Relevant bibliographies by topics / Histamine receptor antagonism

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  2. Dissertations / Theses
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  4. Book chapters
  5. Conference papers

Academic literature on the topic 'Histamine receptor antagonism'

Author: Grafiati
Published: 7 June 2025
Last updated: 2 August 2025

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Journal articles on the topic "Histamine receptor antagonism"

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Neely, C. F., I. Matot, D. Haile, J. Nguyen, and V. Batra. "Tone-dependent responses of histamine in feline pulmonary vascular bed." American Journal of Physiology-Heart and Circulatory Physiology 268, no. 2 (1995): H653—H661. http://dx.doi.org/10.1152/ajpheart.1995.268.2.h653.

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Under conditions of controlled pulmonary blood flow and constant left atrial pressure, histamine produced tone-dependent responses in the pulmonary vascular (PV) bed of intact-chest, spontaneously breathing cats. At low, baseline PV tone, histamine produced dose-dependent increases in mean lobar arterial pressure that were antagonized by the selective histamine H1-receptor antagonist, diphenhydramine. The cyclooxygenase inhibitor, meclofenamate, and the thromboxane A2 (TxA2) receptor antagonist, SQ-29548, had no effect on these vasoconstrictor responses of histamine. After an increase in PV to
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Mocking, Tamara A. M., Maurice C. M. L. Buzink, Rob Leurs, and Henry F. Vischer. "Bioluminescence Resonance Energy Transfer Based G Protein-Activation Assay to Probe Duration of Antagonism at the Histamine H3 Receptor." International Journal of Molecular Sciences 20, no. 15 (2019): 3724. http://dx.doi.org/10.3390/ijms20153724.

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Duration of receptor antagonism, measured as the recovery of agonist responsiveness, is gaining attention as a method to evaluate the ‘effective’ target-residence for antagonists. These functional assays might be a good alternative for kinetic binding assays in competition with radiolabeled or fluorescent ligands, as they are performed on intact cells and better reflect consequences of dynamic cellular processes on duration of receptor antagonism. Here, we used a bioluminescence resonance energy transfer (BRET)-based assay that monitors heterotrimeric G protein activation via scavenging of rel
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Leth, R., B. Elander, U. Haglund, L. Olbe, and E. Fellenius. "Histamine H2-receptor of human and rabbit parietal cells." American Journal of Physiology-Gastrointestinal and Liver Physiology 253, no. 4 (1987): G497—G501. http://dx.doi.org/10.1152/ajpgi.1987.253.4.g497.

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The histamine H2-receptor on the human parietal cell has been characterized by using dose-response curves and the negative logarithm of the molar concentration of an antagonist (pA2) analyses of cimetidine antagonism of betazole, histamine, and impromidine stimulation in isolated human and rabbit gastric glands. To evaluate the in vitro results, betazole-stimulated gastric acid secretion with and without cimetidine was also studied in healthy subjects. In the in vivo model, individual dose-response curves were shifted to the right with increasing cimetidine concentrations, but this was counter
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Miller, Thomas R., David G. Witte, Lynne M. Ireland, et al. "Analysis of Apparent Noncompetitive Responses to Competitive H1-Histamine Receptor Antagonists in Fluorescent Imaging Plate Reader-Based Calcium Assays." Journal of Biomolecular Screening 4, no. 5 (1999): 249–58. http://dx.doi.org/10.1177/108705719900400506.

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We have examined the utility of high throughput fluorescent imaging plate reader (FLIPR)-based calcium assays for pharmacological characterization of G-protein coupled receptors (GPCRs) using recombinant and native human H1-histamine receptors (H1-HR), expressed in HEK293 and HeLa S3 cells, respectively, as model systems. For stably transfected HEK293 cell lines, the potency of histamine for elevating intracellular calcium increased (pD2, 7.13 and 7.86) with increased H1-HR density (about 0.8 and 14 pmol/mg protein, respectively), though histamine binding affinities were similar. The classic H
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Pfanzagl, Beatrix, Roswitha Pfragner, and Erika Jensen-Jarolim. "The Transient Receptor Potential Vanilloid 4 Agonist RN-1747 Inhibits the Calcium Response to Histamine." Pharmacology 104, no. 3-4 (2019): 166–72. http://dx.doi.org/10.1159/000501144.

