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Relevant bibliographies by topics / Benzamidine derivative

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Dissertations / Theses
Book chapters
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Academic literature on the topic 'Benzamidine derivative'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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Journal articles on the topic "Benzamidine derivative"

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Eick, Sigrun, Wolfgang Pfister, Uta Stürzebecher, Sigrid Jarema, and Jörg Stürzebecher. "Inhibitors of benzamidine type influence the virulence properties of Porphyromonas gingivalis strains." Acta Biochimica Polonica 50, no. 3 (2003): 725–34. http://dx.doi.org/10.18388/abp.2003_3663.

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Synthetic inhibitors of benzamidine type have been found to have inhibiting effects on arginine specific cysteine proteinases of P. gingivalis. The purpose of our study was to assess the effects of these inhibitors on the virulence properties of two P. gingivalis strains, the reference strain ATCC 33277 and JH16-1, a clinical isolate obtained from a patient with severe periodontitis. The inhibitors tested were pentamidine, benzamidine, three bis-benzamidine derivatives with a pentamidine-related structure, one bis-benzamidine derivative with another structure, and one arginine derivative as a

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Sa’ad, Mohammad Auwal, Ramasamy Kavitha, Shivkanya Fuloria, Neeraj Kumar Fuloria, Manickam Ravichandran, and Pattabhiraman Lalitha. "Synthesis, Characterization and Biological Evaluation of Novel Benzamidine Derivatives: Newer Antibiotics for Periodontitis Treatment." Antibiotics 11, no. 2 (2022): 207. http://dx.doi.org/10.3390/antibiotics11020207.

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Periodontal disease (PD) is complex polymicrobial disease which destroys tooth-supporting tissue. Although various synthetic inhibitors of periodontitis-triggering pathogens have been recognized, their undesirable side effects limit their application. Hence, the present study intended to perform the synthesis, characterization, antimicrobial evaluation, and cytotoxicity analysis of novel benzamidine analogues (NBA). This study involved the synthesis of novel imino bases of benzamidine (4a–c), by reacting different aromatic aldehydes with 2-(4-carbamimidoylphenoxy) acetohydrazide (3), which was

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Jain, A., M. A. Sa'ad, S. Ugrappa, et al. "Synthesis, Characterization and Biological Evaluation of New Benzamidine Derivatives: Antibiotics for Periimplantitis Causing Pathogen." Asian Journal of Chemistry 35, no. 8 (2023): 1927–31. http://dx.doi.org/10.14233/ajchem.2023.28022.

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Periimplantitis (PI) is complex polymicrobial disease, which destroys implant-supporting tissue. Although facts suggest several synthetic inhibitors of periimplantitis causing bacteria (PCB), but the undesirable side effects of them limits their application. Hence, current investigation was intended to carry out the synthesis, characterization, in vitro antimicrobial evaluation and cytotoxicity (cell viability) analysis of new benzamidine derivatives (NBDs) against periimplantitis causing bacteria. Present study involved synthesis of 2-(4-((4-substituted)carbamothioyl)phenoxy)-N-(4-substituted

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Nishimura, Yasuhiko, Wataru Yasui, Kazuhiro Yoshida, Toshiya Matsuyama, Kiyohiko Dohi, and Eiichi Tahara. "A Serine Protease-inhibitory Benzamidine Derivative Inhibits the Growth of Human Colon Carcinoma Cells." Japanese Journal of Cancer Research 83, no. 7 (1992): 723–28. http://dx.doi.org/10.1111/j.1349-7006.1992.tb01972.x.

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Kantlehner, Willi, Jochen Mezger, Ralf Kreß, and Wolfgang Frey. "Orthoamide und Iminiumsalze, XCII. Synthese und Reaktionen von Orthoamiden aus ethinylierten Terpenderivatena." Zeitschrift für Naturforschung B 73, no. 7 (2018): 437–55. http://dx.doi.org/10.1515/znb-2018-0011.

