Relevant bibliographies by topics / Indole-2

Contents

  1. Journal articles
  2. Dissertations / Theses
  3. Books
  4. Book chapters
  5. Conference papers
  6. Reports

Academic literature on the topic 'Indole-2'

Author: Grafiati
Published: 5 June 2025
Last updated: 1 August 2025

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic 'Indole-2.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "Indole-2"

1

Elmakki, Mohammed A. E., Orbett Teboho Alexander, Gertruida J. S. Venter, Johan Andries Venter, and Andreas Roodt. "Structural Study of Model Rhodium(I) Carbonylation Catalysts Activated by Indole-2-/Indoline-2-Carboxylate Bidentate Ligands and Kinetics of Iodomethane Oxidative Addition." Inorganics 10, no. 12 (2022): 251. http://dx.doi.org/10.3390/inorganics10120251.

Full text
Abstract:
The rigid-backbone bidentate ligands Indoline-2-carboxylic acid (IndoliH) and Indole-2-carboxylic acid (IndolH) were evaluated for rhodium(I). IndoliH formed [Rh(Indoli)(CO)(PPh3)] (A2), while IndolH yielded the novel dinuclear [Rh1(Indol’)(CO)(PPh3)Rh2(CO)(PPh3)2] (B2) complex (Indol’ = Indol2−), which were characterized by SCXRD. In B2, the Rh1(I) fragment [Rh1(Indol’)(CO)(PPh3)] (bidentate N,O-Indol) exhibits a square-planar geometry, while Rh2(I) shows a ‘Vaska’-type trans-[O-Rh2(PPh3)2(CO)] configuration (bridging the carboxylate ‘oxo’ O atom of Indol2−). The oxidative addition of MeI to
APA, Harvard, Vancouver, ISO, and other styles
2

Sharma, Upendra, Inder Kumar, and Rakesh Kumar. "Recent Advances in the Regioselective Synthesis of Indoles via C–H Activation/Functionalization." Synthesis 50, no. 14 (2018): 2655–77. http://dx.doi.org/10.1055/s-0037-1609733.

Full text
Abstract:
Indole is an important heterocyclic motif that occurs ubiquitously in bioactive natural products and pharmaceuticals. Immense efforts have been devoted to the synthesis of indoles starting from the Fisher indole synthesis to the recently developed C–H activation/functionalization-based methods. Herein, we have reviewed the progress made on the regioselective synthesis of functionalized indoles, including 2-substituted, 3-substituted and 2,3-disusbstituted indoles, since the year 2010.1 Introduction2 Metal-Catalyzed Synthesis of 2-Substituted Indoles3 Metal-Catalyzed Synthesis of 3-Substituted
APA, Harvard, Vancouver, ISO, and other styles
3

Kumar, Anil, and Ganesh Shelke. "Sc(OTf)3-Catalyzed Oligomerization of Indole: One-Pot Synthesis of 2-[2,2-Bis(indol-3-yl)ethyl]anilines and 3-(Indolin-2-yl)indoles." Synthesis 49, no. 18 (2017): 4321–26. http://dx.doi.org/10.1055/s-0036-1588181.

Full text
Abstract:
Oligomerization of substituted indoles and N-methylindoles was investigated in the presence of catalytic amounts of scandium triflate in dichloromethane. Two types of indole oligomer, 2-[2,2-bis(indol-3-yl)ethyl]anilines and 3-(indolin-2-yl)indoles were obtained based on the substituent on indole ring. This study constitutes the first example of Sc(OTf)3-catalyzed oligomerization of indoles and gave good yield of 2-[2,2-bis(indol-3-yl)ethyl]anilines and 3-(indolin-2-yl)indoles.
APA, Harvard, Vancouver, ISO, and other styles
4

CHAUBAN, Vishal, Sbivkanya FULORIA, Neeraj K. FULORIA, Syed R. HASHIM, and Sokindra KUMAR. "SYNTHESIS, CHARACTERIZATION AND COMPARATIVE SCREENING OF SOME NEWER 2-PHENYL INDOLE AND 5-CHLORO-2-PHENYL INDOLE DERIVATIVES." SOUTHERN BRAZILIAN JOURNAL OF CHEMISTRY 20, no. 20 (2012): 69–76. http://dx.doi.org/10.48141/sbjchem.v20.n20.2012.71_revista_2012a.pdf.

