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Journal articles on the topic 'Amino-substituted'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Widler, Leo, Knut A. Jaeggi, and Jonathan R. Green. "Amino-Substituted GEM-Bisphosphonates." Phosphorus, Sulfur, and Silicon and the Related Elements 144, no. 1 (1999): 5–8. http://dx.doi.org/10.1080/10426509908546168.

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2

Mathew, Abraham E., Robert K. Y. Zee-Cheng, and C. C. Cheng. "Amino-substituted p-benzoquinones." Journal of Medicinal Chemistry 29, no. 9 (1986): 1792–95. http://dx.doi.org/10.1021/jm00159a041.

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3

Barlin, GB, FL Tian, B. Kotecka, and KH Rieckmann. "Potential Antimalarials. XVI. 4'-Chloro-3-[7″-chloro(and trifluoromethyl)quinolin-4″-yl]amino-5-(substituted amino)methylbiphenyl-4-ols and 4'-Bromo(and 3'-trifluoromethyl)-3-(substituted amino)methyl-5-(7″-trifluoromethylquinolin-4″-yl)aminobiphenyl-2-ols." Australian Journal of Chemistry 45, no. 11 (1992): 1845. http://dx.doi.org/10.1071/ch9921845.

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Twenty-four mono-Mannich bases of the general formulae 4'-chloro-3-[7″-chloro(and trifluoro-methyl)quinolin-4'-yl]amino-5-(substituted amino)methylbiphenyl-4-ols and 4'-bromo(and 3'- trifluoromethyl-3(substituted amino)methyl-5(7″-trifluoromethylquinolin-4″-yl) aminobiphenyl-2-ols have been prepared by condensation of the 4-chloro heterocycle with 5-amino-3-(N-substituted amino)methyl-4'-chlorobiphenyl-4-ols or 5-amino-3-(N-substituted amino)methyl- 4'-bromo(or 3'-trifluoromethyl)biphenyl-2-ols. The antimalarial activity of these products in in vitro tests against Plasmodium falciparum reveals

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4

Hussain, Sabir, Jyoti Sharma, and Mohd Amir. "Synthesis and Antimicrobial Activities of 1,2,4-Triazole and 1,3,4-Thiadiazole Derivatives of 5-Amino-2-Hydroxybenzoic Acid." E-Journal of Chemistry 5, no. 4 (2008): 963–68. http://dx.doi.org/10.1155/2008/924734.

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Various 4-amino-2-[4-(4-substituted phenyl)-5-sulfanyl-4H-1,2,4-triazol-3-yl] phenol (4a-c), 4-amino-2-{4-amino-5-[(4-substituted phenyl)amino]-4H-1,2,4-triazol-3-yl} phenol (5a-c) and 4-amino-2-{5-[(4-substituted phenyl)amino]-1,3,4-thiadiazole-2-yl} phenol (6a-g) were synthesized and evaluated for their antibacterial and antifungal activity. The compounds showed significant antibacterial activity againstS. aureus(gram-positive) andE.coli(gram-negative) bacteria and antifungal activity againstA. nigerfungi using cup plate technique

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5

Padmaja, Pannala, Pedavenkatagari Narayana Reddy, and Bijaya Ketan Sahoo. "A Green Approach to the Synthesis of Novel Indole Substituted 2-Amino- 4,5-dihydro-3-furancarbonitriles in Water." Letters in Organic Chemistry 16, no. 3 (2019): 209–14. http://dx.doi.org/10.2174/1570178615666180917104820.

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2-Amino-4,5-dihydro-3-furancarbonitriles (ADFCs) have attracted much attention due to their utility as valuable synthetic intermediates for the preparation of a series of acyclic and cyclic organic compounds. On the other hand, indoles substituted with furans are highly interesting compounds displaying a wide range of biological and pharmaceutical activities. However, to the best of our knowledge, indole substituted 2-amino-4,5-dihydro-3-furancarbonitriles have not been previously reported. A new and efficient synthesis of indole substituted 2-amino-4,5-dihydro-3-furancarbonitriles has been de

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6

Jain, Sonika, Anamika Sharma, Meenakshi Agrawal, Swapnil Sharma, Jaya Dwivedi, and D. Kishore. "Synthesis and Antimicrobial Evaluation of Some Novel Trisubstituted s-Triazine Derivatives Based on Isatinimino, Sulphonamido, and Azacarbazole." Journal of Chemistry 2013 (2013): 1–9. http://dx.doi.org/10.1155/2013/925439.