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Abstract β-Ionone and camphor were ethynylated to give the alkynols 14, 16, 17 which can be transformed to the alkynolethers 5b, 5i, 5j, 5k, 5l, 5m by treatment with dimethylsulfate and chlorotrimethylsilane, respectively. From the alkynolethers 5h, 5i, 5j/5k, 5l/5m the orthoamide derivatives 4h, 4i, 4j/4k, 4l/4m can be prepared by treatment with N,N,N′,N′,N″,N″-hexamethylguanidinium chloride (8) in the presence of sodium hydride. The orthoamides 4h, 4i react with the sulfonamide 30 under condensation yielding the N-sulfonylated acrylamidines 31, 32. From the orthoamide 4h and p-nitroaniline t

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Salchert, Katrin, Marie-Françoise Gouzy, Maja Glorius, Anett Kühn, Mirko Nitschke, and Carsten Werner. "Immobilization of an anticoagulant benzamidine derivative: Effect of spacer arms and carrier hydrophobicity on thrombin binding." Acta Biomaterialia 1, no. 4 (2005): 441–49. http://dx.doi.org/10.1016/j.actbio.2005.04.001.

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Letari, Ornella, Catherine Booth, Albino Bonazzi, et al. "Efficacy of CR3294, a new benzamidine derivative, in the prevention of 5-fluorouracil-induced gastrointestinal mucositis and diarrhea in mice." Cancer Chemotherapy and Pharmacology 66, no. 5 (2009): 819–27. http://dx.doi.org/10.1007/s00280-009-1224-1.

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Jaafar, Mohammed Thamer, Luma Majeed Ahmed, and Rahman Tama Haiwal. "Synthesis, Characterization, and Electrochemical Study of Novel Porphyrin Derivatives as Corrosion Inhibitors for Carbon Steel in HCl Solutions." Indonesian Journal of Chemistry 24, no. 2 (2024): 379. http://dx.doi.org/10.22146/ijc.87682.

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This study involves the synthesis of some porphyrins derivatives, these are termed as 4,4',4'',4'''-(porphyrin-5,10,15,20-tetrayl)tetrakis(N-(6-aminoacridin-3-yl)benzamide) (3a), 4,4',4'',4'''-(porphyrin-5,10,15,20-tetrayl)tetrakis(N-(5-methoxybenzo[d]thiazol-2-yl)benzamide) (3b), 4,4'-(10,20-bis(3-hydroxyphenyl)porphyrin-5,15-diyl)bis(N-(6-aminoacridin-3yl)benzamide) (5a), and 4,4'-(10,20-bis(3-hydroxyphenyl)porphyrin-5,15-diyl)bis(N-(benzo[d]thiazol-2-yl)benzamide) (5b). These derivatives were synthesized using open circuit potential (OCP) and potentiodynamic polarization (PDP) in 0.1 M HCl

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PLESCIA, Janet, and Dario C. ALTIERI. "Activation of Mac-1 (CD11b/CD18)-bound factor X by released cathepsin G defines an alternative pathway of leucocyte initiation of coagulation." Biochemical Journal 319, no. 3 (1996): 873–79. http://dx.doi.org/10.1042/bj3190873.

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Leucocyte initiation of coagulation preserves the haemostatic balance and may aberrantly contribute to vascular injury. In addition to the extrinsic activation mediated by tissue factor: factor VIIa, monocytes express an alternative procoagulant response after binding of the zymogen factor X to the integrin Mac-1 (CD11b/CD18). Here, factor X-activating activity was found in purified monocyte granules, and coincided with size-chromatographed fractions containing cathepsin G. In contrast, elastase-containing granule fractions did not activate factor X. In the presence of Ca2+ ions, purified cath

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Li, Yawen, Ming-Kuan Chyan, Donald K. Hamlin, Holly Nguyen, Eva Corey, and D. Scott Wilbur. "Oxidation of p-[125I]Iodobenzoic Acid and p-[211At]Astatobenzoic Acid Derivatives and Evaluation In Vivo." International Journal of Molecular Sciences 23, no. 18 (2022): 10655. http://dx.doi.org/10.3390/ijms231810655.

