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Journal articles on the topic 'Salicylamido'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Malakhova, Anna Yu, and Vladimir N. Kuklin. "Synthesis, the structure of arylsalicylic amides, which have anthelmintic activity." Butlerov Communications 57, no. 3 (2019): 58–70. http://dx.doi.org/10.37952/roi-jbc-01/19-57-3-58.

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Salicylamides (N-aryl-substituted hydroxybenzamides): well-known organic compounds with diverse biological activity, which were originally investigated as antimicrobial and antifungal substances. Salicylamides have also been used as anthelmintic or molluscicidal agents in human and veterinary medicine. The most famous is 5,2'-dichloro-4'-nitrosalicylamide (niclosamide, yomezan – Germany), resynthesized in the USSR under the name of fenasal, which is effective in treating diphyllobothriasis and hymenolepidosis and has molluscicidal properties. The works of domestic and foreign scientists F.S. M

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2

Makhaeva, Galina F., Nadezhda V. Kovaleva, Elena V. Rudakova, et al. "Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer’s Disease." International Journal of Molecular Sciences 24, no. 3 (2023): 2285. http://dx.doi.org/10.3390/ijms24032285.

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A series of previously synthesized conjugates of tacrine and salicylamide was extended by varying the structure of the salicylamide fragment and using salicylic aldehyde to synthesize salicylimine derivatives. The hybrids exhibited broad-spectrum biological activity. All new conjugates were potent inhibitors of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) with selectivity toward BChE. The structure of the salicylamide moiety exerted little effect on anticholinesterase activity, but AChE inhibition increased with spacer elongation. The most active conjugates were salicylimine de

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3

Atlasovich, Fabi�n, Jos� A. Santom�, and Horacio N. Fern�ndez. "Photoreactive fatty acid analogues that bind to the rat liver fatty-acid binding protein: 11-(5?-azido-salicylamido)-undecanoic acid derivatives." Molecular and Cellular Biochemistry 120, no. 1 (1993): 15–23. http://dx.doi.org/10.1007/bf00925980.

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4

Scott, Richard W., Michael J. Costanzo, Katie B. Freeman, et al. "Optimized Fully-Synthetic Salicylamide Heparin Antagonists Have Greater Efficacy Versus LMWHs and Display Improved Hemodynamic Responses as Compared to Protamine." Blood 116, no. 21 (2010): 191. http://dx.doi.org/10.1182/blood.v116.21.191.191.

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Abstract Abstract 191 A series of salicylamides, fully synthetic cationic foldamers designed to disrupt the binding of the pentasaccharide unit of heparin to antithrombin III, were found to be potent neutralizers of the activity of unfractionated heparin (UFH) and low molecular weight heparins (LMWHs). A compound from this series, PMX-60056, is currently in human clinical trials for neutralization of UFH and LMWHs. PMX-60056 potently neutralizes UFH and LMWHs but is not as efficacious versus fondaparinux (FPX). The goal of the present research was to 1) identify back-up compounds to optimize a

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5

Jesaitis, A. J., G. M. Bokoch, J. O. Tolley, and R. A. Allen. "Lateral segregation of neutrophil chemotactic receptors into actin- and fodrin-rich plasma membrane microdomains depleted in guanyl nucleotide regulatory proteins." Journal of Cell Biology 107, no. 3 (1988): 921–28. http://dx.doi.org/10.1083/jcb.107.3.921.

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Subcellular fractions were prepared from human neutrophils desensitized at 15 degrees C with stimulatory doses of the photoaffinity derivative F-Met-Leu-Phe-N epsilon-(2-(rho-azido[125I]salicylamido)ethyl-1,3'- dithio-propionyl)-Lys. The covalently labeled receptors were found in a membrane fraction of higher density than those from cells preexposed to ligand at 4 degrees C but not desensitized. The denser fraction (rho approximately equal to 1.155 g/cc) was the cellular locus of the membrane associated cytoskeletal proteins, actin, and fodrin, as detected immunologically on western blots. The

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6

Farat, Oleg, Svetlana Varenichenko, Ekaterina Zaliznaya, and Victor Markov. "REARRANGEMENT OF SUBSTITUTED 1,3-BENZOXAZINES INTO XANTHENE-TYPE COMPOUNDS." Ukrainian Chemistry Journal 86, no. 2 (2020): 111–22. http://dx.doi.org/10.33609/0041-6045.86.2.2020.111-122.

