Log in

Relevant bibliographies by topics / 4-oxadiazole derivatives containing R-phenyl moiety

Contents

Journal articles

Academic literature on the topic '4-oxadiazole derivatives containing R-phenyl moiety'

Author: Grafiati

Published: 7 June 2025

Last updated: 2 August 2025

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic '4-oxadiazole derivatives containing R-phenyl moiety.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "4-oxadiazole derivatives containing R-phenyl moiety"

1

Markov, Andrey V., Aleksandra V. Sen’kova, Irina I. Popadyuk та ін. "Novel 3′-Substituted-1′,2′,4′-Oxadiazole Derivatives of 18βH-Glycyrrhetinic Acid and Their O-Acylated Amidoximes: Synthesis and Evaluation of Antitumor and Anti-Inflammatory Potential In Vitro and In Vivo". International Journal of Molecular Sciences 21, № 10 (2020): 3511. http://dx.doi.org/10.3390/ijms21103511.

Full text

Abstract:

A series of novel 18βH-glycyrrhetinic acid (GA) derivatives containing 3′-(alkyl/phenyl/pyridin(-2″, -3″, and -4″)-yl)-1′,2′,4′-oxadiazole moieties at the C-30 position were synthesized by condensation of triterpenoid’s carboxyl group with corresponding amidoximes and further cyclization. Screening of the cytotoxicity of novel GA derivatives on a panel of tumor cell lines showed that the 3-acetoxy triterpenoid intermediates—O-acylated amidoxime 3a-h—display better solubility under bioassay conditions and more pronounced cytotoxicity compared to their 1′,2′,4′-oxadiazole analogs 4f-h (median IC

APA, Harvard, Vancouver, ISO, and other styles

2

Wang, Lei, Xia Zhou, Hui Lu, Xianfu Mu, and Linhong Jin. "Synthesis and Antibacterial Evaluation of Novel 1,3,4-Oxadiazole Derivatives Containing Sulfonate/Carboxylate Moiety." Molecules 25, no. 7 (2020): 1488. http://dx.doi.org/10.3390/molecules25071488.

Full text

Abstract:

In order to discover new lead compounds with high antibacterial activity, a series of new derivatives were designed and synthesized by introducing a sulfonate or carboxylate moiety into the 1,3,4-oxadiazole structure. Antibacterial activity against two phytopathogens, Xanthomonas oryzae pv. oryzae (Xoo) and Xanthomonas axonopodis pv. citri (Xac), was assayed in vitro. The preliminary results indicated that ten compounds including 4a-1-4a-4 and 4a-11-4a-16 had good antibacterial activity against Xoo, with EC50 values ranging from 50.1-112.5 µM, which was better than those of Bismerthiazol (253.

APA, Harvard, Vancouver, ISO, and other styles

3

Adimule, Vinayak, Sudha Medapa, AdarshaHaraballi Jagadeesha, LalitaSanjeev Kumar, and Prakash Kumar Rao. "Synthesis, characterization and cytotoxic evaluation of novel derivatives of 1, 3, 4-oxadiazole containing 5-phenyl thiophene moiety." IOSR Journal of Pharmacy and Biological Sciences 9, no. 5 (2014): 42–48. http://dx.doi.org/10.9790/3008-09544248.

Full text

APA, Harvard, Vancouver, ISO, and other styles

4

*Ashwini, H. Pagare, and Anwar R. Shaikh Dr. "CONVENTIONAL SYNTHESIS AND STRUCTURAL ELUCIDATION OF NEWER 1,3,4-OXADIAZOLE DERIVATIVES BIO FUNCTIONING AS ANTI-BACTERIAL AND ANTI-FUNGAL." World Journal of Pharmaceutical Science and Research 4, no. 1 (2025): 836–44. https://doi.org/10.5281/zenodo.14940193.

Full text

APA, Harvard, Vancouver, ISO, and other styles

5

Li, Feng-Yun, Jing-Bo Liu, Jia-Ning Gong, and Gen Li. "(R)-2-Phenyl-4,5-Dihydrothiazole-4-Carboxamide Derivatives Containing a Diacylhydrazine Group: Synthesis, Biological Evaluation, and SARs." Molecules 24, no. 24 (2019): 4440. http://dx.doi.org/10.3390/molecules24244440.

