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Journal articles on the topic 'Phenylthiazole'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

Bhuiyan, M. H., and A. F. M. H. Rahman. "Synthesis and Antimicrobial Evaluation of Some Thiazole Derivatives." Journal of Scientific Research 3, no. 1 (2010): 111. http://dx.doi.org/10.3329/jsr.v3i1.5419.

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Reaction of 2-amino-4-phenylthiazole with various aromatic aldehydes afforded 2-arylideneamino-4-phenylthiazoles. On the other hand treatment of 2-amino-4-phenylthiazole with several acyl halides furnished N-(thiazol-2-yl)-amides. The synthesized compounds have been screened for their antimicrobial activity against Bacillus cereus, Bacillus subtilis, Staphylococcus aureus, Shigella dysenteriae, Salmonella typhi, Pseudomonous sp. bacteria and Aspergillus niger, Penicillium notatum, Aspergillus funiculosus, Collectrichum corchori Ikata (Yoshida) and Curvularia lunata fungi respectively. Some of

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2

Fouda, Abdel Aziz, A. Abdel Nazeerb, and K. M. Abdel Khalek. "Corrosion Inhibition of Zinc Using Some Phenylthiazole Derivatives in Hydrochloric acid Solutions." JOURNAL OF ADVANCES IN CHEMISTRY 12, no. 7 (2013): 425–40. http://dx.doi.org/10.24297/jac.v12i7.2798.

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The inhibitive action of some phenylthiazole derivatives namely: 2-acetylamino-5-p-bromophenylazo-4-phenylthiazole (BPT), 2-acetylamino-5-p-methylphenylazo-4-phenylthiazole (MPT), 2-acetylamino-5-p-methoxyphenylazo-4-phenylthiazole (XPT) and 2-acetylamino-5-p-nitrophenylazo-4-phenylthiazole (NPT), on zinc corrosion in 0.2 M HCl has been studied using weight loss, potentiodynamic polarization, electrochemical impedance spectroscopy (EIS)and electrochemical frequency modulation (EFM) measurements. The results showed that the dissolution rate of zinc decreases with increasing the phenylthiazole d

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3

Fouda, Abdel Aziz, A. Abdel Nazeerb, and K. M. Abdel Khalek. "Corrosion Inhibition of Zinc Using Some Phenylthiazole Derivatives in Hydrochloric acid Solutions." JOURNAL OF ADVANCES IN CHEMISTRY 4, no. 2 (2008): 425–40. http://dx.doi.org/10.24297/jac.v4i2.2704.

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The inhibitive action of some phenylthiazole derivatives namely: 2-acetylamino-5-p-bromophenylazo-4-phenylthiazole (BPT), 2-acetylamino-5-p-methylphenylazo-4-phenylthiazole (MPT), 2-acetylamino-5-p-methoxyphenylazo-4-phenylthiazole (XPT) and 2-acetylamino-5-p-nitrophenylazo-4-phenylthiazole (NPT), on zinc corrosion in 0.2 M HCl has been studied using weight loss, potentiodynamic polarization, electrochemical impedance spectroscopy (EIS)and electrochemical frequency modulation (EFM) measurements. The results showed that the dissolution rate of zinc decreases with increasing the phenylthiazole d

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4

Zhu, ShaoPing, Yuan Chen, Jun Sun, YuTing Yang, and ChuanJun Yue. "Synthesis, Characterization, Thermochromism, and Photochromism of Aromatic Aldehyde Hydrazone Derivatives." Journal of Chemistry 2016 (2016): 1–8. http://dx.doi.org/10.1155/2016/8460462.

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The Schiff bases N-(5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (1), N-(4′-chloro-5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (2), and N-(4′-nitro-5-phenylthiazole-2-yl)-2-hydroxylnaphthaldehydehydrazone (3) were synthesized. These compounds were characterized by using IR,1H NMR,13C NMR, and MS. The photochromism of the compounds was investigated by IR and UV-visible spectrometry which is time variable under irradiation of 254 nm UV light. The thermochromism of the compounds was studied using temperature-variable IR, UV-visible spectrometry, TG, and differential scann

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5

Au-Alvarez, O., R. C. Peterson, A. Acosta Crespo, et al. "2-Amino-4-phenylthiazole." Acta Crystallographica Section C Crystal Structure Communications 55, no. 5 (1999): 821–23. http://dx.doi.org/10.1107/s0108270199001961.

