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Journal articles on the topic '2-amino benzamide'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Kushwaha, Mr Abhay, Dr Shailesh Jain, Mr Ajay Kumar, Mr Ritesh Raj, Dr Phool Singh Yaduwanshi, and Dr Dhanraj Patidar. "An Overall Review of Different Derivatives That Activate Glucokinase Enzyme Having Multiple Actions to Treat Type 2 Diabetes." International Journal of Pharmaceutical Research and Applications 10, no. 1 (2025): 358–67. https://doi.org/10.35629/4494-1001358367.

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Different derivatives like3,6-disubstituted2- pyridine carboxamide derivatives, Phenylethyl benzamide derivatives, Carboxypyridine benzamide derivatives, Pyrazole benzamide derivatives, Quinazoline-2,4 dione analogs, Ketopiperazine analogs, Cycloalkyl-fused Nthiazol-2-yl-benzamides derivatives, 1,4- disubstituted indazoles derivatives, 2,5,6- trisubstituted indole derivatives, Azaindole derivatives andPyrimidone derivatives was designed, synthesized and evaluated the pharmacological activity in mice. Such compounds activate the glucokinase by interaction between glucokinase activators and gluc

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2

Journal, Baghdad Science. "Synthesis of New Amide and ThioUrease Compounds." Baghdad Science Journal 4, no. 3 (2007): 430–37. http://dx.doi.org/10.21123/bsj.4.3.430-437.

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The reaction of some new Schiff bases ( 2-[(2-Amino – ethylimino)-methyl]-R , 2-({2-[(R-benzylidene)-amino]-ethylimino}-methyl)-R with Benzoyl chloride or Acetyl chloride were carried out. Subsequent reactions of these products N-(2-Amino-ethyl)-N-[Chloro-(R) –methyl]-benzamide or N-(2-{?-[chloro-(R) –methyl]-amino}-ethyl)-N-[chloro-(R) –methyl]- benzamide with thiourea afforded thioureas compounds. The synthesized compounds were confirmed by their IR,UV,spectra and C.H.N. analysis.

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3

Garg, Ajay Kumar, Ranjan Kumar Singh, Vaibhav Saxena, Saurabh Kr Sinha, and Sanjay Rao. "Synthesis, Characterization, and Anti-inflammatory activity of Some Novel Oxazole Derivatives." Journal of Drug Delivery and Therapeutics 13, no. 1 (2023): 26–28. http://dx.doi.org/10.22270/jddt.v13i1.5719.

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A series of novel oxazole derivatives (A, A1, A2) were synthesized starting from acetone and urea. The compound (A) was obtained by heating it with acetophenone and urea in iodine. Compound (A) on treatment with 4-amino benzaldehyde (Z)-N-(4-amino benzylidine)-4-((E)-Penta-2, 4-diene-2) oxazole-2-amine afforded (A1). Acylation of compound (A) with 4-amino benzoyl chloride to obtain the corresponding N-(4 phenyl oxazole-2- yl)- benzamide (A2). The structures of compounds have been established employing FTIR and 1H-NMR spectral analysis. All oxazole derivatives were evaluated for anti-inflammato

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4

Pokotylo, Ihor O., Pavlo V. Zadorozhnii, Vadym V. Kiselev, Oxana V. Okhtina, and Aleksandr V. Kharchenko. "Some New Heterocyclisations Based on N-(2,2-dichloro-1-isothiocyanatoethyl)benzamide Derivatives." Acta Chemica Iasi 27, no. 1 (2019): 65–72. http://dx.doi.org/10.2478/achi-2019-0005.

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Abstract Based on the readily available N-(2,2-dichloro-1-(2-(4-methylbenzoyl)-hydrazine-1-carbothioamido)ethyl)benzamide, the corresponding N-(2,2-dichloro-1-((5-(p-tolyl)-1,3,4-oxadiazol-2-yl)amino)ethyl)benzamide and 5-(p-tolyl)-1,3,4-thiadiazol-2-amine were obtained. The products were received in acceptable yields and were isolated from the reaction mixture without any particular difficulty. The structure of the compounds obtained was confirmed by 1H, 13C NMR spectroscopy and mass spectrometry data.

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5

Selvakumaran, N., R. Karvembu, Seik Weng Ng, and Edward R. T. Tiekink. "3-({[Bis(2-methylpropyl)carbamothioyl]amino}carbonyl)benzamide." Acta Crystallographica Section E Structure Reports Online 69, no. 7 (2013): o1183. http://dx.doi.org/10.1107/s1600536813017455.

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6

Gaston, Lewis A., Martin A. Locke, Steven C. Wagner, Robert M. Zablotowicz, and Krishna N. Reddy. "Sorption of Bentazon and Degradation Products in Two Mississippi Soils." Weed Science 44, no. 3 (1996): 678–82. http://dx.doi.org/10.1017/s0043174500094522.