Full text
Abstract:
Biologically active phenyl indole and chloro phenyl indole derivatives were efficiently synthesized. The reaction of 2-phenyl-1H-indole A and 5-chloro-2-phenyl-1H-indole B, with chloroacetylchloride yielded 2-chloro-1-(2-phenyl-1H-indol-1-yl)ethanone 1 and 2-chloro-1-(5-chloro-2-phenyl-1H-indol-1-yl)ethanone 4 respectively. Compound 1 and 4 on Friedal Crafts cyclization in presence of aluminium chloride and nitrobenzene yielded indolo[2,1 -alfa]isoquinolin-6(5H)-one 2 and 10-chloroindolo [2,1-alfa]isoquinolin-6(5H)-one 5 respectively, which upon hydrolysis afforded 2-(2-(1H-indol-2-yl)phenyl)a
APA, Harvard, Vancouver, ISO, and other styles
5

Aksenov, Alexander V., Nicolai A. Aksenov, Elena V. Aleksandrova, et al. "Direct Conversion of 3-(2-Nitroethyl)-1H-Indoles into 2-(1H-Indol-2-yl)Acetonitriles." Molecules 26, no. 20 (2021): 6132. http://dx.doi.org/10.3390/molecules26206132.

Full text
Abstract:
The recently discovered [4+1]-spirocyclization of nitroalkenes to indoles provided a convenient new approach to 2-(1H-indol-2-yl)acetonitriles. However, this reaction was complicated by the formation of inert 3-(2-nitroethyl)-1H-indole byproducts. Herein, we offer a workaround this problem that allows for effective transformation of the unwanted byproducts into acetonitrile target molecules.
APA, Harvard, Vancouver, ISO, and other styles
6

Riar, G. K., D. Utreja, A. Kalia, and S. Kaur. "Synthesis and antipathogenic evaluation of isatin-indole Schiff bases as potent nematicidal and agrochemical agents." INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY 35, no. 02 (2025): 295. https://doi.org/10.59467/ijhc.2025.35.295.

Full text
Abstract:
N-alkylated Schiff bases of isatin-indole were synthesized through the reaction of isatin hydrazide with indole-3-carbaldehyde followed by N-alkylation. The synthesized isatin-indole Schiff bases were evaluated for their in vitro antimicrobial activity against the pathogenic bacteria Dickeya sp. and Streptomyces sp., as well as the fungi Fusarium oxysporum and Rhizoctonia solani. In addition, their nematicidal potential was assessed against the tomato parasite Meloidogyne incognita through egg hatch inhibition and J2 mortality assays. The compounds were further evaluated for their inhibitory a
APA, Harvard, Vancouver, ISO, and other styles
7

Golantsov, Nikita, Alexey Festa, Alexey Varlamov, and Leonid Voskressensky. "Revision of the Structure and Total Synthesis of Topsentin C." Synthesis 49, no. 11 (2017): 2562–74. http://dx.doi.org/10.1055/s-0036-1588731.

Full text
Abstract:
An efficient synthetic approach to access (indol-3-yl)ethane-1,2-diamines with a protecting group at the indole N atom from readily available 3-(2-nitrovinyl)indoles is reported. This approach includes solvent-free conjugate addition of O-pivaloylhydroxylamines to 1-Boc-3-(2-nitrovinyl)indoles followed by mild reduction of the adducts. The obtained (indol-3-yl)ethane-1,2-diamines are convenient synthetic precursors for several classes of marine alkaloids. The first total synthesis of racemic topsentin C, a secondary metabolite from Hexadella sp., based on this approach is reported. The initial
APA, Harvard, Vancouver, ISO, and other styles
8

Xu, Xiaobing, Jianchao Liu, Lin Lu, Furong Wang, and Biaolin Yin. "Pd-catalyzed regioselective intramolecular direct arylation of 3-indolecarboxamides: access to spiro-indoline-3,3′-oxindoles and 5,11-dihydro-6H-indolo[3,2-c]quinolin-6-ones." Chemical Communications 53, no. 55 (2017): 7796–99. http://dx.doi.org/10.1039/c7cc02256e.