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6

Stokes, Emily C., Emily E. Langdon-Jones, Lara M. Groves, et al. "Cationic, luminescent cyclometalated iridium(iii) complexes based on substituted 2-phenylthiazole ligands." Dalton Transactions 44, no. 18 (2015): 8488–96. http://dx.doi.org/10.1039/c4dt03054k.

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7

D., C. DASH, K. BEHERA R., M. SEN (Miss), and M. MEHER F. "Synthesis and Characterisation of some Transition Metal Complexes of 4-Substituted-2-thiazolylhydrazones of Salicylaldehyde and 2-Hydroxyacetophenone." Journal of Indian Chemical Society Vol. 68, Dec 1991 (1991): 663–64. https://doi.org/10.5281/zenodo.6134555.

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Post-Graduate Department of Chemistry, Sambalpur University, Jyoti Vihar, Burla-788 019 <em>Manuscript received 27 April 1988, revised 21 November 1991, accepted 6 December 1991</em> THE communication reports the synthesis and structural studies on the complexes of Co<sup>II</sup>, Ni<sup>II</sup> and Cu<sup>ll</sup> with some hydrazone derivatives containing thiazole moiety and a OH group near the condensation site, such as 2-salicylideneiminoamino-4- phenylthiazole (SPTH), 2-salicylideneiminoamino-4-bromophenylthiazole (SBPTH), 2-α-methylsalicyli-deneiminoamino-4- phenylthiazole (MSPTH

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8

Zhao, Jiang, Xiaojie Chen, Jianglan Wu, Maoyang Jian, Guijiang Zhou, and Zhenguo Chi. "Fluoro-benzenesulfonyl-functionalized 2-phenylthiazole-type iridium(iii) complexes for efficient solution-processed organic light-emitting diodes." Journal of Materials Chemistry C 8, no. 30 (2020): 10390–400. http://dx.doi.org/10.1039/d0tc02250k.

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9

Bhuiyan, Md Mosharef Hossain, Mohammed M. Matin, AFM Hafizur Rahman, and Md Rabiul Alam. "Synthesis and Biological Evaluation of Sugar Induced Thiazole Derivatives." Chittagong University Journal of Science 41, no. 1 (2021): 68–84. http://dx.doi.org/10.3329/cujs.v41i1.51915.

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The starting materials, 2-amino-4-phenylthiazole and 2-amino-4,5,6,7-tetrahydrobenzo[d]thiazole, were prepared by reacting thiourea with acetophenone and cyclohexanone in the presence of iodine under heating on a water bath with occasional stirring, respectively. Reaction of 2-amino-4-phenylthiazole and 2-amino-4,5,6,7-tetrahydrobenzo[d]thiazole with various sugars afforded corresponding N-glycoside derivatives in good yields. The structures of the synthesized N-glycosides derivatives have been established on the basis of their IR and NMR spectral data. The obtained compounds were screened for

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10

Mayhoub, Abdelrahman S., Mansoora Khaliq, Carolyn Botting, Ze Li, Richard J. Kuhn, and Mark Cushman. "An investigation of phenylthiazole antiflaviviral agents." Bioorganic & Medicinal Chemistry 19, no. 12 (2011): 3845–54. http://dx.doi.org/10.1016/j.bmc.2011.04.041.

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11

Ai, Hong-Lian, Bao-Bao Shi, Wei Li, et al. "Bipolarithizole A, an antifungal phenylthiazole-sativene merosesquiterpenoid from the potato endophytic fungus Bipolaris eleusines." Organic Chemistry Frontiers 9, no. 7 (2022): 1814–19. http://dx.doi.org/10.1039/d1qo01887f.

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Bipolarithizole A (1) is a phenylthiazole-sativene sesquiterpenoid hybrid isolated from the fungus Bipolaris eleusines. It shows anti-pathogenic fungi activity against Rhizoctonia solani with an MIC value of 16 μg mL−1.

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12

Omara, Mariam, Mohamed Hagras, Mohamed M. Elsebaie, et al. "Exploring novel aryl/heteroaryl-isosteres of phenylthiazole against multidrug-resistant bacteria." RSC Advances 13, no. 29 (2023): 19695–709. http://dx.doi.org/10.1039/d3ra02778c.

