Relevant bibliographies by topics / Pyridone analogues

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  2. Dissertations / Theses
  3. Books
  4. Book chapters
  5. Conference papers

Academic literature on the topic 'Pyridone analogues'

Author: Grafiati
Published: 19 February 2023
Last updated: 31 July 2025

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Journal articles on the topic "Pyridone analogues"

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Tang, Yao, Nvjiang Wu, Junyu Xu, Xiaopo Zhang, Youbin Li, and Xuesong Wang. "Metal-Free Cascade Formation of C–C and C–N Bond for the Construction of 3-Cyano-2-Pyridones with Insecticidal Properties." Molecules 29, no. 12 (2024): 2792. http://dx.doi.org/10.3390/molecules29122792.

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A straightforward and efficient methodology has been developed for the synthesis of 3-cyano-2-pyridones via the C–C and C–N bond formation processes. A total of 51 diverse 3-cyano-2-pyridone derivatives were obtained in moderate to excellent yields. This reaction featured advantages such as a metal-free process, wide functional group tolerance, simple operation, and mild conditions. A plausible mechanism for the reaction was proposed. 3-cyano-2-pyridones as ricinine analogues for insecticidal properties were evaluated, and the compound 3ci (LC50 = 2.206 mg/mL) showed the best insecticidal prop
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Yang, Yinghua, Lianli Sun, Shengyi Dong, et al. "Synthesis of the pyridone analogues of territrem B." Mendeleev Communications 18, no. 4 (2008): 186–87. http://dx.doi.org/10.1016/j.mencom.2008.07.004.

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Kaur, Ishwinder, Gopal P. Jadhav, Peter M. Fischer, and Gerlof Sebastiaan Winkler. "The Discovery of Substituted 5-(2-Hydroxybenzoyl)-2-Pyridone Analogues as Inhibitors of the Human Caf1/CNOT7 Ribonuclease." Molecules 29, no. 18 (2024): 4351. http://dx.doi.org/10.3390/molecules29184351.

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The Caf1/CNOT7 nuclease is a catalytic component of the Ccr4-Not deadenylase complex, which is a key regulator of post-transcriptional gene regulation. In addition to providing catalytic activity, Caf1/CNOT7 and its paralogue Caf1/CNOT8 also contribute a structural function by mediating interactions between the large, non-catalytic subunit CNOT1, which forms the backbone of the Ccr4-Not complex and the second nuclease subunit Ccr4 (CNOT6/CNOT6L). To facilitate investigations into the role of Caf1/CNOT7 in gene regulation, we aimed to discover and develop non-nucleoside inhibitors of the enzyme
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Hwang, Gil Tae, Aaron M. Leconte, and Floyd E. Romesberg. "Polymerase Recognition and Stability of Fluoro-Substituted Pyridone Nucleobase Analogues." ChemBioChem 8, no. 13 (2007): 1606–11. http://dx.doi.org/10.1002/cbic.200700308.

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Capps, Nigel K., Gareth M. Davies, David Loakes, Richard W. McCabe та Douglas W. Young. "Synthesis of bicyclic pyridone and dihydropyridone analogues of β-lactam antibiotics". J. Chem. Soc., Perkin Trans. 1, № 12 (1991): 3077–86. http://dx.doi.org/10.1039/p19910003077.

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Rubovič, Peter, Andriy Pysanenko, Jozef Lengyel, Dana Nachtigallová, and Michal Fárník. "Biomolecule Analogues 2-Hydroxypyridine and 2-Pyridone Base Pairing on Ice Nanoparticles." Journal of Physical Chemistry A 120, no. 27 (2016): 4720–30. http://dx.doi.org/10.1021/acs.jpca.5b11359.

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Haffner, Curt D., Caroline J. Diaz, Aaron B. Miller, et al. "Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)." Bioorganic & Medicinal Chemistry Letters 18, no. 15 (2008): 4360–63. http://dx.doi.org/10.1016/j.bmcl.2008.06.067.

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Tauraitė, Daiva, Rytis Ražanas, Algirdas Mikalkėnas, Saulius Serva, and Rolandas Meškys. "Synthesis of Pyridone-based Nucleoside Analogues as Substrates or Inhibitors of DNA Polymerases." Nucleosides, Nucleotides and Nucleic Acids 35, no. 4 (2016): 163–77. http://dx.doi.org/10.1080/15257770.2015.1122197.

