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Journal articles on the topic 'Boronic Acids/pharmacology'

Author: Grafiati

Published: 2 June 2025

Last updated: 31 July 2025

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1

Arvanitis, Costa, Trevor Rook, and Ian Macreadie. "Mechanism of Action of Potent Boron-Containing Antifungals." Current Bioactive Compounds 16, no. 5 (2020): 552–56. http://dx.doi.org/10.2174/1573407215666190308152952.

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Background: Boron is unusual to organic chemists, yet boron interacts greatly with organic biochemicals and has considerable bioactivity, especially as an antifungal and insecticide. The bestknown bioactive boron compounds are boric acid, its salt borax, and the closely related boronic acids. A newcomer is tavaborole (trade name Kerydin), recently developed and approved in 2014 for topical treatment of onychomycosis, a fungal infection of nails and the nail bed. It is timely to review the literature and explore the way in which these compounds may work. Methods: The focus of this review is to

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2

Han, Young Taek. "A Concise Synthesis of Rhodanthpyrone A and B, Natural 4-(Hydroxyphenyl)-substituted α-Pyrones". Natural Product Communications 12, № 1 (2017): 1934578X1701200. http://dx.doi.org/10.1177/1934578x1701200127.

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A concise synthesis of rhodanthpyrone A and B was accomplished via a Suzuki coupling reaction. To find the conditions appropriate to install hydroxyphenyl moieties to the α-pyrone skeleton, a model study was conducted using commercially available boronic acids. It was revealed that the hydroxy moiety of the phenylboronic acids should be concealed when reacted with labile 4-tosyl α-pyrone. Consequently, rhodanthpyrone A and B could be synthesized in high yields by Suzuki reaction using TIPS-protected arylboronic acids. This procedure provided a concise and versatile route for the synthesis of r

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3

Bassini, Emanuele, Stefano Gazzotti, Filomena Sannio та ін. "Isonitrile-Based Multicomponent Synthesis of β-Amino Boronic Acids as β-Lactamase Inhibitors". Antibiotics 9, № 5 (2020): 249. http://dx.doi.org/10.3390/antibiotics9050249.

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The application of various isonitrile-based multicomponent reactions to protected (2-oxoethyl)boronic acid (as the carbonyl component) is described. The Ugi reaction, both in the four components and in the four centers–three components versions, and the van Leusen reaction, proved effective at providing small libraries of MIDA-protected β-aminoboronic acids. The corresponding free β-aminoboronic acids, quantitatively recovered through basic mild deprotection, were found to be quite stable and were fully characterized, including by 11B-NMR spectroscopy. Single-crystal X-ray diffraction analysis

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4

Bosch, Eric, and Nate Schultheiss. "Facile Synthesis of Diarylpyrazines Using Suzuki Coupling of Dichloropyrazines with Aryl Boronic Acids." HETEROCYCLES 60, no. 8 (2003): 1891. http://dx.doi.org/10.3987/com-03-9789.

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5

Hayama, Noboru. "Asymmetric Hetero-Michael Additions to α,β-Unsaturated Carboxylic Acids by Multifunctional Boronic Acid Catalysts". YAKUGAKU ZASSHI 141, № 3 (2021): 293–301. http://dx.doi.org/10.1248/yakushi.20-00214.

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6

Matteson, Donald S. "α-Amido boronic acids: A synthetic challenge and their properties as serine protease inhibitors". Medicinal Research Reviews 28, № 2 (2007): 233–46. http://dx.doi.org/10.1002/med.20105.

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7

Kumar, Sandeep, and Arvind M. Kayastha. "Inhibition studies of soybean (Glycine max) urease with heavy metals, sodium salts of mineral acids, boric acid, and boronic acids." Journal of Enzyme Inhibition and Medicinal Chemistry 25, no. 5 (2009): 646–52. http://dx.doi.org/10.3109/14756360903468155.

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8

Hargrove, Amanda E., Andrew D. Ellington, Eric V. Anslyn, and Jonathan L. Sessler. "Chemical Functionalization of Oligodeoxynucleotides with Multiple Boronic Acids for the Polyvalent Binding of Saccharides." Bioconjugate Chemistry 22, no. 3 (2011): 388–96. http://dx.doi.org/10.1021/bc100376x.

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9

Boyd, Derek R., Narain D. Sharma, Peter A. Goodrich, et al. "Enantiopurity and absolute configuration determination of arenecis-dihydrodiol metabolites and derivatives using chiral boronic acids." Chirality 30, no. 1 (2017): 5–18. http://dx.doi.org/10.1002/chir.22764.

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10

Gorovoy, Alexey S., Olga Gozhina, John-Sigurd Svendsen та ін. "Syntheses and anti-tubercular activity ofβ-substituted andα,β-disubstituted peptidylβ-aminoboronates and boronic acids". Journal of Peptide Science 19, № 10 (2013): 613–18. http://dx.doi.org/10.1002/psc.2537.