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A study directed towards exploring the temperature-dependent reactivity of the chlorine atoms of 2,4,6-trichloro-s-triazine (TCT) in the nucleophilic displacement reaction, allowed a facile replacement of its chlorine atoms in succession with (i) N-amino methyl substituted isatin-3-hydrazones, (ii) N1-substituted-4-amino benzene sulphonamides, and (iii) 8-amino-4-oxo-N-benzyl-azacarbazole to produce the corresponding 2,4,6-trisubstituted-s-triazine, namely; 2-(N-amino methyl substituted isatin-3-hydrazinyl)-4-(N1-substituted-4′-amino benzenesulfonamidyl)-6-(8′-amino-4′-oxo-N-benzylazacarbazoly

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7

Srivastav, Manish, MD Salahuddin, and S. M. Shantakumar. "Synthesis and Anti-inflammatory Activity of Some Novel 3-(6-Substituted-1, 3-benzothiazole-2-yl)-2-[{(4-substituted phenyl) amino} methyl] quinazolines-4 (3H)-ones." E-Journal of Chemistry 6, no. 4 (2009): 1055–62. http://dx.doi.org/10.1155/2009/507052.

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A series of novel 3-(6-substituted-1, 3-benzothiazole-2-yl)-2-[{(4-substituted phenyl) amino} methyl] quinazolines-4(3H)-ones were synthesized by treating 2-(chloromethyl)-3-(6-substituted-1, 3-benzothiazole-2-yl) quinazoline-4-(3H)-one (IIa-d) with various substituted amine. The compounds (IIa-d) prepared by treating 2-[(chloroacetyl) amino] benzoic acid with different 2-amino-6-substituted benzothiazole. Elemental analysis, IR,1HNMR and mass spectral data confirmed the structure of the newly synthesized compounds. Synthesized quinazolines-4-one derivative were investigated for their anti-inf

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8

Archana. "SYNTHESIS AND EVALUATION OF SOME NEWER QUINAZOLINONYL SUBSTITUTED BENZOXAZEPINYL / BENZOTHIAZEPINYL INDOLES AS POTENT ANTICONVULSANT AGENTS." INDIAN DRUGS 56, no. 03 (2019): 18–24. http://dx.doi.org/10.53879/id.56.03.11538.

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new series of 3-[3-amino-2-methyl-6-substituted quinazolin-4(3H)-onyl chalconyl)-2-substituted indoles (3-8), 3-[3-Amino-2-methyl-6- substituted quinazolin-4(3H) -onyl-benzoxazepin/benzo -thiazepin- 2-yl] -2-substituted indoles (9-20) and 3-[3-amino-2-methyl-6-substituted quinazolin-4(3H) -onyl-3- (sub-stituted phenylaminomethylene) -benzoxazepin/benzothizepin-2-yl] -2-substitutedindoles (21-44) were synthesised and evaluated for anticonvulsant activity. All these compounds were screened in vivo, for their anticonvulsant activity and acute toxicity. Coumpund 44 , 3-[3-amino-2-methyl-6-bromoqui

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9

Keshk, Eman M., Emad M. El-Telbani, and H. Abdel-Rahman. "Synthesis of Some New Furocoumarins and their Usage in Peptide Synthesis." Zeitschrift für Naturforschung B 58, no. 12 (2003): 1237–41. http://dx.doi.org/10.1515/znb-2003-1214.

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1,5-Benzodiazepin-2-ones (3a - d) were obtained fromω-carbethoxy visnaginone or ω-carbethoxy khellinone and substituted 1,2-phenylenediamines. Reactions of active nitriles such as malononitrile and ethyl cyanoacetate with substituted 6-dimethylaminomethylene furocoumarins (4a,b) are described. Additionally, reaction of substituted 6-dimethylaminomethylene furocoumarins with different amino acids gave furochromen-6-ylidenemethyl amino acids (7 - 9). Compound 7 was coupled with glycine ethyl ester to form amino acetic acid ethyl ester (10).

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10

El-Naggar, Mohamed, Abdel-Nasser El-Shorbagi, Dina H. Elnaggar, Abd El-Galil E. Amr, Mohamed A. Al-Omar, and Elsayed A. Elsayed. "Synthesis, Characterization, and Cytotoxic Evaluation of Some Newly Substituted Diazene Candidates." Journal of Chemistry 2018 (November 1, 2018): 1–9. http://dx.doi.org/10.1155/2018/3626824.

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A series of azocompounds containing methyl salicylate 4a–k and 1-naphthyl moiety 6–8 was synthesized and tested as anticancer agents. Nitrosation of methyl 5-amino-2-hydroxybenzoate or 1-aminonaphthalene by using NaNO2 in the presence of HCl afforded diazonium salt derivatives 2 and 5, which were treated with substituted imino or substituted amino derivatives, to give the corresponding substituted amino-pent-2-en-3-yl-diazenylbenzoate 4a–k or 2-substituted-1-(naphthalen-1-yl)diazene derivatives 6a–h, 7a,b, and 8a,b. All the synthesized compounds were elucidated by elemental analysis and spectr

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11

Holle, Sigrid, and Peter W. Jolly. "Amino-substituted cyclopentadienyl cobalt complexes." Journal of Organometallic Chemistry 605, no. 2 (2000): 157–67. http://dx.doi.org/10.1016/s0022-328x(00)00244-8.

