Relevant bibliographies by topics / Piperidine synthesis

Contents

  1. Journal articles
  2. Dissertations / Theses
  3. Books
  4. Book chapters
  5. Conference papers
  6. Reports

Academic literature on the topic 'Piperidine synthesis'

Author: Grafiati
Published: 4 June 2021
Last updated: 2 February 2022

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Journal articles on the topic "Piperidine synthesis"

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Šilhánková, Alexandra, Karel Šindelář, Karel Dobrovský, Ivan Krejčí, Jarmila Hodková, and Zdeněk Polívka. "Synthesis of New L-Proline Amides with Anticonvulsive Effect." Collection of Czechoslovak Chemical Communications 61, no. 7 (1996): 1085–92. http://dx.doi.org/10.1135/cccc19961085.

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Series of heterocyclic L-proline amides were prepared from BOC-L-proline and heterocyclic amines (mostly substituted piperazines and morpholines) via active ester with hydroxysuccinimide. 4-(4-Fluorobenzoyl)piperidine afforded L-proline 4-(4-(4-(4-fluorobenzoyl)piperidin-1-yl)benzoyl)piperidine (7b) simultaneously with expected L-proline 4-(4-fluorobenzoyl)piperidide (7a). D-Proline N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)amide (2) was prepared starting from D-proline. The amides were tested by methods of biochemical and behavioural pharmacology.
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Jílek, Jiří, Miroslav Rajšner, Vladimír Valenta, et al. "Synthesis of piperidine derivatives as potential analgetic agents." Collection of Czechoslovak Chemical Communications 55, no. 7 (1990): 1828–53. http://dx.doi.org/10.1135/cccc19901828.

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Reaction of N-(1-(2-phenylethyl)-4-piperidinyl)propionanilide (I) with phosphorus pentasulfide gave the thioamide VI. Acylation of N-(1-(2-phenylethyl)-4-piperidinyl)aniline with 2-(methoxy)acetic and 2-(methylthio)acetic anhydrides afforded the amides II and III. Treatment of 4-anilino-1-benzylpiperidine-4-methanol with thionyl chloride gave the spirocyclic sulfurous acid ester amide XIV. Reduction of the hydrochloride of ethyl 3-(1-ethoxycarbonyl-4-phenylimino-3-piperidinyl)propionate (XXII) with sodium cyanoborohydride gave the perhydro-1,6-naphthyridine derivative XIX, a model compound in
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Klegraf, Ellen, and Horst Kunz. "Stereoselective Synthesis of 3-Substituted and 3,4-Disubstituted Piperidine und Piperidin-2-one Derivatives." Zeitschrift für Naturforschung B 67, no. 4 (2012): 389–405. http://dx.doi.org/10.1515/znb-2012-0413.

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The stereoselective synthesis of 3-substituted and 3,4-disubstituted piperidine and piperidin-2-one derivatives was achieved starting from 2-pyridone. After N-galactosylation and subsequent O-silylation, nucleophilic addition of organometallic reagents proceeded with high regio- and stereoselectivity at 4-position. Substituents at position 3 were stereoselectively introduced by reaction of electrophiles with amide enolates of the N-galactosyl-2-piperidones.
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Tilve, Santosh, Sandesh Bugde, and Prajesh S.Volvoikar. "Protecting-Group-Directed Regio- and Stereoselective Oxymercuration–Demercuration: Synthesis of Piperidine Alkaloids Containing 1,2- and 1,3-Amino Alcohol Units." Synthesis 50, no. 05 (2017): 1113–22. http://dx.doi.org/10.1055/s-0036-1589523.

