydrolytic cleavage of the heterocycle to a β-hydroxyketone followed by reduction affords the target 6-deoxy-higher sugar. Two ω-unsaturated monosaccharide derivatives, 3-<I>O</I>-benzyl-5,6-dideoxy-1,2,<I>O</I>-isopropylidene-α-<SUB>D</SUB>-<I>xylo</I>-hex-5-en

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19

Fritsch, Luma. "Síntese de novos cristais líquidos derivados de base de schiff com núcleo isoxazolina/isoxazol." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2015. http://hdl.handle.net/10183/129750.

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Esta dissertação apresenta a síntese e caracterização espectroscópica e térmica de duas novas series de bases de Schiff líquido cristalinas contendo o anel isoxazolina e isoxazol. Foram sintetizados 22 bases de Schiff da série (E)-N-[4-(alquiloxi)benzilideno]-4-[5-(X)-4,5-dihidroisoxazol-3-il]anilinas (8c-i) e 22 bases de Schiff da série (E)-N-[4-(alquiloxi)benzilideno]-4-[5-(X)-isoxazol-3-il]anilinas (8c´-i´). Em ambas as séries, o grupo X é CH3 para 8c/8c’; Cl para 8d/8d’; Br para 8e/8e’; H para 8f/8f’; n-Butila; para 8h/8h’ e 2-Etilhexila para 8i/8i’. O substituinte alquiloxila em ambas as

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20

BEZERRA, JÚNIOR Natanael da Silva. "Síntese e avaliação da atividade citotóxica de novos derivados tiossemicarbazônicos isoxazolínicos aza-bicíclicos." Universidade Federal de Pernambuco, 2016. https://repositorio.ufpe.br/handle/123456789/22669.

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SANTOS, Adriano Carlos Vieira dos. "Síntese e avaliação da atividade antimicrobiana de 3-aril-2-isoxazolina [5,4-d]pirrolidinas na forma de base livre e de seus sais cloridratos." Universidade Federal de Pernambuco, 2014. https://repositorio.ufpe.br/handle/123456789/11770.

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Submitted by Ramon Santana (ramon.souza@ufpe.br) on 2015-03-10T18:47:31Z No. of bitstreams: 2 DISSERTAÇÃO Adriano Carlos Vieira dos Santos.pdf: 4334924 bytes, checksum: fb764c055d3256c9ebc2045d717205ac (MD5) license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5)<br>Made available in DSpace on 2015-03-10T18:47:31Z (GMT). No. of bitstreams: 2 DISSERTAÇÃO Adriano Carlos Vieira dos Santos.pdf: 4334924 bytes, checksum: fb764c055d3256c9ebc2045d717205ac (MD5) license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5) Previous issue date: 2014-05-30<br>A quími

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22

Mancuso, Vincent. "Nouvelle voie de synthèse de bêta-aminocétones via les Delta4-isoxazolines." Doctoral thesis, Universite Libre de Bruxelles, 1990. http://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/213161.

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23

MARQUES, Ronmilson Alves. "Síntese de 3-aril-2-isoxazolinas Aza-bicíclicas, Potenciais Anti-inflamatórios." Universidade Federal de Pernambuco, 2013. https://repositorio.ufpe.br/handle/123456789/10735.

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Submitted by Ramon Santana (ramon.souza@ufpe.br) on 2015-03-05T14:59:20Z No. of bitstreams: 2 Dissertaçao Romilson Marques.pdf: 2036007 bytes, checksum: f115cf2424502d94f10d7887506d0249 (MD5) license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5)<br>Made available in DSpace on 2015-03-05T14:59:20Z (GMT). No. of bitstreams: 2 Dissertaçao Romilson Marques.pdf: 2036007 bytes, checksum: f115cf2424502d94f10d7887506d0249 (MD5) license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5) Previous issue date: 2013-08<br>Comumente, os anti-inflamatórios não ester

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Lee, Ja Young. "Synthese neuartiger Furanomycin-Analoga und Versuche zur Synthese von Bis-([alpha]-Aminosäuren) über Bis(isoxazoline) /." Waabs : GCA-Verl, 2005. http://deposit.ddb.de/cgi-bin/dokserv?id=2760965&prov=M&dok_var=1&dok_ext=htm.

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25

Sharma, Prawin Kumar. "Greener approach to the synthesis of some novel class of isoxazolidine and isoxazoline derivatives using N-methyl and N-phenyl-a-chloro nitrones." Thesis, University of North Bengal, 2016. http://ir.nbu.ac.in/handle/123456789/1884.