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12

Burck, Sebastian, Dietrich Gudat, Falk Lissner, Kalle Nättinen, Martin Nieger, and Thomas Schleid. "2-Amino-substituted 1,3,2-Diazaphospholenes." Zeitschrift für anorganische und allgemeine Chemie 631, no. 13-14 (2005): 2738–45. http://dx.doi.org/10.1002/zaac.200500120.

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13

Walstra, P., W. P. Trompen, and J. Th Hackmann. "Amino-substituted glyoximes and furoxans." Recueil des Travaux Chimiques des Pays-Bas 87, no. 4 (2010): 452–60. http://dx.doi.org/10.1002/recl.19680870413.

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14

Appel, Rolf, and Michael Poppe. "A Stable Amino-Substituted Phosphaalkyne." Angewandte Chemie International Edition in English 28, no. 1 (1989): 53–54. http://dx.doi.org/10.1002/anie.198900531.

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15

Ju Liu, Ju Liu, Jian Tao Shi Jian Tao Shi, Xue Chen Hao Xue Chen Hao, Yu Tong Liu Yu Tong Liu, Shi Ding Shi Ding, and Yang Wang and Ye Chen Yang Wang and Ye Chen. "Synthesis of New Substituted 2-amino-4H-benzo[h]chromene-3-carbonitrile Derivatives." Journal of the chemical society of pakistan 41, no. 5 (2019): 888. http://dx.doi.org/10.52568/000795/jcsp/41.05.2019.

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A series of novel substituted 2-amino-4H-benzo[h]chromene-3-carbonitrile derivatives was synthesised by condensation of different halogen derivatives with the hydroxy-group of 2-amino-8-hydroxy-4-styryl- 4H-benzo[h]chromene-3-carbonitrile and 2-amino-8-hydroxy-4- phenethyl-4H-benzo-[h]chromene-3-carbonitrile, which were prepared from cinnamaldehyde, malononitrile and naphthalene-1,6-diol through Knoevenagel condensation and cyclization reaction and then reduction with hydrogen in the presence of Pd/C at room temperature. Each intermediates and target compounds were obtained in good yields.

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16

Mandour, Adel, Eslam El-Sawy, Manal Ebaid, and Seham Hassan. "Synthesis and potential biological activity of some novel 3-[(N-substituted indol-3-yl)methyleneamino]-6-amino-4-aryl-pyrano(2,3-c)pyrazole-5-carbonitriles and 3,6-diamino-4-(N-substituted indol-3-yl)pyrano(2,3-c)pyrazole-5-carbonitriles." Acta Pharmaceutica 62, no. 1 (2012): 15–30. http://dx.doi.org/10.2478/v10007-012-0007-0.

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Synthesis and potential biological activity of some novel 3-[(N-substituted indol-3-yl)methyleneamino]-6-amino-4-aryl-pyrano(2,3-c)pyrazole-5-carbonitriles and 3,6-diamino-4-(N-substituted indol-3-yl)pyrano(2,3-c)pyrazole-5-carbonitriles Starting from N-substituted indole-3-carboxaldehydes (1a-g) a series of new 3-[(N-substituted indol-3-yl)methyleneamino]-6-amino-4-aryl-pyrano(2,3-c)pyrazole-5-carbonitriles (3a-g and 4a-g) have been synthesized via the acid catalyzed condensation reaction of 1a-g with 3-amino-5-pyrazolone, followed by the reaction with arylidene malononitriles. A series of ne

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17

Lyčka, Antonín, Libuše Havlíčková, Alois Koloničný, and Josef Jirman. "15N NMR study of amino-imino tautomerism in derivatives of 1,4-bis(substituted amino)-9,10-anthraquinones and 1,4-bis(substituted amino)-2,3-dihydro-9,10-anthraquinones." Collection of Czechoslovak Chemical Communications 52, no. 3 (1987): 736–41. http://dx.doi.org/10.1135/cccc19870736.

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The 15N chemical shifts and 1J(15N, H) coupling constants of 1,4-bis(substituted amino)-9,10-anthraquinones and 1,4-bis(substituted amino)-2,3-dihydro-9,10-anthraquinones indicate that these derivatives exist as true aminoderivatives except for 1,4-bis(phenylamino)-2,3-dihydro-9,10-anthraquinone which forms a tautomeric mixture of the amino and imino forms in deuteriochloroform and hexadeuteriodimethyl sulphoxide.

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18

Kharlamova, Alisa D., Anton S. Abel, Alexei D. Averin, et al. "Mono- and Diamination of 4,6-Dichloropyrimidine, 2,6-Dichloropyrazine and 1,3-Dichloroisoquinoline with Adamantane-Containing Amines." Molecules 26, no. 7 (2021): 1910. http://dx.doi.org/10.3390/molecules26071910.

