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Journal articles on the topic 'Phenylthiazoyl'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Mamedov, Vakhid A., Yakov A. Levin, Evgeniya K. Trutneva, et al. "Functionalized 4-methyl-5-phenylthiazole and 1,3-bis(4'-methyl-5'-phenylthiazol-2'-yl)benzene. Approaching thiazole macrocycles." Arkivoc 2004, no. 12 (2005): 47–69. http://dx.doi.org/10.3998/ark.5550190.0005.c06.

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2

Fouda, Abdel Aziz, A. Abdel Nazeerb, and K. M. Abdel Khalek. "Corrosion Inhibition of Zinc Using Some Phenylthiazole Derivatives in Hydrochloric acid Solutions." JOURNAL OF ADVANCES IN CHEMISTRY 12, no. 7 (2013): 425–40. http://dx.doi.org/10.24297/jac.v12i7.2798.

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The inhibitive action of some phenylthiazole derivatives namely: 2-acetylamino-5-p-bromophenylazo-4-phenylthiazole (BPT), 2-acetylamino-5-p-methylphenylazo-4-phenylthiazole (MPT), 2-acetylamino-5-p-methoxyphenylazo-4-phenylthiazole (XPT) and 2-acetylamino-5-p-nitrophenylazo-4-phenylthiazole (NPT), on zinc corrosion in 0.2 M HCl has been studied using weight loss, potentiodynamic polarization, electrochemical impedance spectroscopy (EIS)and electrochemical frequency modulation (EFM) measurements. The results showed that the dissolution rate of zinc decreases with increasing the phenylthiazole d

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3

Fouda, Abdel Aziz, A. Abdel Nazeerb, and K. M. Abdel Khalek. "Corrosion Inhibition of Zinc Using Some Phenylthiazole Derivatives in Hydrochloric acid Solutions." JOURNAL OF ADVANCES IN CHEMISTRY 4, no. 2 (2008): 425–40. http://dx.doi.org/10.24297/jac.v4i2.2704.

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The inhibitive action of some phenylthiazole derivatives namely: 2-acetylamino-5-p-bromophenylazo-4-phenylthiazole (BPT), 2-acetylamino-5-p-methylphenylazo-4-phenylthiazole (MPT), 2-acetylamino-5-p-methoxyphenylazo-4-phenylthiazole (XPT) and 2-acetylamino-5-p-nitrophenylazo-4-phenylthiazole (NPT), on zinc corrosion in 0.2 M HCl has been studied using weight loss, potentiodynamic polarization, electrochemical impedance spectroscopy (EIS)and electrochemical frequency modulation (EFM) measurements. The results showed that the dissolution rate of zinc decreases with increasing the phenylthiazole d

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4

Sarangi, P. K. N., J. Sahoo, S. K. Paidesetty, and G. P. Mohanta. "SYNTHESIS, SPECTRAL CHARACTERIZATION AND ANTICANCER EVALUATION OF NEW DIAZENYL SCHIFF BASE DERIVATIVES." INDIAN DRUGS 54, no. 02 (2017): 20–28. http://dx.doi.org/10.53879/id.54.02.10877.

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A series of several diazenyl Schiff base derivatives were designed and synthesized through azo coupling of diazotised primary amines with the novel synthesized Schiff base ligand (E)-N-((2-chloroquinolin-3-yl) methylene)-4-phenylthiazol-2-amine. All the synthesized compounds have been analysed by different spectral techniques such as elemental analysis, 1H NMR, FT-IR, UV-Vis and LC-MS for their structural confirmation. The above conjugates have been studied for their solvent effects by treating them with different solvents. The results of in vitro cytotoxic study of the synthesized compounds a

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5

Abdel-Wahab, Bakr F., Benson M. Kariuki, Hanan A. Mohamed, and Gamal A. El-Hiti. "Catalyst-Free Synthesis of Novel 4-(Benzofuran-2-yl)-N-phenylthiazol-2(3H)-imines, Crystal Structure Elucidation, and the Effect of Phenyl Substitution on Crystal Packing." Crystals 13, no. 8 (2023): 1239. http://dx.doi.org/10.3390/cryst13081239.

