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Relevant bibliographies by topics / Pyridines, pharmacology

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Academic literature on the topic 'Pyridines, pharmacology'

Author: Grafiati

Published: 4 June 2021

Last updated: 29 July 2025

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Journal articles on the topic "Pyridines, pharmacology"

1

Laxmi, Dandamudi Sri, Suryadevara V. Vardhini, Venkata R. Guttikonda, Mandava V. B. Rao, and Manojit Pal. "Synthesis of 2-substituted Furo[3,2-b]pyridines Under Pd/C-Cu Catalysis Assisted by Ultrasound: Their Evaluation as Potential Cytotoxic Agents." Anti-Cancer Agents in Medicinal Chemistry 20, no. 8 (2020): 932–40. http://dx.doi.org/10.2174/1871520620666200311102304.

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Background: Compounds containing furo[3,2-b]pyridine framework have shown interesting pharmacological properties, including anticancer activities. Though these compounds are generally synthesized via the heteroannulation processes involving acetylenic derivatives, some of them are complex. Objective: The study aimed to explore a series of 2-substituted furo[3,2-b]pyridines for their cytotoxic properties against cancer cell lines in vitro. Methods: We developed a convenient synthesis of 2-substituted furo[3,2-b]pyridines via sequential (i) C-C coupling followed by (ii) C-O bond-forming reaction

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2

Abdelrazek, Fathy M., Sobhi M. Gomha, Mohamed E. B. Shaaban, et al. "One-Pot Three-Component Synthesis and Molecular Docking of Some Novel 2-Thiazolyl Pyridines as Potent Antimicrobial Agents." Mini-Reviews in Medicinal Chemistry 19, no. 6 (2019): 527–38. http://dx.doi.org/10.2174/1389557518666181019124104.

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Background: Thiazoles and pyridines are versatile synthetic scaffolds possessing wide spectrum of biological effects including potential antimicrobial activity. Objective: In the efforts to develop suitable antimicrobia drugs, medicinal chemists have focused on thiazole derivatives. A novel series of 2-thiazolyl pyridines was prepared in a one-pot three-component reaction using 2-bromoacetyl pyridine as a starting precursor. Method: Structure of the synthesized compounds was elucidated by spectral data (FT-IR, 1H NMR, 13C NMR, and mass) and elemental analyses. The prepared compounds were scree

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3

Khalili, Faeze, Sara Akrami, Malihe Safavi, et al. "Design, Synthesis, In vitro Cytotoxic Activity Evaluation, and Study of Apoptosis Inducing Effect of New Styrylimidazo[1,2-a]Pyridines as Potent Anti-Breast Cancer Agents." Anti-Cancer Agents in Medicinal Chemistry 19, no. 2 (2019): 265–75. http://dx.doi.org/10.2174/1871520618666180903100835.

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Background: This paper reports synthesis, cytotoxic activity, and apoptosis inducing effect of a novel series of styrylimidazo[1,2-a]pyridine derivatives. Objective: In this study, anti-cancer activity of novel styrylimidazo[1,2-a]pyridines was evaluated. Methods: Styrylimidazo[1,2-a]pyridine derivatives 4a-o were synthesized through a one-pot three-component reaction of 2-aminopyridines, cinnamaldehydes, and isocyanides in high yield. All synthesized compounds 4a-o were evaluated against breast cancer cell lines including MDA-MB-231, MCF-7, and T-47D using MTT assay. Apoptosis was evaluated b

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Szafran, Miroslaw, and Zofia Dega-Szafran. "Complexes of Carboxylic Acids with Pyridines and Pyridine N-Oxides." HETEROCYCLES 37, no. 1 (1994): 627. http://dx.doi.org/10.3987/rev-93-sr5.

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5

Enguehard-Gueiffier, Cecile, and Alain Gueiffier. "Recent Progress in the Pharmacology of Imidazo[1,2-a]pyridines." Mini-Reviews in Medicinal Chemistry 7, no. 9 (2007): 888–99. http://dx.doi.org/10.2174/138955707781662645.

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6

Hagen, A., and V. Hagen. "Cardiotonic and vasodilator activity of some novel 3-cyano-2-oxaalkylamino-5-(4-pyridinyl)-pyridines." European Journal of Pharmacology 183, no. 3 (1990): 775. http://dx.doi.org/10.1016/0014-2999(90)92581-3.

