Relevant bibliographies by topics / 4-thiadiazole derivatives

Contents

  1. Journal articles
  2. Book chapters
  3. Conference papers

Academic literature on the topic '4-thiadiazole derivatives'

Author: Grafiati
Published: 4 June 2025
Last updated: 1 August 2025

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic '4-thiadiazole derivatives.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "4-thiadiazole derivatives"

1

A. Ameen, Husam, and Ahlam J. Qasir. "Synthesis and Preliminary Antimicrobial Study of 2-Amino-5-Mercapto-1,3,4-Thiadiazole Derivatives." Iraqi Journal of Pharmaceutical Sciences ( P-ISSN 1683 - 3597 E-ISSN 2521 - 3512) 21, no. 1 (2017): 98–104. http://dx.doi.org/10.31351/vol21iss1pp98-104.

Full text
Abstract:
Nitrogen heterocycles are of a special interest because they constitute an important class of natural and non natural products, many of which exhibit useful biological activities.Among these nitrogen heterocycles are 1, 3, 4-thiadiazole containing compounds. The therapeutic effects of these derivatives have been well studied for a number of pathological conditions including inflammation, pain, or hypertension. Moreover, synthesis of thiadiazoles has attracted wide-spread attention due to their diverse applications as antibacterial, anticancer, antifungal anti-inflammatory and antidepressant ag
APA, Harvard, Vancouver, ISO, and other styles
2

Singh, S., and Amandeep Kaur. "SYNTHESIS AND ANTICANCER ACTIVITY OF NOVEL 2-BENZYL-6- (SUBSTITUTED PHENYL)-IMIDAZO[2,1-B] [1,3,4] THIADIAZOLE DERIVATIVES." INDIAN DRUGS 56, no. 04 (2019): 13–20. http://dx.doi.org/10.53879/id.56.04.11454.

Full text
Abstract:
A new series of 2-benzyl-6-(substituted phenyl)-imidazo[2,1-b][1,3,4] thiadiazoles (S1-S8) was synthesized as potential anti-cancer agents. These compounds were evaluated for their anticancer activity against various cancer cell lines. The anticancer activity data reveals that the compounds S1 (2-benzyl- 6-phenylimidazo[2,1-b][1,3,4]thiadiazole) showed maximum growth inhibition against CNS cancer cell lines while the compounds S2 (2-benzyl-6-(4-chlorophenyl) imidazo[2,1-b][1,3,4] thiadiazole) and S3 (2-benzyl-6-(2,4-dichlorophenyl)imidazo[2,1-b][1,3,4] thiadiazole) showed maximum inhibition ag
APA, Harvard, Vancouver, ISO, and other styles
3

Rakhmonov, R., Sh Sharipov, M. Odilzoda, B. Safarov, A. Kobilzoda, and A. Abdurakhmonov. "SYNTHESIS AND FUNCTIONALIZATION OF SOME PARA-R-PHENYLIMIDAZO[2,1-B][1,3,4]- THIADIAZOLE DERIVATIVES." East European Scientific Journal 1, no. 4(68) (2021): 54–61. http://dx.doi.org/10.31618/essa.2782-1994.2021.1.68.15.

Full text
Abstract:
The article describes the synthesis of new modifications of derivatives of 6-phenyl-, 6-piodophenyl- and 6-p-bromophenylimidazo[2,1-b][1,3,4]-thiadiazoles - N -((6-(4-iodophenyl)-2-R-imidazo[2,1-b][1,3,4]-thiadiazol-5-yl)methyl)-alkyl/ heterylamine based on the Mannich reaction, bromination 2((ethylsulfonyl)methyl)-6-phenylimidazo[2,1-b][1,3,4]-thiadiazole and the structure of the resulting compounds was established on the basis of IR spectroscopy. It was shown that the presence of substituents at the 2-nd position of the thiadiazole fragment and substituents at the 5th and 6th positions of th
APA, Harvard, Vancouver, ISO, and other styles
4

Zain Alabdeen, Khalid. "The Activity of 1,3,4 Thiadiazole Derivatives on the Soluble Oils." Journal of Petroleum Research and Studies 2, no. 1 (2021): 59–88. http://dx.doi.org/10.52716/jprs.v2i1.34.