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CAPPS, N. K., G. M. DAVIES, D. LOAKES, R. W. MCCABE та D. W. YOUNG. "ChemInform Abstract: Synthesis of Bicyclic Pyridone and Dihydropyridone Analogues of β- Lactam Antibiotics." ChemInform 23, № 13 (2010): no. http://dx.doi.org/10.1002/chin.199213234.

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Murgatroyd, Christopher, Lisa Pirrie, Fanny Tran, Terry K. Smith, Nicholas J. Westwood, and Catherine S. Adamson. "Structure-Activity Relationships of the Human Immunodeficiency Virus Type 1 Maturation Inhibitor PF-46396." Journal of Virology 90, no. 18 (2016): 8181–97. http://dx.doi.org/10.1128/jvi.01075-16.

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ABSTRACTHIV-1 maturation inhibitors are a novel class of antiretroviral compounds that consist of two structurally distinct chemical classes: betulinic acid derivatives and the pyridone-based compound PF-46396. It is currently believed that both classes act by similar modes of action to generate aberrant noninfectious particles via inhibition of CA-SP1 cleavage during Gag proteolytic processing. In this study, we utilized a series of novel analogues with decreasing similarity to PF-46396 to determine the chemical groups within PF-46396 that contribute to antiviral activity, Gag binding, and th
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Dissertations / Theses on the topic "Pyridone analogues"

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Karis, Nils David. "Design and Synthesis of 1,3-Disubstitiuted-2-Pyridones as a New Class of Glycogen Phosphorylase Inhibitors." Thesis, Griffith University, 2009. http://hdl.handle.net/10072/365791.

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Glycogen Phosphorylase (GP) is the regulatory enzyme that catalyses the first step in glycogen degradation and is a potential enzyme target for therapeutic intervention in the treatment of diabetes. The 16 amino acid C-terminal sequence of human Gl is the only known targeting subunit that binds to GPa. Blocking the interactions between Gl and GPa should reduce high blood glucose levels in a diabetic person. A segment of the 16 amino acid segment was chosen for a small molecule peptidomimetric approach, and de nova design from this segment identified the pyridone ring as apotential scaffold. Th
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Dufour, Fabien Kirsch Gilbert. "Synthèse en série carbazolique, analogues d' ellipticine, et dihydrocarbazolocarbazolzq." [S.l.] : [s.n.], 2007. ftp://ftp.scd.univ-metz.fr/pub/Theses/2007/Dufour.F.SMZ0731.pdf.

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Schmitt, Benoît. "5,6,7,8-tétrahydro-1,6-naphtyridines : dérivés et analogues structuraux." Université Louis Pasteur (Strasbourg) (1971-2008), 2004. http://www.theses.fr/2004STR13210.

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Crawford, Julia Ann. "A study of synthetic routes to pyridine-stretched nucleoside analogues." Thesis, Keele University, 2004. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.414756.

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An introduction to the use of oligonucleotides as antigene or antisense therapeutic agents is presented. This includes an analysis of the major areas of structural change implemented to improve the stability, specificity, nuclease resistance and cellular delivery of oligonucleotides. The synthetic aspect of the project concerns the preparation of two novel 'pyridinestretched' heterocyclic bases principally designed to improve base stacking. The first of these, 8-amino-3 -(2-deoxy-J3-D-ribofuranosyl)-imidazo [4' ,5': 5 ,6]pyrido[2,3-d]pyrimidine, is a stretched adenosine analogue which may be s
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Lee, Jasmine. "The design and preparation of pyridoxal 5'-phosphate analogues." Thesis, Abertay University, 2002. https://rke.abertay.ac.uk/en/studentTheses/2576be85-8cca-4f11-89ab-f1159fa57f94.

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Chioua, Rachid. "Synthèse, structure et réactivité de dérivés de la 1H-pyrazolo[3,4-c]pyridine. Analogues acycliques de nucléosides." Montpellier 1, 1992. http://www.theses.fr/1992MON13526.

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Houdaibi, Khalid. "Contribution à la synthèse de nouvelles molécules herbicides analogues au pyridate." Doctoral thesis, Universite Libre de Bruxelles, 2000. http://hdl.handle.net/2013/ULB-DIPOT:oai:dipot.ulb.ac.be:2013/211773.