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A one-pot reaction of an equimolar mixture of 4-methoxyaniline, phenyl isothiocyanate, and 2-bromoacetylbenzofuran in absolute ethanol in the absence of any catalysts afforded 4-(benzofuran-2-yl)-3-(4-methoxyphenyl)-N-phenylthiazol-2(3H)-imine with an 83% yield. Under similar conditions, 4-flouroaniline provided a mixture of the expected 4-(benzofuran-2-yl)-3-(4-fluorophenyl)-N-phenylthiazol-2(3H)-imine and unexpected 4-(benzofuran-2-yl)-N-(4-fluorophenyl)-3-phenylthiazol-2(3H)-imine at an overall 73% yield. The structures of the synthesized heterocycles were confirmed using NMR spectroscopy.

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6

Zhu, ShaoPing, Yuan Chen, Jun Sun, YuTing Yang, and ChuanJun Yue. "Synthesis, Characterization, Thermochromism, and Photochromism of Aromatic Aldehyde Hydrazone Derivatives." Journal of Chemistry 2016 (2016): 1–8. http://dx.doi.org/10.1155/2016/8460462.

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The Schiff bases N-(5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (1), N-(4′-chloro-5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (2), and N-(4′-nitro-5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (3) were synthesized. These compounds were characterized by using IR,1H NMR,13C NMR, and MS. The photochromism of the compounds was investigated by IR and UV-visible spectrometry which is time variable under irradiation of 254 nm UV light. The thermochromism of the compounds was studied using temperature-variable IR, UV-visible spectrometry, TG, and differential scann

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7

Luo, Yong, Yongxia Zhu, Kai Ran, et al. "Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents." MedChemComm 6, no. 6 (2015): 1036–42. http://dx.doi.org/10.1039/c4md00573b.

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8

Luo, Yong, Yongxia Zhu, Kai Ran, et al. "Correction: Synthesis and biological evaluation of N-(4-phenylthiazol-2-yl)cinnamamide derivatives as novel potential anti-tumor agents." MedChemComm 6, no. 7 (2015): 1404. http://dx.doi.org/10.1039/c5md90027a.

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9

Stokes, Emily C., Emily E. Langdon-Jones, Lara M. Groves, et al. "Cationic, luminescent cyclometalated iridium(iii) complexes based on substituted 2-phenylthiazole ligands." Dalton Transactions 44, no. 18 (2015): 8488–96. http://dx.doi.org/10.1039/c4dt03054k.

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10

D., C. DASH, K. BEHERA R., M. SEN (Miss), and M. MEHER F. "Synthesis and Characterisation of some Transition Metal Complexes of 4-Substituted-2-thiazolylhydrazones of Salicylaldehyde and 2-Hydroxyacetophenone." Journal of Indian Chemical Society Vol. 68, Dec 1991 (1991): 663–64. https://doi.org/10.5281/zenodo.6134555.

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Post-Graduate Department of Chemistry, Sambalpur University, Jyoti Vihar, Burla-788 019 <em>Manuscript received 27 April 1988, revised 21 November 1991, accepted 6 December 1991</em> THE communication reports the synthesis and structural studies on the complexes of Co<sup>II</sup>, Ni<sup>II</sup> and Cu<sup>ll</sup> with some hydrazone derivatives containing thiazole moiety and a OH group near the condensation site, such as 2-salicylideneiminoamino-4- phenylthiazole (SPTH), 2-salicylideneiminoamino-4-bromophenylthiazole (SBPTH), 2-α-methylsalicyli-deneiminoamino-4- phenylthiazole (MSPTH

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11

Au-Alvarez, O., R. C. Peterson, A. Acosta Crespo, et al. "2-Amino-4-phenylthiazole." Acta Crystallographica Section C Crystal Structure Communications 55, no. 5 (1999): 821–23. http://dx.doi.org/10.1107/s0108270199001961.

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12

Zhao, Jiang, Xiaojie Chen, Jianglan Wu, Maoyang Jian, Guijiang Zhou, and Zhenguo Chi. "Fluoro-benzenesulfonyl-functionalized 2-phenylthiazole-type iridium(iii) complexes for efficient solution-processed organic light-emitting diodes." Journal of Materials Chemistry C 8, no. 30 (2020): 10390–400. http://dx.doi.org/10.1039/d0tc02250k.