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N-heteroaryl substituted adamantane-containing amines are of substantial interest for their perspective antiviral and psychotherapeutic activities. Chlorine atom at alpha-position of N-heterocycles has been substituted by the amino group using convenient nucleophilic substitution reactions with a series of adamantylalkylamines. The prototropic equilibrium in these compounds was studied using NMR spectroscopy. The introduction of the second amino substituent in 4-amino-6-chloropyrimidine, 2-amino-chloropyrazine, and 1-amino-3-chloroisoquinoline was achieved using Pd(0) catalysis.

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19

Vijay, Kumar Salvi, Pemawat Gangotri, Bapna Archita, and L. Talesara G. "Synthesis, characterization and antimicrobial activity of substituted 3-(phthalazine-1-ylamino)alkanoic acid containing imidoxy moiety." Journal of Indian Chemical Society Vol. 86, May 2009 (2009): 491–97. https://doi.org/10.5281/zenodo.5810168.

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Synthetic Organic Chemistry Research Laboratory, Department of Chemistry, M. L. Sukhadia University, Udaipur-313 001, Rajasthan, India <em>E-mail</em> : gtalesara@yahoo.com <em>Manuscript received 12 May 2008, revised 16 January 2009, accepted 20 January 2009</em> Hydrozinolysis of phthalyl derivatives of amino acid la-c afforded [(4-oxo-3,4-dihydrophthalazine-1- yl)amino]substituted acetic acid 2a-c, which on reaction with POCI<sub>3</sub>/PCI<sub>5</sub> gave ((4-chlorophahalazine-1-yl)amino]substituted acetic acid 3a-c. This when condensed with <em>N</em>-hydroxyphthalimide/ N-hydroxysuccin

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20

Berkessel, Albrecht, Serap Eröksüz, and Jörg Neudörfl. "Kinetic Resolution of 5-Substituted Oxazinones with Bifunctional Chiral Base/Squaramide Organocatalysts." Synlett 28, no. 11 (2017): 1278–81. http://dx.doi.org/10.1055/s-0036-1588852.

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5-Substituted oxazinones provide N-protected β2-amino acid esters upon alcoholytic ring opening. Thus far, this access to enantiopure β2-amino acids has been restricted to the use of enzymes (hydrolases) as catalysts for the kinetic resolution of racemic 5-substituted oxazinones, and branched alkyl or ortho-substituted aryl groups on the substrate oxazinone’s 5-position were typically not tolerated. We herein report that certain bifunctional chiral base/squaramide organocatalysts, in particular those derived from cis-1,2-diaminocyclohexane or 9-amino-9-epi-quinine, allow the first organocataly

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21

Mistry, K. M., and K. R. Desai. "Synthesis of Novel Heterocyclic 4-Thiazolidinone Derivatives and their Antibacterial Activity." E-Journal of Chemistry 1, no. 4 (2004): 189–93. http://dx.doi.org/10.1155/2004/590439.

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4-Thiazolidinones have been prepared by the reaction of various substituted Schiff bases 3 with Thioglycolic acid and Thiolactic acid. The intermediate Schiff bases 3 were synthesized by the condensation of various substituted 2-amino benzothiazole 1 with 1-(4'-methyl Phenyl)-3-methyl-5-pyrazolone 2. The starting compound substituted 2-amino benzothiazoles were prepared from various substituted amines via substituted phenyl thiourea. The structures of the compounds have been confirmed by elemental analysis and spectral analysis. The antibacterial activity of the compounds has also been screene

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22

L'abbé, Gerrit, Maria Bruynseels, Linda Beenaerts, Anna Vandendriessche, Pieter Delbeke, and Suzanne Toppet. "Synthesis of 1-Amino-5-(Substituted)Amino-1,2,3-Triazoles." Bulletin des Sociétés Chimiques Belges 98, no. 5 (2010): 343–47. http://dx.doi.org/10.1002/bscb.19890980509.

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23

Kumar, Sanjeev. "Synthesis of Some 2-Amino-5-Substituted-1,3,4-Oxadiazoles Through the Electrooxidation of Semicarbazone." Journal of the Korean Chemical Society 53, no. 2 (2009): 159–65. http://dx.doi.org/10.5012/jkcs.2009.53.2.159.

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24

Omar, Parvin Mirdamat. "METABOLISM OF NEUROMEDIATORY AMINO ACIDS IN DIFFERENT BRAIN DIVISIONS." Deutsche internationale Zeitschrift für zeitgenössische Wissenschaft 60 (July 18, 2023): 16–17. https://doi.org/10.5281/zenodo.8161055.

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The morpho-functional differentiation and maturation of different departments of the brain are accompanied by changes in the amount of number of biologically active substances, amino acids, proteins, and lipids. When studying the protein metabolism occurring in nerve tissue, it was determined that this tissue contains many substituted and non-substituted amino acids and enzymes involved in amino acid metabolism. These indicate that amino acid metabolism and protein biosynthesis occur with particular intensity in nervous tissue.

