Relevant bibliographies by topics / 2-a]pyridine analogues

Contents

  1. Journal articles
  2. Dissertations / Theses
  3. Conference papers

Academic literature on the topic '2-a]pyridine analogues'

Author: Grafiati
Published: 4 June 2021
Last updated: 5 February 2022

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic '2-a]pyridine analogues.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "2-a]pyridine analogues"

1

Schmitt, Martine, Jean-Jacques Bourguignon, Gordon B. Barlin, and Les P. Davies. "Imidazo[1,2-b]pyridazines. XXIII Some 5-Deaza Analogues. Syntheses of Some 2-Aryl-6-(chloro, methoxy or unsubstituted)-3- (variously substituted)imidazo[1,2-a]pyridines and Their Affinity for Central and Mitochondrial Benzodiazepine Receptor." Australian Journal of Chemistry 50, no. 7 (1997): 719. http://dx.doi.org/10.1071/c97004.

Full text
Abstract:
The syntheses of ethyl {2′-aryl-6′-(chloro, methoxy and unsubstituted)imidazo[1,2-a]pyridin-3′-yl}-2- (acylamino, acetoxy and hydroxy)acetates, 3-benzamidomethyl-2-benzoyl-6-(chloro and methoxy)imidazo-[1,2-a]pyridines, 3-amino-6-chloro-2-phenylimidazo[1,2-a]pyridine and ethyl 2-(2′-phenylimidazo[1,2-a]pyridin-3′-yl)acetate are reported. The ability of these compounds to displace [3H]diazepam from central and mitochondrial (peripheral-type) benzodiazepine receptors has been examined. Ethyl 2-benzamido-2-{6′-chloro-2′-(4′′-chlorophenyl)imidazo[1,2-a]pyridin-3′-yl} acetate (21) was selective for
APA, Harvard, Vancouver, ISO, and other styles
2

Maskey, Rajendra P., Felix Huth, Iris Grün-Wollny, and Hartmut Laatsch. "2-Alkyl-3,4-dihydroxy-5-hydroxymethylpyridine Derivatives: New Natural Vitamin B6 Analogues from a Terrestrial Streptomyces sp." Zeitschrift für Naturforschung B 60, no. 1 (2005): 63–66. http://dx.doi.org/10.1515/znb-2005-0110.

Full text
Abstract:
The ethyl acetate extract of the strain Streptomyces sp. GW23/1540 has yielded four new 2-alkyl-5-(hydroxymethyl)pyridine-3,4-diols, 5-hydroxymethyl-2-isopropyl-pyridine-3,4-diol (1a), 5-hydroxymethyl-2-propyl-pyridine-3,4-diol (1b), 2-sec-butyl-5-hydroxymethyl-pyridine-3,4-diol (1c), and 5-hydroxymethyl-2-isobutyl-pyridine-3,4-diol (1d). Similarly, the strain Streptomyces sp. GW63/1571 afforded 2-sec-butyl-5-hydroxymethyl-pyridine-3,4-diol (1c) and another new natural product, (3aS, 7aR)-3a-hydroxy-3a,4,7,7a-tetrahydro-1-benzofuran-2(3H)-on e (3), together with anthranilic acid, anthranilamid
APA, Harvard, Vancouver, ISO, and other styles
3

Shilin, S., Z. Voitenko, and M. Nechai. "SYNTHETIC PYRIDINE SUBSTITUTED AMINO ACIDS AND THEIR DERIVATIVES." Bulletin of Taras Shevchenko National University of Kyiv. Chemistry, no. 1(56) (2019): 22–25. http://dx.doi.org/10.17721/1728-2209.2019.1(56).5.