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Background: Sensitization of transient receptor potential (TRP) cation channels probably contributes to intestinal hypersensitivity, a hallmark of gastrointestinal disorders. Histamine acting via histamine 1 receptor (H1R) to open TRP cation channels might also be involved. Method: The enterochromaffin cell line P-STS, responsive to histamine via H1R, was used as model to study possible synergism between histamine and TRP vanilloid 4 (TRPV4) pathways. Results: The TRPV4 antagonist RN-1734, but not HC-067047, inhibited the cytoplasmic calcium response to histamine in P-STS cells. However, also
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Balemans, D., J. Aguilera-Lizarraga, M. V. Florens, et al. "Histamine-mediated potentiation of transient receptor potential (TRP) ankyrin 1 and TRP vanilloid 4 signaling in submucosal neurons in patients with irritable bowel syndrome." American Journal of Physiology-Gastrointestinal and Liver Physiology 316, no. 3 (2019): G338—G349. http://dx.doi.org/10.1152/ajpgi.00116.2018.

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Previously, we showed histamine-mediated sensitization of transient receptor potential (TRP) vanilloid 1 (TRPV1) in patients with irritable bowel syndrome (IBS). Sensitization of TRP ankyrin 1 (TRPA1) and TRP vanilloid 4 (TRPV4) are also involved in aberrant pain perception in preclinical models of somatic pain. Here, we hypothesize that in parallel with TRPV1, histamine sensitizes TRPA1 and TRPV4, contributing to increased visceral pain in patients with IBS. Rectal biopsies were collected from patients with IBS and healthy subjects (HS) to study neuronal sensitivity to TRPA1 and TRPV4 agonist
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Aihara, Takeshi, Yusuke Nakamura, Makoto M. Taketo, Minoru Matsui, and Susumu Okabe. "Cholinergically stimulated gastric acid secretion is mediated by M3 and M5 but not M1 muscarinic acetylcholine receptors in mice." American Journal of Physiology-Gastrointestinal and Liver Physiology 288, no. 6 (2005): G1199—G1207. http://dx.doi.org/10.1152/ajpgi.00514.2004.

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Muscarinic acetylcholine receptors play an important role in the regulation of gastric acid secretion stimulated by acetylcholine; nonetheless, the precise role of each receptor subtype (M1–M5) remains unclear. This study examined the involvement of M1, M3, and M5 receptors in cholinergic regulation of acid secretion using muscarinic receptor knockout (KO) mice. Gastric acid secretion was measured in both mice subjected to acute gastric fistula production under urethane anesthesia and conscious mice that had previously undergone pylorus ligation. M3 KO mice exhibited impaired gastric acid secr
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Black, James. "Drugs from emasculated hormones: The principle of syntopic antagonism." Bioscience Reports 9, no. 3 (1989): 253–72. http://dx.doi.org/10.1007/bf01114681.

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Black, James. "Drugs from Emasculated Hormones: The Principle of Syntopic Antagonism." Bioscience Reports 24, no. 4-5 (2004): 302–22. http://dx.doi.org/10.1007/s10540-005-2736-5.

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DiBaise, J. K. "Nocturnal acid breakthrough and histamine-2 receptor antagonism." American Journal of Gastroenterology 97, no. 7 (2002): 1595. http://dx.doi.org/10.1111/j.1572-0241.2002.05890.x.

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Dissertations / Theses on the topic "Histamine receptor antagonism"

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Mercer, Amanda Denise. "Stereochemical studies of H₁-receptor histamine antagonists." Thesis, University of Bath, 1989. https://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.439288.

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Cooper, David Gwyn. "Structure-activity in pyridine-containing histamine receptor antagonists." Thesis, Imperial College London, 1987. http://hdl.handle.net/10044/1/38269.

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Dulabh, R. "Histamine and H2-receptor antagonist interactions in the respiratory tract of the guinea pig." Thesis, University of Hertfordshire, 1985. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.304132.