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Jourdan, Fabrice. "Synthèse, études physicochimique et pharmacologique d'inhibiteurs potentiels de la transcriptase inverse comprenant différents analogues de nucléosides cycliques et acycliques thiéno et dihydrothiénopyrimidiniques, différentes pyridin-2-ones et pyrido[3,2-ƒ]pyrollo[1,2-a]diazépines." Caen, 1996. http://www.theses.fr/1996CAEN4018.

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Lepretre, Jean-Claude. "Synthèse et étude électrochimique de sels de pyridinium 3,5- disubstitués modèles du NAD+ : réactivité et comportement de leurs analogues réduits." Grenoble 1, 1992. http://www.theses.fr/1992GRE10032.

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L'etude electrochimique de composes 1-alkyl-3,5-dialkylcarbamido-pyridinium montre que ces especes se comportent comme des modeles du nad#+ (nicotinamide adenine dinucleotide forme oxydee). Sur differents materiaux d'electrodes, leur reduction donne deux types de produits: tout d'abord des dimeres 4,4, en general au nombre de trois qui sont des isomeres de conformation dont la structure a ete determinee par rmn. Ensuite les 1,4-dihydropyridines dont la proportion evolue selon la cathode utilisee. Nous avons pu montrer que certaines conditions de travail (variant selon le modele etudie) permett
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Nicolaÿ, Jean-François. "Synthèse asymétrique d'alcaloides pipéridiniques, composés analogues des coccinellines et de l'anatoxine-A." Paris 11, 1989. http://www.theses.fr/1989PA112365.

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Une méthode générale de synthèse asymétrique d'alcaloides piperidiniques a récemment été mise au point dans notre laboratoire. Elle repose sur la préparation d'un synthon chiral équivalent réactionnel de dihydro-1,4-pyridine. Cette méthode a été appliquée à la synthèse d'alcaloides extraits des secrétions de coccinelles et possédant une structure perhydroazaphénalène. Plusieurs composes analogues, enantiomériquement purs, ont ete obtenus. La préparation de composes tricycliques, par ailleurs également précurseurs potentiels d'alcaloides de type poranthéridine, a été effectuée. Enfin, la synthè
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Books on the topic "Pyridone analogues"

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Holder, Alvin A. Dipicolinic acid, its analogues and derivatives: Aspects of their coordination chemistry. Nova Science Publishers, 2011.

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Book chapters on the topic "Pyridone analogues"

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Duffy, Colm. "Synthesis and Biological Evaluation of Pyridine-Containing Lipoxin A4 Analogues." In Heteroaromatic Lipoxin A4 Analogues. Springer Berlin Heidelberg, 2012. http://dx.doi.org/10.1007/978-3-642-24632-6_4.

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Gangjee, Aleem, Farahnaz Mavandadi, and Sherry F. Queener. "Synthesis and Biological Activity of Tricyclic, Conformationally Restricted Analogs of Lipophilic Pyrido[2,3-d]-Pyrimidine Antifolates." In Advances in Experimental Medicine and Biology. Springer US, 1993. http://dx.doi.org/10.1007/978-1-4615-2960-6_88.

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Gangjee, Aleem, Anil Vasudevan, and Sherry F. Queener. "Bicyclic Conformationally Restricted Analogs of Nonclassical Pyrido[2,3-d] Pyrevddines as Potential Inhibitors of Dihydrofolate Reductases." In Advances in Experimental Medicine and Biology. Springer US, 1993. http://dx.doi.org/10.1007/978-1-4615-2960-6_90.

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D. Adesina, Adebimpe. "The Chemistry of Benzo and Carbocyclic Derivatives of Pyridine." In Exploring Chemistry with Pyridine Derivatives [Working Title]. IntechOpen, 2022. http://dx.doi.org/10.5772/intechopen.108127.

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The chemistry of pyridine and its derivatives is of considerable importance in the synthesis of intermediates leading to biologically active compounds and novel materials. Generally, derivatives of pyridine are stable and relatively unreactive but can be attacked by electrophiles at ring nitrogen and certain carbon atoms. Pyridines undergo radical substitution reactions preferentially at the 2-position. Simple pyridines and their benzo derivatives are weak bases that form salts with strong acids. Various Lewis acids form complexes with pyridine and its benzo derivatives. The quaternization of
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Davies, David T. "Six-membered ring heterocycles containing one oxygen atom." In Aromatic Heterocyclic Chemistry. Oxford University Press, 1992. http://dx.doi.org/10.1093/hesc/9780198556602.003.0009.