Full text
Abstract:
This paper reports on the synthesis of new derivatives of ε-aminocaproic and γ-aminobutyric acid modified with a pyridin-2-yl substituent at the ω-position of the main chain. The hemostatic activity of both ε-aminocaproic acid itself and its various synthetic analogues is widely known. Likewise, numerous γ-aminobutyric acid derivatives are strong neurotransmitters extensively used in the treatment of the nervous system disorders. No less popular are biologically active substances containing a pyridine or piperidine fragment; among which there are antibiotics, antimalarial, anti-sclerotic and a
APA, Harvard, Vancouver, ISO, and other styles
4

Majamaa, K., T. M. Turpeenniemi-Hujanen, P. Latipää, et al. "Differences between collagen hydroxylases and 2-oxoglutarate dehydrogenase in their inhibition by structural analogues of 2-oxoglutarate." Biochemical Journal 229, no. 1 (1985): 127–33. http://dx.doi.org/10.1042/bj2290127.

Full text
Abstract:
Inhibition of lysyl hydroxylase and prolyl 3-hydroxylase was studied with 23 selected aromatic and aliphatic structural analogues of 2-oxoglutarate and the results were compared with those previously reported for prolyl 4-hydroxylase. All the compounds inhibited the hydroxylases competitively with respect to 2-oxoglutarate and noncompetitively with respect to Fe2+ and the peptide substrate. The inhibition patterns for the three collagen hydroxylases were basically similar, but certain differences in detail emerged. One systematic difference was that lysyl hydroxylase had a higher Ki for almost
APA, Harvard, Vancouver, ISO, and other styles
5

Patel, Navin, Sabir Pathan, and Hetal I. Soni. "3,4-Dihydropyrimidin-2(1H)-One Analogues: Microwave irradiated Synthesis with Antimicrobial and Antituberculosis Study." Current Microwave Chemistry 6, no. 1 (2019): 61–70. http://dx.doi.org/10.2174/2213335606666190724093305.

Full text
Abstract:
Background: For rapid and sustainable synthesis, microwave irradiation method is serviceable. This present study deals with the preparation of oxadiazole and pyridine bearing 1,2,3,4- tetrahydro pyrimidine derivatives by microwave irradiation. Objective: The present study aims to carry out rapid synthesis of chloro-acetamides of oxadiazoles of Biginelli product and amino cyano derivative of pyridine by microwave-assisted heating. Our efforts are focused on the introduction of chemical diversity in the molecular framework in order to synthesize pharmacologically interesting compounds. Methods::
APA, Harvard, Vancouver, ISO, and other styles
6

SLEATH, P. R., A. L. HANDLON, and N. J. OPPENHEIMER. "ChemInform Abstract: Pyridine Coenzyme Analogues. Part 3. Synthesis of Three NAD+ Analogues Containing a 2′-Deoxy-2′-Substituted Nicotinamide Arabinofuranosyl Moiety." ChemInform 22, no. 41 (2010): no. http://dx.doi.org/10.1002/chin.199141250.

Full text
APA, Harvard, Vancouver, ISO, and other styles
7

Kutniewska, Sylwia E., Katarzyna N. Jarzembska, Radosław Kamiński, Anton J. Stasyuk, Daniel T. Gryko, and Michał K. Cyrański. "Structural, energetic and spectroscopic studies of new luminescent complexes based on 2-(2′-hydroxyphenyl)imidazo[1,2-a]pyridines and 1,2-phenylenediboronic acid." Acta Crystallographica Section B Structural Science, Crystal Engineering and Materials 74, no. 6 (2018): 725–37. http://dx.doi.org/10.1107/s2052520618015469.

Full text
Abstract:
Three new blue-luminescent complexes of selected imidazo[1,2-a]pyridine derivatives and 1,2-phenylenediboronic acid have been synthesized and structurally characterized using single-crystal X-ray diffraction. Additionally, the crystal structures of two of the (N,O)-donor compounds have been evaluated for the first time. The crystal packing and molecular motifs observed in the studied crystals have been thoroughly analysed, including computational studies, and are also discussed within the context of analogous systems reported in the literature. It appears that the new compounds form different
APA, Harvard, Vancouver, ISO, and other styles
8

Lin, Nan-Horng, Yihong Li, Yun He, et al. "Synthesis and structure–activity relationships of 5-substituted pyridine analogues of 3-[2-((S)-pyrrolidinyl)methoxy]pyridine, A-84543." Bioorganic & Medicinal Chemistry Letters 11, no. 5 (2001): 631–33. http://dx.doi.org/10.1016/s0960-894x(01)00030-0.