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26

AGUIAR, Hellen Rayanna Tôrres de Sousa. "Síntese e avaliação da atividade citotóxica de 3-carboxamidas-2-isoxazolinas azabicíclicas." Universidade Federal de Pernambuco, 2013. https://repositorio.ufpe.br/handle/123456789/24360.

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Submitted by Alice Araujo (alice.caraujo@ufpe.br) on 2018-04-17T20:10:19Z No. of bitstreams: 1 DISSERTAÇÃO Hellen Rayanna Tôrres de Sousa.pdf: 1104206 bytes, checksum: d3954e6cc348b627ea44b745ab57d3ba (MD5)<br>Made available in DSpace on 2018-04-17T20:10:19Z (GMT). No. of bitstreams: 1 DISSERTAÇÃO Hellen Rayanna Tôrres de Sousa.pdf: 1104206 bytes, checksum: d3954e6cc348b627ea44b745ab57d3ba (MD5) Previous issue date: 2013-08-30<br>O método mais usado para síntese de novos fármacos é a modificação molecular. Esse método consiste em tomar uma substância conhecida, como modelo ou protótipo e a p

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Rosa, Rafaela Raupp da. "Isoxazolinas e isoxazóis como reais candidatos na preparação de cristais líquidos polares." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2018. http://hdl.handle.net/10183/180639.

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A presente tese descreve a síntese e caracterização de 10 novas séries de moléculas na forma de banana contendo os anéis isoxazolina e isoxazol como reais candidatos na preparação de cristais líquidos polares. Foram avaliados parâmetros estruturais tais como o tipo de função conectora do centro curvado com os braços mesogênicos, a natureza do heterociclo e a sua posição relativa ao núcleo. A síntese dos compostos contou com a metodologia de preparação do anel isoxazolina, a cicloadição [3+2] 1,3-dipolar entre alcenos e óxidos de nitrila, os quais foram gerados pelas oximas preparadas a partir

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Mota, Fernanda Virginia Barreto. "Estudo das atividades anti-inflamatória e antinociceptiva de novos derivados isoxazolinaacilhidrazonas." Universidade Federal de Pernambuco, 2013. https://repositorio.ufpe.br/handle/123456789/11417.

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Lee, Ja Young. "Synthese neuartiger Furanomycin-Analoga und Versuche zur Synthese von Bis-([alpha]-Aminosäuren [alpha-Aminosäuren]) über Bis(isoxazoline)." Waabs GCA, 2004. http://deposit.ddb.de/cgi-bin/dokserv?id=2760965&prov=M&dok_var=1&dok_ext=htm.

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Ritter, Olga Maria Schimidt. "Síntese e caracterização de novos materiais líquido-cristalinos derivados de bifenilcarboxilatos e 3,5-isoxazolinas." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2005. http://hdl.handle.net/10183/6327.

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Este trabalho mostra a síntese de novos materiais poliméricos utilizando como unidade mesogênica anéis bifenilas, com um grupo espaçador de onze unidades metilênicas, com uma cadeia polimérica acrilato e que apresentam como grupo terminal uma porção quiral sintetizada a partir de L-isoleucina. Os monômeros apresentaram comportamento enantiotrópico mesofases esmética C e A quiral. Do mesmo modo, os polímeros apresentaram mesofase esmética A estável no aquecimento e no resfriamento. Foi realizado também a síntese de poliacrilatos tendo presente como grupo de ligação na unidade mesogênica o anel

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ARAÚJO, NETA Marlene Saraiva de. "Síntese de novas 4-acil-semicarbazidas e 1,2,4-triazóis isoxazolínicos com potenciais atividades biológicas." UNIVERSIDADE FEDERAL DE PERNAMBUCO, 2014. https://repositorio.ufpe.br/handle/123456789/14989.

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Submitted by Isaac Francisco de Souza Dias (isaac.souzadias@ufpe.br) on 2016-01-25T17:16:38Z No. of bitstreams: 2 license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5) DISSERTAÇÃO DE MESTRADO - MARLENE SARAIVA DE ARAÚJO NETA.pdf: 2177316 bytes, checksum: ba8286fc22cd5e5e207b9fa533be39e5 (MD5)<br>Made available in DSpace on 2016-01-25T17:16:38Z (GMT). No. of bitstreams: 2 license_rdf: 1232 bytes, checksum: 66e71c371cc565284e70f40736c94386 (MD5) DISSERTAÇÃO DE MESTRADO - MARLENE SARAIVA DE ARAÚJO NETA.pdf: 2177316 bytes, checksum: ba8286fc22cd5e5e207b9fa533be39e5 (MD5) Prev

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Lima, Dias Cabral Nadia. "Síntese e avaliação do potencial biológico de novos derivados N-fenacilados do aza-biciclo pirrolidino [3,2-d] isoxazolina." Universidade Federal de Pernambuco, 2005. https://repositorio.ufpe.br/handle/123456789/3497.