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Bentazon degradation in soil typically proceeds with development of bound residue. Low sorption of bentazon suggests that this residue consists of degradation products; however, there is little data on the sorption behavior of these products. This study was undertaken to determine the sorption of bentazon and the degradation products 2-amino-N-isopropyl benzamide, 2-aminobenzoic acid, andN-methyl bentazon in Dundee silt loam and Sharkey clay, two common agricultural soils of the Mississippi Delta. Greater sorption of bentazon and degradation products in the Sharkey soil was related to finer te

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7

Konovalova, S. A., A. P. Avdeenko, V. I. Lubenets, O. Z. Komarovska-Porokhnyavets, I. Yu Yakymenko, and E. N. Lysenko. "BIOLOGICAL ACTIVITY OF N-{3-[(4-METHYLBENZENE-1- SULFONYL)IMINO]-6-OXOCYCLOHEXA-1,4-DIEN-1-YL}ARYLAMIDES AND THEIR DERIVATIVES." Odesa National University Herald. Chemistry 26, no. 1(77) (2021): 37–47. http://dx.doi.org/10.18524/2304-0947.2021.1(77).226136.

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N-{3-[(4-Methylbenzene-1-sulfonyl)imino]-6-oxocyclohexa-1,4-dien-1-yl}arylamides and their derivatives were synthesized by the reaction of the corresponding N-(4-oxocyclohexa-2,5-dien-1-ylidene)arylsulfonamides with N-chloramides. The biological activity of the synthesized compounds was studied on test cultures of Escherichia coli 67, Staphylococcus aureus 209-p, Mycobacterium luteum VKM B-868 and fungi Candida tenuis VKM Y-70, Aspergillus niger VKM F-1119 by the method of diffusion of substances into agar on a solid nutrient medium. The degree of activity of the test compounds was determined

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8

Belz, Tyson, Saleh Ihmaid, Jasim Al-Rawi, and Steve Petrovski. "Synthesis Characterization and Antibacterial, Antifungal Activity of N-(Benzyl Carbamoyl or Carbamothioyl)-2-hydroxy Substituted Benzamide and 2-Benzyl Amino-Substituted Benzoxazines." International Journal of Medicinal Chemistry 2013 (October 31, 2013): 1–20. http://dx.doi.org/10.1155/2013/436397.

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New N-(benzyl carbamothioyl)-2-hydroxy substituted benzamides 13, 20, and 21 were synthesized using sodium bicarbonate and benzyl amine with 2-thioxo-substituted-1,3-benzoxazines 6, 10a, b, 11c, and 12a–n. The 2-thioxo-substituted-1,3-oxazines 6, 10a-b, 11d 12a–n, and 26 were converted to the corresponding 2-methylthio-substituted-1,3-oxazines 14a–l and 24 which were then converted to 2-benzyl amino-substituted-benzoxazines 15a–i by refluxing with benzylamine. Products 15a, b, e, f, and g were also synthesized by boiling the corresponding N-(benzyl carbamothioyl)-2-hydroxy substituted benzamid

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9

Zhang, Yan, Jian-Quan Liu, and Xiang-Shan Wang. "An efficient synthesis of 16H-dibenzo[2,3:6,7][1,4]oxazepino[5,4-b]quinazolin-16-ones via an Ullmann reaction catalyzed by CuI." Organic & Biomolecular Chemistry 16, no. 10 (2018): 1679–85. http://dx.doi.org/10.1039/c8ob00005k.

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16H-Dibenzo[2,3:6,7][1,4]oxazepino[5,4-b]quinazolin-16-ones were obtained from the available reactants 2-amino-N-(2-hydroxyphenyl)benzamide and 2-bromobenzaldehyde via an Ullmann reaction catalyzed by CuI.

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Haller, Joseph P., Warunee Thaenghin, Wannipa Un-chai, and Kenneth J. Haller. "Inductive and supramolecular effects in 2-amino-N-(2-hydroxyphenyl)benzamide." Acta Crystallographica Section A Foundations and Advances 73, a2 (2017): C685. http://dx.doi.org/10.1107/s205327331708888x.

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11

Balewski, Łukasz, and Anita Kornicka. "Synthesis of the Guanidine Derivative: N-{[(7-(4,5-Dihydro-1H-imidazol-2-yl)-2-(p-tolyl)-6,7-dihydro-2H-imidazo[2,1-c][1,2,4]triazol-3(5H)-ylidene)amino](phenylamino)methylene}benzamide." Molbank 2021, no. 3 (2021): M1246. http://dx.doi.org/10.3390/m1246.

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The guanidine derivative N-{[(7-(4,5-dihydro-1H-imidazol-2-yl)-2-(p-tolyl)-6,7-dihydro-2H-imidazo[2,1-c][1,2,4]triazol-3(5H)-ylidene)amino](phenylamino)methylene}benzamide (3) has been obtained by the reaction of one measure of N-{[7-(4,5-dihydro-1H-imidazol-2-yl)-2-(p-tolyl)-6,7-dihydro-2H-imidazo[2,1-c][1,2,4]triazol-3(5H)-ylidene]carbamothioyl}benzamide (2) with one measure of aniline in the presence of mercury(II) chloride and triethylamine in anhydrous dimethylformamide. The structure of product 3 was confirmed by 1H and 13C-NMR, infrared spectroscopy, and elemental analysis.