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Twenty-three compounds of novel phenylthiazole derivatives were synthesized utilizing the Suzuki coupling reaction. Antibacterial activity in an in vivo model against MRSA USA300 was evaluated, as it reduced the burden of MRSA USA300 in skin-infected mice.

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13

Mamedov, Vakhid A., Yakov A. Levin, Evgeniya K. Trutneva, et al. "Functionalized 4-methyl-5-phenylthiazole and 1,3-bis(4'-methyl-5'-phenylthiazol-2'-yl)benzene. Approaching thiazole macrocycles." Arkivoc 2004, no. 12 (2005): 47–69. http://dx.doi.org/10.3998/ark.5550190.0005.c06.

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14

Nagaladinne, Nizamuddin, Abdul Ahad Hindustan, and Devanna Nayakanti. "Design, Synthesis and Molecular Modelling Studies of 1-Methyl-3-(4-Substituted phenyl-1,3- thiazol-2-yl)-2-(pyridin-3-yl)-2,3-dihydroquinazolin-4(1H)-ones as Potent Anticancer Agents." Asian Journal of Chemistry 32, no. 12 (2020): 3067–74. http://dx.doi.org/10.14233/ajchem.2020.22930.

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The present study involves the design, synthesis, characterization and molecular docking studies of biologically active quinazolin-4-ones, which were synthesized by condensing 2-amino-4-substituted phenylthiazole with N-methylbenzoxazin-4-one. The N-methylbenzoxazin-4-one and 2-amino-4- substituted phenylthiazole were synthesized from N-methylanthranilic acid and substituted ketones, respectively. The ADME properties determined the synthetic accessibility of quinazolin-4-ones by in silico Swiss ADME. The colorectal anticancer screening was done by using cell HT-29 human colorectal adenocarcino

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15

Pulat, Sultan, Inho Yang, Jihye Lee, et al. "Anithiactin D, a Phenylthiazole Natural Product from Mudflat-Derived Streptomyces sp., Suppresses Motility of Cancer Cells." Marine Drugs 22, no. 2 (2024): 88. http://dx.doi.org/10.3390/md22020088.

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Anithiactin D (1), a 2-phenylthiazole class of natural products, was isolated from marine mudflat-derived actinomycetes Streptomyces sp. 10A085. The chemical structure of 1 was elucidated based on the interpretation of NMR and MS data. The absolute configuration of 1 was determined by comparing the experimental and calculated electronic circular dichroism (ECD) spectral data. Anithiactin D (1) significantly decreased cancer cell migration and invasion activities at a concentration of 5 μM via downregulation of the epithelial-to-mesenchymal transition (EMT) markers in A549, AGS, and Caco-2 cell

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16

Tian, Yao, Jinchao Shi, Xiaoqian Deng, et al. "Design, Synthesis, and Antifungal Activity of Some Novel Phenylthiazole Derivatives Containing an Acylhydrazone Moiety." Molecules 28, no. 20 (2023): 7084. http://dx.doi.org/10.3390/molecules28207084.

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Crop fungal diseases pose a serious threat to global crop production and quality. Developing new and efficient fungicides is an important measure to control crop diseases. Phenylthiazole was found to be an excellent antifungal skeleton based on our previous study on the structural optimization and biological activity of the natural product thiasporine A. To find new fungicides, 45 phenylthiazole derivatives containing an acylhydrazone moiety were designed and synthesized by the principle of active substructure splicing. Forty-two of the forty-five compounds are novel, except for compounds E1,

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17

Seleem, Mohammed A., Ahmed M. Disouky, Haroon Mohammad, et al. "Second-Generation Phenylthiazole Antibiotics with Enhanced Pharmacokinetic Properties." Journal of Medicinal Chemistry 59, no. 10 (2016): 4900–4912. http://dx.doi.org/10.1021/acs.jmedchem.6b00233.

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18

Y., Jadegoud, B. Ijare Omkar, N. Mallikarjuna N., D. Angadi S., and H. M. Mruthyunjayaswamy B. "Synthesis and antimicrobial activity of copper-, cobalt- and nickel(II) complexes with Schiff bases." Journal of Indian Chemical Society Vol. 79, Dec 2002 (2002): 921–24. https://doi.org/10.5281/zenodo.5847948.