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An efficient synthesis of naturally occurring 1,2- and 1,3-amino alcohol unit containing 2-substituted piperidine alkaloids and their analogues has been developed from l-pipecolinic acid. The protocol describes the regio- and stereoselective oxymercuration–demercuration of 2-alkenyl piperidines based on protecting groups to give piperidine alkaloids as a key step.
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López-Rodríguez, Alberto, Gema Domínguez, and Javier Pérez-Castells. "Synthesis of Novel Iminosugar Derivatives Based on a 2-Azabi­cyclo[4.1.0]heptane Skeleton." Synthesis 49, no. 20 (2017): 4606–12. http://dx.doi.org/10.1055/s-0036-1589109.

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Iminosugars are good starting points for the development of different kinds of drugs. Many are polyhydroxylated piperidines that behave as biomimetics of their corresponding pyranoses analogues. In the interaction with carbohydrate processing enzymes, selectivity is a crucial issue and the benefits of introducing a cyclopropane bridge in a piperidine structure is demonstrated. The synthesis of novel bicyclic piperidine-based iminosugars using a sulfur ylide cyclopropanation as the key synthetic step is described.
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Pelletier, Guillaume, Léa Constantineau-Forget, and André B. Charette. "Directed functionalization of 1,2-dihydropyridines: stereoselective synthesis of 2,6-disubstituted piperidines." Chem. Commun. 50, no. 52 (2014): 6883–85. http://dx.doi.org/10.1039/c4cc02220c.

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A practical and highly stereoselective approach to access 2,6-disubstituted piperidines using an amidine auxiliary is reported. These were reduced to the saturated piperidine rings with high diastereoselectivity.
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Du, Rui, Liangliang Han, Zhongqiang Zhou, and Victor Borovkov. "Efficient Synthesis of Novel Quinolinone Derivatives via Catalyst-free Multicomponent Reaction." Letters in Organic Chemistry 17, no. 5 (2020): 403–7. http://dx.doi.org/10.2174/1570178616666190828092728.

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The synthesis of 3-(aryl(piperidin-1-yl)methyl)-4-hydroxyquinolin-2(1H)-one derivatives via catalyst-free multicomponent reaction is described. The reaction of 4-hydroxyquinolin-2(1H)-one, piperidine, and 4-chlorobenzaldehyde was carried out in different solvents and under solvent-free conditions at room temperature. The best solvent in terms of the yield and reaction time was found to be dichloromethane. Most substituted benzaldehydes reacted with 4-hydroxyquinolin-2(1H)-one and piperidine to afford corresponding products in good-to-excellent yields. Aldehydes with electronwithdrawing groups
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Guzmán-Rodríguez, Sergio, Jesús Chávez-Reyes, Priscila Vázquez-León, et al. "1-Boc-Piperidine-4-Carboxaldehyde Prevents Binge-Eating Behaviour and Anxiety in Rats." Pharmacology 106, no. 5-6 (2021): 305–15. http://dx.doi.org/10.1159/000513376.

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<b><i>Background:</i></b> Piperidines are biogenic amines studied mainly in toxicology because they were initially found as alkaloids from peppers and insect venoms. Piperidines are also produced in the human body, and their actions seem to be related to wakefulness/sleep and other cognitive phenomena. Piperidines have been minimally characterized for therapeutic applications. In this context, 1-Boc-piperidine-4-carboxaldehyde (1-Boc-piperidine) is a piperidine-derivative molecule with no mechanism of action reported, although its uses include the synthesis of GPR119 se
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Matulevičiūtė, Gita, Eglė Arbačiauskienė, Neringa Kleizienė, et al. "Synthesis and Characterization of Novel Methyl (3)5-(N-Boc-piperidinyl)-1H-pyrazole-4-carboxylates." Molecules 26, no. 13 (2021): 3808. http://dx.doi.org/10.3390/molecules26133808.