Full text
Abstract:
We report regioselective intramolecular direct C-3 and C-2 arylations of the indole rings of 3-indolecarboxamides for diastereospecific production of spiro-indoline-3,3′-oxindoles and 5,11-dihydro-6H-indolo[3,2-c]quinolin-6-ones, respectively, under different reaction conditions.
APA, Harvard, Vancouver, ISO, and other styles
9

Padmaja, Pannala, Pedavenkatagari Narayana Reddy, and Bijaya Ketan Sahoo. "A Green Approach to the Synthesis of Novel Indole Substituted 2-Amino- 4,5-dihydro-3-furancarbonitriles in Water." Letters in Organic Chemistry 16, no. 3 (2019): 209–14. http://dx.doi.org/10.2174/1570178615666180917104820.

Full text
Abstract:
2-Amino-4,5-dihydro-3-furancarbonitriles (ADFCs) have attracted much attention due to their utility as valuable synthetic intermediates for the preparation of a series of acyclic and cyclic organic compounds. On the other hand, indoles substituted with furans are highly interesting compounds displaying a wide range of biological and pharmaceutical activities. However, to the best of our knowledge, indole substituted 2-amino-4,5-dihydro-3-furancarbonitriles have not been previously reported. A new and efficient synthesis of indole substituted 2-amino-4,5-dihydro-3-furancarbonitriles has been de
APA, Harvard, Vancouver, ISO, and other styles
10

Short, Spencer, Steven Rhodes, Vishakha S. Bhave, Ryoga Hojo, and Mukund Jha. "Metal-Free Hydroamination of Alkynes: A Mild and Concise Synthesis of Thiazolo[3,2-a]indoles and their Cytotoxic Activity." Synthesis 51, no. 22 (2019): 4263–70. http://dx.doi.org/10.1055/s-0039-1690680.

Full text
Abstract:
A metal-free, mild and efficient method for the synthesis of thiazolo[3,2-a]indoles has been developed starting from indoline-2-thiones. The reaction methodology involves first the formation of thermally labile 2-(prop-2-ynylthio)-1H-indole intermediates, which undergo base-mediated intramolecular hydroamination to produce the title compounds in excellent yields.
APA, Harvard, Vancouver, ISO, and other styles
More sources

Dissertations / Theses on the topic "Indole-2"

1

Wang, Yu-Pu Ph D. Massachusetts Institute of Technology. "I. [2 +2] Cycloaddition and benzannulation of 2-iodoynamides and application to the construction of highly substituted indoles : II. Synthesis of furo[2,3-g]thieno[2,3-e]indole via a benzannulation strategy." Thesis, Massachusetts Institute of Technology, 2015. http://hdl.handle.net/1721.1/101556.

Full text
Abstract:
Thesis: Ph. D., Massachusetts Institute of Technology, Department of Chemistry, 2015.<br>Cataloged from PDF version of thesis.<br>Includes bibliographical references.<br>The synthesis and reactions of 2-iodoynamides were investigated. 2-Iodoynamides undergo efficient and regioselective [2 + 2] cycloaddition with ketene to produce cyclobutenones that are useful synthetic building blocks. Reaction of 2-iodoynamides and vinylketenes generated in situ from cyclobutenones proceeds via a pericyclic cascade mechanism to produce highly substituted 2-iodoanilines. Tandem strategies for the synthesis of
APA, Harvard, Vancouver, ISO, and other styles
2

Shattat, Ghassan F. "Synthesis and pharmacological evaluation of novel ethyl-1H-indole-2-carboxamides as potential cardiovascular agents." Thesis, Coventry University, 2004. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.403613.