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The alpha particle-emitting radionuclide astatine-211 (211At) is of interest for targeted radiotherapy; however, low in vivo stability of many 211At-labeled cancer-targeting molecules has limited its potential. As an alternative labeling method, we evaluated whether a specific type of astatinated aryl compound that has the At atom in a higher oxidation state might be stable to in vivo deastatination. In the research effort, para-iodobenzoic acid methyl ester and dPEG4-amino acid methyl ester derivatives were prepared as HPLC standards. The corresponding para-stannylbenzoic acid derivatives wer

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Dissertations / Theses on the topic "Benzamidine derivative"

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Fuller, S. J. "The mode of antibacterial action of 2-thiocyanatobenzamide and some of its derivatives." Thesis, University of Nottingham, 1986. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.371122.

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Bukataru, J. S. "The study of the derivatives of 2-benzamide-2-(2-oxoindolin-3-iliden) acetic acid on the antihypoxic activity under the conditions of hypobaric hypoxia." Thesis, Буковинський державний медичний університет, 2014. http://dspace.bsmu.edu.ua:8080/xmlui/handle/123456789/7915.

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Lin, Wan-Li, and 林萬里. "Development and biological characterization of 99m-Tc-labeled benzamide derivatives as imaging probes for melanoma." Thesis, 2014. http://ndltd.ncl.edu.tw/handle/74227584925641149880.

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碩士<br>國立陽明大學<br>生物醫學影像暨放射科學系<br>102<br>Malignant melanoma is one of the most lethal cancers due to its high cellular proliferation rate and the early occurrence of metastases. Melanoma is usually treated by surgery and support with radiotherapy and chemotherapy with metastasis, and late stage melanoma is lack of effective treatment, the development of new melanoma imaging probes is quite essential. Purpose: To synthesize 99mTc labeled benzamide derivatives, 5-Tc, 9-Tc and 12-Tc, are characterized to exhibit high binding to melanin and high hydrophilic for imaging melanoma tumors. Methods: The

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Chen, Yang-Yi, and 陳楊翊. "Development and biological characterization of 123/131I-labeled benzamide derivatives as novel theranostics for melanoma." Thesis, 2019. http://ndltd.ncl.edu.tw/handle/6yj24f.

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HAN-CHIH, CHANG, and 張瀚之. "Design and Synthesis of Amide/Amine Bridged Benzamide Derivatives and Establishing Their IKK Beta Inhibitory Activity." Thesis, 2014. http://ndltd.ncl.edu.tw/handle/36780066380948995417.

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碩士<br>東海大學<br>化學系<br>103<br>NF-κB (nuclear factor kappa-light-chain-enhancer of activated B cells) is a protein complex that controls transcription of DNA. When it is activated excessively, enhanced expression of pro-inflammatory cytokines such as TNF-α, lead to inflammatory and autoimmune diseases. The target was IKKβ, which play an key role in NF-κB signal pathway. We selected WY5107, which was designed from our Lab and has good inhibitory activity of IKKβ. In order to achieve better IKKβ inhibitory activity, we synthesis different bridges link WY5107 and another IKKβ inhibitor, IMD-0354, as

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Wheelhouse, Richard T., Terence C. Jenkins, Sharon A. Jennings, and Dimitrios Pletsas. "Design, Synthesis and Evaluation of Novel Biarylpyrimidines ¿ a New Class of Ligand for Unusual Nucleic Acid Structures." 2006. http://hdl.handle.net/10454/3150.