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The rearrangement patterns of new 1,3-benzoxazines derivatives obtained by condensation of substituted salicylamides with cyclic ketones under the influence of Vilsmeier-Haack reagent has been studied. The influence of angel strain in a 4-membered spirocycle prevents the rearrangement of spiro [1,3-benzoxazine-2,1'-cyclobutan]-4(3H)-one under the action of a formylating agent. 1,3-Benzoxazines derivatives with ring sizes from 5- to 8-membered under the action of a formylating agent have formed formylxanthene derivative. Their formation reaction rate depends on the presence of electronegativity

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7

Pospíšil, Stanislav, Věra Přikrylová, Jan Němeček, and Jaroslav Spížek. "Oxidation and amidation of salicylate by Streptomyces species." Canadian Journal of Microbiology 42, no. 8 (1996): 867–69. http://dx.doi.org/10.1139/m96-111.

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Seven streptomycete strains were tested for biotransformation of salicylate. The products were identified by nuclear magnetic resonance spectroscopy and three types of conversion were found. Streptomyces cinnamonensis and Streptomyces spectabilis formed gentisate and salicylamide concurrently. Streptomyces rimosus transformed salicylate to salicylamide. Streptomyces lividans, Streptomyces coelicolor, Streptomyces griseus and Streptomyces avermitilis produced only gentisate. Time course studies of salicylate conversion by thin-layer chromatography and high pressure liquid chromatography showed

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8

Abdel-Rahman, Mohamed S., Alluru S. Reddi, Frederick A. Curro, Rita M. Turkall, Abdelrazak M. Kadry, and Julia A. Hansrote. "Bioavailability of aspirin and salicylamide following oral co-administration in human volunteers." Canadian Journal of Physiology and Pharmacology 69, no. 10 (1991): 1436–42. http://dx.doi.org/10.1139/y91-215.

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BC® powder (I) is a commercially available analgesic containing the active ingredients aspirin and salicylamide. The kinetics of I, BC® powder minus aspirin (II), and BC® powder minus salicylamide (III) were evaluated in 13 volunteers. Ten minutes after administration of I, aspirin reached a maximum concentration of 12.9 μg/mL, while salicylamide concentration reached a peak value of 3.4 μg/mL. However, when III was administered, aspirin was not detected at 10 min and only reached a concentration of 0.4 μg/mL at 2 and 6 h. Furthermore, the area under the plasma concentration versus time curve

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9

Yao, Shu-Feng, Zhao-Sheng Cai, Xu-Juan Huang, and Lan-Xuan Song. "Preparation of Salicylic Nitrile through Direct Catalytic Dehydration of Salicylamide with Immobilized Phosphoric Acid as Catalyst." Asian Journal of Chemistry 32, no. 5 (2020): 1082–86. http://dx.doi.org/10.14233/ajchem.2020.22545.

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Salicylic nitrile was prepared through direct catalytic dehydration of salicylamide under high temperature using immobilized phosphoric acid as catalyst. The catalytic performances of different catalysts were evaluated according to the analytic results of GC-MS, and the feasibility about the preparation of salicylic nitrile by direct catalytic dehydration of salicylamide was investigated according to the composition of product determinated by GC analysis (area nomalization). Experimental results indicated the comprehensive property of silica gel supported phosphoric acid was the best one among

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10

Zarei, Ali Reza, Abbas Afkhami, and Nahid Sarlak. "Simultaneous Spectrophotometric Determination of Paracetamol and Salicylamide in Human Serum and Pharmaceutical Formulations by a Differential Kinetic Method." Journal of AOAC INTERNATIONAL 88, no. 6 (2005): 1695–701. http://dx.doi.org/10.1093/jaoac/88.6.1695.