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Series of methyl 3- and 5-(N-Boc-piperidinyl)-1H-pyrazole-4-carboxylates were developed and regioselectively synthesized as novel heterocyclic amino acids in their N-Boc protected ester form for achiral and chiral building blocks. In the first stage of the synthesis, piperidine-4-carboxylic and (R)- and (S)-piperidine-3-carboxylic acids were converted to the corresponding β-keto esters, which were then treated with N,N-dimethylformamide dimethyl acetal. The subsequent reaction of β-enamine diketones with various N-mono-substituted hydrazines afforded the target 5-(N-Boc-piperidinyl)-1H-pyrazol
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Mill, Sibel, and Claude Hootelé. "A revised structure for the piperidine alkaloid andrachamine." Canadian Journal of Chemistry 74, no. 12 (1996): 2434–43. http://dx.doi.org/10.1139/v96-272.

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A new method for the synthesis of trans-2,6-disubstituted piperidine derivatives is described. The transformation of cyclic α-methoxycarbamates 5 and 6 affords trans ketones 17 and 18. The synthesis of diols 1–4 from 17 and 18 has shown that the structure proposed in the literature for the piperidine alkaloid andrachamine is incorrect. A reexamination of the original spectral data of this alkaloid suggested that it is a meso 2,6-disubstituted piperidine derivative. Unambiguous syntheses of 23 and 24 and comparison with a sample of andrachamine have established that this alkaloid possesses stru
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Dissertations / Theses on the topic "Piperidine synthesis"

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Lewis, Neil. "Asymmetric piperidine synthesis." Thesis, University of Nottingham, 1995. http://eprints.nottingham.ac.uk/13293/.

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It has been demonstrated that bakers' yeast reduction of 1-tert-butyl-2-methyl 3-oxo-piperidine-1,2-dicarboxylate gives (2R, 3S), 1-tert-butyl-2-methyl 3-hydroxy-piperidine-1,2-dicarboxylate in 80% chemical yield with >99% d.e. and >97% e.e. Also bakers' yeast reduction of 1-tert-butyl-3-ethyl 4-oxo-piperidine-1,3-dicarboxylate gives (3R, 4S), 1-tert-butyl-3-ethyl4-hydroxy-piperidine-1,3-dicarboxylate in 74% chemical yield with >99% d.e. and >93% e.e. The optical purity and absolute configurations of the hydroxy-ester derivatives were determined by conversion into the corresponding chiral bis-
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Taylor, Sarah Alison. "Sulfur-mediated pyrrolidine and piperidine synthesis." Thesis, University of Cambridge, 2007. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.613286.

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Mosts, R. C. "Studies in the synthesis of piperidine alkaloids." Thesis, University of Essex, 1987. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.379495.

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Lenagh-Snow, Gabriel Matthew Jack. "The synthesis of azetidine and piperidine iminosugars from monosaccharides." Thesis, University of Oxford, 2012. http://ora.ox.ac.uk/objects/uuid:207235d5-2ea5-4724-92fd-924fa0ccd4ed.

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Iminosugars are polyhydroxylated alkaloids, and can be generally defined as sugar mimetics in which the endocyclic oxygen atom has been replaced with a basic nitrogen. A common affect of this atomic substitution is to bestow these compounds with the ability to inhibit various sugarprocessing enzymes; most significantly the glycosidases (glycoside hydrolases) which areintimately involved in a huge array of biological functions. Compounds which inhibit these enzymes concordantly possess much potential as medicinal agents for the treatment of a variety of diseases. Several iminosugars have alread
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Adams, David Roger. "Studies in the synthesis of piperidine alkaloids." Thesis, University of Exeter, 1990. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.236570.

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Eskici, Mustafa. "Asymmetric piperidine synthesis via 1,3-cyclic sulfates." Thesis, University of Bristol, 2001. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.368215.

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Adriaenssens, Louis. "Stereoselective synthesis of piperidines." Thesis, Connect to e-thesis to view edited abstract. Move to record for print version, 2008. http://theses.gla.ac.uk/49/.

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Abdelsalam, Mansour. "Synthesis of piperidines using organometallic chemistry." Thesis, University of Sheffield, 2013. http://etheses.whiterose.ac.uk/4069/.