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7

De Munno, Angela, Vincenzo Bertini, Nevio Picci, Francesca Iemma, and Marco Pocci. "Synthesis of Pluriaminated Pyridines." HETEROCYCLES 48, no. 6 (1998): 1203. http://dx.doi.org/10.3987/com-98-8144.

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8

Lila, Amr S. Abu, Marwa H. Abdallah, El-Sayed Khafagy, et al. "Design, synthesis and cytotoxic evaluation of 2-amino-4- aryl-6-substituted pyridine-3,5-dicarbonitrile derivatives." Tropical Journal of Pharmaceutical Research 20, no. 10 (2021): 2127–33. http://dx.doi.org/10.4314/tjpr.v20i10.16.

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Purpose: To synthesize novel pyridine derivatives and evaluate their efficiency as potent inhibitors of cyclin dependent kinase 2 (CDK2) enzyme for cancer therapy.Methods: Pyridine scaffold were synthesized using one-pot multicomponent condensation reaction of arylidine with different primary amines. The cytotoxic potential of the new compounds was assessed using various cell lines. Furthermore, molecular docking studies based on the crystal structure of CDK2 was carried out to determine the possible binding modes that influence the anticancer activities.Results: The results indicate that one-

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9

R. Katritzky, Alan, Jose M. Ayrrecoechea, and Luis M. Vazquez de Miguel. "Ortho-lithiation of 2-(Benzothiazol-2-ylthio)pyridine. Preparation of 2,3-Disubstituted Pyridines." HETEROCYCLES 26, no. 2 (1987): 427. http://dx.doi.org/10.3987/r-1987-02-0427.

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10

Sanapalli, Bharat Kumar Reddy, Akram Ashames, Dilep Kumar Sigalapalli, Afzal B. Shaik, Richie R. Bhandare, and Vidyasrilekha Yele. "Synthetic Imidazopyridine-Based Derivatives as Potential Inhibitors against Multi-Drug Resistant Bacterial Infections: A Review." Antibiotics 11, no. 12 (2022): 1680. http://dx.doi.org/10.3390/antibiotics11121680.

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Fused pyridines are reported to display various pharmacological activities, such as antipyretic, analgesic, antiprotozoal, antibacterial, antitumor, antifungal, anti-inflammatory, and antiapoptotic. They are widely used in the field of medicinal chemistry. Imidazopyridines (IZPs) are crucial classes of fused heterocycles that are expansively reported on in the literature. Evidence suggests that IZPs, as fused scaffolds, possess more diverse profiles than individual imidazole and pyridine moieties. Bacterial infections and antibacterial resistance are ever-growing risks in the 21st century. Onl

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Dissertations / Theses on the topic "Pyridines, pharmacology"

1

Gueiffier, Alain. "Hétérocyclisation en série imidazo [1,2-a] pyridinique : synthèse, structure, pharmacologie." Montpellier 1, 1989. http://www.theses.fr/1989MON13505.

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2

Gezginci, Mikail Hakan. "Synthesis and in vitro antimycobacterial activity of some pyridine and pyrazinecarboxylic acid isosteres." Diss., The University of Arizona, 1999. http://hdl.handle.net/10150/284057.

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Tuberculosis has been one of the most commonly encountered infectious diseases of humans throughout history. The discovery and introduction of effective treatments in the 1940s resulted in a decline of the incidence of the disease until the 1980s, which marked a sharp turn in this trend with an increase in the number of reported cases in the world. The prevalence of mycobacterial infections in poorer nations and centers of urban decay, and especially in immunologically compromised patients indicates the need for new and better treatments. In this study, to contribute to the worldwide effort to

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3

Colgin, Neil. "Synthetic approaches to novel pyridine and indole derivatives as potential agents for the treatment of neurodegenerative disorders." Thesis, University of Sunderland, 2009. http://sure.sunderland.ac.uk/4064/.