Full text
Abstract:
That Thiadiazoles derivative is biologically active as antimicrobial agents in cooling fluids.
 Derivatives of 1, 3, 4- thiadiazole have prepared:
 
 2-amino-3-[(2-amino-1, 3, 4-thiadiazol-5-yl) dithio] propanoic acid.
 2-(2-Carbethoxyamino-1, 3, 4-thiadiazol-5-yl)-thio acetic acid.
 [(5-amino-1,3,4-thiadiazol-2-yl) dithio] acetic acid
 
 The synthesized compounds have been used as antimicrobial against the microorganisms which have been found in the cooling fluid of industrial
 purposes by using media culture the results showed that the compounds 1 and
APA, Harvard, Vancouver, ISO, and other styles
5

Zhao, Yuxiang, Peter J. McCarthy, and Cyril Párkányi. "Synthesis and In Vitro Evaluation of Novel Acyclic and Cyclic Nucleoside Analogs with a Thiadiazole Ring." ISRN Organic Chemistry 2013 (March 5, 2013): 1–10. http://dx.doi.org/10.1155/2013/159164.

Full text
Abstract:
The synthesis of six thiadiazole nucleoside analogs is reported: 5-diacetylamino-1,2,4-thiadiazol-3-one (1), 5-amino-2- (tetrahydrofuran-2-yl)-1,2,4-thiadiazol-3-one (2), 5-amino-3-[(2′-hydroxyethoxy)methyl]-1,3,4-thiadiazol-2-one (3), 5-amino-3-(4′-hydroxy-2′-hydroxymethyl-butyl)-1,3,4-thiadiazole-2-thione (4), (R)-5-amino-3-(2′,3′-dihydroxypropyl)-1,3,4-thiadiazole-2-thione (5), and (S)-5-amino-3-(2′,3′-dihydroxypropyl)-1,3,4-thiadiazole-2-thione (6). The synthesis, characterization, and properties of these new synthesized thiadiazole derivatives are discussed. A dimerization of 5-amino-3H-1
APA, Harvard, Vancouver, ISO, and other styles
6

Yu, Lu, Lingling Xiao, Pei Li, Jiyan Chi, Jie Li, and Shuming Tan. "Synthesis and Bioactivity Evaluation of Novel Thiochroman-4-One Derivatives Incorporating Carboxamide and 1, 3, 4-Thiadiazole Thioether Moieties." Journal of Chemistry 2022 (February 26, 2022): 1–7. http://dx.doi.org/10.1155/2022/5354088.

Full text
Abstract:
A series of novel thiochroman-4-one derivatives incorporating carboxamide and 1, 3, 4-thiadiazole thioether moieties were synthesized. Bioassay results indicated that the EC50 values of compound 6-chloro-N-(5-(methylthio)-1, 3, 4-thiadiazol-2-yl)-4-oxothiochromane-2-carboxamide (5a) against Xanthomonas oryzae pv. Oryzae (Xoo) and Xanthomonas axonopodis pv. Citri (Xac) were 24 and 30 μg/mL, respectively, which were even better than those of bismerthiazol and thiadiazole copper. Meanwhile, compound 6-methyl-4-oxo-N-(5-(propylthio)-1, 3, 4-thiadiazol-2-yl)thiochromane-2-carboxamide (5m) showed a
APA, Harvard, Vancouver, ISO, and other styles
7

Ergena, Asrat, Yerra Rajeshwar, and Gebremedhin Solomon. "Synthesis and Diuretic Activity of Substituted 1,3,4-Thiadiazoles." Scientifica 2022 (April 8, 2022): 1–9. http://dx.doi.org/10.1155/2022/3011531.