Full text
APA, Harvard, Vancouver, ISO, and other styles
3

Yip, Choi-wan, and 葉彩雲. "Degradation of N-heterocyclic aromatics indole and 2-methylindole by bacteria from wetland sediment and characterization of the bacteriainvolved." Thesis, The University of Hong Kong (Pokfulam, Hong Kong), 2005. http://hub.hku.hk/bib/B36383156.

Full text
APA, Harvard, Vancouver, ISO, and other styles
4

Yip, Choi-wan. "Degradation of N-heterocyclic aromatics indole and 2-methylindole by bacteria from wetland sediment and characterization of the bacteria involved." Click to view the E-thesis via HKUTO, 2005. http://sunzi.lib.hku.hk/hkuto/record/B36383156.

Full text
APA, Harvard, Vancouver, ISO, and other styles
5

Koulibaly, Issa. "Automatisation et optimisation de la synthèse du ((pyridyl-4)-2 ethyl)-3 indole, précurseur d'un antidépresseur." Paris 6, 1986. http://www.theses.fr/1986PA066413.

Full text
Abstract:
Dans le cadre des recherches concernant l'application des techniques d'automatisation et des méthodes d'optimisation, sur les procédés de fabrications industrielles de produits pharmaceutiques, nous avons choisi l'automatisation et l'optimisation de la synthèse d'un précurseur de l'indalpine, qui est un produit pharmaceutique important par ses propriétés d'antidépresseur. Nous montrons, dans la première partie de ce travail, qu'il est possible d'automatiser, à l'échelle du laboratoire, et pour un cout réduit, une synthèse organique complexe à l'aide d'un automate de bas de gamme et de capteurs
APA, Harvard, Vancouver, ISO, and other styles
6

Koulibaly, Issa. "Automatisation et optimisation de la synthèse du (pyridyl-4)-2 éthyl)-3 indole, précurseur d'un antidépresseur." Grenoble 2 : ANRT, 1986. http://catalogue.bnf.fr/ark:/12148/cb37598826w.

Full text
APA, Harvard, Vancouver, ISO, and other styles
7

Ciccolini, Cecilia. "Synthesis of Mono and Poly-Heterocycles starting from 1,2-Diaza-1,3-Dienes (or precursors) as Building Blocks." Doctoral thesis, Urbino, 2020. http://hdl.handle.net/11576/2674162.

Full text
APA, Harvard, Vancouver, ISO, and other styles
8

Estevão, Mónica Alexandra Silva. "Síntese de uma biblioteca de derivados de indole com potencial actividade antioxidante e inibição selectiva da COX‐2." Master's thesis, FCT - UNL, 2008. http://hdl.handle.net/10362/1444.

Full text
Abstract:
Os compostos indólicos constituem uma extensa e larga família de compostos presentes em bactérias, plantas e animais, sendo alvo de especial interesse nas áreas tanto da química biológica como na da química medicinal. O triptofano, aminoácido essencial para o Homem, constitui um importante exemplo de derivados de indole. Outros exemplos, derivados desta importante estrutura, são o ácido indole‐3‐acético (hormona presente nas plantas) e a melatonina (hormona segregada pela glândula pineal). Uma importante característica dos compostos derivados do indole é que estes podem ser úteis como fármac
APA, Harvard, Vancouver, ISO, and other styles
9

Calderon, Morales Raul. "The Fischer Indole synthesis in choline chloride.2 zinc chloride ionic liquid and the 1,3 arene-olefin cycloaddition reaction." Thesis, University of Leicester, 2003. http://hdl.handle.net/2381/30075.

Full text
Abstract:
We have utilised the copper(I) triflate catalysed intramolecular [2+2] photocycloaddition reaction to cyclise diene 53 to afford the exo product 54 in 60% yield (Chapter 2). (Fig. 15762A) Using choline chloride.2zinc chloride ionic liquid we have carried out a one pot Fischer Indole synthesis. Phenyl hydrazine 149 was reacted with ethylmethyliketone 298 to give 2,3-dimethyl-indole 273 as the only product in 80% yield. The product 273 was directly sublimed from the ionic liquid. 10 more examples of this reaction was carried out with direct sublimation of the product from the ionic liquid with y
APA, Harvard, Vancouver, ISO, and other styles
10

Dacko, Christopher Andrew. "The synthesis of tryptophan derivatives, 2- and/or 3-substituted indoles, progress toward dilemmaones A-C, and synthetic studies towards fistulosin via palladium-catalyzed reductive N-heteroannulation." Morgantown, W. Va. : [West Virginia University Libraries], 2009. http://hdl.handle.net/10450/10403.