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Hagenow, Stefanie [Verfasser], Holger [Gutachter] Stark, and Holger [Gutachter] Gohlke. "Histamine H3 receptor antagonists with multitargeting properties at GPCRs and enzymes / Stefanie Hagenow ; Gutachter: Holger Stark, Holger Gohlke." Düsseldorf : Universitäts- und Landesbibliothek der Heinrich-Heine-Universität Düsseldorf, 2019. http://d-nb.info/1178112543/34.

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Affini, Anna [Verfasser]. "Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease / Anna Affini." Düsseldorf : Universitäts- und Landesbibliothek der Heinrich-Heine-Universität Düsseldorf, 2019. http://d-nb.info/1190350807/34.

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Zanellato, Fabbri Natalia 1981. "Cloridrato de azelastina e budesonida intranasais (isoladas e associadas) : efeito na obstrução nasal e função pulmonar de pacientes com rinopatia alérgica : modelo de estudo farmacodinâmico para drogas intranasais." [s.n.], 2014. http://repositorio.unicamp.br/jspui/handle/REPOSIP/311758.

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Orientador: Ricardo de Lima Zollner<br>Tese (doutorado) - Universidade Estadual de Campinas, Faculdade de Ciências Médicas<br>Made available in DSpace on 2018-08-24T18:58:24Z (GMT). No. of bitstreams: 1 ZanellatoFabbri_Natalia_D.pdf: 35087770 bytes, checksum: d1d79dc3e2bc0a5a2a05b4261a363a74 (MD5) Previous issue date: 2014<br>Resumo: Apesar das diversas terapias disponíveis para o tratamento da rinite alérgica (RA), muitos pacientes não obtêm alívio dos sintomas com uso de um único fármaco e apresentam frequentemente queixa da manutenção dos sintomas mesmo sob tratamento. Estudos clínicos al
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López, Muñoz Laura. "Homology modeling and structural analysis of the antipsychotic drugs receptorome." Doctoral thesis, Universitat Pompeu Fabra, 2010. http://hdl.handle.net/10803/7228.

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Classically it was assumed that the compounds with therapeutic effect exert their action interacting with a single receptor. Nowadays it is widely recognized that the pharmacological effect of most drugs is more complex and involves a set of receptors, some associated to their positive effects and some others to the side effects and toxicity. Antipsychotic drugs are an example of effective compounds characterized by a complex pharmacological profile binding to several receptors (mainly G protein-coupled-receptors, GPCR). In this work we will present a detailed study of known antipsychotic drug
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Janse, van Rensburg Hendrika Nicolien. "A longitudinal study of the usage of acid reducing medicine using a medicine claims database / Hendrika Nicolien Janse van Rensburg." Thesis, North-West University, 2007. http://hdl.handle.net/10394/1903.

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Acid-related disorders are common, chronic conditions that have considerable impact on a patient's quality of life. In a study conducted by Majumdar et al. (2003:2411) the prevalence of chronic acid-related disorders was 2.3%. Acid-related disorders represent a major financial consideration with respect to the costs of drug prescribing (Whitaker, 1998:6). Health care cost increases each year. This leads to an increased interest in economic evaluation of health care and medical technologies (Anell & Svarvar, 2000:175). Health care providers no longer make treatment decisions independent of the
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Mummaneni, Vanaja. "Oral absorption of histamine-2 receptor antagonists." 1993. http://catalog.hathitrust.org/api/volumes/oclc/68796913.html.

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Ho, Yu-Hsiang, and 何宇祥. "Study on the analysis of H2 histamine receptor antagonists by capillary electrophoresis." Thesis, 2000. http://ndltd.ncl.edu.tw/handle/07802329296156111829.