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13

Bhuiyan, Md Mosharef Hossain, Mohammed M. Matin, AFM Hafizur Rahman, and Md Rabiul Alam. "Synthesis and Biological Evaluation of Sugar Induced Thiazole Derivatives." Chittagong University Journal of Science 41, no. 1 (2021): 68–84. http://dx.doi.org/10.3329/cujs.v41i1.51915.

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The starting materials, 2-amino-4-phenylthiazole and 2-amino-4,5,6,7-tetrahydrobenzo[d]thiazole, were prepared by reacting thiourea with acetophenone and cyclohexanone in the presence of iodine under heating on a water bath with occasional stirring, respectively. Reaction of 2-amino-4-phenylthiazole and 2-amino-4,5,6,7-tetrahydrobenzo[d]thiazole with various sugars afforded corresponding N-glycoside derivatives in good yields. The structures of the synthesized N-glycosides derivatives have been established on the basis of their IR and NMR spectral data. The obtained compounds were screened for

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14

Bhuiyan, M. H., and A. F. M. H. Rahman. "Synthesis and Antimicrobial Evaluation of Some Thiazole Derivatives." Journal of Scientific Research 3, no. 1 (2010): 111. http://dx.doi.org/10.3329/jsr.v3i1.5419.

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Reaction of 2-amino-4-phenylthiazole with various aromatic aldehydes afforded 2-arylideneamino-4-phenylthiazoles. On the other hand treatment of 2-amino-4-phenylthiazole with several acyl halides furnished N-(thiazol-2-yl)-amides. The synthesized compounds have been screened for their antimicrobial activity against Bacillus cereus, Bacillus subtilis, Staphylococcus aureus, Shigella dysenteriae, Salmonella typhi, Pseudomonous sp. bacteria and Aspergillus niger, Penicillium notatum, Aspergillus funiculosus, Collectrichum corchori Ikata (Yoshida) and Curvularia lunata fungi respectively. Some of

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15

Rahaman, Fazlur, Priti Gupta, Prabhat Gautam, et al. "Synthesis, Characterization, Fluorescence and Antimicrobial studies of Cu(II), Co(II), Ni(II), Zn(II) and Cd(II) complexes derived from Schiff’s base (E)-2-(5-chloro-2-hydroxybenzylidene)-N-(4-phenylthiazol-2-yl)hydrazinecarboxamide." Journal of University of Shanghai for Science and Technology 23, no. 09 (2021): 81–111. http://dx.doi.org/10.51201/jusst/21/09518.

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A series of Cu(II), Co(II), Ni(II), Zn(II) and Cd(II) complexes of (E)-2-(5-chloro-2-hydroxybenzylidene)-N-(4-phenylthiazol-2-yl)hydrazinecarboxamide (HL) with ONO donor ligand was synthesized. The ligand (HL) was prepared by the condensation of N-(4-phenylthiazol-2-yl)hydrazinecarboxamide with 5-chloro-2-hydroxybenzaldehyde. The HL and its metal complexes have been characterized using elemental analysis and various spectral techniques such as, FTIR, 1H and 13C NMR, Mass, UV–Visible, ESR, thermal analysis (TGA), magnetic moment, conductivity and powder-XRD. The Powder XRD pattern indicates hex

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16

Ai, Hong-Lian, Bao-Bao Shi, Wei Li, et al. "Bipolarithizole A, an antifungal phenylthiazole-sativene merosesquiterpenoid from the potato endophytic fungus Bipolaris eleusines." Organic Chemistry Frontiers 9, no. 7 (2022): 1814–19. http://dx.doi.org/10.1039/d1qo01887f.

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Bipolarithizole A (1) is a phenylthiazole-sativene sesquiterpenoid hybrid isolated from the fungus Bipolaris eleusines. It shows anti-pathogenic fungi activity against Rhizoctonia solani with an MIC value of 16 μg mL−1.