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Abstract A rapid, simple, and sensitive differential kinetic method is presented for the determinations of acetaminophen (also known as paracetamol) and salicylamide. The method is based on their oxidation reaction by Fe3+ ion in the presence of 1,10-phenanthroline as indicator. The reactions can be monitored spectrophotometrically by measuring the increase in the absorbance of the solution at 510 nm. Two times were selected one in which only paracetamol is oxidized by Fe3+ ion and the other in which both drugs are oxidized by Fe3+ ion. The data were evaluated by the proportional equations met

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11

Jesaitis, A. J., J. O. Tolley, G. M. Bokoch, and R. A. Allen. "Regulation of chemoattractant receptor interaction with transducing proteins by organizational control in the plasma membrane of human neutrophils." Journal of Cell Biology 109, no. 6 (1989): 2783–90. http://dx.doi.org/10.1083/jcb.109.6.2783.

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Isolated purified plasma membrane domains from unstimulated human neutrophils were photoaffinity labeled with F-Met-Leu-Phe-N epsilon-(2-(p-azido-[125I]salicylamido)ethyl- 1,3'-dithiopropionyl)-Lys also referred to as FMLPL-SASD[125I]. Most of the photoaffinity-labeled N-formyl peptide receptors were found in light plasma membrane fraction (PM-L) which has been previously shown to be enriched in guanyl nucleotide binding proteins and the plasma membrane marker alkaline phosphatase (Jesaitis, A. J., G. M. Bokoch, J. O. Tolley, and R. A. Allen. 1988. J. Cell Biol. 107:921-928). Furthermore, the

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12

&NA;. "Aspirin/caffeine/salicylamide." Reactions Weekly &NA;, no. 1359 (2011): 10. http://dx.doi.org/10.2165/00128415-201113590-00030.

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13

&NA;. "Codeine/paracetamol/salicylamide." Reactions Weekly &NA;, no. 567 (1995): 5. http://dx.doi.org/10.2165/00128415-199505670-00016.

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14

&NA;. "Aspirin/caffeine/salicylamide." Reactions Weekly &NA;, no. 1336 (2011): 9. http://dx.doi.org/10.2165/00128415-201113360-00024.

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15

Jeske, Walter, Aleah Brubaker, Dahui Liu, et al. "In Vitro Characterization of the Neutralization of Unfractionated Heparin and Low Molecular Weight Heparin by Novel Salicylamide Derivatives." Blood 110, no. 11 (2007): 1869. http://dx.doi.org/10.1182/blood.v110.11.1869.1869.

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Abstract Introduction: Unfractionated heparin and the low molecular weight heparins (LMWHs) are commonly used in the treatment of acute coronary syndromes, as prophylaxis against deep vein thrombosis and pulmonary embolism and to prevent clotting during interventional and surgical procedures. The neutralization of unfractionated heparin is critical following the completion of coronary bypass surgery to avoid excessive blood loss. Unfractionated heparin can be neutralized by protamine sulfate, a highly cationic peptide that binds to heparin in a charge-dependent manner. However, the use of prot

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16

Jiang, Ye, Fengshan Zhou, Xiaodong Wen, et al. "Terahertz Absorption Spectroscopy of Benzamide, Acrylamide, Caprolactam, Salicylamide, and Sulfanilamide in the Solid State." Journal of Spectroscopy 2014 (2014): 1–9. http://dx.doi.org/10.1155/2014/732802.