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Williams, Jodi Thomas. "Stereoselective piperidine synthesis via ene and carbonyl ene cyclisations." Thesis, Oxford Brookes University, 2003. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.289247.

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Smith, Peter Duncan. "Synthesis of pipecolic acid derivatives via aza-Diels-Alder reactions." Thesis, Heriot-Watt University, 2000. http://hdl.handle.net/10399/552.

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Books on the topic "Piperidine synthesis"

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Williams, Jodi Thomas. Stereoselective piperidine synthesis via ene and carbonyl ene cyclisations. University of Birmingham, 2003.

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Rubiralta, Mario. Piperidine: Structure, preparation, reactivity, and synthetic applications of piperidine and its derivatives. Elsevier, 1991.

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Hutchinson, Ian. The synthesis of 3-substituted-2-(nitromethylene)-piperidines. typescript, 1994.

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Piperidine - Structure, Preparation, Reactivity, and Synthetic Applications of Piperidine and its Derivatives. Elsevier, 1991. http://dx.doi.org/10.1016/c2009-0-12882-9.

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Vinilat͡s︡etilenovye proizvodnye piperidina i polimery na ikh osnove. "Gylym", 1991.

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Book chapters on the topic "Piperidine synthesis"

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Suryavanshi, Padmakar, Vijaykumar Paike, Sandeep More, Rajendra P. Pawar, Sandeep B. Mane, and K. L. Ameta. "Synthesis of Functionalized Piperidine Derivatives Based on Multicomponent Reaction." In Multicomponent Reactions. CRC Press, 2017. http://dx.doi.org/10.1201/9781315369754-11.

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Shnide, Ravindra S. "Design, Synthesis, and Studies of Novel Piperidine Substituted Triazine Derivatives as Potential Anti-Inflammatory and Antimicrobial Agents." In Green Chemistry and Biodiversity. Apple Academic Press, 2019. http://dx.doi.org/10.1201/9780429202599-15.

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Shao, Xia, and Peter J. H. Scott. "Synthesis ofN-[11C]Methyl-4-Piperidinyl Propionate ([11C]PMP)." In Radiochemical Syntheses. John Wiley & Sons, Inc, 2015. http://dx.doi.org/10.1002/9781118834114.ch7.

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Shao, Xia, Keunsam Jang, and Peter J. H. Scott. "Synthesis of 1-(2,4-Dichlorophenyl)-4-Cyano-5-(4-[11C]methoxyphenyl)-N-(Piperidin-1-yl)-1H-Pyrazole-3-Carboxamide ([11C]OMAR)." In Radiochemical Syntheses. John Wiley & Sons, Inc, 2015. http://dx.doi.org/10.1002/9781118834114.ch8.

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Khalid, Hira, Aziz-ur-Rehman, M. Athar Abbasi, et al. "Synthesis, Spectral Analysis and Biological Evaluation of 5-Substituted 1,3,4-Oxadiazole-2-yl-4-(Piperidin-1-ylsulfonyl)Benzyl Sulfide." In Emerging Trends in Chemical Sciences. Springer International Publishing, 2017. http://dx.doi.org/10.1007/978-3-319-60408-4_14.

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Otto, H., D. Kaiser, C. Kempter, and G. Jung. "Formation of piperidides in peptides containing Asp-Gly during Fmoc synthesis, as identified by 2D NMR and tandem MS." In Peptides 1994. Springer Netherlands, 1995. http://dx.doi.org/10.1007/978-94-011-1468-4_105.

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de Laszlo, S. E., B. L. Bush, J. J. Doyle, et al. "The synthesis and use of 3-amino-4-phenyl-2-piperidones and 4-amino-2-benzazepine-3-ones as conformationally restricted phenylalanine isosteres in renin inhibitors." In Peptides. Springer Netherlands, 1990. http://dx.doi.org/10.1007/978-94-010-9060-5_142.