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17

Jemili, Rihab, Joana F. Campos, Nicolas Dumuis, Hervé Rabat, Nadjib Semmar, and Sabine Berteina-Raboin. "Laser synthesis: a solvent-free approach for the preparation of phenylthiazolo[5,4-b]pyridine derivatives." RSC Advances 11, no. 9 (2021): 5003–7. http://dx.doi.org/10.1039/d0ra10094c.

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18

Dinçer, Muharrem, Namık Özdemir, Alaaddin Çukurovalı, and İbrahim Yılmaz. "2-[(4-Phenylthiazol-2-yl)hydrazonomethyl]phenol." Acta Crystallographica Section E Structure Reports Online 61, no. 6 (2005): o1712—o1714. http://dx.doi.org/10.1107/s1600536805014418.

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19

N., K. MANDAL, SINHA R., and P. BANERJEE K. "Synthesis and Biological Activity of Thiazolo and Phenylthiazolo-2-carboxamido-pyrazoline and -isoxazoline Derivatives." Journal of Indian Chemical Society Vol. 64, May 1987 (1987): 318–21. https://doi.org/10.5281/zenodo.6236397.

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P. G. Department of Chemistry, Bhagalpur University, Bhagalpur-812 007 <em>Manuscript received 23 June 1986, accepted 22 April 1987</em> Synthesis and Biological Activity of Thiazolo and Phenylthiazolo-2-carboxamido-pyrazoline and -isoxazoline Derivatives.

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20

Yernale, Nagesh Gunvanthrao, and Mruthyunjayaswamy Bennikallu Hire Mathada. "Synthesis, Characterization, Antimicrobial, DNA Cleavage, andIn VitroCytotoxic Studies of Some Metal Complexes of Schiff Base Ligand Derived from Thiazole and Quinoline Moiety." Bioinorganic Chemistry and Applications 2014 (2014): 1–17. http://dx.doi.org/10.1155/2014/314963.

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A novel Schiff base ligandN-(4-phenylthiazol-2yl)-2-((2-thiaxo-1,2-dihydroquinolin-3-yl)methylene)hydrazinecarboxamide(L)obtained by the condensation ofN-(4-phenylthiazol-2-yl)hydrazinecarboxamide with 2-thioxo-1,2-dihydroquinoline-3-carbaldehyde and its newly synthesized Cu(II), Co(II), Ni(II), and Zn(II) complexes have been characterized by elemental analysis and various spectral studies like FT-IR,1H NMR, ESI mass, UV-Visible, ESR, TGA/DTA, and powder X-ray diffraction studies. The Schiff base ligand(L)behaves as tridentate ONS donor and forms the complexes of type [ML(Cl)2] with square pyr

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21

Omara, Mariam, Mohamed Hagras, Mohamed M. Elsebaie, et al. "Exploring novel aryl/heteroaryl-isosteres of phenylthiazole against multidrug-resistant bacteria." RSC Advances 13, no. 29 (2023): 19695–709. http://dx.doi.org/10.1039/d3ra02778c.

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Twenty-three compounds of novel phenylthiazole derivatives were synthesized utilizing the Suzuki coupling reaction. Antibacterial activity in an in vivo model against MRSA USA300 was evaluated, as it reduced the burden of MRSA USA300 in skin-infected mice.

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22

Nagaladinne, Nizamuddin, Abdul Ahad Hindustan, and Devanna Nayakanti. "Design, Synthesis and Molecular Modelling Studies of 1-Methyl-3-(4-Substituted phenyl-1,3- thiazol-2-yl)-2-(pyridin-3-yl)-2,3-dihydroquinazolin-4(1H)-ones as Potent Anticancer Agents." Asian Journal of Chemistry 32, no. 12 (2020): 3067–74. http://dx.doi.org/10.14233/ajchem.2020.22930.

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The present study involves the design, synthesis, characterization and molecular docking studies of biologically active quinazolin-4-ones, which were synthesized by condensing 2-amino-4-substituted phenylthiazole with N-methylbenzoxazin-4-one. The N-methylbenzoxazin-4-one and 2-amino-4- substituted phenylthiazole were synthesized from N-methylanthranilic acid and substituted ketones, respectively. The ADME properties determined the synthetic accessibility of quinazolin-4-ones by in silico Swiss ADME. The colorectal anticancer screening was done by using cell HT-29 human colorectal adenocarcino

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23

Pulat, Sultan, Inho Yang, Jihye Lee, et al. "Anithiactin D, a Phenylthiazole Natural Product from Mudflat-Derived Streptomyces sp., Suppresses Motility of Cancer Cells." Marine Drugs 22, no. 2 (2024): 88. http://dx.doi.org/10.3390/md22020088.