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Terahertz (THz) absorption spectra of the similarly structured molecules with amide groups including benzamide, acrylamide, caprolactam, salicylamide, and sulfanilamide in the solid phase at room temperature and 7.8 K for salicylamide are reported and compared to infrared vibrational spectral calculations using density functional theory. The results of THz absorption spectra show that the molecules have characteristic bands in the region of 0.2–2.6 THz (~7–87 cm−1). THz technique can be used to distinguish different molecules with amide groups. In the THz region benzamide has three bands at 0.

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17

Galal, Alaaeldin M. F., Maha M. Soltan, Esam R. Ahmed, and Atef G. Hanna. "Synthesis and biological evaluation of novel 5-chloro-N-(4-sulfamoylbenzyl) salicylamide derivatives as tubulin polymerization inhibitors." MedChemComm 9, no. 9 (2018): 1511–28. http://dx.doi.org/10.1039/c8md00214b.

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18

Ali, Reham. "Dual Optical Nanosensor Based on Ormosil Nanoparticles for Monitoring O2 and pH." Biosensors 12, no. 11 (2022): 1011. http://dx.doi.org/10.3390/bios12111011.

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Monitoring O2 and pH has excellent potential in different sensing applications, especially in biological and clinical applications. This report presents a protocol for synthesizing an optical dual nanosensor for those two parameters. The organically modified silica (ormosil) nanoparticles were prepared based on phenytrimethoxysilane in an aqueous solution using an acid-base one-pot strategy. Ormosil was selected as a lipophilic matrix for loading fluorescent O2-sensitive dye platinum(II)-tetrakis-(pentafluorophenyl) porphyrin (Pt-TPFPP), which was quenched in the presence of O2 gas and exhibit

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19

Andrews, PR, JM Gulbis, MN Iskander, MF Mackay, C. Dipaola, and M. Sadek. "Structure and Conformations of GABA-Transaminase Inhibitors. IV. Transition State Analogs." Australian Journal of Chemistry 41, no. 4 (1988): 493. http://dx.doi.org/10.1071/ch9880493.

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Crystal structures of three potential inhibitors [salicylamide derivative C16H15NO4 (5), pyridoxazine C11H16N2O5S (6) and benzoxazone C12H13NO4 (7).H2O] of GABA- transaminase (E.C.2.6.1.19, GABA-T) based on the calculated transition state of GABA-T were determined. The conformational analyses of these structures (non-bonded energies, MNDO,AM1) indicate that they can all fit the transition state in relatively low energy conformations. The crystal structures appear to be close to the calculated minimum energy conformations, except for the salicylamide derivative (5), which features internal hydr

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20

&NA;. "Paracetamol/caffeine/salicylamide/promethazine." Reactions Weekly &NA;, no. 1193 (2008): 23. http://dx.doi.org/10.2165/00128415-200811930-00072.

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21

Lei, Ke-Wei, Jian-Li Lin, Xiao-Hui Wen, and Yun-Song Zhou. "N-(3-Pyridylmethyl)salicylamide." Acta Crystallographica Section E Structure Reports Online 63, no. 6 (2007): o3007. http://dx.doi.org/10.1107/s1600536807022969.

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22

&NA;. "Dexamethasone/glycol salicylate/salicylamide." Reactions Weekly &NA;, no. 1432 (2012): 21. http://dx.doi.org/10.2165/00128415-201214320-00071.

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23

Gohel, Sunil Kumar, Vasanthi Palanisamy, Palash Sanphui, Muthuramalingam Prakash, Girij Pal Singh, and Vladimir Chernyshev. "Isostructural cocrystals of metaxalone with improved dissolution characteristics." RSC Advances 11, no. 49 (2021): 30689–700. http://dx.doi.org/10.1039/d1ra05959a.

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Metaxalone forms isostructural cocrystals with nicotinamide and salicylamide that offer a solubility advantage compared to the native drug. A drug–drug homosynthon is retained in all the cocrystal structures.

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24

Surov, Artem O., Katarzyna A. Solanko, Andrew D. Bond, Annette Bauer-Brandl, and German L. Perlovich. "Cocrystals of the antiandrogenic drug bicalutamide: screening, crystal structures, formation thermodynamics and lattice energies." CrystEngComm 18, no. 25 (2016): 4818–29. http://dx.doi.org/10.1039/c6ce00931j.