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25

Sharma, L. K., S. Kumar, S. Singh, and R. K. P. Singh. "Electrochemical synthesis of 5-substituted-2-amino (substituted amino)-1,3,4-oxadiazoles at the platinum electrode." Russian Journal of Electrochemistry 46, no. 1 (2010): 34–40. http://dx.doi.org/10.1134/s1023193510010040.

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26

Rajeswar Rao, V., M. S. Rao, and T. V. Padmanabha Rao. "A novel synthesis of thiazolyl, imidazothiadiazolyl, and thiadiazinyl-2H-1-benzopyran-2-ones." Collection of Czechoslovak Chemical Communications 51, no. 10 (1986): 2214–21. http://dx.doi.org/10.1135/cccc19862214.

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3-Acetylcoumarins I with arylthiourea in the presence of iodine gave substituted 3-(2-arylamino-4-thiazolyl)-2H-1-benzopyran-2-ones (IIa-IIc). The structures of these products have been confirmed and they were converted into acetyl derivatives (IId-IIf). Condensation of various 3-(2-bromoacetyl)-2H-1-benzopyran-2-ones (III) with 2-amino-6-substituted thiadiazoles IV in the presence of ethanol and dimethylformamide yielded substituted 3-(2-substituted imidazo[2,1-b]thiadiazol-6-yl)-2H-1-benzopyran-2-ones (VI). Reaction of III with 3-substituted 4-amino-5-mercapto-S-triazole VII resulted in the

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27

D.T.Tayade*, R. D. Thombare S.A. Waghmare. "SYNTHESIS OF 3-[4-AMINO-N-SUBSTITUTED-o-ANISAMIDO- 5-YL]AMINO-5-SUBSTITUTED-1,2,4-DITHIAZOLE." Indo American Journal of Pharmaceutical Sciences 04, no. 10 (2017): 3890–94. https://doi.org/10.5281/zenodo.1035231.

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A novel series of 3-{4-Amino-N-[2-(dithethylamino)ethyl-o-anisamido-5-yl}amino-5-substitutedimino-1,2,4- dithiazole was synthesized by the oxidative cyclization of 4-amino-5-substituteddithiobiureto-N-[2- (dithethylamino)ethyl-o-anisamide in chloroform medium by making the use of liquid bromine as oxidizing agent. The products were characterized and justified on the basis of elemental analysis, chemical characteristics and spectral studies. Keywords:3-{4-Amino-N-[2-(dithethylamino)ethyl-o-anisamido-5-yl}amino-5-substituted -imino-1,2,4-dithiazole, 4- amino-5-substituteddithiobiureto-N-[2-(dith

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28

Nemeryuk, Michal P., Andrej L. Sedov, Tamara S. Safonova, Antonín Černý, and Jiří Křepelka. "Transformations of substituted 5-aminopyrimidines under conditions of the diazotization." Collection of Czechoslovak Chemical Communications 51, no. 1 (1986): 215–33. http://dx.doi.org/10.1135/cccc19860215.

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Reaction of nitrous acid with 4-substituted and 4,6-substituted 5-aminopyrimidines Ia-In produces 4-substituted and 4,5-disubstituted 1,2,3-triazoles IIa-IIv,resp. Under similar conditions, 2,5-diaminopyrimidines XIIa-XIId give N(7)-oxides of 2-amino-4-aralkylthiopyrimido[5,4-d]-1,2,3-triazines XIIIa-XIIId, and 5-amino-4-chloropyrimidines In and X give 2-diazocyanoacetamides XIa and XIb resp. Also described are syntheses of 5-formylaminopyrimidines XVa-XVg from glycine ethyl ester via sodium salt XVI.

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29

Diez-Martinez, Alba, and Ramanarayanan Krishnamurthy. "Investigations towards the Synthesis of 5-Amino-l-lyxofuranosides and 4-Amino-lyxopyranosides and NMR Analysis." SynOpen 01, no. 01 (2017): 0029–40. http://dx.doi.org/10.1055/s-0036-1588859.

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The reactivity of trifluoromethanesulfonyl esters derived from l-lyxofuranosides and l-lyxopyranosides was investigated with various 5-aminopyrimidines as nucleophiles with the expectation to synthesize N-substituted 5-amino-ribosugars. The lyxopyranoside forms were found to be unreactive, while the lyxofuranoside forms were found to be reactive with 5-aminopyrimidines, yielding novel N-substituted 5-amino-lyxofuranosides. We report on the synthesis of these novel N-substituted lyxofuranosides and the systematic analyses of NMR data that demonstrate trends within each series: furano-, pyrano-,

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30

Pawar, P. Y., P. M. Gaikwad, and P. H. Balani. "Microwave Assisted Synthesis of N-Substituted-7-hydroxy-4-methyl-2-oxoquinolines as Anticonvulsant Agents." E-Journal of Chemistry 8, no. 2 (2011): 945–51. http://dx.doi.org/10.1155/2011/121476.