Full text
Abstract:
1,3,4-Thiadiazole nuclease, a 5-membered heterocyclic ring system containing two nitrogen and one sulfur atoms in addition to carbon atoms, is compound that showed promising results in the process of searching new diuretic agents. In this study, seven 5- and 2-thioate derivatives of 1, 3, 4-thiadiazoles were synthesized by substitution reaction using acetone as solvent and K2CO3 as a base. The compounds ware then characterized by using IR and NMR spectroscopy. The diuretic activity of the compounds was evaluated on Swiss albino mice by measuring urine volume, urinary pH, and urinary Na+, K+, a
APA, Harvard, Vancouver, ISO, and other styles
8

Ammar Ferman Abbood. "Synthesis, Characterization and Molecular Docking Study of New 1,3,4-Thiadiazole Derivatives." Journal of Wasit for Science and Medicine 17, no. 3 (2024): 26–38. http://dx.doi.org/10.31185/jwsm.503.

Full text
Abstract:
In this study, a series of 5-(5-{(Z)-[(4-R1)methylidene]amino}-1,3,4-thiadiazol-2-yl)benzene-1,2,3-triol (L1-3), and 4-(5-{(Z)-[(4-R1)methylidene]amino}-1,3,4-thiadiazol-2-yl)benzene-1,2-diol (L4-6) compounds were synthesized, where R1 = 4-Nitro, 4-bromo, 4-chloro. The reaction between benzoic acid derivatives and hydrazinecarbothioamide in the basic medium gave the intended products with high yield and purity. The preparation of the compounds was confirmed by spectroscopic measurements in addition to physical properties. The biological properties of the prepared compounds were studied by mole
APA, Harvard, Vancouver, ISO, and other styles
9

JOHNSON, REEJA, JOBY THOMAS KAKKASSERY, Vinod Raphael Palayoor, Ragi Kooliyat, and Vidhya Thomas Kannanaikkal. "Experimental and Theoretical Investigations on the Corrosion Inhibition action of Thiadiazole Derivatives on Carbon Steel in 1M HCl medium." Oriental Journal Of Chemistry 36, no. 6 (2020): 1179–88. http://dx.doi.org/10.13005/ojc/360624.

Full text
Abstract:
Novel thiadiazole derivatives of Schiff bases namely (E)-N-(anthracen-9-ylmethylene)-5-(4-nitrophenyl)-1,3,4-thiadiazol-2-amine (A9CNPTDA) and N-(anthracen-9(10H)-ylidene)-5-(4-nitrophenyl)-1,3,4-thiadiazol-2-amine (ANNPTDA) were synthesized, characterized and corrosion inhibition behaviour, as well as the mechanism of inhibition were investigated by different monitoring techniques like gravimetric measurements, electrochemical impedance spectroscopy, potentiodynamic polarization, quantum chemical and SEM studies. Both of the thiadiazole derivatives showed excellent corrosion inhibitor action
APA, Harvard, Vancouver, ISO, and other styles
10

Shein, Anatoliy B., Mariya D. Plotnikova, and Alexander E. Rubtsov. "PROTECTIVE PROPERTIES OF SOME THIADIAZOLE DERIVATIVES IN SULFURIC ACID SOLUTIONS." IZVESTIYA VYSSHIKH UCHEBNYKH ZAVEDENII KHIMIYA KHIMICHESKAYA TEKHNOLOGIYA 62, no. 7 (2019): 123–29. http://dx.doi.org/10.6060/ivkkt.20196207.5968.

Full text
Abstract:
The work presents the results of the study of some thiadiazole derivatives as corrosion inhibitors for mild steel in 5-20% H2SO4. Gravimetric tests and electrochemical studies were performed on low-carbon steel St3 at ambient temperature. The exposure time of the samples was 24 h. Polarization curves were obtained by potentiodynamic method (v = 1 mV/s) in a three-electrode cell, using the SOLARTRON 1280 C electrochemical measuring complex. The following thiadiazole derivatives were studied: (E)-N,N-dimethyl-4-{[(5-phenyl-1,3,4-thiadiazol-2-yl)imino]methyl}aniline, (E)-5-{[4-(dimethylamino)benz
APA, Harvard, Vancouver, ISO, and other styles
More sources

Book chapters on the topic "4-thiadiazole derivatives"

1

Palekar, Vikrant Sudhakar, and Kulbhushan A. Sasane. "Examining Biological Relevence of Thiazolo Thiadiazole and Thiazolo Thiazole Fused Heterocyles." In Advances in Bioinformatics and Biomedical Engineering. IGI Global, 2024. http://dx.doi.org/10.4018/979-8-3693-7520-4.ch005.