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Two new cocrystals of the antiandrogenic drug bicalutamide with benzamide and salicylamide are reported. Relationships between crystal structures, melting temperatures, aqueous dissolution, formation thermodynamics and crystal lattice energies of the cocrystals are investigated.

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25

Kakkar, Shubhangi, K. Renuka Devi, Michael Svärd, and Åke Rasmuson. "Crystal nucleation of salicylamide and a comparison with salicylic acid." CrystEngComm 22, no. 19 (2020): 3329–39. http://dx.doi.org/10.1039/d0ce00168f.

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Nucleation behaviour of salicylamide in different solvents was determined and compared with salicylic acid, attempting to progress the rationalization of the influence of the solvent and solute on crystal nucleation of organic compounds in solution.

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26

Jeske, Walter, Christine Schroeder, Margaret Prechel, Jeanine M. Walenga, and Mamdouh Bakhos. "Novel Antagonists for Low Molecular Weight Heparin and Heparin-Like Drugs." Blood 114, no. 22 (2009): 2092. http://dx.doi.org/10.1182/blood.v114.22.2092.2092.

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Abstract Abstract 2092 Poster Board II-69 Unfractionated heparin and other heparin derivatives such as low molecular weight heparins (LMWHs) are used for treatment of coagulation diseases and in surgical applications. Currently neutralization is achieved using protamine sulfate, whose cationic properties allow charge-based binding to heparin. However, protamine is unable to completely reverse LMWH's anticoagulant effects and has potential for side-effects. Our objective was to characterize the ability of a series of salicylamide derivatives (PolyMedix Corp, Radnor, PA) to neutralize the activi

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27

Johnstone, Russell D. L., Alistair R. Lennie, Stewart F. Parker, et al. "High-pressure polymorphism in salicylamide." CrystEngComm 12, no. 4 (2010): 1065. http://dx.doi.org/10.1039/b921288d.

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28

Zuo, Youpeng, Xinwei He, Yi Ning, Lanlan Zhang, Yuhao Wu, and Yongjia Shang. "Divergent synthesis of 3,4-dihydrodibenzo[b,d]furan-1(2H)-ones and isocoumarins via additive-controlled chemoselective C–C or C–N bond cleavage." New Journal of Chemistry 42, no. 3 (2018): 1673–81. http://dx.doi.org/10.1039/c7nj03799f.

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29

Gondolova, Gulnar H. "SYNTHESIS AND STUDY OF Zn COMPLEXES WITH N'-ACYL-SALICYLHYDRAZIDES." IZVESTIYA VYSSHIKH UCHEBNYKH ZAVEDENII KHIMIYA KHIMICHESKAYA TEKHNOLOGIYA 62, no. 9 (2019): 27–32. http://dx.doi.org/10.6060/ivkkt.20196209.5902.

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Zn complexes with potentially tridentate (carbonyl and hydroxyl oxygen atoms of the salicylic fragment and nitrogen atom of the amide group) were synthesized by the ligand N'-phthalimido-salicylamide (H2L) and potentially heptadentate (carbonyl and hydroxyl oxygen atoms of the salicylic fragment, two nitrogen atoms of the hydrazide moiety and two oxygen atoms of the carbonyl and carboxyl groups of the maleic fragment) with the ligand N'-maleoal-salicylhydrazide (H4L) with 78% and 86% yield, respectively. The structural features of the N'-phthalimido-salicylamide (H2L) and N'-maleoyl-salicylhyd

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30

Xin, Zhi Jun, Zhong Jia, Dian He, et al. "Study on N-(pyridin-4-Yl) Salicylamides as Antimycobacterial Agents." Advanced Materials Research 634-638 (January 2013): 1371–75. http://dx.doi.org/10.4028/www.scientific.net/amr.634-638.1371.