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11

Kotsakis, S. D., E. Caselli, L. S. Tzouvelekis, E. Petinaki, F. Prati, and V. Miriagou. "Interactions of Oximino-Substituted Boronic Acids and -Lactams with the CMY-2-Derived Extended-Spectrum Cephalosporinases CMY-30 and CMY-42." Antimicrobial Agents and Chemotherapy 57, no. 2 (2012): 968–76. http://dx.doi.org/10.1128/aac.01620-12.

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12

Chao, Jianping, Yangzhi Ling, Xiaofeng Liu, Xuande Luo, and A. M. H. Brodie. "A versatile synthesis of 17-heteroaryl androstenes via palladium-mediated Suzuki cross-coupling with heteroaryl boronic acids." Steroids 71, no. 7 (2006): 585–90. http://dx.doi.org/10.1016/j.steroids.2006.02.004.

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13

Tafi, Andrea, Mariangela Agamennone, Paolo Tortorella, Stefano Alcaro, Carlo Gallina та Maurizio Botta. "AMBER force field implementation of the boronate function to simulate the inhibition of β-lactamases by alkyl and aryl boronic acids". European Journal of Medicinal Chemistry 40, № 11 (2005): 1134–42. http://dx.doi.org/10.1016/j.ejmech.2005.06.011.

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14

Ryu, Ji Hyun, Gyeong Jin Lee, Yu-Ru V. Shih, Tae-il Kim, and Shyni Varghese. "Phenylboronic Acid-polymers for Biomedical Applications." Current Medicinal Chemistry 26, no. 37 (2019): 6797–816. http://dx.doi.org/10.2174/0929867325666181008144436.

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Background: Phenylboronic acid-polymers (PBA-polymers) have attracted tremendous attention as potential stimuli-responsive materials with applications in drug-delivery depots, scaffolds for tissue engineering, HIV barriers, and biomolecule-detecting/sensing platforms. The unique aspect of PBA-polymers is their interactions with diols, which result in reversible, covalent bond formation. This very nature of reversible bonding between boronic acids and diols has been fundamental to their applications in the biomedical area. Methods: We have searched peer-reviewed articles including reviews from

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15

Kotsakis, Stathis D., Vivi Miriagou, Eva Tzelepi та Leonidas S. Tzouvelekis. "Comparative Biochemical and Computational Study of the Role of Naturally Occurring Mutations at Ambler Positions 104 and 170 in GES β-Lactamases". Antimicrobial Agents and Chemotherapy 54, № 11 (2010): 4864–71. http://dx.doi.org/10.1128/aac.00771-10.

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ABSTRACT In GES-type β-lactamases, positions 104 and 170 are occupied by Glu or Lys and by Gly, Asn, or Ser, respectively. Previous studies have indicated an important role of these amino acids in the interaction with β-lactams, although their precise role, especially that of residue 104, remains uncertain. In this study, we constructed GES-1 (Glu104, Gly170), GES-2 (Glu104, Asn170), GES-5 (Glu104, Ser170), GES-6 (Lys104, Ser170), GES-7 (Lys104, Gly170), and GES-13 (Lys104, Asn170) by site-specific mutagenesis and compared their hydrolytic properties. Isogenic comparisons of β-lactam resistanc

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16

Ghosh, Arun K., Zilei Xia, Satish Kovela, et al. "Potent HIV‐1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein‐Ligand X‐ray Structural Studies." ChemMedChem 14, no. 21 (2019): 1863–72. http://dx.doi.org/10.1002/cmdc.201900508.

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17

Zhang, Tianyi, Fu-Ning Hsu, Xiao-Jun Xie, et al. "Reversal of hyperactive Wnt signaling-dependent adipocyte defects by peptide boronic acids." Proceedings of the National Academy of Sciences 114, no. 36 (2017): E7469—E7478. http://dx.doi.org/10.1073/pnas.1621048114.

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Deregulated Wnt signaling and altered lipid metabolism have been linked to obesity, diabetes, and various cancers, highlighting the importance of identifying inhibitors that can modulate Wnt signaling and aberrant lipid metabolism. We have established a Drosophila model with hyperactivated Wnt signaling caused by partial loss of axin, a key component of the Wnt cascade. The Axin mutant larvae are transparent and have severe adipocyte defects caused by up-regulation of β-catenin transcriptional activities. We demonstrate pharmacologic mitigation of these phenotypes in Axin mutants by identifyin

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18

Curini, Massimo, Francesco Epifano, Salvatore Genovese, et al. "Lipoxygenase Inhibitory Activity of Boropinic Acid, Active Principle of Boronia Pinnata." Natural Product Communications 1, no. 12 (2006): 1934578X0600101. http://dx.doi.org/10.1177/1934578x0600101214.