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Taber, Douglass. "The Smith Synthesis of ( + )-Lyconadin A." In Organic Synthesis. Oxford University Press, 2011. http://dx.doi.org/10.1093/oso/9780199764549.003.0086.

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The pentacyclic alkaloid ( + )-lyconadin A 3, isolated from the club moss Lycopodium complanatum, showed modest in vitro cytotoxicity. A key step in the first reported (J. Am. Chem. Soc. 2007, 129, 4148) total synthesis of 3, by Amos B. Smith III of the University of Pennsylvania, was the cyclization of 1 to 2. The pentacyclic alkaloid (+)-lyconadin A 3, isolated from the club moss Lycopodium complanatum, showed modest in vitro cytotoxicity. A key step in the first reported (J. Am. Chem. Soc. 2007, 129, 4148) total synthesis of 3, by Amos B. Smith III of the University of Pennsylvania, was the cyclization of 1 to 2. The pentacyclic skeleton of 3 was constructed around a central organizing piperidine ring 9. This was prepared from the known (and commercial) enantiomerically-pure lactone 4. The akylated stereogenic center of 9 was assembled by diastereoselective hydroxy methylation of the acyl oxazolidinone 5 with s-trioxane, followed by protection. Reduction of the imide to the alcohol led to the mesylate 7, which on reduction of the azide spontaneously cyclized to give, after protection, the piperidine 8. Selective desilylation of the primary alcohol then enabled the preparation of 9. The plan was to assemble the first carbocyclic ring of 3 by intramolecular aldol condensation of the keto aldehyde 15. The enantiomerically-pure secondary methyl substituent of 15 derived from the commercial monoester 10. Activation as the acid fluoride followed by selective reduction led to the volatile lactone 11. Opening of the lactone with H3CONHCH3HCl gave, after protection, the Weinreb amide 12. Alkylation of the derived hydrazone 13, selectively on the methyl group, led, after deprotection, to 15. The intramolecular aldol condensation of 15 did deliver the unstable cyclohexenone 1. Under the acidic conditions of the aldol condensation, the enol derived from the piperidone added in a Michael sense, from the axial direction on the newly-formed ring, to give the trans-fused bicyclic diketone 2.
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Taber, Douglass. "New Methods for the Stereoselective Construction of N-Containing Rings." In Organic Synthesis. Oxford University Press, 2011. http://dx.doi.org/10.1093/oso/9780199764549.003.0053.

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Several methods have been reported for the stereocontrolled preparation of pyrrolidine and piperidine derivatives. Alison J. Frontier of the University of Rochester has observed (Organic Lett. 2007, 9, 4939) that hydrogenation of acyl pyrroles such as 1 gave good control not just around the ring, but also on the sidechain. Chi-Ming Che of the University of Hong Kong has devised ( J. Am. Chem. Soc. 2007, 129, 5828) a catalyst that converted amides such as 3 into the cyclized product 4, also with high diastereocontrol. Jean Ollivier of the Université de Paris-Sud, following the Sato procedure, has applied (Tetrahedron Lett. 2007, 48, 8765) the Kulinkovich reaction to allylated amino acid esters such as 5 , to give, after Fe-mediated fragmentation, the enantiomerically-pure piperidone 7 . Richard C. Hartley of the University of Glasgow has reported (J. Org. Chem. 2007, 72, 10287) what are, remarkably, the first examples of the aza-Petasis-Ferrier reaction, converting an ester such as 9, by carbonyl methylenation followed by Mannich cyclization, into the piperidone 10. Procedures for catalytic enantioselective C-N ring construction have also been developed. Armando Córdova of Stockholm University has shown (Tetrahedron Lett . 2007, 48, 8695) that condensation of 11 with 12 led to 14, which on reduction and hydrolysis delivered the 3-aryl proline 15. In an even simpler case, Santos Fustero of the Universidad de Valencia found (Organic Lett. 2007, 9, 5283) that the aldehyde 16 could cyclize to 17 with high ee. In a different approach (J. Am. Chem. Soc. 2007, 129, 14811), William E. Greenberg and Chi-Huey Wong of Scripps/La Jolla harnessed the power of an enzyme to mediate the addition of 19 to 18, leading to the pyrrolidine 21 . Daniel P. Furkert of the University of Bath has applied (Organic Lett. 2007, 9, 3769) the powerful Itsuno-Corey reduction to the piperidone 22, leading, after SN2’ displacement, to the alkene 23. To construct larger rings, Barry M. Trost of Stanford University has employed (Angew. Chem. Int. Ed. 2007, 46, 6123) his powerful Pd catalyst to effect opening of the racemic aziridine 24, leading, after metathesis, to the amine 27.
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Taber, Douglass F. "C–N Ring Construction: The Fujii/Ohno Synthesis of (–)-Quinocarcin." In Organic Synthesis. Oxford University Press, 2015. http://dx.doi.org/10.1093/oso/9780190200794.003.0056.