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Department of Chemistry, Gulbarga University. Gulbarga-585 106, India <em>E-mail </em>: root@guluni.kar.nic.in         <em>  Fax :</em> 91-08472-21632 <em>Manuscript received 1 January 2002, accepted 12 July 2002</em> A few complexes of Cu<sup>II</sup>, Co<sup>II</sup> and Ni<sup>II</sup> have been prepared by reacting their metal(ll) chlorides with 3-(4'-phenylthiazole-2'-yl)- 1-(2' -hydroxy-l' -iminomcthylphenly)urea and with 3-(4' -phenylthiazole-2' -yl)-1-(2' ,4' -dihydroxy/2' -hydroxy-5' -chloro-1 '-m

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19

Khrustalev, D. P. "Modification of 2-amino-4-phenylthiazole under microwave irradiation." Russian Journal of General Chemistry 79, no. 3 (2009): 515–16. http://dx.doi.org/10.1134/s1070363209030311.

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20

Nalini, Veerapaneni, and Gautam R. Desiraju. "Gas–solid chlorination of 4-phenylthiazole-2(1H)-thione." J. Chem. Soc., Chem. Commun., no. 13 (1987): 1046–48. http://dx.doi.org/10.1039/c39870001046.

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21

Kenzhetaeva, S. O., and L. K. Abulyaissova. "Synthesis of 2-amino-4-phenylthiazole-derived thiuram disulfide." Russian Journal of General Chemistry 83, no. 11 (2013): 2115–16. http://dx.doi.org/10.1134/s1070363213110285.

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22

Kouhkan, Maryam, Ali Souldozi, and Reza Talebi. "In Vitro Antimicrobial Activity of New Substituted Phenylthiazole Derivatives." Iranian Jornal of Toxicology 12, no. 1 (2018): 33–37. http://dx.doi.org/10.29252/arakmu.12.1.33.

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23

Davydova, Yulia А., Taras M. Sokolenko, Yurii G. Vlasenko, and Yurii L. Yagupolskii. "Chemical properties of 5-(1,1,2,2-tetrafluoroethoxy)-4-phenylthiazole derivatives." Chemistry of Heterocyclic Compounds 51, no. 1 (2015): 80–87. http://dx.doi.org/10.1007/s10593-015-1663-z.

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24

Takami, Shizuka, Minori Nishiyama, Masaki Mizuno, Tadatsugu Yamaguchi, Yuichiro Hashimoto, and Tsuyoshi Kawai. "Photochromic Performance of 5-Heteroaryl-4-vinyl-2-phenylthiazole Derivatives." Bulletin of the Chemical Society of Japan 92, no. 10 (2019): 1773–78. http://dx.doi.org/10.1246/bcsj.20190093.

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25

Ezzat, Hany. "SYNTHESIS AND EVALUATION OF NEW PHENYLTHIAZOLE DERVATIVES AS ANTIMICROBIAL AGENTS." Al-Azhar Journal of Pharmaceutical Sciences 60, no. 2 (2019): 59–75. http://dx.doi.org/10.21608/ajps.2019.70240.

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26

Nicolás, Álvaro, Julia G. Quero, Marta Barroso, Zoila Gándara, and Lourdes Gude. "DNA Interactions and Biological Activity of 2,9-Disubstituted 1,10-Phenanthroline Thiosemicarbazone-Based Ligands and a 4-Phenylthiazole Derivative." Biology 13, no. 1 (2024): 60. http://dx.doi.org/10.3390/biology13010060.

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Four 1,10-phenanthroline derivatives (1–4) were synthesized as potential telomeric DNA binders, three substituted in their chains with thiosemicarbazones (TSCs) and one 4-phenylthiazole derivative. The compounds were characterized using NMR, HRMS, FTIR-spectroscopy and combustion elemental analysis. Quadruplex and dsDNA interactions were preliminarily studied, especially for neutral derivative 1, using FRET-based DNA melting assays, equilibrium dialysis (both competitive and non-competitive), circular dichroism and viscosity titrations. The TSC derivatives bind and stabilize the telomeric Tel2

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27

Parvez, M., S. Ali, M. Mazhar, M. H. Bhatti, and M. N. Khokhar. "Aqua[4-(4-chlorophenyl)-2-phenylthiazole-5-acetato-O]trimethyltin(IV)." Acta Crystallographica Section C Crystal Structure Communications 55, no. 8 (1999): 1280–82. http://dx.doi.org/10.1107/s0108270199005120.