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Anithiactin D (1), a 2-phenylthiazole class of natural products, was isolated from marine mudflat-derived actinomycetes Streptomyces sp. 10A085. The chemical structure of 1 was elucidated based on the interpretation of NMR and MS data. The absolute configuration of 1 was determined by comparing the experimental and calculated electronic circular dichroism (ECD) spectral data. Anithiactin D (1) significantly decreased cancer cell migration and invasion activities at a concentration of 5 μM via downregulation of the epithelial-to-mesenchymal transition (EMT) markers in A549, AGS, and Caco-2 cell

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24

Mayhoub, Abdelrahman S., Mansoora Khaliq, Carolyn Botting, Ze Li, Richard J. Kuhn, and Mark Cushman. "An investigation of phenylthiazole antiflaviviral agents." Bioorganic & Medicinal Chemistry 19, no. 12 (2011): 3845–54. http://dx.doi.org/10.1016/j.bmc.2011.04.041.

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25

Tian, Yao, Jinchao Shi, Xiaoqian Deng, et al. "Design, Synthesis, and Antifungal Activity of Some Novel Phenylthiazole Derivatives Containing an Acylhydrazone Moiety." Molecules 28, no. 20 (2023): 7084. http://dx.doi.org/10.3390/molecules28207084.

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Crop fungal diseases pose a serious threat to global crop production and quality. Developing new and efficient fungicides is an important measure to control crop diseases. Phenylthiazole was found to be an excellent antifungal skeleton based on our previous study on the structural optimization and biological activity of the natural product thiasporine A. To find new fungicides, 45 phenylthiazole derivatives containing an acylhydrazone moiety were designed and synthesized by the principle of active substructure splicing. Forty-two of the forty-five compounds are novel, except for compounds E1,

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26

Yu, Yong-Qiang, Yue Wang, Pei-Zhou Ni, and Tao Lu. "6-(Methylsulfanyl)-2-phenylthiazolo[5,4-b]pyridine." Acta Crystallographica Section E Structure Reports Online 63, no. 2 (2007): o968—o969. http://dx.doi.org/10.1107/s1600536807003030.

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27

Chien, James C. W., and S. Ramakrishnan. "Phenylthiazyl polymers with flexible spacers: synthesis and electrical properties." Macromolecules 21, no. 7 (1988): 2007–10. http://dx.doi.org/10.1021/ma00185a020.

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28

Y., Jadegoud, B. Ijare Omkar, N. Mallikarjuna N., D. Angadi S., and H. M. Mruthyunjayaswamy B. "Synthesis and antimicrobial activity of copper-, cobalt- and nickel(II) complexes with Schiff bases." Journal of Indian Chemical Society Vol. 79, Dec 2002 (2002): 921–24. https://doi.org/10.5281/zenodo.5847948.

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Department of Chemistry, Gulbarga University. Gulbarga-585 106, India <em>E-mail </em>: root@guluni.kar.nic.in         <em>  Fax :</em> 91-08472-21632 <em>Manuscript received 1 January 2002, accepted 12 July 2002</em> A few complexes of Cu<sup>II</sup>, Co<sup>II</sup> and Ni<sup>II</sup> have been prepared by reacting their metal(ll) chlorides with 3-(4'-phenylthiazole-2'-yl)- 1-(2' -hydroxy-l' -iminomcthylphenly)urea and with 3-(4' -phenylthiazole-2' -yl)-1-(2' ,4' -dihydroxy/2' -hydroxy-5' -chloro-1 '-m

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29

Limbasiya, Krishna K., Jayesh Babariya, Krushnakumar J. Jilariya, and V. A. Modhavadiya. "SYNTHESIS, CHARACTERIZATION AND BIOLOGICAL EVALUATION OF SOME NOVELTHIAZOL DERIVATIVES OF N-((2-CHLOROPHENYL)DIPHENYLMETHYL)-4-PHENYLTHIAZOL-2-AMINE." Journal of Advanced Scientific Research 13, no. 01 (2022): 305–10. http://dx.doi.org/10.55218/jasr.202213135.