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Made available in DSpace on 2014-06-12T16:31:31Z (GMT). No. of bitstreams: 2 arquivo6103_1.pdf: 1565028 bytes, checksum: 35570c901ad1402b9be60679631dd83b (MD5) license.txt: 1748 bytes, checksum: 8a4605be74aa9ea9d79846c1fba20a33 (MD5) Previous issue date: 2005<br>Diante de trabalhos anteriores do nosso grupo de pesquisas, em que foram obtidos derivados N-(benzoil)-pirrolidino[3,2-d]isoxazolinas 40, com excelentes atividades biológicas, por meio de reações de cicloadição 1,3-dipolar de enecarbamatos e enamidas endocíclicas de 5 membros, vislumbramos a obtenção dos derivados N-(fenacil)-pirr

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Chhetri, Esmita. "Synthesis, characterization and inclusion complexation of some isoxazolidine and isoxazoline derivatives for advanced applications explored by physicochemical approach." Thesis, University of North Bengal, 2021. http://ir.nbu.ac.in/handle/123456789/4343.

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Moschref, Said-Nadjib. "Synthese und Umlagerung von mono-metallierten Bisallylethersystemen und die Synthese von mono-metallierten Isoxazolen." [S.l. : s.n.], 1999. http://deposit.ddb.de/cgi-bin/dokserv?idn=962341290.

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Iannuzzi, M. C. "SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW CTP SYNTHETASE INHIBITORS AS NEW POTENTIAL AGENTS FOR THE TREATMENT OF AFRICAN TRYPANOSOMIASIS." Doctoral thesis, Università degli Studi di Milano, 2012. http://hdl.handle.net/2434/170499.

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Cytidine triphosphate synthetase (CTPS), a glutamine amidotransferase (GAT) responsible for the de novo synthesis of CTP, was recently suggested as a potential drug target for the treatment of Human African Trypanosomiasis, a parasitic disease caused by Trypanosoma brucei. Acivicin, a natural antitumor antibiotic, is a well-known inhibitor of enzymes belonging to the GAT family. Its CTPS inhibitory activity has been related to the observed trypanocidal activity in bloodstream T. brucei cell cultures. The aim of this project was the design and synthesis of Acivicin analogues characterized by

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36

SILVA, Jannieres Darc da. "Síntese de novos derivados naftoquinônicos e avaliação da sua atividade biológica." Universidade Federal de Pernambuco, 2014. https://repositorio.ufpe.br/handle/123456789/25641.

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Submitted by Pedro Barros (pedro.silvabarros@ufpe.br) on 2018-08-08T17:13:01Z No. of bitstreams: 2 license_rdf: 811 bytes, checksum: e39d27027a6cc9cb039ad269a5db8e34 (MD5) DISSERTAÇÃO Jannieres Darc da Silva.pdf: 4262765 bytes, checksum: db979524e7755928a9210a77fd40680b (MD5)<br>Approved for entry into archive by Alice Araujo (alice.caraujo@ufpe.br) on 2018-08-16T22:12:46Z (GMT) No. of bitstreams: 2 license_rdf: 811 bytes, checksum: e39d27027a6cc9cb039ad269a5db8e34 (MD5) DISSERTAÇÃO Jannieres Darc da Silva.pdf: 4262765 bytes, checksum: db979524e7755928a9210a77fd40680b (MD5)<br>Made available i

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Khan, Pasha Moeenuddin. "Application of Pd Catalyzed Alkylation: Synthesis of Bicyclic Furans, Isoxazolines and New Cyclopentane Amino acid Analogs." [Tampa, Fla] : University of South Florida, 2008. http://purl.fcla.edu/usf/dc/et/SFE0002792.

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38

Jurberg, Igor Dias. "Synthesis of Alkynes and New Transformations Catalyzed by Gold(I) Complexes." Palaiseau, Ecole polytechnique, 2010. http://pastel.archives-ouvertes.fr/docs/00/57/00/64/PDF/These_Igor.pdf.