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碩士<br>高雄醫學大學<br>藥學研究所<br>88<br>A simple capillary electrophoretic method was established for the determination of cimetidine, ranitidine, famotidine and nizatidine in tablets. The background buffer was 100 mM sodium dihydrogen phosphate adjusted to pH 3.50. Analysis was run at the voltage of 20 kV and a detection wavelength of 214 nm. The method is sensitive with a detection limit of 10 mM (cimetidine), 20 mM (ranitidine), 20 mM (nizatidine) and 10 mM (famotidine) (S/N=3, hydrodynamic injection 1sec.). The calibration curves were linear over a concentration range of 100-300 mM. Mean recoveries
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Books on the topic "Histamine receptor antagonism"

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E, Pounder R., ed. Histamine H2-receptor antagonists. Science Press, 1990.

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E, Pounder R., ed. Histamine H2-receptor antagonists. Science Press, 1990.

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E, Pounder R., ed. Histamine H2-receptor antagonists. Science Press, 1990.

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1939-, Rocklin Ross E., ed. Histamine and H2 antagonists in inflammation and immunodeficiency. Dekker, 1990.

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R, Simons F. E., ed. Histamine and H1-receptor antagonists in allergic disease. M. Dekker, 1996.

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Heald, Karen Anne. Histamine H2-receptors: Characterisation and preliminary evaluation of their antagonism in the treatment of pepticulceration. University of Birmingham, 1988.

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Divya, Vohora, ed. The third histamine receptor: Selective ligands as potential therapeutic agents in CNS disorders. CRC Press, 2009.

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Walt, Robert P. A comparison of the gastric anti-secretory effects, side effect profile and clinical use of two histamine H [inferior] 2-receptor antagonists. University of Birmingham, 1986.

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Settipane, Guy A. H1 and H2 Histamine Receptors. New England & Regional Allergy, 1988.

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Cardiovascular Effects of Histamine and H2-Receptor Antagonists. Zuckschwerdt, W., 1994.

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Book chapters on the topic "Histamine receptor antagonism"

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Thorlacius, Henrik, Johan Raud, Lennart Lindbom, and Per Hedqvist. "Histamine Potentiates Leukotriene B4-Induced Leukocyte Adhesion: A Potential Role of Histamine1-Receptor Antagonism in Allergic Leukocyte Recruitment." In Advances in Experimental Medicine and Biology. Springer US, 1997. http://dx.doi.org/10.1007/978-1-4899-1810-9_67.

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Schwartz, J. C., J. M. Arrang, M. L. Bouthenet, M. Garbarg, H. Pollard, and M. Ruat. "Histamine Receptors in Brain." In Histamine and Histamine Antagonists. Springer Berlin Heidelberg, 1991. http://dx.doi.org/10.1007/978-3-642-75840-9_15.

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Foreman, J. C. "Histamine H2 Receptors and Lung Function." In Histamine and Histamine Antagonists. Springer Berlin Heidelberg, 1991. http://dx.doi.org/10.1007/978-3-642-75840-9_17.

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Casy, A. F. "Antagonists of H1 Receptors of Histamine: Recent Developments." In Histamine and Histamine Antagonists. Springer Berlin Heidelberg, 1991. http://dx.doi.org/10.1007/978-3-642-75840-9_26.

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Sadek, B., D. Łażewska, S. Hagenow, K. Kieć-Kononowicz, and H. Stark. "Histamine H3R Antagonists: From Scaffold Hopping to Clinical Candidates." In Histamine Receptors. Springer International Publishing, 2016. http://dx.doi.org/10.1007/978-3-319-40308-3_5.

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Sugano, Kentaro. "Histamine H2-receptor antagonists." In Pocket Guide to Gastrointestinal Drugs. John Wiley & Sons, Ltd, 2014. http://dx.doi.org/10.1002/9781118481530.ch3.

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Bloch, Michael H., Michael H. Bloch, Mark A. Geyer, et al. "Histamine Receptor Agonists and Antagonists." In Encyclopedia of Psychopharmacology. Springer Berlin Heidelberg, 2010. http://dx.doi.org/10.1007/978-3-540-68706-1_3306.

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Brimblecombe, Roger W., and C. Robin Ganellin. "Cimetidine and Other Histamine H2-Receptor Antagonists." In Drug Discovery and Development. Humana Press, 1987. http://dx.doi.org/10.1007/978-1-4612-4828-6_13.