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A series of N-(pyridin-4-yl) salicylamides derivatives were prepared through acylation of the corresponding acetylsalicyloyl chlorides with substituted 4-amino-pyridines. These compounds were evaluated in vitro for antimycobacterial activities against Mycobacterium tuberculosis (TB) and Mycobacterium avium (A) by the minimum inhibitory concentrations (MIC) values. Eight of the compounds exhibited lower MIC against A than isoniazide (INH). Meanwhile, four of the compounds exhibited good anti-TB activity, when they were compared with INH. Antimycobacterial activities of N-(pyridin-4-yl) salicyla

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31

Fielding, R. M., J. A. Waschek, D. J. Effeney, A. C. Pogany, S. M. Pond, and T. N. Tozer. "Extrahepatic extraction of salicylamide in dogs." Journal of Pharmacology and Experimental Therapeutics 236, no. 1 (1986): 97–102. https://doi.org/10.1016/s0022-3565(25)38822-1.

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32

Yu, Kuo-Long, Edward Ruediger, Guangxiang Luo, et al. "Novel quinolizidine salicylamide influenza fusion inhibitors." Bioorganic & Medicinal Chemistry Letters 9, no. 15 (1999): 2177–80. http://dx.doi.org/10.1016/s0960-894x(99)00361-3.

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33

Combrink, Keith D., H. Belgin Gulgeze, Kuo-Long Yu, et al. "Salicylamide inhibitors of influenza virus fusion." Bioorganic & Medicinal Chemistry Letters 10, no. 15 (2000): 1649–52. http://dx.doi.org/10.1016/s0960-894x(00)00335-8.

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34

Aisling, Lynch, and Rasmuson Åke. "Crystal Growth of Single Salicylamide Crystals." Crystal Growth & Design 19, no. 12 (2019): 7230–39. http://dx.doi.org/10.1021/acs.cgd.9b01101.

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35

Nordström, Fredrik L., and Åke C. Rasmuson. "Solubility and Melting Properties of Salicylamide." Journal of Chemical & Engineering Data 51, no. 5 (2006): 1775–77. http://dx.doi.org/10.1021/je060178m.

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36

Ribeiro da Silva, Maria D. M. C., and Nuno R. M. Araújo. "Thermochemical studies on salicylaldehyde and salicylamide." Journal of Chemical Thermodynamics 39, no. 10 (2007): 1372–76. http://dx.doi.org/10.1016/j.jct.2007.03.006.

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37

Howell, Stanley R., Lois A. Kotkoskie, Russell L. Dills, and Curtis D. Klaassen. "3-Hydroxylation of Salicylamide in Mice." Journal of Pharmaceutical Sciences 77, no. 4 (1988): 309–13. http://dx.doi.org/10.1002/jps.2600770405.

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38

Isadiartuti, Dewi, Bambang Widjaja, Hendra Wijaya, and Maria Lucia Ardhani Dwi Lestari. "Solubility and Dissolution Study of Salicylamide." Berkala Ilmiah Kimia Farmasi 9, no. 2 (2022): 40–44. http://dx.doi.org/10.20473/bikfar.v9i2.42706.

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Salisilamida termasuk golongan obat AINS (anti inflamasi non steroid)memiliki efek analgesik dan antipiretik mirip dengan asam asetil salisilat, namun di dalam tubuh tidak diubah menjadi salisilat. Dalam penggunaan secara oral,salisilamida tidak menimbulkan radang dan pendarahan pada lambung. Salisilamida merupakan senyawaasam lemah (pKa 8,2) yang kelarutannya dipengaruhi oleh pH lingkungan. Pada pemberian secara oral, salisilamida akan melewati saluran cerna pada rentang pH sekitar 1,5–8,0. Menurut persamaan Noyes-Whitney, disolusi obat akan dipengaruhi oleh kelarutannya. Tujuan penelitian in

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39

Berner, Joachim, Heinz Böhland, Manfred Werner, and Thomas Richter. "Diacetato-bis(salicylamid)-kupfer (II)-Verbindungen." Zeitschrift für Chemie 27, no. 2 (2010): 61–62. http://dx.doi.org/10.1002/zfch.19870270205.