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Sur la plateforme de thèses en ligne Tel on trouve le résumé suivant en français : La synthèse d'alcynes en utilisant des isoxazolones comme précurseurs a été une méthode développée dans notre laboratoire dans ler dernières années. Nous avons appliqué cette méthodologie pour la synthèse de 3-alkynylamides et leur utilisation pour générer des dihydropyrrolones. Nous avons aussi développé de nouvelles réactions catalysées pour complexes d'or(I): la synthèse de 4-oxazol-2-ones à partir de Boc-ynamides, une séquence de transfert 1,5 d'hydrure et cyclisation pour former des éther cycliques et la fo

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39

Springsteel, Mark Francis. "Synthesis of flavones, isoxazolines and related heterocycles : the search for small molecule drugs to treat cystic fibrosis /." For electronic version search Digital dissertations database. Restricted to UC campuses. Access is free to UC campus dissertations, 2003. http://uclibs.org/PID/11984.

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40

Wirtz, Lisa [Verfasser], and Uli [Akademischer Betreuer] Kazmaier. "Entwicklung einer effizienten Synthese von Isoxazolin-Aminosäureesterderivaten : Entwicklung und Anwendung von 7-Dialkyl-Aminocumarin-Fluoreszenz-Labels / Lisa Wirtz. Betreuer: Uli Kazmaier." Saarbrücken : Saarländische Universitäts- und Landesbibliothek, 2012. http://d-nb.info/1052338682/34.

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41

Luitel, Govinda Prasad. "Greener synthesis of some new isoxazolidine and isoxazoline derivatives via 1,3-dipolar cycloaddition reactions and studies of biological activities of the cycloadducts." Thesis, University of North Bengal, 2017. http://ir.nbu.ac.in/handle/123456789/2576.

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42

Soret, Adrien. "Etude de la réactivité d'ylures d'azométhines ou de nitrones avec des 7-oxabicyclo[2. 2. 1]hepta-2,5-diènes : préparation de composés hétérocycliques par réaction de rétro-Diels-Alder." Paris 11, 2007. http://www.theses.fr/2007PA112098.

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Depuis plusieurs années, notre équipe s’intéresse à l’utilisation d’une résine portant des groupes furyles dans diverses stratégies « traceless ». Cette stratégie implique une étape d’accrochage de diénophiles acétyléniques par réaction de Diels-Alder et de décrochage de la résine par réaction rétro-Diels-Alder thermique après fonctionnalisation de l’adduit de cycloaddition. Différentes fonctionnalisations ont déjà été réalisées. Dans un premier temps, nous avons abordé la préparation de dérivés 7-oxa-bicyclo[2. 2. 1]hepta-2,5-diéniques par réaction de Diels-Alder entre des composés acétyléniq

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43

Saraiva, de Araujo Neta Marlène. "Planification, synthèse et activité tripanocide et leishmanicide de nouveaux dérivés hybrides à partir de 2-isoxazoline aza-bicyclique et 5,6,7,8-tétrahydroimidazo[1,2-a]pyrazine." Thesis, Nantes, 2019. http://www.theses.fr/2019NANT1022.

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Neglected diseases reach millions of people around the world. Among these are Chagas disease and Leishmaniasis. Chagas disease is caused by a protozoan, the Trypanosoma cruzi and its main form of transmission is through the faeces of the insect commonly known as barber. Leishmaniasis can be caused by more than 20 types of parasites of the genus Leishmania and there are 3 types of the disease, Cutaneous Leishmaniasis, Cutaneous-Mucous or Tegumentary Leishmaniasis, and Visceral Leishmaniasis. For the treatment of these diseases numerous problems exist, such as the large amount of side effects, l

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Toh, Ophilia Ndi. "Synthesis Towards Fulminic Acid and Its Derivatives in 1, 3-Dipolar Cycloaddition Reactions." Digital Commons @ East Tennessee State University, 2008. https://dc.etsu.edu/etd/1982.

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A new approach to fulminic acid cycloadditions has been developed. At reduced temperatures, fulminic acid is generated in situ and undergoes 1, 3-diploar cycloaddition reactions with dipolarophiles to form isoxazolines and/or its dimers. This procedure represents a novel, safe general method for the one-step generation of fulminic acid, which complements existing potentially explosive protocols.

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45

Moraes, de Almeida Valderes. "Síntese assimétrica de 3-carboxamidas enantiomericamente puras e de hidrazidas e arilhidrazonas, derivadas do novo heterociclo 7-(benzoil)- 2-isoxazolina[5,4-b] pirrolidina. Avaliação das atividades biológicas." Universidade Federal de Pernambuco, 2008. https://repositorio.ufpe.br/handle/123456789/3019.