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Boropinic acid and other natural prenyloxycinnamic and benzoic acids were easily synthesized in high yield by a two-step sequence from the corresponding p-hydroxy aromatic acids and were assayed for radical scavenging activity using the DPPH test and for inhibition of enzymatic lipid peroxidation mediated by soybean 5-lipoxygenase. Compared to other acids and to known antioxidant compounds like BHT, Trolox and ascorbic acid, boropinic acid was far more active in the lipoxygenase test (IC50 = 7.6 ng/mL, p < 0.05). The recorded inhibition value suggested that boropinic acid acted as an enzyme

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19

Spandana, Zanjam, Tadigiri M. Rekha, Mandava V. B. Rao, and Manojit Pal. "One-Pot Synthesis of 5-(Het)Aryl 8-Aminoquinoline Amide Derivatives as Potential Antibacterial / Cytotoxic Agents." Current Bioactive Compounds 16, no. 2 (2020): 142–51. http://dx.doi.org/10.2174/1573407214666180910130225.

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Background: The 8-Aminoquinoline (8-AQ) framework has attracted particular attention in the discovery and development of antimalarial and anti-bacterial agents or drugs. However, the clinical uses of 8-AQ based drugs are often associated with toxic side effects such as methemoglobinemia and hemolytic anemia with deficiency in Glucose-6-Phosphate Dehydrogenase (G6PD) Activity. The 4-aryl- 8-amino(acetamido)quinoline derivatives, on the other hand, have shown antiproliferative activities against cancer cell lines. These reports prompted us to assess the antibacterial and cytotoxic activities of

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20

Karabela, Sophia, Ioannis Psallidas, Taylor Sherrill та ін. "Opposing effects of bortezomib-induced nuclear factor-κB inhibition on chemical lung carcinogenesis." Carcinogenesis 33, № 4 (2012): 859–67. https://doi.org/10.1093/carcin/bgs024.

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Since recent evidence indicates a requirement for epithelial nuclear factor (NF)-κB signaling in lung tumorigenesis, we investigated the impact of the NF-κB inhibitor bortezomib on lung tumor promotion and growth. We used an experimental model in which wild-type mice or mice expressing an NF-κB reporter received intraperitoneal urethane (1 g/kg) followed by twice weekly bortezomib (1 mg/kg) during distinct periods of tumor initiation/progression. Mice were serially assessed for lung NF-κB activation, inflammation and carcinogenesis. Short-term proteasome inhibition with bortezomib did not impa

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21

Marshall, Jennifer R., Juliana N. O’Brien, and Andrew J. Wommack. "Oxidative Coupling of Aryl Boronic Acids with Aryl- and Alkylamines Via Cooperative Photoredox and Copper Catalysis." SSRN Electronic Journal, 2022. http://dx.doi.org/10.2139/ssrn.4140071.

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22

Desai, Bhargav, Rachit S. Patil, Hussain Bhukya, Bharatkumar Z. Dholakiya, and TOGATI NAVEEN. "Copper-Catalyzed Synthesis of Diaryl Sulfones Via Cross-Coupling of Boronic Acids and P-Toluenesulfonyl Hydrazide." SSRN Electronic Journal, 2023. http://dx.doi.org/10.2139/ssrn.4396667.

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23

hosseini-sarvari, mona, and Abdulhamid Dehghani. "Nickel/Tio2-Catalyzed Suzuki–Miyaura Cross-Coupling (Smr) of Aryl Boronic Acids with Aryl Halides in Meoh/H2o." SSRN Electronic Journal, 2022. http://dx.doi.org/10.2139/ssrn.4185056.

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24

"Bimetallic quantum dots (Cu-Pd, Ni-Pd) catalyzed reaction of bromo arenes with alkenes and aryl boronic acids." Indian Journal of Chemistry 62, no. 8 (2023). http://dx.doi.org/10.56042/ijc.v62i8.4769.

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25

Geng, Fenghua, Xiaoxue Liu, Tingwen Wei, et al. "An Alkaline Phosphatase-Induced Immunosensor for Sars-Cov-2 N Protein Based on the in Situ Fluorogenic Self-Assembly between N-Heterocyclic Boronic Acids and Alizarin Red S." SSRN Electronic Journal, 2022. http://dx.doi.org/10.2139/ssrn.4253425.

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26

BAI, RUI, XU-JUAN LIU, Lin-Yu Jiao, ZHUO LI, SHANSHAN LIU, and XIAOXUN MA. "Nabh4-Enabled Heterogeneous Cu-Usy-Catalyzed Chan−Lam Type Coupling between Boronic Acides and Sulfonyl Azides." SSRN Electronic Journal, 2022. http://dx.doi.org/10.2139/ssrn.4091381.

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