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Alzheimer’s Disease (AD), Parkinson’s Disease (PD) and Lewy Body Disease (LBD) are some of the many neurodegenerative disorders associated with dementia, for which there is no ultimate cure. It is widely accepted that central nervous system (CNS) nicotinic acetylcholine receptors (nAChRs) may be strongly implicated in the pathology of these devastating disorders, and that stimulation of nAChRs can enhance cognitive behaviour in animals and humans. Nicotine and other nicotinic receptor binding compounds have, over many years, been explored as potential therapies for disorders such as AD and PD.

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4

Kopp, Marina. "Synthèse de nouvelles guanidinopyridines et arylimidazolines à visées hypoglycémiantes." Caen, 2002. http://www.theses.fr/2002CAEN4063.

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5

Leflemme, Nicolas. "Synthèse, étude physico-chimique et évaluation biologique d'arylpyridines à visée nicotinique." Caen, 2002. http://www.theses.fr/2002CAEN2068.

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Le travail décrit dans cette thèse porte sur la conception, la synthèse, l'étude physico-chimique et l'évaluation biologique de nouveaux ligands des récepteurs cholinergiques nicotiniques de structure chimique arylpyridine. Cette nouvelle famille de composés est issue du programme de recherche "récepteurs nicotiniques" initié récemment au Centre d'Etudes et de Recherche sur le Médicament de Normandie. Après un rappel de généralités à propos des récepteurs cholinergiques nicotiniques, leurs localisations, leurs structures, leurs différents sous-types, leurs rôles biologiques et les ligands les

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N'Guessan, Déto. "Conception, synthèse et évaluation des activités anthelminthiques de nouvelles molécules à support imidazo (1,2-a) pyridine." Thesis, Tours, 2017. http://www.theses.fr/2017TOUR3802.

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Les strongyloses vétérinaires constituent l’une des principales causes de gastroentérites et d’anémie des ovins et caprins à l’origine de lourdes pertes économiques. Cependant, leurs prise en charge par les anthelminthiques existants, est confrontée à la prolifération d’une pharmacorésistance des nématodes incriminés. La première partie de ce travail de thèse présente l’ampleur du problème que pose la résistance des helminthes impliqués dans les strongyloses des petits ruminants. Elle révèle également le profil novateur des imidazo[1,2-a]pyridinyl-phénylacrylonitriles qui est proposé pour pare

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Raynaud, Isabelle. "Etude des relations structure-activité quantitatives (QSAR) des cytokinines : synthèse et activité biologique de nouvelles molécules actives." Angers, 1996. http://www.theses.fr/1996ANGE0022.

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Un modèle statistique de relations structure-activité de type quantitatif des cytokinines, hormones végétales, a été mis au point. Il a été construit à partir de 26 molécules appartenant aux deux principales classes de cytokinines : les pyridylphenylurées et les purines n#6-substituées. Apres l'analyse conformationnelle de ces 26 molécules, différents alignements ont été construits et testes dans COMFA. Finalement, deux modèles ont été sélectionnés. Ils ont été valides par des échantillons-tests de molécules connues. Le meilleur modèle, ORL1, a ensuite servi pour faire des prédictions d'activi

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8

Burns, C. J., E. Fantino, A. K. Powell, et al. "The microtubule depolymerizing agent CYT997 causes extensive ablation of tumor vasculature in vivo." 2011. http://hdl.handle.net/10454/5902.

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The orally active microtubule-disrupting agent (S)-1-ethyl-3-(2-methoxy-4-(5-methyl-4-((1-(pyridin-3-yl)butyl)amino)pyrimidin-2- yl)phenyl)urea (CYT997), reported previously by us (Bioorg Med Chem Lett 19:4639-4642, 2009; Mol Cancer Ther 8:3036-3045, 2009), is potently cytotoxic to a variety of cancer cell lines in vitro and shows antitumor activity in vivo. In addition to its cytotoxic activity, CYT997 possesses antivascular effects on tumor vasculature. To further characterize the vascular disrupting activity of CYT997 in terms of dose and temporal effects, we studied the activity of the com

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Books on the topic "Pyridines, pharmacology"

1

Albrecht, Fleckenstein, ed. Cardiovascular effects of dihydropyridine-type calcium antagonists and agonists. Springer-Verlag, 1985.

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2

Hofmann, F. B. Nicotine Psychopharmacology. Springer Berlin Heidelberg, 2009.

