Relevant bibliographies by topics / 4-tetrahydroacridines

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Academic literature on the topic '4-tetrahydroacridines'

Author: Grafiati
Published: 7 June 2025
Last updated: 2 August 2025

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Journal articles on the topic "4-tetrahydroacridines"

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Silva, Carlos F. M., Teresa Leão, Filipa Dias, et al. "Structure–Activity Relationship Studies of 9-Alkylamino-1,2,3,4-tetrahydroacridines against Leishmania (Leishmania) infantum Promastigotes." Pharmaceutics 15, no. 2 (2023): 669. http://dx.doi.org/10.3390/pharmaceutics15020669.

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Leishmaniasis is one of the most neglected diseases in modern times, mainly affecting people from developing countries of the tropics, subtropics and the Mediterranean basin, with approximately 350 million people considered at risk of developing this disease. The incidence of human leishmaniasis has increased over the past decades due to failing prevention and therapeutic measures—there are no vaccines and chemotherapy, which is problematic. Acridine derivatives constitute an interesting group of nitrogen-containing heterocyclic compounds associated with numerous bioactivities, with emphasis t
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Abdel-Mohsen, M. Soliman, M. Kamel Mohsen, F. Eweas Ahmad, Wietrzyk Joanna, Milczarek Magdalena, and S. Soliman Salwa. "Synthesis, Antiproliferative Activity and Molecular Docking of Some 9-Substituted 1,2,3,4-Tetrahydroacridine Derivatives against Breast Cancer Cell Line." Chemistry Research Journal 3, no. 2 (2018): 26–32. https://doi.org/10.5281/zenodo.13914532.

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Some new and known substituted 1,2,3,4-tetrahydroacridines incorporated at their position nine with various sulfa drug or thiosemicarbazide moieties were synthesized. Biologically, these compounds were investigated for their antiproliferative activity against human breast cancer (MCF-7) cell line and murine fibroblast normal cell line (BALB/3T3). The results were calculated as the IC<sub>50</sub> (inhibitory concentration 50% i.e. the concentration of tested compound which inhibits 50% of the cells population) compared with Cisplatin as control. Furthermore, a docking simulation study was carr
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Zhang, Weiwei, Yiwei Wang, Hui-Jing Li, et al. "Synergistic Inhibition Effect of 9-(4-Chlorophenyl)-1,2,3,4-tetrahydroacridines and Tween-80 for Mild Steel Corrosion in Acid Medium." Journal of Physical Chemistry C 123, no. 23 (2019): 14480–89. http://dx.doi.org/10.1021/acs.jpcc.9b02595.

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4

Farat, Oleg K., Victor I. Markov, Svetlana A. Varenichenko, Victor V. Dotsenko, and Alexander V. Mazepa. "The Vilsmeier–Haack formylation of 2,3-dihydro-4H-1,3-benzoxazin-4-ones and isomeric 1,2-dihydro-4H-3,1-benzoxazin-4-ones: an effective approach to functionalized 2H-/4H-chromenes and tetrahydroacridines." Tetrahedron 71, no. 34 (2015): 5554–61. http://dx.doi.org/10.1016/j.tet.2015.06.069.

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Farat, Oleg K., Victor I. Markov, Svetlana A. Varenichenko, Victor V. Dotsenko, and Alexander V. Mazepa. "ChemInform Abstract: The Vilsmeier-Haack Formylation of 2,3-Dihydro-4H-1,3-benzoxazin-4-ones and Isomeric 1,2-Dihydro-4H-3,1-benzoxazin-4-ones: An Effective Approach to Functionalized 2H-/4H-Chromenes and Tetrahydroacridines." ChemInform 46, no. 48 (2015): no. http://dx.doi.org/10.1002/chin.201548157.

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Smetanin, N. V., and A. V. Mazepa. "Functionalization of N-arylmaleimides by sp3 C–H bonds of hydroacridines(qinolines)." Voprosy Khimii i Khimicheskoi Tekhnologii, no. 6 (December 2020): 165–70. http://dx.doi.org/10.32434/0321-4095-2020-133-6-165-170.