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12

Mabkhot, Yahia Nasser, Assem Barakat, Hazem A. Ghabbour, and Hoong-Kun Fun. "Crystal structure of 2-amino-N-(4-methoxyphenyl)benzamide, C14H14N2O2." Zeitschrift für Kristallographie - New Crystal Structures 231, no. 1 (2016): 203–4. http://dx.doi.org/10.1515/ncrs-2015-0089.

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13

Shablykin, Oleh, Egor Herasymov, Olga Shablykina, and Andrii Kozytsky. "Synthesis of 2-R-5-amino-4-(1H-tetrazol-5-yl)-1,3-oxazoles from 2-R-5-amino-1,3-oxazole-4-carbonitriles." Current Chemistry Letters 14, no. 1 (2025): 233–38. http://dx.doi.org/10.5267/j.ccl.2024.6.003.

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This short communication reports about new 5-amino-4-(1H-tetrazol-5-yl)-1,3-oxazoles which were synthesized by [3+2] cycloaddition of 2-R-5-amino-1,3-oxazole-4-carbonitriles and trimethylsilyl azide with dibutyltin oxide present. The reaction conditions provided high yields of the products, and were tolerant to some active functional fragments in the oxazole substituents (amino, amido, and hydroxy group). In the case of 2-((4-cyano-2-phenyloxazol-5-yl)amino)-N-methylacetamide the by-product (N-((1-(2-(methylamino)-2-oxoethyl)-1H-tetrazol-5-yl)(1H-tetrazol-5-yl)methyl)-benzamide) was formed tog

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14

Zadrazilova, Iveta, Sarka Pospisilova, Karel Pauk, et al. "In VitroBactericidal Activity of 4- and 5-Chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA." BioMed Research International 2015 (2015): 1–8. http://dx.doi.org/10.1155/2015/349534.

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A series of nine substituted 2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides was assessed as prospective bactericidal agents against three clinical isolates of methicillin-resistantStaphylococcus aureus(MRSA) andS. aureusATCC 29213 as the reference and quality control strain. The minimum bactericidal concentration was determined by subculturing aliquots from MIC determination onto substance-free agar plates. The bactericidal kinetics of compounds 5-chloro-2-hydroxy-N-[(2S)-3-methyl-1-oxo-1-{[4-(trifluoromethyl)phenyl]amino}butan-2-yl]benzamide (1f),N-{(2S)-1-[(4-bromophenyl)amino]-3-me

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15

Adhami, Forogh, Nasim Nabilzadeh, Franziska Emmerling, Mina Ghiasi, and Majid Heravi. "Synthesis of thiadiazolobenzamide via cyclization of thioxothiourea and its Ni and Pd complexes." Journal of the Serbian Chemical Society 77, no. 9 (2012): 1211–22. http://dx.doi.org/10.2298/jsc110911052a.

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In this study, the new compound, N-(3-methyl-4- oxo[1,3,4]thiadiazolo[2,3-c][1,2,4]triazin-7-yl) benzamide, could be obtained via two different reactions: 1) reaction of 4-amino-6-Methyl-3- (Methylsulfanyl)-1,2,4-triazin-5-one with benzoyl isothiocyanate under removal of methylmercaptane, 2) reaction of 4-amino-6-Methyl-3-thioxo- 1,2,4-triazin-5-one with benzoyl isothiocyanate under elimination of hydrogen sulfide. In both reactions a new bond between sulfur and nitrogen atoms was formed and a five-membered ring was created. The oxo thiadiazolo benzamide was characterized by IR-, 1HNMR- and 13

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16

Pavlova, V. V., P. V. Zadorozhnii, V. V. Kiselev, A. V. Kharchenko, and O. V. Okhtina. "Modeling of new potential inhibitors of dihydrofolate reductase based on 1,3,4-thiadiazole amidoalkyl derivatives." Voprosy Khimii i Khimicheskoi Tekhnologii, no. 5 (October 2023): 91–97. http://dx.doi.org/10.32434/0321-4095-2023-150-5-91-97.

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Derivatives of 1,3,4-thiadiazole are very important for medical chemistry and pharmacy as potential drug substances. In this work, we carried out molecular docking studies of amidoalkyl derivatives of 1,3,4-thiadiazole: N-(2,2,2-trichloro-1-((5-aryl-1,3,4-thiadiazol-2-yl)amino)ethyl)carboxamides and N-(2,2,2-trichloro-1-((5-(arylamino)-1,3,4-thiadiazol-2-yl)amino)ethyl)carboxamides with dihydrofolate reductase (DHFR). The AutoDock Vina program based on the PyRx 0.8 platform was used for docking. Before docking, the enzyme structure (PDB ID: 1DLS) was prepared using the Chimera 1.14 program, an

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17

Le, Hong, Quynh Do, Mai Doan, et al. "Chemical Composition and Biological Activities of Metabolites from the Marine Fungi Penicillium sp. Isolated from Sediments of Co To Island, Vietnam." Molecules 24, no. 21 (2019): 3830. http://dx.doi.org/10.3390/molecules24213830.