Full text
Abstract:
Aromatic Fused heterocycles containing Nitrogen (N) and Sulfur(S) has extraordinary bioactive behavior due to which they are attracting the interest of chemists worldwide & thus used as a potential material in medicinal/pharmaceutical industries. The nitrogen-sulphur fused heterocycles attracting attention of the researchers due to number of biological and pharmacological activities and observed to exhibit extensive applications in drug discovery and development. The efforts are made to understand biological activity based on position of heteroatom & the substituent present in 5-member
APA, Harvard, Vancouver, ISO, and other styles

Conference papers on the topic "4-thiadiazole derivatives"

1

Dimić, Dušan, Dejan Milenković, Edina Avdović, Goran Kaluđerović, and Jasmina Dimitrić Marković. "MOLECULAR DOCKING AND MOLECULAR DYNAMICS STUDIES OF THE INTERACTION BETWEEN COUMARIN-NEUROTRANSMITTER DERIVATIVES AND CARBONIC ANHYDRASE IX." In 1st INTERNATIONAL Conference on Chemo and BioInformatics. Institute for Information Technologies, University of Kragujevac,, 2021. http://dx.doi.org/10.46793/iccbi21.056d.

Full text
Abstract:
Novel biologically active compounds can be obtained by the structural modification of coumarins. In this contribution, five new derivatives of 4-hydroxycoumarin with tyramine, octopamine, norepinephrine, 3-methoxytyramine, and dopamine were obtained. Their structures were optimized based on the previously obtained crystal structure of the 4-hydroxycoumarin-dopamine derivative. The special emphasis was put on the effect of various substituents on the structure of obtained compounds and intramolecular interactions governing the stability. To investigate their possible antitumor activity, molecul
APA, Harvard, Vancouver, ISO, and other styles
2

Abbas, Haneen Hadi, and Zeid Hassan Abood. "Microwave synthesis and antibacterial assay of new 1,3-thiazolidin-4-one derivatives based on 2-amino-5-mercapto-1,3,4-thiadiazole." In 4TH INTERNATIONAL SCIENTIFIC CONFERENCE OF ALKAFEEL UNIVERSITY (ISCKU 2022). AIP Publishing, 2023. http://dx.doi.org/10.1063/5.0181971.

Full text
APA, Harvard, Vancouver, ISO, and other styles
3

Raj, Vinit, Sudipta Saha, amit rai, Mahendra Singh, Durgesh Kumar, and Anil Kumar Sahdev. "Homology modeling, Molecular Dynamic Simulation and in silico screening of Activator for the Intensification of human sirtuin type 1 (SIRT1) by novel 1, 3, 4-thiadiazole derivatives-A potential antiaging approach." In MOL2NET, International Conference on Multidisciplinary Sciences. MDPI, 2015. http://dx.doi.org/10.3390/mol2net-1-b019.

Full text
APA, Harvard, Vancouver, ISO, and other styles
4

Nikalje, Anna Pratima, Julio Seijas Vázquez, Shailee Tiwari, and Zahid Zaheer. "Ultrasound-promoted One-Pot, Three Component Synthesis Of Novel 5-Amino-2-(4-Chlorophenyl)-7- Substituted Phenyl-8,8a-Dihydro-7H-[1,3,4]Thiadiazolo[3,2-A]Pyrimidine-6-Carbonitrile Derivatives." In The 19th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2015. http://dx.doi.org/10.3390/ecsoc-19-a048.

Full text
APA, Harvard, Vancouver, ISO, and other styles
You might also be interested in the extended bibliographies on the topic '4-thiadiazole derivatives' for particular source types:
Journal articles
We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!

To the bibliography