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The reaction of resorcinol with ethylacetoacetate yielded the 7-hydroxy-4-methyl coumarin (1), which on treatment with benzidine gives 1-(4ʹ-amino-biphenyl-4-yl)-7-hydroxy-4-methyl-1H-quinolin-2-one (2). 1-{4ʹ-[(Substituted benzylidene)-amino]-biphenyl-4-yl}-7-hydroxy-4-methyl-1H-quinolin-2-one (3a-j) were obtained by reacting 1-(4ʹ-amino-biphenyl-4-yl)-7-hydroxy-4-methyl-1H-quinolin-2-one (2) with different substituted aromatic aldehydes in presence of glacial acetic acid by microwave irradiation. The compound 1-{4ɴ-[(substituted benzylidene)-amino]-biphenyl-4-yl}-7-hydroxy-4-methyl-1H-quinol

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31

Cooper, Gary F. "Synthesis of Substituted 1,3-Propanesultams fromN-Substituted 2-Amino Alcohols." Synthesis 1991, no. 10 (1991): 859–60. http://dx.doi.org/10.1055/s-1991-26593.

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32

Shakh, Yuriy, Mykhaylo Slesarchuk, Vadym Syngaevsky, et al. "Interaction of 5-Substituted 1,4-Naphthoquinones and Amino Thiotriazoles: Reaction Ways and Regioselectivity." Chemistry & Chemical Technology 12, no. 2 (2018): 167–75. http://dx.doi.org/10.23939/chcht12.02.167.

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33

Balatoni, Istvan, Johann Hlina, Rainer Zitz, Alexander Pöcheim, Judith Baumgartner та Christoph Marschner. "β-Amino- and Alkoxy-Substituted Disilanides". Molecules 24, № 21 (2019): 3823. http://dx.doi.org/10.3390/molecules24213823.

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Our recent study on formal halide adducts of disilenes led to the investigation of the synthesis and properties of β-fluoro- and chlorodisilanides. The reaction of the functionalized neopentasilanes (Me3Si)3SiSiPh2NEt2 and (Me3Si)3SiSiMe2OMe with KOtBu in the presence of 18-crown-6 provided access to structurally related β-alkoxy- and amino-substituted disilanides. The obtained Et2NPh2Si(Me3Si)2SiK·18-crown-6 was converted to a magnesium silanide and further on to Et2NPh2Si(Me3Si)2Si-substituted ziroconocene and hafnocene chlorides. In addition, an example of a silanide containing both Et2NPh2

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34

Armoush, Nicola, Preeti Syal, and Daniel P. Becker. "Synthesis of Substituted 2‐Amino‐cyclobutanones." Synthetic Communications 38, no. 11 (2008): 1679–87. http://dx.doi.org/10.1080/00397910801981110.

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35

Chavez, David, Megan Breiner, Thomas Myers, and Richard Gilardi. "1,2,4,5-Tetrazinyl-Substituted Amino-1,2,4,5-Tetrazines." Synlett 26, no. 04 (2015): 557–60. http://dx.doi.org/10.1055/s-0034-1379615.

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36

Bargamov, G. G., and M. D. Bargamova. "Polyfluoroalkyl- substituted 1-amino-1,2,3-triazoles." Journal of Fluorine Chemistry 79, no. 1 (1996): 45–47. http://dx.doi.org/10.1016/0022-1139(96)03446-x.

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37

Piao, Ming-Zhu, and Kimiaki Imafuku. "Convenient synthesis of amino-substituted pyranopyranones." Tetrahedron Letters 38, no. 30 (1997): 5301–2. http://dx.doi.org/10.1016/s0040-4039(97)01184-2.

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38

Rádl, Stanislav, Petr Hezký, Jitka Urbánková, Petr Váchal, and Ivan Krejčí. "Synthesis and Analgesic Activity of Some 1-Benzofurans, 1-Benzothiophenes and Indoles." Collection of Czechoslovak Chemical Communications 65, no. 2 (2000): 280–96. http://dx.doi.org/10.1135/cccc20000280.

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3-Unsubstituted 1-benzofurans 1e and 1f, 3-methyl-1-benzofurans 1a-1d, and 3-amino-1-benzofurans 2a-2l, as well as 3-amino-1-benzothiophenes 3a, 3b and 3-aminoindoles 4a-4f, 11a, and 11b were prepared and tested as analgesics. The 3-amino-1-benzofurans 2 were prepared from the corresponding 2-hydroxybenzonitriles 5 and phenacyl bromides 6 via intermediates 7. Similar treatment of 2-sulfanylbenzonitrile (8) provided 3-amino-1-benzothiophenes 3. Appropriately substituted 2-aminobenzonitriles 9 then provided N-substituted 3-aminoindoles 4. 1-(Ethoxycarbonyl)indoles 4e and 4f were successfully dep

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39

Yang, Minmin, and Stewart W. Schneller. "Amino substituted derivatives of 5′-amino-5′-deoxy-5′-noraristeromycin." Bioorganic & Medicinal Chemistry 13, no. 3 (2005): 877–82. http://dx.doi.org/10.1016/j.bmc.2004.10.031.