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Marine microorganisms are an invaluable source of novel active secondary metabolites possessing various biological activities. In this study, the extraction and isolation of the marine sediment Penicillium species collected in Vietnam yielded ten secondary metabolites, including sporogen AO-1 (1), 3-indolecarbaldehyde (2), 2-[(5-methyl-1,4-dioxan-2-yl)methoxy]ethanol (3), 2-[(2R-hydroxypropanoyl)amino]benzamide (4), 4-hydroxybenzandehyde (5), chrysogine (6), 3-acetyl-4-hydroxycinnoline (7), acid 1H-indole-3-acetic (8), cyclo (Tyr-Trp) (9), and 2’,3’-dihydrosorbicillin (10). Their structures we

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18

Xu, Defeng, Xing Xu, and Zhiling Zhu. "A Convenient Synthesis of 4-amino-2-fluoro-N-methyl-benzamide." Journal of Chemical Research 37, no. 10 (2013): 615–16. http://dx.doi.org/10.3184/174751913x13787959772340.

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19

J. Prathyusha and C. Asha Deepti. "SYNTHESIS, ANTIMICROBIAL, AND ANTITUBERCULAR ACTIVITIES OF NOVEL N-PYRAZOLYLBENZAMIDE DERIVATIVES." RASAYAN Journal of Chemistry 15, no. 04 (2022): 2407–16. http://dx.doi.org/10.31788/rjc.2022.1547092.

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The current study investigated the antimicrobial and antitubercular activities of novel N-Pyrazolyl Benzamide derivatives. The study includes the synthesis, characterization, and ligand-based molecular docking of the designed molecules. Synthesis of N-Pyrazolyl Benzamide derivatives involves a two-step process in which 5-amino pyrazole (3) intermediate is produced by the condensation reaction of aryl hydrazine (1) and β-keto nitrile (2) in acidic conditions. The final N-Pyrazolyl Benzamide derivatives (5a-n) were synthesized by the reaction involving amide coupling between 5-amino pyrazole (3)

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20

Almarhoon, Zainab, Kholood A. Dahlous, Rakia Abd Alhameed, Hazem A. Ghabbour, and Ayman El-Faham. "A Simple, Efficient, and Eco-Friendly Method for the Preparation of 3-Substituted-2,3-dihydroquinazolin-4(1H)-one Derivatives." Molecules 24, no. 22 (2019): 4052. http://dx.doi.org/10.3390/molecules24224052.

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A simple, cost-effective method under environmentally benign conditions is a very important concept for the preparation of 2,3-dihydroquinazolin-4(1H)-one derivatives. The present work describes an efficient and eco-friendly protocol for the synthesis of 2-amino-N-(2-substituted-ethyl)benzamide and 3-substituted-2,3-dihydroquinazolin-4(1H)-one derivatives. The novel feature of this protocol is the use of 2-methyl tetrahydrofuran (2-MeTHF) as an eco-friendly alternative solvent to tetrahydrofuran (THF) in the first step. In the second step, methanol in the presence of potassium carbonate as a c

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21

Sagar, Belakavadi K., Hemmige S. Yathirajan, Ravindranath S. Rathore, and Christopher Glidewell. "Four closely related N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)benzamides: order versus disorder, and similar molecular conformations but different modes of supramolecular aggregation, with a new disordered refinement of 2-amino-3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophene." Acta Crystallographica Section C Structural Chemistry 74, no. 1 (2018): 45–53. http://dx.doi.org/10.1107/s2053229617017326.

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Four closely related N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)benzamides, bearing different substituents on the benzamide ring, have been synthesized and structurally characterized. In each of N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-3-fluorobenzamide, C22H18FNO2S, (I), N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-chlorobenzamide, C22H18ClNO2S, (II), N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2,6-difluorobenzamide, C22H17F2NO2S, (III), and N-(3-benzoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-methoxybenzamide, C23H21NO3S, (IV), the last of which

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22

Bassey, Margaret Emmanuel, Imoh Imeh Johnny, Ogechi Queeneth Iwu, Omodot Timothy Umoh, and Augustine Ogenekevwe Ochuko. "Phyto-constituents of the Dichloromethane Extracts of the Bulbs of Selected Genera in the Family Amaryllidaceae." Asian Plant Research Journal 12, no. 3 (2024): 72–91. http://dx.doi.org/10.9734/aprj/2024/v12i3255.

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The analysis of phytoconstituents present in the dichloromethane extract of the bulb of Hippeastrum vittatum (L’Her.) Herb., Proiphys amboinensis (L.) Herb., Urceolina amazonica (Linden) Christenh. & Byng., Hymenocallis littoralis (Jacq.) Salisb., Crinum jagus (J. Thomps.) Dandy and Zephyranthes carinata Herb. by Gas Chromatography-Mass Spectometry (GC-MS) analysis was carried out using standard methods. The Results of the GC-MS analysis of Hippeastrum vittatum, Proiphys amboinensis, Urceolina amazonica, Hymenocallis littoralis, Crinum jagus and Zephyranthes carinata revealed the presence

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23

Aich, Udayananth, Deanna C. Hurum, Lipika Basumallick, et al. "Evaluation of desialylation during 2-amino benzamide labeling of asparagine-linked oligosaccharides." Analytical Biochemistry 458 (August 2014): 27–36. http://dx.doi.org/10.1016/j.ab.2014.03.008.