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In present work we synthesized novel series of thiazole derivatives of N-((2-chlorophenyl)diphenylmethyl)-4- phenylthiazol-2-amine in the presence of dichloromethane and triethylamine in good yield. The different studies indicate that newly synthesized compounds possess moderate to good biological activities. The title compounds have been synthesized with several structural variations. Biological evaluation of all the synthesized compounds has been carried out in vitro for their antibacterial and antifungal efficacy against various bacterial and fungal strains. The structure of synthesized com

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30

Abdallah, Amira E. M., Rafat M. Mohareb, Maher H. E. Helal, and Germeen J. Mofeed. "Synthesis and Anticancer Evaluations of Novel Thiazole Derivatives Derived from 4-Phenylthiazol-2-amine." Acta Chimica Slovenica 68, no. 3 (2021): 604–16. http://dx.doi.org/10.17344/acsi.2020.6446.

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Many novel thiazole derivatives were designed and synthesized using 4-phenylthiazol-2-amine. The reactivity of the latter compound toward different chemical reagents was studied. The structure of the newly synthesized compounds was established based on elemental analysis and spectral data. Furthermore, twenty compounds of the synthesized systems were selected and evaluated in (μM) as significant anticancer agents towards three human cancer cell lines [MCF-7 (breast adenocarcinoma), NCI-H460 (non-small cell lung cancer), and SF-268 (CNS cancer)] and normal fibroblasts human cell line (WI-38). T

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31

Dow, Geoffrey S., Yufeng Chen, Katherine T. Andrews, et al. "Antimalarial Activity of Phenylthiazolyl-Bearing Hydroxamate-Based Histone Deacetylase Inhibitors." Antimicrobial Agents and Chemotherapy 52, no. 10 (2008): 3467–77. http://dx.doi.org/10.1128/aac.00439-08.

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ABSTRACT The antimalarial activity and pharmacology of a series of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors (HDACIs) was evaluated. In in vitro growth inhibition assays approximately 50 analogs were evaluated against four drug resistant strains of Plasmodium falciparum. The range of 50% inhibitory concentrations (IC50s) was 0.0005 to >1 μM. Five analogs exhibited IC50s of <3 nM, and three of these exhibited selectivity indices of >600. The most potent compound, WR301801 (YC-2-88) was shown to cause hyperacetylation of P. falciparum histones, which is a

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32

Seleem, Mohammed A., Ahmed M. Disouky, Haroon Mohammad, et al. "Second-Generation Phenylthiazole Antibiotics with Enhanced Pharmacokinetic Properties." Journal of Medicinal Chemistry 59, no. 10 (2016): 4900–4912. http://dx.doi.org/10.1021/acs.jmedchem.6b00233.

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33

Nicolás, Álvaro, Julia G. Quero, Marta Barroso, Zoila Gándara, and Lourdes Gude. "DNA Interactions and Biological Activity of 2,9-Disubstituted 1,10-Phenanthroline Thiosemicarbazone-Based Ligands and a 4-Phenylthiazole Derivative." Biology 13, no. 1 (2024): 60. http://dx.doi.org/10.3390/biology13010060.

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Four 1,10-phenanthroline derivatives (1–4) were synthesized as potential telomeric DNA binders, three substituted in their chains with thiosemicarbazones (TSCs) and one 4-phenylthiazole derivative. The compounds were characterized using NMR, HRMS, FTIR-spectroscopy and combustion elemental analysis. Quadruplex and dsDNA interactions were preliminarily studied, especially for neutral derivative 1, using FRET-based DNA melting assays, equilibrium dialysis (both competitive and non-competitive), circular dichroism and viscosity titrations. The TSC derivatives bind and stabilize the telomeric Tel2

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34

Liu, Wei-Wei, Ling Wang, Li-Juan Tang, Wei Cao, and Hong-Wen Hu. "2-Phenylindolizine-3-carbaldehyde (4-phenylthiazol-2-yl)hydrazone hydrobromide monohydrate." Acta Crystallographica Section E Structure Reports Online 63, no. 8 (2007): o3518. http://dx.doi.org/10.1107/s1600536807034149.