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40

Kusumoto, Sotaro, Fumiya Kobayashi, Ryo Ohtani, et al. "Creating capsules with cubanes." Dalton Transactions 47, no. 29 (2018): 9575–78. http://dx.doi.org/10.1039/c8dt01911h.

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41

Torregrosa-Chinillach, Alejandro, Alba Sánchez-Laó, Elisa Santagostino, and Rafael Chinchilla. "Organocatalytic Asymmetric Conjugate Addition of Aldehydes to Maleimides and Nitroalkenes in Deep Eutectic Solvents." Molecules 24, no. 22 (2019): 4058. http://dx.doi.org/10.3390/molecules24224058.

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A chiral primary amine-salicylamide is used as an organocatalyst for the enantioselective conjugate addition of α,α-disubstituted aldehydes to maleimides and nitroalkenes. The reactions are performed in deep eutectic solvents as reaction media at room temperature, leading to the corresponding adducts with enantioselectivities up to 88% (for maleimides) and 80% (for nitroalkenes). Catalyst and solvent can be recovered and reused.

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42

Isadiartuti, Dewi, Noorma Rosita, Esti Hendradi, Firdausiah Fania Dwi Putri Putri, and Frida Magdalena. "Solubility and Partition Coefficient of Salicylamide in Various pH Buffer Solutions." Indonesian Journal of Chemistry 21, no. 5 (2021): 1263. http://dx.doi.org/10.22146/ijc.66411.

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The solubility and partition coefficient are essential physicochemical parameters in developing a pharmaceutical dosage form of medicine. In addition, these parameters help to predict the absorption of an active compound in oral or topical dosage forms. Salicylamide, an active ingredient available in oral and topical dosage forms, is a weak acid (pKa 8.2) and is sparingly soluble in water. Meanwhile, its solubility and partition coefficients are influenced by the pH of the environment. The Henderson-Hasselbalch equation is used to predict solubility-pH and partition-pH profiles at various pH s

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43

Jia, Zhong, Dian He, Jian Ping Liang, et al. "Efficient Synthesis of N-(pyridin-4-yl) Salicylamide Derivatives." Advanced Materials Research 803 (September 2013): 72–75. http://dx.doi.org/10.4028/www.scientific.net/amr.803.72.

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A series of N-(pyridin-4-yl) salicylamides derivatives were prepared through acylation of the corresponding acetylsalicyloyl chlorides with substituted 4-amino-pyridines. These compounds might serve as prospective wide-spectrum antimycobacterial substances.

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Torregrosa-Chinillach, Alejandro, Adrien Moragues, Haritz Pérez-Furundarena, Rafael Chinchilla, Enrique Gómez-Bengoa, and Gabriela Guillena. "Enantioselective Michael Addition of Aldehydes to Maleimides Organocatalyzed by a Chiral Primary Amine-Salicylamide." Molecules 23, no. 12 (2018): 3299. http://dx.doi.org/10.3390/molecules23123299.

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A primary amine-salicylamide derived from chiral trans-cyclohexane-1,2-diamine was used as an organocatalyst for the enantioselective conjugate addition of aldehydes, mainly α,α-disubstituted to N-substituted maleimides. The reaction was performed in toluene as a solvent at room temperature. The corresponding enantioenriched adducts were obtained with high yields and enantioselectivities up to 94%. Theoretical calculations were used to justify the stereoinduction.

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El Kheir, Afaf Abou, Saied F. Belal, and Abdulla El Shanwani. "Spectrophotometric Analysis of Mixtures of Acetaminophen, Salicylamide, and Codeine Phosphate in Tablets." Journal of AOAC INTERNATIONAL 68, no. 5 (1985): 1048–50. http://dx.doi.org/10.1093/jaoac/68.5.1048.