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24

Tran Hoai Tu, Nguyen Trung Nhan, and Dang Hoang Phu. "Synthesis of benzamide derivatives and evaluation of their in vitro and in silico tyrosinase inhibitory activities." Vietnam Journal of Science and Technology 62, no. 4 (2024): 660–69. http://dx.doi.org/10.15625/2525-2518/18302.

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In this research, six benzamide derivatives were traditionally synthesized using hydrazine, carbazide, and hydroxylamine derivatives through the pre- or in situ activation of the carboxylic acid functionality. Their chemical structures were identified as N′-phenylbenzohydrazide, N′-(2,4-dinitrophenyl)benzohydrazide, N′-(benzoyloxy)benzamide, N-dibenzoylurea, 2-amino-5-(4-phenyl)-1,3,4-thiadiazole, and benzohydrazide based on the interpretation of NMR spectroscopic data. Among these products, N′-phenylbenzohydrazide and N-(benzoyloxy)benzamide showed potent tyrosinase inhibitory activity with t

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25

Marini, Richard P., Ross E. Byers, and Donald L. Sowers. "Growth Regulators and Herbicides for Delaying Apple Fruit Abscission." HortScience 24, no. 6 (1989): 957–59. http://dx.doi.org/10.21273/hortsci.24.6.957.

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Abstract Various chemicals were applied to whole-tree, quarter-tree, or single-limb units to determine their efficacy for delaying apple (Malus domestica Borkh.) fruit abscission. NAA and the herbicides fenoprop, dicamba, triclopyr, lontrel, fluroxypyr, and chloroxuron delayed fruit abscission. Benzoic acid, calcium acetate; the growth regulators lactidichlor ethyl, mefluidide, BA, GA4+7, and chlormequat; and the herbicides pronamide, pendimethalin, chloramben, and DCPA did not delay fruit abscission. Chemical names used: benzoic acid,3,6-dichloro-2-methoxy,2-ethoxy, 1-methyl,2-oxoethylester (

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Hoffelner, Beate Sandra, Stanislav Andreev, Nicole Plank, and Pierre Koch. "Photocaging of Pyridinylimidazole-Based Covalent JNK3 Inhibitors Affords Spatiotemporal Control of the Binding Affinity in Live Cells." Pharmaceuticals 16, no. 2 (2023): 264. http://dx.doi.org/10.3390/ph16020264.

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The concept of photocaging represents a promising approach to acquire spatiotemporal control over molecular bioactivity. To apply this strategy to pyridinylimidazole-based covalent JNK3 inhibitors, we used acrylamido-N-(4-((4-(4-(4-fluorophenyl)-1-methyl-2-(methylthio)-1H-imidazol-5-yl)pyridin-2-yl)amino)phenyl)benzamide (1) as a lead compound to design novel covalent inhibitors of JNK3 by modifying the amide bond moiety in the linker. The newly synthesized inhibitors demonstrated IC50 values in the low double-digit nanomolar range in a radiometric kinase assay. They were further characterized

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Senthilkumar, Gopal, Chinnusamy Umarani, and Dhurairaj Satheesh. "Synthesis, Spectral Characterization, Antibacterial, Antifungal and Anticancer Evaluation of N-[4-(1,3-Benzothiazol-2-ylcarbamoyl)phenyl]pyrazine-2-carboxamide." Asian Journal of Organic & Medicinal Chemistry 6, no. 2 (2021): 102–6. http://dx.doi.org/10.14233/ajomc.2021.ajomc-p320.

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A new organic compound, N-[4-(1,3-benzothiazol-2-ylcarbamoyl)-phenyl]pyrazine-2-carboxamide was synthesized through the reaction between 4-amino-N-(benzo[d]thiazol-2-yl)benzamide and pyrazine-2-carboxylic acid. The synthesized compound has been characterized by spectroscopic techniques such as 1H NMR, 13C NMR, FT-IR and mass spectroscopy. The synthesized compound was screened to antibacterial (Staphylococcus aureus, Klebsiella pneumonia and Escherichia coli), antifungal (Candida albicans and Aspergillus niger) activities. The anticancer activity of the title compound was also evaluated against

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KATO, Shiro, Toshiya MORIE, Kazunori OHNO, Naoyuki YOSHIDA, Toyokichi YOSHIDA, and Shunsuke NARUTO. "Synthesis and Gastroprokinetic Activity of 2-Amino-N-((4-benzyl-2-morpholinyl)methyl)benzamide Derivatives." CHEMICAL & PHARMACEUTICAL BULLETIN 43, no. 4 (1995): 582–87. http://dx.doi.org/10.1248/cpb.43.582.

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Skibiński, Robert, and Łukasz Komsta. "Application of Curve Resolution Algorithms in the Study Drug Photodegradation Kinetics—The Example of Moclobemide." Journal of AOAC INTERNATIONAL 95, no. 3 (2012): 708–12. http://dx.doi.org/10.5740/jaoacint.sge_skibinski.