Full text
Abstract:
Thesis (Ph. D.)--West Virginia University, 2009.<br>Title from document title page. Document formatted into pages; contains xxvi, 324 p. : ill. (some col.). Includes abstract. Includes bibliographical references (p. 186-198).
APA, Harvard, Vancouver, ISO, and other styles
More sources

Books on the topic "Indole-2"

1

Leusink, Frederik Ronald. Novel syntheses of azaindoles and indoles: Electrocyclization of the 6p electron-systems of unsaturatedly substituted pyrroles; [4+2]cycloadditions of 2,3-dimethylene-2,3-dihydropyrroles. [s.n.], 1993.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
2

RAHMAN. Indole Alkaloids (Frontiers in Natural Product Research Series Vol. 2). Taylor & Francis, 1998.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
3

Eitel, Manfred. Cycloadditionsreaktionen von 2-Vinylindolen mit CC-Dienophilen zur Synthese selektiv funktionalisierter [b]anellierter Indole und Carbazole. 1990.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
4

Houlihan, William J. Indoles, Part 2. Wiley & Sons, Incorporated, John, 2009.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
5

Pediatric Collections: Infectious Diseases, Part 2: Indolent Head Scratchers. American Academy of Pediatrics, 2025. https://doi.org/10.1542/9781610028295.

Full text
Abstract:
The second part of this 2-part series on infectious disease, “Part 2: Indolent Head Scratchers,” presents cases of patients not in imminent danger, but sick with puzzling symptoms and histories. Some of these cases have a prolonged clinical course, while others are just plain weird. Some cases present with common findings seen every day in clinical practice, but hide something rare and elusive under the surface, which comes into focus as the case progresses. Some of the diagnoses have been missed or overlooked for quite some time, given the indolent nature of the disease and cognitive biases.
APA, Harvard, Vancouver, ISO, and other styles
6

Erfanian-Abdoust, Houshang. [4 + 2]-Cycloadditionen von Carbo- und Hetero-Dienophilen an Pyrano- und Pyrido[3,4-b]indol-3-onen: Ein neuer Zugang zu selektiv funktionalisierten [b]anellierten Indolen und Carbazolen. 1991.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
7

Kim, Myung-Hwa. [4 + 2]-Cycloadditionen von 2- und 3-Vinylindolen mit Heterodienophilen zu neuen heterocyclisch [b]anellierten und funktionalisierten Indolen. 1991.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
8

Sebag-Montefiore, David, Mark Harrison, and Rob Glynne-Jones. Squamous carcinoma of the anus. Oxford University Press, 2013. http://dx.doi.org/10.1093/med/9780199696567.003.0008.

Full text
Abstract:
Squamous cell cancer (SCC) of the anus is a rare cancer whose incidence appears to be increasing. Anal cancers are more common in women than men ( 1 , 2 ) and just under half the patients are over the age of 65. An indolent natural history and a low rate of distant metastases ( 3 , 2 ) determine locoregional control as the primary aim of treatment. The relative 5-year survival rate is 62 % ( 4 ) , and has changed little for patients treated in the last two decades.
APA, Harvard, Vancouver, ISO, and other styles
9

Rampersad, Nicole Claudia. New indolyl phosphines: Synthesis and characterization of 2-diphenylphosphine-3-methylindole and di(1H-3-indolyl)methane-(2,12)-phenylphosphine : . 2001.

Find full text
APA, Harvard, Vancouver, ISO, and other styles
10

Freieck, Harald. 2a,3,4,5-tetrahydro-1H-benz[cd]indol-2-on als Baustein zur Synthese dopaminerger Substanzen. 1999.