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35

Khrustalev, D. P. "Modification of 2-amino-4-phenylthiazole under microwave irradiation." Russian Journal of General Chemistry 79, no. 3 (2009): 515–16. http://dx.doi.org/10.1134/s1070363209030311.

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36

Nalini, Veerapaneni, and Gautam R. Desiraju. "Gas–solid chlorination of 4-phenylthiazole-2(1H)-thione." J. Chem. Soc., Chem. Commun., no. 13 (1987): 1046–48. http://dx.doi.org/10.1039/c39870001046.

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37

Kenzhetaeva, S. O., and L. K. Abulyaissova. "Synthesis of 2-amino-4-phenylthiazole-derived thiuram disulfide." Russian Journal of General Chemistry 83, no. 11 (2013): 2115–16. http://dx.doi.org/10.1134/s1070363213110285.

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38

Kouhkan, Maryam, Ali Souldozi, and Reza Talebi. "In Vitro Antimicrobial Activity of New Substituted Phenylthiazole Derivatives." Iranian Jornal of Toxicology 12, no. 1 (2018): 33–37. http://dx.doi.org/10.29252/arakmu.12.1.33.

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39

Davydova, Yulia А., Taras M. Sokolenko, Yurii G. Vlasenko, and Yurii L. Yagupolskii. "Chemical properties of 5-(1,1,2,2-tetrafluoroethoxy)-4-phenylthiazole derivatives." Chemistry of Heterocyclic Compounds 51, no. 1 (2015): 80–87. http://dx.doi.org/10.1007/s10593-015-1663-z.

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40

McCluskey, Adam, Matthew Finn, Maria Bowman, Roger Smith, and Paul A. Keller. "2,7-Dimethylthiazolo[4,5-d]pyradazine-4-(5H)-thione: A Corticotrophin-Releasing Hormone Type 1 Receptor Agonist." Australian Journal of Chemistry 53, no. 12 (2000): 905. http://dx.doi.org/10.1071/ch99015.

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Thiazoles, including 2,7-dimethylthiazolo[4,5-d]pyradazine-4-(5H)-thione (4b) and the corresponding 5-phenylthiazolo[4,5-d]pyradazine-4-methylthiol (5a), were synthesized as part of an ongoing investigation into corticotrophin-releasing hormone (CRH) type 1 receptor activity. Subsequent screening indicated the successful discovery of receptor agonists. Assay results indicated a 52 and 3% increase in β-endorphin release after the administration of 100 M (4b) and (5a), respectively. It is believed that this represents the first evidence of this class of compounds displaying CRH type 1 receptor a

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41

Gahtori, Prashant, Surajit Kumar Ghosh, Brijesh Singh, Udaya Pratap Singh, Hans Raj Bhat, and Archana Uppal. "Synthesis, SAR and antibacterial activity of hybrid chloro, dichloro-phenylthiazolyl-s-triazines." Saudi Pharmaceutical Journal 20, no. 1 (2012): 35–43. http://dx.doi.org/10.1016/j.jsps.2011.05.003.

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He, Li-Min, Ai-Xi Hu, Gao Cao, and Jun-Jun Peng. "Ethyl 2-methyl-1-(4-phenylthiazol-2-yl)-1H-benzimidazole-6-carboxylate." Acta Crystallographica Section E Structure Reports Online 63, no. 8 (2007): o3643. http://dx.doi.org/10.1107/s1600536807036483.

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43

Subramanian, Arun Prabhu, Rathakrishnan Samiyappan, Balakrishnan Anitha, Gandhimathi Kaliyamoorthi Ayyadurai, and Jayaprakash Rajendran. "Theoretical and Pharmacological Investigations of Phenylthiazol-2, 4 Dihydroxybenzaldehyde Condensed Schiff Base." Biomedical and Pharmacology Journal 17, no. 4 (2024): 2535–49. https://doi.org/10.13005/bpj/3046.