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28

Sadigova, S. E., A. M. Magerramov, and M. A. Allakhverdiev. "Synthesis of Schiff bases and oxazolidines from 2-amino-4-phenylthiazole." Russian Journal of Organic Chemistry 44, no. 12 (2008): 1821–23. http://dx.doi.org/10.1134/s107042800812018x.

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29

Subhashini, N. J. P., Jampaiah Amanaganti, and Shivaraj. "Synthesis and antibacterial activity of 2-(3-acylphenyl)amino-4-phenylthiazole." Russian Journal of General Chemistry 85, no. 3 (2015): 686–88. http://dx.doi.org/10.1134/s1070363215030275.

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30

Khrustalev, D. P., A. A. Suleimenova, and S. D. Fazylov. "Synthesis of 2-amino-4-phenylthiazole under conditions of microwave irradiation." Russian Journal of Applied Chemistry 81, no. 5 (2008): 900. http://dx.doi.org/10.1134/s1070427208050376.

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31

Souldozi, Ali, Ali Ramazani, Ali Reza Dadrass, Katarzyna Ślepokura, and Tadeusz Lis. "Efficient One-Pot Synthesis of Alkyl 2-(Dialkylamino)-4-phenylthiazole-5-carboxylates and Single-Crystal X-Ray Structure of Methyl 2-(Diisopropylamino)-4-phenylthiazole-5-carboxylate." Helvetica Chimica Acta 95, no. 2 (2012): 339–48. http://dx.doi.org/10.1002/hlca.201100322.

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32

Zhang, Zhi-Hua, Hong-Mei Wu, Sai-Nan Deng, et al. "Design, Synthesis, and Anticancer Activities of Novel 2-Amino-4-phenylthiazole Scaffold Containing Amide Moieties." Journal of Chemistry 2018 (October 18, 2018): 1–8. http://dx.doi.org/10.1155/2018/4301910.

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Appropriately substituted 2-amino-4-phenylthiazole derivatives were designed and synthesized according to the structural characteristics of crizotinib. The obtained compounds were characterized using 1H NMR, 13C NMR, and HRMS. The target compounds 5a–o were evaluated for their in vitro antiproliferative activity against A549, HeLa, HT29, and Karpas299 human cancer cell lines. Based on results of biological studies, some of these compounds exhibited significant antiproliferative activity. Compound 5b possessed outstanding growth inhibitory effects on the four cell lines, especially for HT29 cel

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33

Sal’keeva, L. K., P. Voitichek, E. K. Taishibekova, et al. "Unusual phosphorylation of 2-amino-4-phenylthiazole with phosphorous acid ester amides." Russian Journal of General Chemistry 84, no. 12 (2014): 2477–79. http://dx.doi.org/10.1134/s1070363214120275.

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34

Ieda, Hidenori, Hiroyuki Fujiwara, and Yoshio Fuchita. "Synthesis and reactivity of the five-membered cycloaurated complexes of 2-phenylthiazole." Inorganica Chimica Acta 319, no. 1-2 (2001): 203–6. http://dx.doi.org/10.1016/s0020-1693(01)00432-7.

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35

Chen, K. Q., M. Q. Song, W. L. Wu, et al. "Synthesis, Characterization, Crystal Structure, and Antitumor Activity of 2-Phenylthiazole–Coumarin Derivatives." Russian Journal of Organic Chemistry 58, no. 9 (2022): 1341–47. http://dx.doi.org/10.1134/s1070428022090214.

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36

Yahia, Eman, Haroon Mohammad, Tamer M. Abdelghany, Eman Fayed, Mohamed N. Seleem, and Abdelrahman S. Mayhoub. "Phenylthiazole antibiotics: A metabolism-guided approach to overcome short duration of action." European Journal of Medicinal Chemistry 126 (January 2017): 604–13. http://dx.doi.org/10.1016/j.ejmech.2016.11.042.

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37

Avanish, Kumar, and Kumar Rajesh. "ChemInform Abstract: Synthesis of Schiff′s Bases of 2-Amino-4-phenylthiazole." ChemInform 42, no. 48 (2011): no. http://dx.doi.org/10.1002/chin.201148253.