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The catalyst-free sp3 C–H functionalization of tetrahydroacridine(quinolines) derivatives has been achieved using a Michael-type reaction with N-arylmaleimides. This method enables the facile synthesis of biologically important N-aryl bearing tetrahydroacridine(quinolines) moieties in a single step with high yields. The reaction occurs under non-catalytic conditions by heating of hydroacridines(quinolines) in DMSO within 4 h at 100–1200C. The reaction between starting compounds allows synthesizing (3S/4R)-3-[(3R/4S)-9-chloroacridine(quinoline)-4-yl]-1(-N-aryl)pyrrolidine-2,5-diones with a good
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7

Walker, TM, B. Starr, BB Dewhurst, and C. Atterwill. "Potential neurotoxicity of a novel aminoacridine analogue." Human & Experimental Toxicology 14, no. 6 (1995): 469–74. http://dx.doi.org/10.1177/096032719501400601.

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1 A class of compounds, 9-aminoacridines, have long been known to be reversible inhibitors of acetyl cholinesterase (AChE - EC 3.1.1.7), the most familiar of which is 9-amino-1,2,3,4-tetrahydroacridine (Tacrine). 2 A novel aminoacridine was synthesised: - 2-tertiary butyl-9-amino-1,2,3,4-tetrahydroacridine (2tBuTHA). 3 In vitro comparisons of the acetylcholinesterase inhibitory potential and neurotoxicity compared to Tacrine were performed using a chemically differentiated neuroblastoma cell line (Neuro 2A). 2tBuTHA, but not Tacrine, was cytotoxic to the neural cell following 20 h exposure, de
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8

Odabaşoğlu, Mustafa, Muharrem Kaya, Orhan Büyükgüngör, and Yılmaz Yıldırır. "10-(4-Bromophenyl)-9-(4-methoxyphenyl)-3,3,6,6-tetramethyl-3,4,6,7-tetrahydroacridine-1,8(2H,5H,9H,10H)-dione." Acta Crystallographica Section E Structure Reports Online 63, no. 5 (2007): o2162—o2164. http://dx.doi.org/10.1107/s1600536807014729.

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9

Chen, Yan, Wen-Juan Hao, Zi-Qiang Tang, Bo Jiang, and Chun-Mei Li. "10-(4-Chlorophenyl)-9-(4-methoxyphenyl)-3,3,6,6-tetramethyl-3,4,6,7-tetrahydroacridine-1,8(2H,5H,9H,10H)-dione." Acta Crystallographica Section E Structure Reports Online 63, no. 10 (2007): o3934. http://dx.doi.org/10.1107/s1600536807042365.

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10

Patočka, Jiří, Daniel Jun, and Kamil Kuča. "In vitro Inactivation of Rat Brain Acetylcholinesterase by DSP-4 and Its Derivatives OS-21 and OS-23 and Protective Activity of Tacrine (9-Amino-1,2,3,4-tetrahydroacridine)." Acta Medica (Hradec Kralove, Czech Republic) 48, no. 3-4 (2005): 145–48. http://dx.doi.org/10.14712/18059694.2018.42.

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Tertiary N-haloethylamines are able to cyclize to the corresponding aziridinium ions. The inhibitory activity of the DSP-4 (N-(o-brombenzyl)-N-ethyl-2-chlorethylamine) and its two derivatives OS-21 (N-benzyl-N-ethyl-2-chloroethylamine) and OS-23 (N-fenylethyl-N-ethyl-2-chloroethylamine) was studied toward rat brain acetylcholinesterase (AChE) in vitro. The influence of the THA (tacrine; 9–amino-1,2,3,4–tetrahydroacridine) on AChE inhibition by these substances was also evaluated. The results demonstrated that all of three aziridinium compounds formed in solution caused a timeand concentration-
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Book chapters on the topic "4-tetrahydroacridines"

1

"Rational design, synthesis and biological evaluation of dual- binding reversible inhibitors of cholinesterase’s with mild inhibitory potency toward monoamine oxidase B." In Book of Abstracts - RAD 2025 Conference. RAD Centre, Niš, Serbia, 2025. https://doi.org/10.21175/rad.abstr.book.2025.21.3.

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Alzheimer’s disease (AD) is neurodegenerative disease that is the cause of 60-70% of dementia cases. The major symptoms of AD involve progressive decline of cognitive and motor skills, caused by neuropathological changes, including elevation of oxidative stress, shrinkage of neurons, formation of Aβ plaques and neurofibrillary tangles in the central nervous system (CNS) and disruption of glutamatergic and cholinergic neurotransmission systems. In AD, the nerve terminal disruption is observed in immediate vicinity of Aβ plaques. Peripheral ionic site of AChE promotes aggregation of Aβ peptides
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