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Abstract A simple and accurate spectrophotometric procedure for the analysis of a mixture of acetaminophen, salicylamide, and codeine phosphate is described. Determination of the first 2 components depends on pHinduced differential spectral changes of their nitroso derivatives. The third component is assayed by the acid dye method. The proposed procedure was successfully applied to the analysis of laboratory-made and commercial tablets containing the ternary drug mixture

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Torregrosa-Chinillach, Alejandro, and Rafael Chinchilla. "Asymmetric Conjugate Addition of Ketones to Maleimides Organocatalyzed by a Chiral Primary Amine-Salicylamide." Molecules 27, no. 19 (2022): 6668. http://dx.doi.org/10.3390/molecules27196668.

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Enantioenriched substituted succinimides are interesting compounds, and their asymmetric organocatalytic synthesis by the conjugated addition of ketones to maleimides has been scarcely explored. This study shows the enantioselective conjugate addition of ketones to maleimides organocatalyzed by a simple primary amine-salicylamide derived from a chiral trans-cyclohexane-1,2-diamine, which provides the desired succinimides in good to excellent yields (up to 98%) and with moderate to excellent enantioselectivities (up to 99%).

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Pudjiastuti, Pratiwi, Siti Wafiroh, Esti Hendradi, et al. "Disintegration, In vitro Dissolution, and Drug Release Kinetics Profiles of k-Carrageenan-based Nutraceutical Hard-shell Capsules Containing Salicylamide." Open Chemistry 18, no. 1 (2020): 226–31. http://dx.doi.org/10.1515/chem-2020-0028.

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AbstractThe release of drugs from solid drug delivery materials has been studied intently in recent years. Quantitative analyses achieved from in vitro dissolution becomes easier if a zero-order mathematical model is used. Non-gelatin nutraceutical hard-shell capsules of zero size (approximately 0.7-0.8 cm) were produced from carrageenan-based natural polymers, namely carrageenan-alginate (CA) and carrageenan-starch (CS). Disintegration, dissolution and zero-order drug release kinetics of hard-shell capsules containing 100 mg of salicylamide were studied. The disintegration time of CA and CS w

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Abdallah, El, C. Si-Moussa, S. Hanini, and M. Laidi. "Application of PC-SAFT and cubic equations of state for the correlation of solubility of some pharmaceutical and statin drugs in SC-CO2." Chemical Industry and Chemical Engineering Quarterly 19, no. 3 (2013): 449–60. http://dx.doi.org/10.2298/ciceq120407005e.

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In this work, the solubilities of some anti-inflammatory (nabumetone, phenylbutazone and salicylamide) and statin drugs (fluvastatin, atorvastatin, lovastatin, simvastatin and rosuvastatin) were correlated using the Perturbed-Chain Statistical Associating Fluid Theory (PC-SAFT) with one-parameter mixing rule and commonly used cubic equations of state Peng-Robinson (PR) and Soave-Redlich-Kwong (SRK) combining with van-der Waals-1 parameter (VDW1) and van-der Waals-2 parameters (VDW2) mixing rules. The experimental data for studied compounds were taken from literature at temperature and pressure

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KUSHIYA, MAMI, RYUICHI HASEGAWA, TETSUO KOMURO, and HIROSHI ISAKA. "Depression of salicylamide glucuronidation by bacterial lipopolysaccharide." CHEMICAL & PHARMACEUTICAL BULLETIN 35, no. 1 (1987): 416–20. http://dx.doi.org/10.1248/cpb.35.416.

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Fuster Mestre, Y., L. Lahuerta Zamora, and J. Martı́nez Calatayud. "Direct flow injection chemiluminescence determination of salicylamide." Analytica Chimica Acta 394, no. 2-3 (1999): 159–63. http://dx.doi.org/10.1016/s0003-2670(99)00290-1.

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