Find full text
APA, Harvard, Vancouver, ISO, and other styles

Book chapters on the topic "Indole-2"

1

Firooznia, Fariborz, Robert F. Kester, and Steven J. Berthel. "[2+2], [3+2] and [2+2+2] Cycloaddition Reactions of Indole Derivatives." In Topics in Heterocyclic Chemistry. Springer Berlin Heidelberg, 2010. http://dx.doi.org/10.1007/7081_2010_53.

Full text
APA, Harvard, Vancouver, ISO, and other styles
2

Winkelmann, J. "Diffusion of indole (1); carbon dioxide (2)." In Gases in Gases, Liquids and their Mixtures. Springer Berlin Heidelberg, 2007. http://dx.doi.org/10.1007/978-3-540-49718-9_1272.

Full text
APA, Harvard, Vancouver, ISO, and other styles
3

Kester, Robert F., Steven J. Berthel, and Fariborz Firooznia. "[4+2] Cycloaddition Reactions of Indole Derivatives." In Topics in Heterocyclic Chemistry. Springer Berlin Heidelberg, 2010. http://dx.doi.org/10.1007/7081_2010_55.

Full text
APA, Harvard, Vancouver, ISO, and other styles
4

Gallego, Mar Gómez, and Miguel A. Sierra. "Level 1 — Case 2 Sulfenylation of Indole." In Organic Reaction Mechanisms. Springer Berlin Heidelberg, 2004. http://dx.doi.org/10.1007/978-3-642-18788-9_2.

Full text
APA, Harvard, Vancouver, ISO, and other styles
5

Wohlfarth, Ch. "Viscosity of the mixture (1) 1H-indole; (2) 2-methylnaphthalene." In Supplement to IV/18. Springer Berlin Heidelberg, 2008. http://dx.doi.org/10.1007/978-3-540-75486-2_1778.

Full text
APA, Harvard, Vancouver, ISO, and other styles
6

Winkelmann, J. "Diffusion of indole (1); carbon dioxide (2); hexane (3)." In Gases in Gases, Liquids and their Mixtures. Springer Berlin Heidelberg, 2007. http://dx.doi.org/10.1007/978-3-540-49718-9_1710.

Full text
APA, Harvard, Vancouver, ISO, and other styles
7

Pardasani, R. T., and P. Pardasani. "Magnetic properties of indole-2-carboxylatodiruthenium(II, III) complex." In Magnetic Properties of Paramagnetic Compounds. Springer Berlin Heidelberg, 2015. http://dx.doi.org/10.1007/978-3-662-45972-0_425.

Full text
APA, Harvard, Vancouver, ISO, and other styles
8

Wohlfarth, Ch. "Viscosity of the mixture (1) 1H-indole; (2) isoquinoline." In Supplement to IV/18. Springer Berlin Heidelberg, 2008. http://dx.doi.org/10.1007/978-3-540-75486-2_1777.

Full text
APA, Harvard, Vancouver, ISO, and other styles
9

Negishi, Tomoe, Sakae Arimoto, Chiharu Nishizaki, and Hikoya Hayatsu. "Inhibition of the Genotoxicity of 3-Amino-1-Methyl-5H- Pyrido[4,3-b]Indole (Trp-P-2) in Drosophila by Chlorophyll." In Antimutagenesis and Anticarcinogenesis Mechanisms II. Springer US, 1990. http://dx.doi.org/10.1007/978-1-4615-9561-8_29.

Full text
APA, Harvard, Vancouver, ISO, and other styles
10

Swathi, K., M. Chaitanya, B. Murugesan, and B. Karan Kumar. "Synthesis, Anti-inflammatory Activity, and In Silico Studies of Some New 3-({P-Dimethylamino}benzylidenehydrazinylidene)-1,3-dihydro-2H-indole-2-one Derivatives." In GeNeDis 2020. Springer International Publishing, 2021. http://dx.doi.org/10.1007/978-3-030-78787-5_43.