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3

Hoffmeister, F., A. Fleckenstein, C. Van Breemen, and R. Groß. Cardiovascular Effects of Dihydropyridine-Type Calcium Antagonists and Agonists. Springer London, Limited, 2013.

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4

Hoffmeister, F., A. Fleckenstein, C. Van Breemen, and R. Groß. Cardiovascular Effects of Dihydropyridine-Type Calcium Antagonists and Agonists. Springer, 2011.

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5

Fleckenstein, A., C. Van Breemen, and R. Grob. Cardiovascular Effects of Dihydropyridine-Type Calcium Antagonists and Agonists (Bayer-Symposium//(Proceedings)). Springer, 1985.

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6

Cardiovascular Effects of Dihydropyridine-Type Calcium Antagonists and Agonists. Springer, 2011.

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7

Jacobson, Kenneth A., and Joel Linden. Pharmacology of Purine and Pyrimidine Receptors. Elsevier Science & Technology Books, 2011.

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Book chapters on the topic "Pyridines, pharmacology"

1

Enna, S. J., and David B. Bylund. "Pyridine-3-Aldehyde." In xPharm: The Comprehensive Pharmacology Reference. Elsevier, 2007. http://dx.doi.org/10.1016/b978-008055232-3.63164-2.

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2

Singh, Sonia, Nitin Agrawal, and Isha Mishra. "Pharmacology and Phytochemistry of Coriander." In Ethnopharmacological Investigation of Indian Spices. IGI Global, 2020. http://dx.doi.org/10.4018/978-1-7998-2524-1.ch014.

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Coriander, named as Coriandrum sativum Linn, belongs to the family Umbelliferae and is one of the most popular and well-known spices/condiments and herbal medicines. The essential oils and fatty oils are the two major active chemical constituents present in the plant. The other minor ingredients found to be present are monoterpenes hydrocarbons i-e limonene, γ-terpinene, α-pinene, p-cymene, borneol, citronellol, camphor, geraniol, and geraniol acetate and abd heterocyclic components such as pyrazine, pyridine, thiazole, furan and tetrahudrofuran derivatives, isocoumarins, coriandrin, dihydroco

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Singh, Sonia, Nitin Agrawal, and Isha Mishra. "Pharmacology and Phytochemistry of Coriander." In Research Anthology on Recent Advancements in Ethnopharmacology and Nutraceuticals. IGI Global, 2022. http://dx.doi.org/10.4018/978-1-6684-3546-5.ch037.

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Coriander, named as Coriandrum sativum Linn, belongs to the family Umbelliferae and is one of the most popular and well-known spices/condiments and herbal medicines. The essential oils and fatty oils are the two major active chemical constituents present in the plant. The other minor ingredients found to be present are monoterpenes hydrocarbons i-e limonene, γ-terpinene, α-pinene, p-cymene, borneol, citronellol, camphor, geraniol, and geraniol acetate and abd heterocyclic components such as pyrazine, pyridine, thiazole, furan and tetrahudrofuran derivatives, isocoumarins, coriandrin, dihydroco

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4

Strunz, George M., and John A. Findlay. "Chapter 3 Pyridine and Piperidine Alkaloids." In The Alkaloids: Chemistry and Pharmacology. Elsevier, 1985. http://dx.doi.org/10.1016/s0099-9598(08)60194-7.

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Conference papers on the topic "Pyridines, pharmacology"

1

Ungur, Nicon, Aurelian Gulea, and Tatiana Erhan. "Synthesis and study of the same hydrazincarbothioamides as privilege pharmacophores in pharmacology." In Scientific seminar with international participation "New frontiers in natural product chemistry". Institute of Chemistry, Republic of Moldova, 2023. http://dx.doi.org/10.19261/nfnpc.2023.ab05.

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Hydrazinecarbothioamides represent a privileged class of pharmacophores in pharmacology, thanks to an impressive number of derivatives that exhibit outstanding antimicrobial, anticancer and antifungal properties [1]. The presence of electron donor atoms such as N(nitrogen) and S(sulfur) substantially widen the spectrum of use. In the framework of theoretical studies on the structure of biologically active compounds with valuable properties were highlighted following common structural elements such as substitution of a hydrogen atom from the nitrogen atom (N) with the benzene ring, the introduc

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