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Made available in DSpace on 2014-06-12T16:26:16Z (GMT). No. of bitstreams: 2 arquivo2109_1.pdf: 2735340 bytes, checksum: 9eec1389edfda8071ea76404501b0077 (MD5) license.txt: 1748 bytes, checksum: 8a4605be74aa9ea9d79846c1fba20a33 (MD5) Previous issue date: 2008<br>Coordenação de Aperfeiçoamento de Pessoal de Nível Superior<br>Em estudos prévios, 2-isoxazolinas aza-bicíclicas foram obtidos por nosso grupo de pesquisa, dando origem a núcleos como o 2-isoxazolina[5,4-b]piperidina e 2-isoxazolina[5,4- b]pirrolidina. Amidas N-benzoiladas derivadas dessas substâncias, apresentaram-se biologicamen

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46

Toldo, Josene Maria. "Estudo teórico da reação de cicloadição [3+2] 1,3-dipolar para formação do anel isoxazolina utilizando teoria do funcional da densidade e modelos implícitos de solvente." reponame:Biblioteca Digital de Teses e Dissertações da UFRGS, 2013. http://hdl.handle.net/10183/70459.

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As reações de cicloadição 1,3-dipolar são uma poderosa ferramenta para a síntese de uma variedade de anéis heterocíclicos de cinco membros. A cicloadição de óxidos de nitrila à olefinas, em particular, é de considerável interesse para a obtenção de isoxazolinas, que são intermediários versáteis na síntese de produtos naturais e de materiais com potencial aplicação como cristais líquidos. A Teoria do Funcional da Densidade foi utilizada para estudar o mecanismo da reação cicloadição [3+2] 1,3-dipolar que ocorre, inicialmente, entre o óxido de benzonitrila e o ácido vinilacético. Para tal, foram

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47

Becker, Tobias [Verfasser], Wilhelm [Gutachter] Boland, Georg Gutachter] Pohnert, and Wittko [Gutachter] [Francke. "3-Nitropropanoic acid and isoxazolin-5-one derived glucosides in chrysomelina larvae : synthesis, biosynthesis, occurrence and toxicity / Tobias Becker ; Gutachter: Wilhelm Boland, Georg Pohnert, Wittko Francke." Jena : Friedrich-Schiller-Universität Jena, 2017. http://d-nb.info/1177602245/34.

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48

Motei, Rachid. "Nouveaux complexes de fer pour la modélisation du site actif des hydrogénases [FeFe] ou pour la commutation & Synthèse et caractérisation d'aminoesters isoxazoliniques." Thesis, Brest, 2017. http://www.theses.fr/2017BRES0160.

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Dans la première partie de ce travail, nous avons réalisé une étude préliminaire qui avait pour objectif d’étendre la série de complexes dinucléaires du fer [Fe2(CO)4(k2-P2N2)(μ-dithiolate)], comprenant des ligands diphosphine de type P2N2, à des complexes possédant un pont azadithiolate en vue d’étudier leur comportement en milieu acide et le rôle des différentes bases présentes dans la seconde sphère de coordination de ces composés. Les nouveaux complexes [Fe2(CO)6(k2-PPh2NR2)(μ-adtBn)] (R = Ph, Bn)) ont été obtenus par réaction entre le précurseur [Fe2(CO)6(μ-adtBn)] et les diphosphines cyc

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49

Bathich, Yaser. "Synthesis of branched amino polyols and amino hydroxy acids stereoselective addition of C-nucleophiles to isoxazolines and isoxazolinium salts and assignment of configurations /." [S.l. : s.n.], 2006. http://nbn-resolving.de/urn:nbn:de:bsz:93-opus-26179.

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Jurberg, Igor. "Synthèse d´Alcynes et Nouvelles Réactions catalysées par Complexes d´or(I)." Phd thesis, Ecole Polytechnique X, 2010. http://pastel.archives-ouvertes.fr/pastel-00570064.

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La synthèse d'alcynes en utilisant des isoxazolones comme précurseurs a été une méthode développée dans notre laboratoire dans ler dernières années. Nous avons appliqué cette méthodologie pour la synthèse de 3-alkynylamides et leur utilisation pour générer des dihydropyrrolones. Nous avons aussi développé de nouvelles réactions catalysées pour complexes d'or(I): la synthèse de 4-oxazol-2-ones à partir de Boc-ynamides, une séquence de transfert 1,5 d'hydrure et cyclisation pour former des éther cycliques et la formation de dérivés de cinnolines. Nous avons aussi développé un étude mecanistique

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