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The ability of thiazole derivatives to alter the activity of numerous metabolic enzymes suggests that they have promising therapeutic applications. Their antimicrobial, antifungal, anti-inflammatory, antioxidant, and antiproliferative properties were also established. The Schiff base, which was formed by combining 2, 4-dihydrxy benzaldehyde with phenyl thiazole amine, was studied using UV, FTIR, 1H, and 13C-NMR. The significant absorption (283 nm) and vibrational peaks at 1625 cm-1 were observed for the imine group. The compound was confirmed by the presence of a free proton and carbon peak fo

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44

Takami, Shizuka, Minori Nishiyama, Masaki Mizuno, Tadatsugu Yamaguchi, Yuichiro Hashimoto, and Tsuyoshi Kawai. "Photochromic Performance of 5-Heteroaryl-4-vinyl-2-phenylthiazole Derivatives." Bulletin of the Chemical Society of Japan 92, no. 10 (2019): 1773–78. http://dx.doi.org/10.1246/bcsj.20190093.

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Ezzat, Hany. "SYNTHESIS AND EVALUATION OF NEW PHENYLTHIAZOLE DERVATIVES AS ANTIMICROBIAL AGENTS." Al-Azhar Journal of Pharmaceutical Sciences 60, no. 2 (2019): 59–75. http://dx.doi.org/10.21608/ajps.2019.70240.

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Zhang, Zhi-Hua, Hong-Mei Wu, Sai-Nan Deng, et al. "Design, Synthesis, and Anticancer Activities of Novel 2-Amino-4-phenylthiazole Scaffold Containing Amide Moieties." Journal of Chemistry 2018 (October 18, 2018): 1–8. http://dx.doi.org/10.1155/2018/4301910.

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Appropriately substituted 2-amino-4-phenylthiazole derivatives were designed and synthesized according to the structural characteristics of crizotinib. The obtained compounds were characterized using 1H NMR, 13C NMR, and HRMS. The target compounds 5a–o were evaluated for their in vitro antiproliferative activity against A549, HeLa, HT29, and Karpas299 human cancer cell lines. Based on results of biological studies, some of these compounds exhibited significant antiproliferative activity. Compound 5b possessed outstanding growth inhibitory effects on the four cell lines, especially for HT29 cel

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A., K. SINGH, ROY BANI, and P. SINGH R. "Bidentate Pyrimidine-2-thiols as Spectrophotometric Reagents for Palladium and Osmium-Determination in Alloys, Minerals and Catalysts." Journal of Indian Chemical Society Vol. 62, Apr 1985 (1985): 316–18. https://doi.org/10.5281/zenodo.6324802.

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Department of Chemistry, University of Delhi, Delhi-110 007 <em>Manuscript received 23 July 1984, accepted 29 April 1985</em> 1-Pyridyl and 1-(4'-phenylthiazolyI)-4,4,6-trimethyl-1<em>H</em>,4<em>H</em>-pyrimidine-2-thiol (abbreviated as PyTPT and PhTPT, respectively) have been synthesised and studied for the photometric determination of palladium and osmium The reagents are highly selective as other transition and platinum group metals do not interfere. Optimum conditions for both these determinations have been established. The methods have been employed for the determination of pall

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Sal’keeva, L. K., E. V. Minayeva, M. T. Nurmaganbetova, B. Z. Kokzhalova, and A. I. Mantel’. "Glycidol esters from diethylamido-(4-phenylthiazolyl-2-amido)-ketophosphonates and their chemical modification." Russian Journal of General Chemistry 79, no. 4 (2009): 755–58. http://dx.doi.org/10.1134/s1070363209040136.

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Schmidt, Boris. "P2-130: Phenylthiazolyl-hydrazides: A lead for tau aggregation inhibitors and tau imaging?" Alzheimer's & Dementia 4 (July 2008): T408—T409. http://dx.doi.org/10.1016/j.jalz.2008.05.1203.

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Mabkhot, Yahia N., Hazem A. Ghabbour, and Faiz A. Al-aizari. "Crystal structure of 2-(4-methyl-3-phenylthiazol-2(3H)-ylidene)malononitrile, C13H9N3S." Zeitschrift für Kristallographie - New Crystal Structures 232, no. 3 (2017): 451–52. http://dx.doi.org/10.1515/ncrs-2016-0313.

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