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38

Hosny, Yomna, Nader S. Abutaleb, Mariam Omara, et al. "Modifying the lipophilic part of phenylthiazole antibiotics to control their drug-likeness." European Journal of Medicinal Chemistry 185 (January 2020): 111830. http://dx.doi.org/10.1016/j.ejmech.2019.111830.

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39

Souldozi, Ali, Ali Ramazani, Ali Reza Dadrass, Katarzyna Slepokura, and Tadeusz Lis. "ChemInform Abstract: Efficient One-Pot Synthesis of Alkyl 2-(Dialkylamino)-4-phenylthiazole-5-carboxylates and Single Crystal X-Ray Structure of Methyl 2-(Diisopropylamino)-4-phenylthiazole-5-carboxylate." ChemInform 43, no. 26 (2012): no. http://dx.doi.org/10.1002/chin.201226132.

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40

Shi, Da-Hua, Zong-Ming Tang, Xiao-Dong Ma, et al. "Synthesis, Crystal Structure and Biological Evaluation of Novel 2-Phenylthiazole Derivatives as Multi-Targeting Agents to Treat Alzheimer's Disease." Journal of Chemical Research 41, no. 9 (2017): 551–55. http://dx.doi.org/10.3184/174751917x15045169836217.

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Three novel 2-phenylthiazole derivatives were synthesised and characterised by spectroscopic techniques. The structure of the synthesised compounds was unambiguously confirmed by a single-crystal X-ray diffraction analysis of ethyl 2-(4-{[5-(4-benzylpiperidin-1-yl)pentyl]oxy}phenyl)thiazole-4-carboxylate. All of the compounds presented good cholinesterase-inhibition activities and ethyl 2-(4-{[5-(4-benzylpiperidin-1-yl)pentyl]oxy}phenyl)thiazole-4-carboxylate showed the best acetylcholinesterase-inhibition and butyrylcholinesterase-inhibition abilities with IC50 values of 5.19 μM and 5.83 μM.

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41

Shi, Da-Hua, Xiao-Dong Ma, Yu-Wei Liu, et al. "Synthesis, Crystal Structure and Biological Evaluation of Novel 2-Phenylthiazole Derivatives as Butyrylcholinesterase Inhibitors." Journal of Chemical Research 42, no. 7 (2018): 366–70. http://dx.doi.org/10.3184/174751918x15314837408346.

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To find novel butyrylcholinesterase inhibitors, three novel 2-phenylthiazole derivatives were synthesised. The synthesised compounds were characterised by NMR and single-crystal X-ray diffraction analysis. Hirshfeld surface analysis and two-dimensional fingerprint plots of the compounds were used as a theoretical approach to assess the driving force for crystal structure formation via the intermolecular interactions in the crystal lattices of the synthesised compounds. Among the three compounds, N-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro- 1H-pyrazol-4-yl)-2-(4-methoxyphenyl)thiazole-4-carboxam

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42

Mukesh, Bugalia, B. Puranik Sangamesh, Saraswat Rohit, Jhajharia Mahesh, and Sharma Prashant. "Synthesis of Thiazoles and 1,3,4-Thiadiazoles Bearing Spectral Studies, Biological Evaluation and Structure Activity relationship." International Journal of Engineering Research & Science 6, no. 7 (2020): 21–33. https://doi.org/10.5281/zenodo.4095165.

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<strong>Abstract</strong><strong>—</strong> A novel series of thiazole based-1,3,4-thiadiazoles were designed and prepared via the reaction of the 2-(4-methyl-2-phenylthiazole-5-carbonyl)-N-phenylhydrazinecarbothioamide with the appropriate hydrazonoyl chlorides. The structures of the newly synthesized compounds were established based on spectroscopic evidences and their alternative syntheses. Thirteen new 1,3,4-thiadiazoles have been evaluated for their anticancer activity against liver carcinoma cell line (HepG2). Also, their structure activity relationship (SAR) was studied. The 1,3,4

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43

Cao, Lei, Jingwei Sun, Qiang Liu, et al. "Synthesis and Biological Activity of 5-Amino-4-methyl-N-phenylthiazole-2-carboxamide." Chinese Journal of Organic Chemistry 37, no. 11 (2017): 3031. http://dx.doi.org/10.6023/cjoc201705029.