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Tsutomu Katsuki of Kyushu University devised (Org. Lett. 2012, 14, 4658) a Ru catalyst for the enantioselective aziridination of vinyl ketones such as 1. David W.C. MacMillan of Princeton University added (J. Am. Chem. Soc. 2012, 134, 11400) 3 to the alkene 4 under single electron conditions to give 5 with high stereocontrol. Barry M. Trost of Stanford University effected (J. Am. Chem. Soc. 2012, 134, 4941) the Pd-catalyzed addition of 7 to an imine 6 to give the pyrrolidine 8. More recently, he used (J. Am. Chem. Soc. 2013, 135, 2459) this approach to construct pyrrolidines containing defined quaternary centers. Christoph Schneider of the Universität Liepzig employed (Org. Lett. 2012, 14, 5972) an organocatalyst to control the relative and absolute configuration not only of the nitrogen-containing ring, but also of the stereogenic center on the sidechain of the pyrrolidone 11. Wei Wang of Lanzhou University also used (Adv. Synth. Catal. 2012, 354, 2635) an organocatalyst to assemble the pyrrolidine 14bearing two stereogenic centers. Using a gold catalyst, Constantin Czekelius of the Freie Universität Berlin constructed (Angew. Chem. Int. Ed. 2012, 51, 11149) the pyrrolidine 16 having a defined quaternary center. Motomu Kanai of the University of Tokyo used (J. Am. Chem. Soc. 2012, 134, 17019) a Cu catalyst to prepare both pyrrolidines and piperidines by condensing the precursor protected aminal 17 with a ketone 18. Wolfgang Kroutil of the University of Graz effected (Angew. Chem. Int. Ed. 2012, 51, 6713) selective enzymatic reductive amination of the methyl ketone of 20 to give, after cyclization and hydrogenation, the 2,6-dialkyl piperidine 21. Ramakrishna G. Bhat of the Indian Institute of Science Education and Research showed (J. Org. Chem. 2012, 77, 11349) that the reductive cyclization of the amino acid derivative could proceed with high diastereoselectivity to give 23. Peter O’Brien of the University of York and Iain Coldham of the University of Sheffield prepared (J. Am. Chem. Soc. 2012, 134, 5300) both pyrrolidines and piperidines by metalation of an aryl derivative such as 24, followed by alkylation. Shital K. Chattopadhyay of the University of Kalyani cyclized (J. Org. Chem. 2012, 77, 11056) the nitrone 26 to 27 with high diastereoselectivity.
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Conference papers on the topic "Piperidine synthesis"

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Méndez, Leonor Yamile Vargas, and Vladimir V. Kouznetsov. "Simple preparation of new piperidine derivatives as AChE inhibitors for pest control." In 14th Brazilian Meeting on Organic Synthesis. Editora Edgard Blücher, 2013. http://dx.doi.org/10.5151/chempro-14bmos-r0250-2.