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This chapter describes six-membered ring heterocycles containing one oxygen atom. The pyrilium cation, 2-pyrone, 4-pyrone, and their benzo-fused analogues, the benzopyrilium cation, coumarin, and chromone, are the parent structures of a series of six-membered ring heterocycles containing one oxygen atom. The impetus for research in this area comes from the enormous number of plant-derived natural products based on the benzopyrilium, coumarin, and chromone structures. The pyrylium cation is the oxygen analogue of pyridine and is a six π-electron aromatic system. Nevertheless, being a cation, it
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Abbaspour Tehrani, K., and N. De Kimpe. "Photochemical Isomerization of Pyridines." In Heteroatom Analogues of Aldehydes and Ketones. Georg Thieme Verlag KG, 2004. http://dx.doi.org/10.1055/sos-sd-027-00288.

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Perseghini, M., and A. Togni. "Synthesis of 4-(Dimethylamino)pyridine Analogues via Racemate Resolution." In Compounds with Transition Metal-Carbon pi-Bonds and Compounds of Groups 10-8 (Ni, Pd, Pt, Co, Rh, Ir, Fe, Ru, Os). Georg Thieme Verlag KG, 2001. http://dx.doi.org/10.1055/sos-sd-001-00889.

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Pilli, R. A., and G. B. Rosso. "N-Acylation of Imines, Pyridines, and Related Compounds." In Heteroatom Analogues of Aldehydes and Ketones. Georg Thieme Verlag KG, 2004. http://dx.doi.org/10.1055/sos-sd-027-00388.

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Saunders, John. "Proton pump inhibitors as gastric acid secretion inhibitors." In Top Drugs. Oxford University Press, 2000. http://dx.doi.org/10.1093/hesc/9780198501008.003.0005.

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This chapter tackles omeprazole which had been characterized as a gastric acid-pump inhibitor, blocking the final step of acid production and thus curbing acid production by all stimulatory mechanisms. The chapter first explains the omeprazole cycle, noting that the omeprazole’s mechanism of action is not entirely straightforward and is dependent on a subtle balance of chemical reactivity, controlled by the nature of substituents in the pyridine ring, and enzymatic transformation under the physiological conditions prevailing in the gut and liver. The chapter then explains the process by which
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Shanawad, S. S., Sureshappa K. Sajjan, Shridhar A H, and Vidyagayatri Marrakkur. "PHOTOPHYSICAL AND BIOLOGICAL STUDIES ON NEWLY SYNTHESIZED NOVEL ARYLSUBSTITUTED PYRAZOLONE ANALOGUE." In Futuristic Trends in Chemical, Material Sciences & Nano Technology Volume 2 Book 12. Iterative International Publishers, Selfypage Developers Pvt Ltd, 2023. http://dx.doi.org/10.58532/v2bs12p4ch1.

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In the present work, a new pyrazoles derivative namely ethyl 2-(2- (ethoxycarbonyl)hept-1-en-3-yl)6,7-dihydro3-hydroxy-2Hpyrazolo[4,3c]Pyridine5(4H)carboxylate (EP P) was synthesized and studied their biological and photophysical properties. The EEP structure was confirmed by 1H NMR, FT-IR and LCMS analyses. EPP show good inhibitor properties for S. aureus and C. albicans. The photophysical properties are estimated using density functional theory in gaussian-9w software. The ground state dipole moment, HOMO-LUMO and molecular electrostatic potential map are estimated using basis set B3LYP-311G
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Conference papers on the topic "Pyridone analogues"

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Felczak, Krzysztof, and Krzysztof W. Pankiewicz. "Rehab of NAD-dependent enzymes with NAD-based inhibitors; synthesis of methylenebis(phosphonate) analogues of pyridone-3-carboxamide adenine dinucleotides." In XVth Symposium on Chemistry of Nucleic Acid Components. Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, 2011. http://dx.doi.org/10.1135/css201112204.

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Wysocka, Alicja, Agnieszka Galanty, and Wiktor Kasprzyk. "Novel oxidized 2-pyridone analogs, properties and prospects." In 3rd International PhD Student’s Conference at the University of Life Sciences in Lublin, Poland: ENVIRONMENT – PLANT – ANIMAL – PRODUCT. Publishing House of The University of Life Sciences in Lublin, 2024. http://dx.doi.org/10.24326/icdsupl3.b005.