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40

D.K. Gautam and I. Singh. "A NEW SERIES OF 1,3,4-THIADIAZOLE SUBSTITUTED AZETIDINONE AND THIAZOLIDINONE DERIVATIVES AND THEIR ANTIMICROBIAL ACTIVITY." RASAYAN Journal of Chemistry 17, no. 01 (2024): 176–82. http://dx.doi.org/10.31788/rjc.2024.1718308.

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The new series of 2-({[5-(3-chloro-2-oxo-4-substituted-phenylazetidin-1-yl)-1,3,4-thiadiazol-2- yl]methyl}amino)benzoic acid (13-20) and 2-({[5-(4-oxo-2- substituted-phenyl-1,3-thiazolidin-3-yl)- 1,3,4- thiadiazol-2-yl]methyl}amino)benzoic acid (21-28) have been synthesized from 2-[({5-[(benzylideneamino]- 1,3,4- thiadiazol-2-yl }methyl)amino]-benzoic acid (5-12). All these synthesized compounds were tested for their antimicrobial activity and established by spectroscopic data, and elemental analyses.

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41

Gupta, Apoorva, and Anand K. Halve. "Synthesis & Antifungal Screening of Novel Azetidin-2-ones." Open Chemistry Journal 2, no. 1 (2015): 1–6. http://dx.doi.org/10.2174/1874842201502010001.

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A new series of 4-[3-chloro-2-(4-hydroxy-3-methoxybenzyllidene)-4-oxoazetidin-1-yl]amino-N-(substituted)benzenesulfonamide, 4-{3-chloro-2-[5-methoxy-2-nitro-4-(prop-2-en-1-yloxy)benz yllidene]-4-oxoazetidin-1-yl}]amino}-N-(substituted)benzenesulfonamide and 4-{3-chloro-2-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)benzylidene]-4-oxoazetidin-1-yl}amino}-N-(substituted) benzenesulfonamide were synthesized using appropriate synthetic route. The chemical structures of all the synthesized compounds were deduced on the basis of elemental analysis and spectroscopic data. The antifungal activity of the syn

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42

Yengoyan, Aleksandr P., Vergush A. Pivazyan, Emma A. Ghazaryan, and Zhermen A. Azaryan. "Synthesis of Novel 2-Amino-substituted 6-Methyl-pyrimidin-4-ol Derivatives and Their Biological Evaluation." Letters in Organic Chemistry 16, no. 7 (2019): 575–83. http://dx.doi.org/10.2174/1570178615666181025120951.

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A series of novel derivatives based on 2-amino-substituted 4-methylpyrimidin-4-ols were synthesized by simple, accessible and efficient methods. 4-N-triazolyl derivatives were obtained from the corresponding 4-chloro derivatives, and O-substituted products, including compounds with a combination of the pyrimidine and oxadiazole rings in the molecule, were synthesized from the sodium salts of 2-amino-substituted pyrimidin-4-ols. The synthesized compounds showed a pronounced stimulating action on plants growth. Their growth stimulant activities were in the range of 46-93% compared to heteroauxin

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43

Šinkovec, Rok, Uroš Grošelj, Benjamin Prek, et al. "A simple synthesis of dimethyl 2-[(Z)-3-amino-1-oxo-1-(substituted)but-2-en-2-yl]fumarates: potential intermediates in the synthesis of polysubstituted five- and six-membered heterocycles." Zeitschrift für Naturforschung B 71, no. 6 (2016): 677–82. http://dx.doi.org/10.1515/znb-2016-0017.

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AbstractIn this communication, a simple synthesis of dimethyl 2-[(Z)-3-amino-1-oxo-1-(substituted)but-2-en-2-yl]fumarates is described. Methyl ketones were transformed by treatment with N,N-dimethylacetamide dimethyl acetal (DMADMA) into 3-dimethylamino-1-(substituted)but-2-en-1-ones, followed by treatment with ammonium acetate into (Z)-3-amino-1-(substituted)but-2-en-1-ones and addition to dimethyl acetylenedicarboxylate. These novel polysubstituted butadienes are potential intermediates for the metal-free preparation of polysubstituted five- and six-membered heterocycles.

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44

(Miss), MAITREYEE DEBI. "Synthesis of some 2,4-Diamino-6-substituted-aminopyrimidines and some related 5 - Arylazopyrimidines." Journal of Indian Chemical Society Vol. 64, Oct 1987 (1987): 612–15. https://doi.org/10.5281/zenodo.6198779.

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Department of Chemical Technology, University Colleges of Science and Technology, University of Calcutta, Calcutta-700 009 <em>Manuscript received 12 February 1986, revised 6 April 1987, accepted 7 August 1987</em> Synthesis of some 2,4-diamino-6-(substituted-amino)pyrimidines (2) and 2,4- diamino-5-(substituted-phenylazo)-6-(substituted-amino)pyrimidines (3) are described. Compounds 2a — e were synthesised by condensation of 2,4-diamino-6-chloropyrimi-dine (1) with the appropriate aromatic amines, and compounds 3a —u by coupling 2  with diazotised arylamines.