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No<br>Biarylpyrimidines are characterized as selective ligands for higher-order nucleic acid structures. A concise and efficient synthesis has been devised incorporating Suzuki biaryl cross-coupling of dihalopyrimidines. Two ligand series are described based on the parent thioether 4,6-bis[4-[[2-(dimethylamino)ethyl]mercapto]-phenyl]pyrimidine (la) and amide 4,6-bis(4[(2-(dimethylamino)ethyl)carboxamido]phenyl)pyrimidine (2a) compounds. In UV thermal denaturation studies with the poly(dA)·[poly(dT)]2 triplex structure, thioethers showed stabilization of the triplex form (¿Tm ¿ 20 °C). In contr

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Book chapters on the topic "Benzamidine derivative"

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Stürzebecher, Jörg, Helmut Vieweg, and Dagmar Prasa. "Inhibition of Glandular and Plasma Kallikrein by Benzamidine Derivatives." In Recent Progress on Kinins. Birkhäuser Basel, 1992. http://dx.doi.org/10.1007/978-3-0348-7321-5_25.

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Protais, P., M. Vasse, I. Dubuc, et al. "Dopaminergic Behavioral Responses and Classes of Binding Sites Distinguished by Discriminant Benzamide Derivatives." In Dopaminergic Systems and their Regulation. Palgrave Macmillan UK, 1986. http://dx.doi.org/10.1007/978-1-349-07431-0_9.

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Bockaert, J., L. Fagni, M. Sebben, and A. Dumuis. "Pharmacological Characterization of Brain 5-HT4 Receptors: Relationship between the Effects of Indole, Benzamide and Azabicycloalkybenzimidazolone Derivatives." In Serotonin: Molecular Biology, Receptors and Functional Effects. Birkhäuser Basel, 1991. http://dx.doi.org/10.1007/978-3-0348-7259-1_20.

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Stein, Lybak, and Ronald W. Pero. "Evaluation of the DNA damage and inhibition of DNA repair caused by the benzamide derivative Metoclopramide in human peripheral mononuclear leukocytes." In ADP-Ribosylation Reactions. Springer New York, 1992. http://dx.doi.org/10.1007/978-1-4419-8718-1_43.

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Stanovnik, B., and J. Svete. "By Elimination of Benzamide from Methyl 3-(Benzoylamino)-4,5-dihydro-3-pyrazole-3-carboxylate Derivatives." In Five-Membered Hetarenes with Two Nitrogen or Phosphorus Atoms. Georg Thieme Verlag KG, 2002. http://dx.doi.org/10.1055/sos-sd-012-00211.

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Argyropoulos, N. G. "1,6,6aλ-Trithia-3-azapentalenes by Oxygen–Sulfur Exchange Reactions of (1,2-Dithiol-3-ylidene)benzamide Derivatives." In Five-Membered Hetarenes with Three or More Heteroatoms. Georg Thieme Verlag KG, 2004. http://dx.doi.org/10.1055/sos-sd-013-00078.

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Conference papers on the topic "Benzamidine derivative"

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Cisneros, David, Eduardo Cueto, Tania Medina, et al. "Synthesis and SAR studies of a new trypanosome alternative oxidase inhibitors: imidazoline and benzamidine derivatives." In 7th International Electronic Conference on Medicinal Chemistry. MDPI, 2021. http://dx.doi.org/10.3390/ecmc2021-11520.

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Ienascu, Ioana M. C., Adina Cata, and Mariana N. Stefanut. "Antioxidant capacity of some new N-(2-bromophenyl)-2-hydroxy-benzamide derivatives." In 2017 E-Health and Bioengineering Conference (EHB). IEEE, 2017. http://dx.doi.org/10.1109/ehb.2017.7995376.

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Nikalje, Anna Pratima, Shailee Tiwari, Sumaiya Siddiqui, and Julio Seijas Vázquez. "Microwave-assisted Facile Synthesis And Anticancer Evaluation Of N-((5-(substituted Methylene Amino)- 1,3,4-thiadiazol-2-yl)methyl) Benzamide Derivatives." In The 20th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2016. http://dx.doi.org/10.3390/ecsoc-20-a010.

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