Full text
APA, Harvard, Vancouver, ISO, and other styles

Conference papers on the topic "Indole-2"

1

Tiuleanu, Pavel, Ivan Marenin, and Andrei Shchekotikhin. "Synthesis and evaluation of new 2-azolylindoles - derivatives of indole-2-carboxylic." In Conferința științifică națională cu participare internațională "Integrare prin cercetare și inovare", dedicată Zilei Internaționale a Științei pentru Pace și Dezvoltare. Moldova State University, 2025. https://doi.org/10.59295/spd2024n.91.

Full text
Abstract:
Indole-2-carboxylic acid is a promising scaffold for the design of new compounds with application in biological studies and medicine practice. Its derivatives have shown a wide range of biological activity: antiviral, antifungal, antibacterial, anti-inflammatory. As part of the presented study, the method for preparation of alkyl derivatives of acetoacetic ester has been optimized. These derivatives are intermediates for the synthesis of indole-2-carboxylic acid esters according to the Japp-Klingemann/Fisher methodology. Several methods for the transformation of indole-2-carboxylic acid ester
APA, Harvard, Vancouver, ISO, and other styles
2

Zou, Wen-Sheng, Hong Zhang, Shuang Jia, Wu-Fu Zhu, and Shan Xu. "3-(2-chloro-5-fluoropyrimidin-4-yl)-1-methyl-1H-indole." In 2017 2nd International Conference on Biological Sciences and Technology (BST 2017). Atlantis Press, 2018. http://dx.doi.org/10.2991/bst-17.2018.35.

Full text
APA, Harvard, Vancouver, ISO, and other styles
3

Savchuk, Maria I., Dmitry S. Kopchuk, Alexey P. Krinochkin, et al. "Preparation of indole-containing 3-(2-pyridyl)-1,2,4-triazines as tryptamine derivatives." In PROCEEDINGS OF THE 3RD INTERNATIONAL CONFERENCE ON AUTOMOTIVE INNOVATION GREEN ENERGY VEHICLE: AIGEV 2018. Author(s), 2019. http://dx.doi.org/10.1063/1.5087380.

Full text
APA, Harvard, Vancouver, ISO, and other styles
4

Menéndez, J., Vellaisamy Sridharan, Subbu Perumal, and Carmen Avendaño. "Bischler Indole Synthesis under Microwave Irradiation: A Solvent-Free Synthesis of 2-Arylindoles." In The 9th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2005. http://dx.doi.org/10.3390/ecsoc-9-01632.

Full text
APA, Harvard, Vancouver, ISO, and other styles
5

yang, shiyi, Kaijun Chen, Min Zhang, et al. "4-Indole-2-Arylaminopyrimidine identifies lysosomal cathepsin L activation critical for acute lung injury." In ERS International Congress 2023 abstracts. European Respiratory Society, 2023. http://dx.doi.org/10.1183/13993003.congress-2023.pa1257.

Full text
APA, Harvard, Vancouver, ISO, and other styles
6

Blasko, Gy, G. Blasko, G. Sas, and Cs Szantay. "MODULATION OF THROMBIN-MEDIATED REACTIONS IN HAEMOSTASIS- BY TREQUINSIN AND ITS ANALOGUES." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643432.

Full text
Abstract:
A new pyrimido/6,1-a/-isoquinoline derivative ,/Ref.1 / developed by Hoechst and named Trequinsine has been reported to be a powerful inhibitor of cAMP phosphodiesterase and platelet aggregation having a potency nearly similar to prostacyclin. We synthesized Trequins-in (1), its indole derivative (4) , as well as their precursors (2 3) and subjected them to a study in order to evaluate their effects on haemostasis. Surprisingly they exhibited a modulatory effect only on reactions mediated mainly by thrombin. They inhibited platelet aggregation (ICc:q for Trequinsin: 13 + 2.5 ng/ml, for indole
APA, Harvard, Vancouver, ISO, and other styles
7

Shaw, Subrata, James Chris Tarr, Nicholas Pelz, et al. "Abstract 4331: Discovery of potent 2-Indole-acylsulfonamide Mcl-1 inhibitors using structure guided fragment-based methods." In Proceedings: AACR 107th Annual Meeting 2016; April 16-20, 2016; New Orleans, LA. American Association for Cancer Research, 2016. http://dx.doi.org/10.1158/1538-7445.am2016-4331.