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Thurmond, Robin L., Jennifer Venable, Brad Savall, et al. "Clinical Development of Histamine H4 Receptor Antagonists." In Handbook of Experimental Pharmacology. Springer International Publishing, 2017. http://dx.doi.org/10.1007/164_2016_130.

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Dunford, Paul J., and Robin L. Thurmond. "Histamine H4 receptor antagonists." In New Drugs and Targets for Asthma and COPD. KARGER, 2010. http://dx.doi.org/10.1159/000320818.

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Conference papers on the topic "Histamine receptor antagonism"

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Ritter, Arthur, Christine M. Genua, Janardan Yadav, Swamy Laxminarayan, and David Kristol. "Active analog approach to Histamine HI receptor antagonists." In 1992 14th Annual International Conference of the IEEE Engineering in Medicine and Biology Society. IEEE, 1992. http://dx.doi.org/10.1109/iembs.1992.5760929.

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Ritter, Gerula, Yadav, Laxminarayan, and Kristol. "Active Analog Approach To Histamine H1 Receptor Antagonists." In Proceedings of the Annual International Conference of the IEEE Engineering in Medicine and Biology Society. IEEE, 1992. http://dx.doi.org/10.1109/iembs.1992.589633.

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Lumley, P., E. W. Collington, P. Hallett, et al. "THE EFFECTS OF GR32191, A NEW THROMBOXANE RECEPTOR BLOCKING DRUG,ON PLATELETS AND VASCULAR SMOOTH MUSCLE IN VITRO." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643754.

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The effect of a new thromboxane receptor blocking drug GR32191 ([1R-[1α(Z),2β,3β,5α]]-(+)-7-[5-[[(1,1"-biphenyl)-4-yl]methoxy] -3-hydroxy-2-(l-piperidinyl)cyclopentyl]-4-heptenoic acid,hydrochloride) has been examined upon platelets and vascular smooth muscle. In human platelet-rich plasma (PRP), aggregation to thromboxane(Tx) A2, PGH2, arachidonic acid, collagen andU-46619 was antagonised by GR32191 (IC50 range 2-36 nM).Primary aggregation (PRP treated with aspirin 10 pM) to ADP, 5-HT and adrenaline were unaffected by concentrations of GR32191 up to 10 pM. In human PRP, U-46619-induced aggreg
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Alfon, Jose, Sonia Sanchez-Gomez, Carolina Salcedo, et al. "Efficacy Of UR-63325, A New Histamine H4 Receptor Antagonist, In House Dust Mite-Induced Mouse Asthma Models." In American Thoracic Society 2011 International Conference, May 13-18, 2011 • Denver Colorado. American Thoracic Society, 2011. http://dx.doi.org/10.1164/ajrccm-conference.2011.183.1_meetingabstracts.a1302.

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Choi, Won-Il, Jihyeon Jeong, and Choong Won Lee. "Association between antacid proton pump inhibitors and histamine 2 receptor antagonists) and incidence of lung cancer: a population-based cohort analysis." In ERS International Congress 2021 abstracts. European Respiratory Society, 2021. http://dx.doi.org/10.1183/13993003.congress-2021.pa1731.

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Al-Hazzani, Waleed, Farhan Alenzi, Roman Jaeschke, Paul Moayyedi, and Deborah J. Cook. "Proton Pump Inhibitors Versus Histamine 2 Receptor Antagonists For Stress Ulcer Prophylaxis In Critically Ill Patients: A Systematic Review And Meta-Analysis." In American Thoracic Society 2012 International Conference, May 18-23, 2012 • San Francisco, California. American Thoracic Society, 2012. http://dx.doi.org/10.1164/ajrccm-conference.2012.185.1_meetingabstracts.a2562.

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Shirinsky, I., and V. Shirinsky. "SAT0491 Use of histamine h1-receptor antagonists is associated with decreased prevalence of radiographic knee osteoarthritis: a cross-sectional analysis of osteoarthritis initiative data." In Annual European Congress of Rheumatology, 14–17 June, 2017. BMJ Publishing Group Ltd and European League Against Rheumatism, 2017. http://dx.doi.org/10.1136/annrheumdis-2017-eular.2658.

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