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Burtoloso, Antonio C. B. "α,β-Unsaturated Diazoketones as Useful Platforms in the Synthesis of Pyrrolidine, Piperidine and Indolizidine Alkaloids". У 15th Brazilian Meeting on Organic Synthesis. Editora Edgard Blücher, 2013. http://dx.doi.org/10.5151/chempro-15bmos-young5.

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Khalid, Hira. "Synthesis of Bioactive Sulfonamides Bearing Piperidine Nucleus with Talented Activity Against Cholinesterase." In The 16th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2012. http://dx.doi.org/10.3390/ecsoc-16-01064.

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Sravya, G., N. Bakthavatchala Reddy, and Grigory V. Zyryanov. "Synthesis, structural elucidation and bioassay of morpholine/thiomorpholine and piperidine containing oxazoles." In PROCEEDINGS OF INTERNATIONAL CONFERENCE ON RECENT TRENDS IN MECHANICAL AND MATERIALS ENGINEERING: ICRTMME 2019. AIP Publishing, 2020. http://dx.doi.org/10.1063/5.0018089.

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Wang, Min, Wenhui Wang, Qidong Tang, and Shan Xu. "Synthesis of tert-butyl 4-((2-methoxy-4-(methoxycarbonyl) phenoxy) methyl) piperidine-1-carboxylate." In 2015 2nd International Workshop on Materials Engineering and Computer Sciences. Atlantis Press, 2015. http://dx.doi.org/10.2991/iwmecs-15.2015.46.

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Lin, Shuangjie, Xiao Leng, Xiaoji Wang, and Shuangping Huang. "Synthetic study towards (+)-vertine and (+)-lythrine synthesis of the intermediate of benzyl-2-(1-methoxy-1,3-dioxobutan-2-yl)piperidine-1-carboxylate." In 2015 2nd International Conference on Machinery, Materials Engineering, Chemical Engineering and Biotechnology. Atlantis Press, 2016. http://dx.doi.org/10.2991/mmeceb-15.2016.165.

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Kong, Dejia, Yuxing Zhang, Tongsheng Xu, Yuanzhang Zhou, Pengwu Zheng, and Shan Xu. "Synthesis of Tert-butyl-4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)piperidine-1-carboxylate." In 2016 4th International Conference on Machinery, Materials and Computing Technology. Atlantis Press, 2016. http://dx.doi.org/10.2991/icmmct-16.2016.153.

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Rosset, Isac G., та Antonio C. B. Burtoloso. "Synthesis of Piperidines from Z-α,β-Unsaturated Diazoketones". У 15th Brazilian Meeting on Organic Synthesis. Editora Edgard Blücher, 2013. http://dx.doi.org/10.5151/chempro-15bmos-bmos2013_2013915103424.

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Wang, Caolin, Yuanbiao Tu, Jiaqian Han, and Yuping Guo. "Synthesis of 1-(2-(piperidin-1-yl)ethyl)-1H-pyrrole-2-carbaldehyde." In 2016 7th International Conference on Education, Management, Computer and Medicine (EMCM 2016). Atlantis Press, 2017. http://dx.doi.org/10.2991/emcm-16.2017.114.

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10

Couture, Axel, Eric Deniau, Pierre Grandclaudon, and Stéphane Lebrun. "Synthesis of Cyclic Enehydrazides by Ring-Closure Metathesis. Application to the Enantioselective Synthesis of 2-Alkyl and Aryl Piperidines." In The 10th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2006. http://dx.doi.org/10.3390/ecsoc-10-01385.

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Reports on the topic "Piperidine synthesis"

1

Banks, Harold D. Piperidine Synthesis. Defense Technical Information Center, 1992. http://dx.doi.org/10.21236/ada258925.

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