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Abstract The photodegradation of moclobemide was studied in methanolic media. Ultra-HPLC (UHPLC)/MS/MS analysis proved decomposition to 4-chlorobenzamide as a major degradation product and small amounts of Ro 16-3177 (4-chloro-N-[2-[(2-hydroxyethyl)amino] ethyl]benzamide) and 2-[(4-chlorobenzylidene)amino]-N-[2-ethoxyethenyl]ethenamine. The methanolic solution was investigated spectrophotometrically in the UV region, registering the spectra during 30 min of degradation. Using reference spectra and a multivariate chemometric method (multi- variate curve resolution-alternating least squares), th

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Nishimura, Teruyuki, Tomoharu Iino, Morihiro Mitsuya, et al. "Identification of novel and potent 2-amino benzamide derivatives as allosteric glucokinase activators." Bioorganic & Medicinal Chemistry Letters 19, no. 5 (2009): 1357–60. http://dx.doi.org/10.1016/j.bmcl.2009.01.053.

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Xu, Defeng, Xing Xu, and Zhiling Zhu. "ChemInform Abstract: A Convenient Synthesis of 4-Amino-2-fluoro-N-methyl-benzamide." ChemInform 45, no. 24 (2014): no. http://dx.doi.org/10.1002/chin.201424075.

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C., B. MAHTO. "Complexes of 2-Methoxy-4-amino-5-chloro-N-[ 2-(diethylamino)ethyl]benzamide with Metal Ions." Journal of Indian Chemical Society Vol. 62, Oct 1985 (1985): 731–33. https://doi.org/10.5281/zenodo.6322687.

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Department of Chemistry, Gopalganj College, Gopalganj, Bihar <em>Manuscript received 13 February 1984, revised 24 June 1985, accepted 11 September 1985</em> The complexes of 2-methoxy-.4-amino-5-chloro-N-[2-(diethylamino)ethyl]benzamide (L) with the metal ions of the types ML<sub>2</sub>X<sub>2</sub> (M- Ni<em><sup>ll</sup></em>, Cd<em><sup>ll</sup></em>, Fe<em><sup>ll</sup></em>, Co<em><sup>II</sup></em>, Mn<em><sup>lI</sup></em> and Zn<em><sup>ll</sup></em>; X - \({1\ \over 2}\)\(SO_4^{2-}\), Cl<sup>-</sup>or NO\(_3^-\)), ML<sub>2</sub>X<sub>2</sub> (M - Cu<em><sup>ll</sup></e

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33

A Ben Hadj Amor, A. Ben Hadj Amor, and A. Mezni and R. Abderrahim A Mezni and R Abderrahim. "Synthesis, Characterization, Enhanced Solubility and Antioxidant Activity of the Inclusion Compound of 2-Amino-N-o-tolyl-benzamide and Beta Cyclodextrin." Journal of the chemical society of pakistan 46, no. 1 (2024): 93. http://dx.doi.org/10.52568/001427/jcsp/46.01.2024.

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The objectives of this research, were to study the effect of beta cyclodextrin on the enhancement of the solubility and the antioxidant activity of 2-Amino-N-o-tolyl-benzamide (ATB). ATB was obtained by a new synthesis method and used to form inclusion compound macromolecule with -CD. The characterization of the ATB and the complex were subsequently established by FT-IR; 1H NMR; 13C NMR; NMR 2D spectra and XRD. The optical activity was measured. The interaction of β-CD and ATB was also analyzed by UV-Vis spectroscopy in order to determine the formation constant. The stoichiometry of the compl

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Kanyonyo, Martial R., Jacques H. Poupaert, and Didier M. Lambert. "Anticonvulsant Profile of 4-Amino-(2-methyl-4-aminophenyl)benzamide in Mice and Rats." Pharmacology & Toxicology 82, no. 1 (1998): 47–50. http://dx.doi.org/10.1111/j.1600-0773.1998.tb01397.x.

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Bigge, J. C., T. P. Patel, J. A. Bruce, P. N. Goulding, S. M. Charles, and R. B. Parekh. "Nonselective and Efficient Fluorescent Labeling of Glycans Using 2-Amino Benzamide and Anthranilic Acid." Analytical Biochemistry 230, no. 2 (1995): 229–38. http://dx.doi.org/10.1006/abio.1995.1468.

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Durant, F., P. Renard, V. De Beys та G. Evrard. "Molecular Structure of Benzamide Neuroleptics IV. Amino-4, Bromo-5, Methoxy-2 π-π (Chloro-2 Phenylmethyl)-8 Aza-8 Bicyclo [ 3.2.1] Octyl-3°] Benzamide (exo)". Bulletin des Sociétés Chimiques Belges 93, № 10 (2010): 923–24. http://dx.doi.org/10.1002/bscb.19840931013.

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KATO, S., T. MORIE, K. OHNO, N. YOSHIDA, T. YOSHIDA, and S. NARUTO. "ChemInform Abstract: Synthesis and Gastroprokinetic Activity of 2-Amino-N-((4-benzyl-2- morpholinyl)methyl)benzamide Derivatives." ChemInform 26, no. 45 (2010): no. http://dx.doi.org/10.1002/chin.199545194.