Full text

Abstract:

A series of (R)-2-phenyl-4,5-dihydrothiazole-4-carboxamide derivatives containing a diacylhydrazine moiety were designed and synthesized. Their structures were confirmed by melting points, 1H NMR, 13C NMR, and elemental analysis (EA). Their antifungal and insecticidal activities were evaluated. The antifungal activity result indicated that most title compounds against Cercospora arachidicola, Alternaria solani, Phytophthora capsici, and Physalospora piricola exhibited apparent antifungal activities at 50 mg/L, and better than chlorothalonil or carbendazim. The EC50 values of (R)-N’-benzoyl-2-(

APA, Harvard, Vancouver, ISO, and other styles

6

Liu, Jingbo, Fengyun Li, Yuanhong Wang, Haoxuan Zhang, Yuxin Li, and Zhengming Li. "Synthesis, biological activities, and 3D-QSAR studies of (R)-2-phenyl-4,5-dihydrothiazole-4-carboxamide derivatives containing a sulfonohydrazide moiety." Medicinal Chemistry Research 29, no. 3 (2020): 495–503. http://dx.doi.org/10.1007/s00044-020-02499-3.

Full text

APA, Harvard, Vancouver, ISO, and other styles

7

Liu, Jingbo, Fengyun Li, Yuanhong Wang, et al. "Synthesis, biological activities and 3D-QSAR studies of (R)-2-phenyl-4,5-dihydrothiazole-4-carboxamide derivatives containing a sulfur ether moiety." Chinese Chemical Letters 30, no. 3 (2019): 668–71. http://dx.doi.org/10.1016/j.cclet.2018.11.001.

Full text

APA, Harvard, Vancouver, ISO, and other styles

8

Irfan, Ali, Shah Faisal, Ameer Fawad Zahoor, et al. "In Silico Development of Novel Benzofuran-1,3,4-Oxadiazoles as Lead Inhibitors of M. tuberculosis Polyketide Synthase 13." Pharmaceuticals 16, no. 6 (2023): 829. http://dx.doi.org/10.3390/ph16060829.

Full text

Abstract:

Benzofuran and 1,3,4-oxadiazole are privileged and versatile heterocyclic pharmacophores which display a broad spectrum of biological and pharmacological therapeutic potential against a wide variety of diseases. This article reports in silico CADD (computer-aided drug design) and molecular hybridization approaches for the evaluation of the chemotherapeutic efficacy of 16 S-linked N-phenyl acetamide moiety containing benzofuran-1,3,4-oxadiazole scaffolds BF1–BF16. This virtual screening was carried out to discover and assess the chemotherapeutic efficacy of BF1–BF16 structural motifs as Mycobac

APA, Harvard, Vancouver, ISO, and other styles

9

Ölmez, Nevin Arıkan, and Faryal Waseer. "New Potential Biologically Active Compounds: Synthesis and Characterization of Urea and Thiourea Derivativpes Bearing 1,2,4-oxadiazole Ring." Current Organic Synthesis 17, no. 7 (2020): 525–34. http://dx.doi.org/10.2174/1570179417666200417112106.

Full text

Abstract:

Background: Urea, thiourea, and 1,2,4-oxadiazole compounds are of great interest due to their different activities such as anti-inflammatory, antiviral, analgesic, fungicidal, herbicidal, diuretic, antihelminthic and antitumor along with antimicrobial activities. Objective: In this work, we provide a new series of potential biologically active compounds containing both 1,2,4-oxadiazole and urea/thiouprea moiety. Materials and Methods: Firstly, 5-chloromethyl-3-aryl-1,2,4-oxadiazoles (3a-j) were synthesized from the reaction of different substituted amidoximes (2a-j) and chloroacetyl chloride i

APA, Harvard, Vancouver, ISO, and other styles

10

Bhat, Mashooq Ahmad, Mohamed A. Al-Omar, Ahmed M. Naglah, Atef Kalmouch, and Abdullah Al-Dhfyan. "Synthesis and Characterization of Novel Biginelli Dihydropyrimidinone Derivatives Containing Imidazole Moiety." Journal of Chemistry 2019 (May 13, 2019): 1–7. http://dx.doi.org/10.1155/2019/3131879.

Full text

Abstract:

Enaminone, (2E)-1-[4-(1H-imidazol-1-yl) phenyl]-4-methylpent-2-en-1-one (II) was synthesized by refluxing 1-[4-(1H-imidazol-1-yl) phenyl] ethan-1-one (I) with dimethylforamide dimethylacetal (DMF–DMA) under solvent-free condition for 12 hours. Finally, the dihydropyrimidinone derivatives containing imidazole moiety (1–15) were obtained by reacting enaminone, (2E)-1-[4-(1H-imidazol-1-yl) phenyl]-4-methylpent-2-en-1-one (II) with urea and different substituted benzaldehydes in the presence of glacial acetic acid. Dihydropyrimidinone derivatives containing imidazole moiety were synthesized in exc

APA, Harvard, Vancouver, ISO, and other styles

More sources

We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!