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44

Sayyah, S. M., M. M. EL-Deeb, and S. S. Abdel-Rehim. "ELECTROPOLYMERIZATION OF 2-AMINO-4-PHENYLTHIAZOLE AND CHARACTERIZATION OF THE OBTAINED POLYMER FILMS." International Journal of Polymeric Materials 53, no. 11 (2004): 941–58. http://dx.doi.org/10.1080/00914030490502454.

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45

Shi, Da-Hua, Xiao-Dong Ma, Zong-Ming Tang, et al. "Synthesis, characterization, crystal structure and urease-inhibition activities of three 2-phenylthiazole derivatives." Journal of Molecular Structure 1173 (December 2018): 81–91. http://dx.doi.org/10.1016/j.molstruc.2018.06.096.

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Liu, Guoxing, Guilai Liu, Madhumita Chatterjee та ін. "Influence of γ-Secretase Inhibitor 24-Diamino-5-Phenylthiazole DAPT on Platelet Activation". Cellular Physiology and Biochemistry 38, № 2 (2016): 726–36. http://dx.doi.org/10.1159/000443029.

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Background/Aims: DAPT (24-diamino-5-phenylthiazole) inhibits γ-secretase, which cleaves the signaling molecule CD44, a negative regulator of platelet activation and apoptosis. CD44 is a co-receptor for macrophage migration inhibitory factor (MIF) an anti-apoptotic pro-inflammatory cytokine expressed and released from blood platelets. Whether DAPT influences platelet function, remained, however, elusive. Activators of platelets include collagen related peptide (CRP). The present study thus explored whether DAPT modifies the stimulating effect of CRP on platelet function. Methods: Platelets isol

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Aliabadi, Alireza, Fazel Shamsa, Seyed Nasser Ostad, et al. "Synthesis and biological evaluation of 2-phenylthiazole-4-carboxamide derivatives as anticancer agents." European Journal of Medicinal Chemistry 45, no. 11 (2010): 5384–89. http://dx.doi.org/10.1016/j.ejmech.2010.08.063.

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V., Mishra. "Coordination polymers of copper( II) imides with polymeric heterocyclic Schiff bases of thiazole derivatives." Journal of India Chemical Society Vol. 79, Apr 2002 (2002): 374–75. https://doi.org/10.5281/zenodo.5849358.

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Department of Post- Graduate Studies in Chemistry, Nehru College, Chhibramau-209 721, India <em>Manuscript received 29 September 2000. revised 26 July 2001. accepted 1 September 2001</em> Two polymeric ligands, L<sub>1</sub> and L<sub>2</sub> were synthesized by polymerizing new heterocyclic Schiff bases 2-hydroxy-1-benzylidene-2-amino· 4-phenylthiazole and 2-hydroxy-1-benzylidene-2-amino-4-phenyl-5-phenylazothiazole, with 1,6-dichlorohexane. L<sub>1</sub>. L<sub>2</sub> gave solid chelates with copper( II) phthalimide or succinimide. The metal ion is coordinated through nitrogen of imi

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Tian, Yuan, Ni An, Wenru Li, et al. "Discovery of Ureido-Substituted 4-Phenylthiazole Derivatives as IGF1R Inhibitors with Potent Antiproliferative Properties." Molecules 29, no. 11 (2024): 2653. http://dx.doi.org/10.3390/molecules29112653.

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The existing kinase inhibitors for hepatocellular carcinoma (HCC) have conferred survival benefits but are hampered by adverse effects and drug resistance, necessitating the development of novel agents targeting distinct pathways. To discover potent new anti-HCC compounds, we leveraged scaffold hopping from Sorafenib and introduced morpholine/piperidine moieties to develop ureido-substituted 4-phenylthiazole analogs with optimized physicochemical properties and binding interactions. Notably, compound 27 exhibited potent cytotoxicity against HepG2 cells (IC50 = 0.62 ± 0.34 μM), significantly ex

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Ashry, El, Sammer Yousuf, Hayat Hassan, Magdy Zahran, and Ali Hebishy. "Synthesis and Single-Crystal X-Ray Diffraction Studies of an Arylidenethiosemicarbazone and Hydrazonyl-phenylthiazole." Letters in Organic Chemistry 11, no. 2 (2014): 101–8. http://dx.doi.org/10.2174/15701786113106660065.

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