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Patrick A., Robertson, Villani Luigi, Martin Danielle, and Robertson Evan G. "Laser spectroscopy of nicotine and related analogues : perturbations and puckering in pyridine and pyrrolidine rings." In Asian Spectroscopy Conference 2020. Institute of Advanced Studies, Nanyang Technological University, 2020. http://dx.doi.org/10.32655/asc_8-10_dec2020.4.

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Hussein, Ola, Feras Alali, Ala‐Eddin Al Mustafa, and Ashraf Khalil. "Development of Novel Chalcone Analogs as Potential Multi-Targeted Therapies for Castration-Resistant Prostate Cancer." In Qatar University Annual Research Forum & Exhibition. Qatar University Press, 2021. http://dx.doi.org/10.29117/quarfe.2021.0114.

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Prostate cancer (PCa) is the second most frequently diagnosed malignancy, as well as a leading cause of cancer-related mortality in men globally. Despite the initial response to hormonal targeted therapy, the majority of patients ultimately progress to a lethal form of the disease, castration-resistant prostate cancer (CRPC). Therefore, the objective of this study was to discover and develop novel treatment modalities for CRPC. Chalcones are among the highly attractive scaffolds being investigated for their antitumor activities. A library of 26 chalcone analogs were designed, synthesized and e
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Трофимов, Б., B. Trofimov, Н. Гусарова, and N. Gusarova. "The development of original methodologies of directed synthesis of le-Carbs their analogs and precursors base donacetylene and its derivatives." In Topical issues of translational medicine: a collection of articles dedicated to the 5th anniversary of the day The creation of a department for biomedical research and technology of the Irkutsk Scientific Center Siberian Branch of RAS. INFRA-M Academic Publishing LLC., 2017. http://dx.doi.org/10.12737/conferencearticle_58be81ec92d17.

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New reactions, which have been discovered and continue to be developed in A.E. Favorsky Irkutsk institute of chemistry SB RAS on the basis of acetylene, a product of oil, gas and coal processing and multi-faceted building block for organic synthesis, have been considered. These reactions provide for the shortest routes to construction of fundamental heterocyclic scaffolds (pyrroles, imidazoles, pyrazoles, indoles, pyridines, dihydropyridines, etc.) with desirable and optimum combination of functional pharmacophoric groups and fragments, which are responsible for antiviral (HIV, flu), antitumor
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Hussein, Ola, Feras Alali, Ala-Eddin Al Moustafa, and Ashraf Khalil. "Design, Synthesis and Biological Evaluation of Novel Chalcone Analogs as Potential Therapeutic Agents for Castration-Resistant Prostate Cancer." In Qatar University Annual Research Forum & Exhibition. Qatar University Press, 2020. http://dx.doi.org/10.29117/quarfe.2020.0179.

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Prostate cancer (PCa) is the second most frequently diagnosed malignancy, as well as a leading cause of cancer-related mortality in men globally. Despite the initial response to hormonal targeted therapy, the majority of patients ultimately progress to a lethal form of the disease, termed as castration-resistant prostate cancer (CRPC), which currently lacks curative therapeutic options and is associated with poor prognosis. Therefore, the development of novel treatment modalities for PCa is urgently needed. Chalcones, also known as 1,3-diphenyl-2-propen-1-ones, are among the highly attractive
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Montaño, Rocío, and Murali Venkata Unnamatla. "Efficient and rapid conversion of 3-amino imidazo[1,2-a] pyridin-2-yl)-4H-chromene-4-ones to its corresponding thio analogues using Lawesson’s reagent ." In The 22nd International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2018. http://dx.doi.org/10.3390/ecsoc-22-05668.

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Marchand, Pascal, Thierry Besson, Yvonnick Loidreau, Marie-Renée Nourrisson, Corinne Fruit, and Cécile Corbière. "Synthesis of potential bioactive benzo-, pyrido-, or pyrazinothieno[3,2-<em>d</em>]pyrimidin- 4-amine analogs of MPC-6827." In 6th International Electronic Conference on Medicinal Chemistry. MDPI, 2020. http://dx.doi.org/10.3390/ecmc2020-07391.

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