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45

Koner, Abhishek, Spencer C. Serin, Gregor Schnakenburg, Brian O. Patrick, Derek P. Gates, and Rainer Streubel. "Exploring the chemistry of backbone amino(chloro)phosphanyl-substituted imidazole-2-thiones." Dalton Transactions 46, no. 31 (2017): 10504–14. http://dx.doi.org/10.1039/c7dt01859b.

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46

Zhou, Jin, Canliang Fang, Ying Liu та ін. "Visible-light-induced cleavage of 4-α-amino acid substituted naphthalimides and its application in DNA photocleavage". Organic & Biomolecular Chemistry 13, № 13 (2015): 3931–35. http://dx.doi.org/10.1039/c5ob00302d.

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4-α-Amino acid substituted naphthalimides can be photocleaved at the C–N bond between the 4-amino and the amino acid residue under visible light irradiation, releasing a fluorophore, 4-aminonaphthalimide.

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47

Gera, Ankur, Chander Mohan, and Sandeep Arora. "Synthesis of Phthaloylglycyl Hydrazide Derivatives: Selective Protection of Phthalimide Group from Hydrazinolysis." Current Organic Synthesis 15, no. 6 (2018): 839–45. http://dx.doi.org/10.2174/1570179415666180601083256.

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Background: N-phthalimide amino acid hydrazide is a class of compounds that have the potential therapeutic use. In general, hydrazinolysis of N-substituted amino acid(s) ester removes the ester group and yields the corresponding hydrazide. However, in case if N-substitution group is phthalimide, phthalimide group is cleaved and not the ester group. The resulted compound, therefore, is amino acid ester rather than Nphthalimide amino acid hydrazide. The above class of compounds, because of susceptibility of phthalimide group to hydrazinolysis, has previously been synthesized by a lengthy three-s

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48

Bakherad, Mohammad, Vahid Keley, and Amir H. Amin. "Synthesis of a Novel Heterocyclic Ring System: Imidazo[3,2-D] [1,2,4]Triazolo[3,4-B][1,3,4]Thiadiazine." Journal of Chemical Research 2008, no. 11 (2008): 633–34. http://dx.doi.org/10.3184/030823408x371236.

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Synthesis of the novel compounds 3-substituted-6-arylimidazo[3,2-d][1,2,4]triazolo[3,4-b][1,3,4]thiadiazines was achieved by the reaction of 6-amino-3-substituted-7H-[1,2,4]triazolo[3,4-jb][1,3,4]thiadiazines with 4-substituted-phenacyl bromides in refluxing ethanol.

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49

Alpatova, Victoria M., Evgeny G. Rys, Elena G. Kononova, and Valentina A. Ol'shevskaya. "Synthesis of new representatives of A₃B-type carboranylporphyrins based on meso-tetra(pentafluorophenyl)porphyrin transformations." Beilstein Journal of Organic Chemistry 20 (April 12, 2024): 767–76. http://dx.doi.org/10.3762/bjoc.20.70.

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A carboranylporphyrin of A3B-type bearing a single pentafluorophenyl ring was prepared through the regioselective nucleophilic aromatic substitution reaction of the p-fluorine atoms in 5,10,15,20-tetrakis(pentafluorophenyl)porphyrin with 9-mercapto-m-carborane. The reaction of this porphyrin with sodium azide led to the selective substitution of the p-fluorine atom in the pentafluorophenyl substituent with an azide functionality which upon reduction with SnCl2 resulted in the formation of the corresponding porphyrin with an amino group. Pentafluorophenyl-substituted A3B-porphyrins were studied

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50

Janeba, Zlatko, Antonín Holý, and Milena Masojídková. "Synthesis of Acyclic Nucleoside and Nucleotide Analogs Derived from 6-Amino-7H-purine-8(9H)-thione and 8-(Methylsulfanyl)adenine." Collection of Czechoslovak Chemical Communications 65, no. 11 (2000): 1698–712. http://dx.doi.org/10.1135/cccc20001698.

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Reaction of 8-bromoadenine derivatives 1 with thiourea in ethanol or butanol was used for the synthesis of the corresponding N9-substituted 6-amino-7H-purine-8(9H)-thiones 2. 8-(Methylsulfanyl)adenine derivatives 3 were prepared by reaction of thiones 2 with iodomethane in 1 M sodium methoxide or in aqueous 1.5 M potassium hydroxide. Alkylation of 6-amino-7H-purine-8(9H)-thione (2a) proceeds preferentially on the sulfur atom. Under similar conditions, alkylation of 8-(methylsulfanyl)adenine (3a) with diverse alkylation agents afforded N9-substituted adenine derivatives 3 and 6, and N3-substitu

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