Full text
APA, Harvard, Vancouver, ISO, and other styles
9

Ginocchietti, Gabriella, Ugo Mazzucato, and Anna Spalletti. "Protonation effect on the excited state behaviour of some aza-analogues ofEE-distyrylbenzene." International Journal of Photoenergy 6, no. 4 (2004): 241–50. http://dx.doi.org/10.1155/s1110662x04000315.

Full text
Abstract:
The photobehaviour of four aza-analogues ofEE-distyrylbenzene bearing the heteroatom in the two side rings [1,4-di-(2-pyridylethenyl)benzene] or in the central ring [2,5-di-(phenylethenyl)pyridine, 2,6-di(phenylethenyl)pyridine and the corresponding diene, 2,6-di(phenylbutadienyl)pyridine] has been investigated in aqueous solutions at pH 2 and 9, where the molecules are in mono-protonated and neutral forms, respectively. The type of conjugation, linear for the first two compounds and crossed for the others, is particularly important in determining the spectral and photochemical properties. The
APA, Harvard, Vancouver, ISO, and other styles
10

Boyode, B. P., M. Sinet, A. Farese, et al. "Synthesis and Antiviral Evaluation of Fluorinated Dipyridodiazepinones and Dipyridodiazepines (Nevirapine Derivatives)." Antiviral Chemistry and Chemotherapy 6, no. 3 (1995): 162–68. http://dx.doi.org/10.1177/095632029500600305.

Full text
Abstract:
The synthesis of trifluoromethyldipyridodiazepinones, which are analogues of nevirapine, one of the non-nucleoside inhibitors of the HIV-1 RT enzyme, is described. The condensation of 3-amino-2-chloro-4-tri-fluoromethyl pyridine with 2-chloronicotinoyl chloride followed by a cyclization with cyclopropylamine provided the corresponding trifluoromethylated dipyridodiazepinone. Similarly, the dipyridodiazepine analogues were synthesized by condensation of 3-amino-2-chloro-4-trifluoromethylpyridine with the O-mesyl derivative of 2-chloro-3-pyridincarbinol followed by reaction with cyclopropylamine
APA, Harvard, Vancouver, ISO, and other styles
More sources

Dissertations / Theses on the topic "2-a]pyridine analogues"

1

Nicolaÿ, Jean-François. "Synthèse asymétrique d'alcaloides pipéridiniques, composés analogues des coccinellines et de l'anatoxine-A." Paris 11, 1989. http://www.theses.fr/1989PA112365.

Full text
Abstract:
Une méthode générale de synthèse asymétrique d'alcaloides piperidiniques a récemment été mise au point dans notre laboratoire. Elle repose sur la préparation d'un synthon chiral équivalent réactionnel de dihydro-1,4-pyridine. Cette méthode a été appliquée à la synthèse d'alcaloides extraits des secrétions de coccinelles et possédant une structure perhydroazaphénalène. Plusieurs composes analogues, enantiomériquement purs, ont ete obtenus. La préparation de composes tricycliques, par ailleurs également précurseurs potentiels d'alcaloides de type poranthéridine, a été effectuée. Enfin, la synthè
APA, Harvard, Vancouver, ISO, and other styles
2

Nordqvist, Anneli. "Hit Identification and Hit Expansion in Antituberculosis Drug Discovery : Design and Synthesis of Glutamine Synthetase and 1-Deoxy-D-Xylulose-5-Phosphate Reductoisomerase Inhibitors." Doctoral thesis, Uppsala universitet, Avdelningen för organisk farmaceutisk kemi, 2011. http://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-155428.