Full text
APA, Harvard, Vancouver, ISO, and other styles
8

Jabbar, Alyaa, and Yasameen K. Al-Majedy. "Synthesis and bio-evaluation of 2-Methyl Indole-3-carboxaldehyde derivatives as potential lanosterol 14-demethylase inhibitors." In 4TH INTERNATIONAL CONFERENCE ON INNOVATION IN IOT, ROBOTICS AND AUTOMATION (IIRA 4.0). AIP Publishing, 2025. https://doi.org/10.1063/5.0255335.

Full text
APA, Harvard, Vancouver, ISO, and other styles
9

Manabe, S., H. Yanagisawa, S. Ishikawa, et al. "TRYPTOPHAN PYROLYSIS PRODUCTS FOUND IN COOKED FOODS INHIBIT HUMAN PLATELET AGGREGATION BY INHIBITING CYCLOOXYGENASE." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643402.

Full text
Abstract:
Humans are exposed to numerous toxic compounds in foods. During the past decade, several carcinogenic heterocyclic amines have been reported to be present in the cooked foods. Recently, we reported that some of the carcinogenic heterocyclic amines isolated from foods were present in human plasma. In order to know the effects of the carcinogens isolated from foods on the cell function, we investigated the effects of the carcinogenic heterocyclic amines including Trp-P-1(3-amino-l,4-dimethyl-5H-pyrido❘4,3-b❘indole) and Trp-P-2(3-amino-1-methyl-5H-pyrido❘4,3-b❘indole) on human platelet aggregatio
APA, Harvard, Vancouver, ISO, and other styles
10

Azev, Yu A., O. S. Koptyaeva, O. S. Eltsov, Yu A. Yakovleva, T. A. Pospelova, and V. A. Bakulev. "Benzaldehyde phenylhydrazones as c-nucleophiles for functionalization of quinoxaline-2-one. Unusual transformations of indole-3-carbaldehyde phenylhydrazones." In PROCEEDINGS OF INTERNATIONAL CONFERENCE ON RECENT TRENDS IN MECHANICAL AND MATERIALS ENGINEERING: ICRTMME 2019. AIP Publishing, 2020. http://dx.doi.org/10.1063/5.0018799.

Full text
APA, Harvard, Vancouver, ISO, and other styles

Reports on the topic "Indole-2"

1

Chamovitz, A. Daniel, and Georg Jander. Genetic and biochemical analysis of glucosinolate breakdown: The effects of indole-3-carbinol on plant physiology and development. United States Department of Agriculture, 2012. http://dx.doi.org/10.32747/2012.7597917.bard.

Full text
Abstract:
Genetic and biochemical analysis of glucosinolate breakdown: The effects of indole-3-carbinol on plant physiology and development Glucosinolates are a class of defense-related secondary metabolites found in all crucifers, including important oilseed and vegetable crops in the Brassica genus and the well-studied model plant Arabidopsis thaliana. Upon tissue damage, such as that provided by insect feeding, glucosinolates are subjected to catalysis and spontaneous degradation to form a variety of breakdown products. These breakdown products typically have a deterrent effect on generalist herbivor
APA, Harvard, Vancouver, ISO, and other styles
2

Steele, W. V., and R. D. Chirico. Thermodynamics and the hydrodenitrogenation of indole: Part 1, Thermodynamic properties of indoline and 2-methylindole: Part 2, Gibbs energies of reaction in the hydrodenitrogenation of indole: Part 3, Thermodynamic equilibria and comparison with literature kinetic. Office of Scientific and Technical Information (OSTI), 1989. http://dx.doi.org/10.2172/6124014.

Full text
APA, Harvard, Vancouver, ISO, and other styles
You might also be interested in the extended bibliographies on the topic 'Indole-2' for particular source types:
Journal articles Dissertations / Theses
We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!

To the bibliography