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38

Paromov, Artyom, Irina Shchurova, Alla Rogova, Irina Bagryanskaya, and Dmitriy Polovyanenko. "Acid-Catalyzed Condensation of Benzamide with Glyoxal, and Reaction Features." Molecules 27, no. 3 (2022): 1094. http://dx.doi.org/10.3390/molecules27031094.

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Scholars from around the world have been attempting to simplify and cheapen the synthetic method for the promising high-energy compound CL-20 for decades. The lack of understanding of the formation mechanisms of hexaazaisowurtzitane derivatives―CL-20 precursors―is a barrier to solving the said problems. Here, we report the results from an in-depth study into the acid-catalyzed condensation between benzamide and glyoxal in a molar ratio of 2:1 in polar protic and aprotic solvents. Sixteen compounds were isolated and identified, of which eight were synthesized for the first time. A geminal diol,

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Lee, Chaewon, Boreum Song, Eunsu Kim, et al. "68Ga-labeled fluorinated benzamide derivatives for positron emission tomography imaging of melanoma." PLOS ONE 20, no. 2 (2025): e0317489. https://doi.org/10.1371/journal.pone.0317489.

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Malignant melanoma tends to aggressively metastasize, resulting in it being a potentially lethal form of skin cancer with high mortality rates. The advanced stages of melanoma have a very poor prognosis because of the high tendency for metastasis, and there is therefore, a strong desire to develop efficient technology for the early detection of melanoma. The benzamide structure, which contains aromatic ring and amine group, exhibits a high affinity for melanin, making it a promising agent for targeting melanoma in diagnostic and therapeutic applications. In this study, we synthesized a fluorin

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Diouf, O., M. Bourhim, D. M. Lambert, J. H. Poupaert, J. P. Stables, and J. Vamecq. "Anticonvulsant and neurotoxicological properties of 4-amino-N-(2-ethylphenyl)benzamide, a potent ameltolide analogue." Biomedicine & Pharmacotherapy 51, no. 3 (1997): 131–36. http://dx.doi.org/10.1016/s0753-3322(97)86911-9.

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Marquezin, Cássia Alessandra, Izaura Yoshico Hirata, Luiz Juliano, and Amando Siuiti Ito. "Spectroscopic characterization of 2-amino-N-hexadecyl-benzamide (AHBA), a new fluorescence probe for membranes." Biophysical Chemistry 124, no. 2 (2006): 125–33. http://dx.doi.org/10.1016/j.bpc.2006.06.002.

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42

Moreno-Fuquen, Rodolfo, Kevin Arango-Daraviña, Diana Becerra, Juan-Carlos Castillo, Alan R. Kennedy, and Mario A. Macías. "Catalyst- and solvent-free synthesis of 2-fluoro-N-(3-methylsulfanyl-1H-1,2,4-triazol-5-yl)benzamide through a microwave-assisted Fries rearrangement: X-ray structural and theoretical studies." Acta Crystallographica Section C Structural Chemistry 75, no. 3 (2019): 359–71. http://dx.doi.org/10.1107/s2053229619002572.

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An efficient approach for the regioselective synthesis of (5-amino-3-methylsulfanyl-1H-1,2,4-triazol-1-yl)(2-fluorophenyl)methanone, C10H9FN4OS, (3), from the N-acylation of 3-amino-5-methylsulfanyl-1H-1,2,4-triazole, (1), with 2-fluorobenzoyl chloride has been developed. Heterocyclic amide (3) was used successfully as a strategic intermediate for the preparation of 2-fluoro-N-(3-methylsulfanyl-1H-1,2,4-triazol-5-yl)benzamide, C10H9FN4OS, (4), through a microwave-assisted Fries rearrangement under catalyst- and solvent-free conditions. Theoretical studies of the prototropy process of (1) and t

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43

Dorn, Angelika, Dieter Schollmeyer, and Stefan A. Laufer. "N-{2-Methyl-5-[(5-oxo-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-2-yl)amino]phenyl}benzamide." Acta Crystallographica Section E Structure Reports Online 66, no. 7 (2010): o1867. http://dx.doi.org/10.1107/s1600536810024256.

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Valverde, Lauro Figueroa, Francisco DIaz Cedillo, Eduardo Pool GOmez, Maria LOpez Ramos, and Abelardo Camacho Luis. "Design and Synthesis of N-(2-{[(2-Hydroxy-naphtalen-1-yl)-phenyl-methyl]-amino}-ethyl)-3,4-dinitro-benzamide." Oriental Journal Of Chemistry 29, no. 1 (2013): 17–22. http://dx.doi.org/10.13005/ojc/290103.

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., Pavlo V. Zadorozhnii Ihor O. Pokotylo Vadym V. Kiselev Aleksandr V. Kharchenko Oxana V. Okhtina. "MOLECULAR DOCKING STUDIES OF N-(1-(BENZO[d]THIAZOL-2-YLAMINO)-2,2,2-TRICHLOROETHYL)-CARBOXAMIDES AS А2A RECEPTOR POTENTIAL ANTAGONISTS". INDO AMERICAN JOURNAL OF PHARMACEUTICAL SCIENCES 06, № 01 (2019): 1345–51. https://doi.org/10.5281/zenodo.2544020.