Full text
Abstract:
Since the discovery of Mycobacterium tuberculosis (Mtb) as the bacterial agent causing tuberculosis, the permanent eradication of this disease has proven challenging. Although a number of drugs exist for the treatment of tuberculosis, 1.7 million people still die every year from this infection. The current treatment regimen involves lengthy combination therapy with four different drugs in an effort to combat the development of resistance. However, multidrug-resistant and extensively drug-resistant strains are emerging in all parts of the world. Therefore, new drugs effective in the treatment o
APA, Harvard, Vancouver, ISO, and other styles
3

Chaulet, Charlotte. "Synthèse et étude du mécanisme d'action de nouveaux analogues de la thalidomide, dérivés du noyau 1H-pyrrolo (2, 3-b) pyridine, sur la modulation des cellules NK et la production des cytokines TNF-a et IL-6." Thesis, Tours, 2010. http://www.theses.fr/2010TOUR3802/document.

Full text
Abstract:
La thalidomide est un sédatif hypnotique mis sur le marché pour la première fois en Allemagne en octobre 1957 et largement vendu par la suite dans 46 pays sous 51 noms commerciaux différents. Il fut également utilisé comme antiémétique chez les femmes enceintes et, dès le jour de Noël de l’année 1956, un premier enfant atteint de phocomélie naissait, six mois avant la mise sur le marché. La thalidomide fut retirée de la vente fin 1961, du fait de ses effets dévastateurs sur le développement fœtal. De nombreux mécanismes d’action de la thalidomide dans l’embryopathie ont été rapportés, notammen
APA, Harvard, Vancouver, ISO, and other styles
4

Jourdan, Fabrice. "Synthèse, études physicochimique et pharmacologique d'inhibiteurs potentiels de la transcriptase inverse comprenant différents analogues de nucléosides cycliques et acycliques thiéno et dihydrothiénopyrimidiniques, différentes pyridin-2-ones et pyrido[3,2-ƒ]pyrollo[1,2-a]diazépines." Caen, 1996. http://www.theses.fr/1996CAEN4018.

Full text
APA, Harvard, Vancouver, ISO, and other styles

Conference papers on the topic "2-a]pyridine analogues"

1

Hussein, Ola, Feras Alali, Ala-Eddin Al Moustafa, and Ashraf Khalil. "Design, Synthesis and Biological Evaluation of Novel Chalcone Analogs as Potential Therapeutic Agents for Castration-Resistant Prostate Cancer." In Qatar University Annual Research Forum & Exhibition. Qatar University Press, 2020. http://dx.doi.org/10.29117/quarfe.2020.0179.

Full text
Abstract:
Prostate cancer (PCa) is the second most frequently diagnosed malignancy, as well as a leading cause of cancer-related mortality in men globally. Despite the initial response to hormonal targeted therapy, the majority of patients ultimately progress to a lethal form of the disease, termed as castration-resistant prostate cancer (CRPC), which currently lacks curative therapeutic options and is associated with poor prognosis. Therefore, the development of novel treatment modalities for PCa is urgently needed. Chalcones, also known as 1,3-diphenyl-2-propen-1-ones, are among the highly attractive
APA, Harvard, Vancouver, ISO, and other styles
2

Montaño, Rocío, and Murali Venkata Unnamatla. "Efficient and rapid conversion of 3-amino imidazo[1,2-a] pyridin-2-yl)-4H-chromene-4-ones to its corresponding thio analogues using Lawesson’s reagent ." In The 22nd International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2018. http://dx.doi.org/10.3390/ecsoc-22-05668.

Full text
APA, Harvard, Vancouver, ISO, and other styles
You might also be interested in the extended bibliographies on the topic '2-a]pyridine analogues' for particular source types:
Journal articles
We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!

To the bibliography