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Relevant bibliographies by topics / Actinobacteria ; Quinolone antibacterial agents – Synthesis

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Journal articles
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Academic literature on the topic 'Actinobacteria ; Quinolone antibacterial agents – Synthesis'

Author: Grafiati

Published: 4 June 2021

Last updated: 12 February 2022

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Journal articles on the topic "Actinobacteria ; Quinolone antibacterial agents – Synthesis"

1

Jinbo, Yoshikazu, Hirosato Kondo, Masahiro Taguchi, Yoshimasa Inoue, Fumio Sakamoto, and Goro Tsukamoto. "Synthesis and Antibacterial Activity of Thiazolopyrazine-Incorporated Tetracyclic Quinolone Antibacterial Agents. 2." Journal of Medicinal Chemistry 37, no. 17 (1994): 2791–96. http://dx.doi.org/10.1021/jm00043a018.

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2

Cooper, Curt S., Michael D. Tufano, Pamela K. Donner, and Daniel T. W. Chu. "The synthesis and in vitro antibacterial activity of conformationally restricted quinolone antibacterial agents." Bioorganic & Medicinal Chemistry 4, no. 8 (1996): 1307–15. http://dx.doi.org/10.1016/0968-0896(96)00106-x.

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3

Chu, Daniel T. W., Prabhavathi B. Fernandes, and Andre G. Pernet. "Synthesis and biological activity of benzothiazolo[3,2-a]quinolone antibacterial agents." Journal of Medicinal Chemistry 29, no. 8 (1986): 1531–34. http://dx.doi.org/10.1021/jm00158a037.

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4

Patel, Mehul M., and Laxman J. Patel. "Design, Synthesis, Molecular Docking, and Antibacterial Evaluation of Some Novel Flouroquinolone Derivatives as Potent Antibacterial Agent." Scientific World Journal 2014 (2014): 1–10. http://dx.doi.org/10.1155/2014/897187.

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Objective. Quinolone moiety is an important class of nitrogen containing heterocycles widely used as key building blocks for medicinal agents. It exhibits a wide spectrum of pharmacophores and has bactericidal, antiviral, antimalarial, and anticancer activities. In view of the reported antimicrobial activity of various fluoroquinolones, the importance of the C-7 substituents is that they exhibit potent antimicrobial activities. Our objective was to synthesize newer quinolone analogues with increasing bulk at C-7 position of the main 6-fluoroquinolone scaffold to produce the target compounds wh

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5

Fedorowicz, Joanna, Jarosław Sączewski, Agnieszka Konopacka, et al. "Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents." European Journal of Medicinal Chemistry 179 (October 2019): 576–90. http://dx.doi.org/10.1016/j.ejmech.2019.06.071.

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6

Fu, Hai-Gen, Zhi-Wen Li, Xin-Xin Hu, et al. "Synthesis and Biological Evaluation of Quinoline Derivatives as a Novel Class of Broad-Spectrum Antibacterial Agents." Molecules 24, no. 3 (2019): 548. http://dx.doi.org/10.3390/molecules24030548.

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Nineteen new quinoline derivatives were prepared via the Mannich reaction and evaluated for their antibacterial activities against both Gram-positive (G+) and Gram-negative (G−) bacteria, taking compound 1 as the lead. Among the target compounds, quinolone coupled hybrid 5d exerted the potential effect against most of the tested G+ and G− strains with MIC values of 0.125–8 μg/mL, much better than those of 1. Molecular-docking assay showed that compound 5d might target both bacterial LptA and Top IV proteins, thereby displaying a broad-spectrum antibacterial effect. This hybridization strategy

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7

Daneshtalab, Mohsen, and Abeer Ahmed. "Nonclassical Biological Activities of Quinolone Derivatives." Journal of Pharmacy & Pharmaceutical Sciences 15, no. 1 (2011): 52. http://dx.doi.org/10.18433/j3302n.

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Quinolones are considered as a big family of multi-faceted drugs; their chemical synthesis is flexible and can be easily adapted to prepare new congeners with rationally devised structures. This is shown by the description of many thousands of derivatives in the literature. Scientists could accurately describe their QSAR, which is essential for effective drug design. This also gave them the chance to discover new and unprecedented activities, which makes quinolones an endless source of hope and enables further development of new clinically useful drugs. Quinolones are among the most comm

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8

Khamkhenshorngphanuch, Thitiphong, Kittipat Kulkraisri, Alongkorn Janjamratsaeng, et al. "Synthesis and Antimicrobial Activity of Novel 4-Hydroxy-2-quinolone Analogs." Molecules 25, no. 13 (2020): 3059. http://dx.doi.org/10.3390/molecules25133059.

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Alkyl quinolone has been proven to be a privileged scaffold in the antimicrobial drug discovery pipeline. In this study, a series of new 4-hydroxy-2-quinolinone analogs containing a long alkyl side chain at C-3 and a broad range of substituents on the C-6 and C-7 positions were synthesized. The antibacterial and antifungal activities of these analogs against Staphylococcus aureus, Escherichia coli, and Aspergillus flavus were investigated. The structure-activity relationship study revealed that the length of the alkyl chain, as well as the type of substituent, has a dramatic impact on the anti

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9

Michael, Joseph P., Charles B. de Koning, Gladys D. Hosken, and Trevor V. Stanbury. "Reformatsky reactions with N-arylpyrrolidine-2-thiones: synthesis of tricyclic analogues of quinolone antibacterial agents." Tetrahedron 57, no. 47 (2001): 9635–48. http://dx.doi.org/10.1016/s0040-4020(01)00964-4.

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10

Kamal, Ahmed, S. Ahmed, M. A. Khan, Rajesh Shetty, B. Siddhardha, and U. Murty. "Synthesis and Biological Evaluation of a New Series of Benzothiazole-Quinolone Hybrids as Antibacterial Agents." Letters in Drug Design & Discovery 5, no. 5 (2008): 353–57. http://dx.doi.org/10.2174/157018008784912072.

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Dissertations / Theses on the topic "Actinobacteria ; Quinolone antibacterial agents – Synthesis"

1

Salvaggio, Flavia. "Synthesis of biologically active quinolone natural products extracted from the actinomycete Pseudonocardia sp. CL38489." Thesis, University of Cambridge, 2014. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.648770.

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2

Ndaba, Hlengiwe Glenrose. "Microwave as an energy source in the synthesis of 2-aryl-4-quinolone alkaloids and naphthyridines." Thesis, 2011. http://hdl.handle.net/10321/704.

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Thesis submitted in fulfilment of the requirements for the Degree of Masters of Technology: Organic Chemistry, Durban University of Technology, 2011.<br>One of the greatest medical challenges facing mankind is the Human Immunodeficiency Virus/Acquired Immunodeficiency Syndrome (HIV/AIDS) which has now become a major epidemic with more than 40 million people infected worldwide. Of equal concern is its implication in high mortality and the onset of a number of opportunist mycobacterial infections, principally tuberculosis. In spite of the discovery of some relatively effective antiretroviral

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