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<em>In this work, using the ArgusLab 4.0.1 software package, we carried out in silico modeling of A<sub>2A</sub> receptor antagonists. We proposed N-(1-(benzo[d]thiazol-2-ylamino)-2,2,2-trichloroethyl)carboxamides as potential biologically active substances. According to the results of molecular docking, all of the analyzed benzo[d]thiazol-2-amine derivatives were superior to ZM-241385 in the strength of the complex formed with the receptor. N-(1-(benzo[d]thiazol-2-ylamino)-2,2,2-trichloroethyl)-4-methylbenzamide, N-(1-(benzo[d]thiazol-2-ylamino)-2,2,2-trichloroethyl)-1-naphthamide and N-(2,2,

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Pindjakova, Dominika, Eliska Pilarova, Karel Pauk, et al. "Study of Biological Activities and ADMET-Related Properties of Salicylanilide-Based Peptidomimetics." International Journal of Molecular Sciences 23, no. 19 (2022): 11648. http://dx.doi.org/10.3390/ijms231911648.

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A series of eleven benzylated intermediates and eleven target compounds derived from salicylanilide were tested against Staphylococcus aureus ATCC 29213 and Enterococcus faecalis ATCC 29212 as reference strains and against three clinical isolates of methicillin-resistant S. aureus (MRSA) and three isolates of vancomycin-resistant E. faecalis. In addition, the compounds were evaluated against Mycobacterium tuberculosis H37Ra and M. smegmatis ATCC 700084. The in vitro cytotoxicity of the compounds was assessed using the human monocytic leukemia cell line THP-1. The lipophilicity of the prepared

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47

Mostafa, Gamal A. E., Ahmed H. Bakheit, Mohamed H. Al-Agamy, Rashad Al-Salahi, Essam A. Ali, and Haitham Alrabiah. "Synthesis of 4-Amino-N-[2 (diethylamino)Ethyl]Benzamide Tetraphenylborate Ion-Associate Complex: Characterization, Antibacterial and Computational Study." Molecules 28, no. 5 (2023): 2256. http://dx.doi.org/10.3390/molecules28052256.

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The 4-amino-N-[2 (diethylamino) ethyl] benzamide (procainamide)-tetraphenylborate complex was synthesized by reacting sodium tetraphenyl borate with 4-amino-N-[2 (diethylamino) ethyl] benzamide, chloride salt, and procainamide in deionized water at room temperature through an ion-associate reaction (green chemistry) at room temperature, and characterized by several physicochemical methods. The formation of ion-associate complex between bio-active molecules and/or organic molecules is crucial to comprehending the relationships between bioactive molecules and receptor interactions. The solid com

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48

Al-Soud, Yaseen A., Najim A. Al-Masoudi, Hossam H. Al-Suod, and Christophe Pannecouque. "Nitroimidazoles Part 8. Synthesis and Anti-HIV Activity of New 4-Nitroimidazole Derivatives Using the Suzuki Cross-Coupling Reaction." Zeitschrift für Naturforschung B 67, no. 9 (2012): 925–34. http://dx.doi.org/10.5560/znb.2012-0185.

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The development of new HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs) offers the possibility of generating structures of increased potency. To this end, a series of 1-(1-benzyl-2-ethyl- 4-nitro-1H-imidazol-5-yl)-4-(1,1'-biaryl)-4-yl-piperazine derivatives (6a-l) was synthesized via the Suzuki coupling reaction. Analogously, coupling of the acid derivative 5, prepared from 4, with various amino acid methyl esters in the presence of HOBt/DCC reagents afforded the benzamide derivatives 8-11. The newly synthesized compounds were assayed against HIV-1 and HIV-2 in MT- 4 cells. All com

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Al-Hazam, Hanan A., Zeki A. Al-Shamkani, Najim A. Al-Masoudi, Bahjat A. Saeed, and Christophe Pannecouque. "New chalcones and thiopyrimidine analogues derived from mefenamic acid: microwave-assisted synthesis, anti-HIV activity and cytotoxicity as antileukemic agents." Zeitschrift für Naturforschung B 72, no. 4 (2017): 249–56. http://dx.doi.org/10.1515/znb-2016-0223.

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AbstractThe development of new HIV non-nucleoside reverse transcriptase inhibitors offers the possibility of generating structures of increased potency. To this end, coupling of mefenamic acid (4) with 4-amino-acetophenone (6) in the presence of dicyclohexylcarbodiimide and dimethylaminopyridine (DMAP) reagents afforded 4-(acetyphenyl)-2-((2,3-dimethylphenyl)amino)benzamide (7). Analogously, treatment of mefenamyl chloride (5) prepared from 4 with 6 under microwave irradiation (MWI) afforded 7. A new series of substituted chalconyl-incorporated amide derivatives of mefenamic acid 8–13 were syn

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50

Ruys, Luc, and Etienne Schacht. "Synthesis of 4-[N- [2-(Methacryloyloxy) Ethoxycarbonyl) ]Amino-N′-[2- (Diethylamino) Ethyl]Benzamide; A Novel Polymerizable Derivative of Procainamide." Bulletin des Sociétés Chimiques Belges 93, no. 2 (2010): 159–60. http://dx.doi.org/10.1002/bscb.19840930211.

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