Log in

Relevant bibliographies by topics / Schiffs Bases 4-Thiazolidinone Derivatives Anti-Convulsant Activity

Contents

Journal articles

Academic literature on the topic 'Schiffs Bases 4-Thiazolidinone Derivatives Anti-Convulsant Activity'

Author: Grafiati

Published: 5 June 2025

Last updated: 2 August 2025

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic 'Schiffs Bases 4-Thiazolidinone Derivatives Anti-Convulsant Activity.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "Schiffs Bases 4-Thiazolidinone Derivatives Anti-Convulsant Activity"

1

Dr., Faizan Sayeed1* Abdul Sayeed1 MD Akram1 Mohd Waseem Akram2. "DESIGN, SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW SUBSTITUTED THIAZOLIDIN-4- ONE DERIVATIVES." Indo American Journal of Pharmaceutical Sciences 04, no. 08 (2017): 2461–72. https://doi.org/10.5281/zenodo.846845.

Full text

Abstract:

4-thiazolidinones are among t h e most extensively investigated class of organic compounds. Thiazolidin-4-one has been considered as magic moiety, which is a core structure in various synthetic pharmaceuticals displaying a broad spectrum of biological activities.They are widely used as anti-inflammatory, anticonvulsant, analgesic, antimicrobial,anti-HIV,CNS depressant, carcinostatic, antihypertensive and cytotoxic. In view of the wide spectrum activities of condensed 4-thiazolidinones, it was thought worthwhile to undertake the synthesis of heterocyclic systems in which 4-thiazolidinone nucleu

APA, Harvard, Vancouver, ISO, and other styles

2

Dr.Faizan, Sayeed* Abdul Sayeed1 MD Akram Mohd Waseem Akram. "ANALGESIC AND ANTI INFLAMMATORY ACTIVITY OF NEW SUBSTITUTED THIAZOLIDIN-4-ONE DERIVATIVES." Indo American Journal of Pharmaceutical Sciences 04, no. 08 (2017): 2449–60. https://doi.org/10.5281/zenodo.846843.

Full text

Abstract:

4-thiazolidinones are among t he most extensively investigated class of organic compounds. Thiazolidin-4-one has been considered as magic moiety, which is a core structure in various synthetic pharmaceuticals displaying a broad spectrum of biological activities.They are widely used as anti-inflammatory, anticonvulsant, analgesic, antimicrobial,anti-HIV,CNS depressant, carcinostatic, antihypertensive and cytotoxic. In view of the wide spectrum activities of condensed 4-thiazolidinones, itwas thought worthwhile to undertake the synthesis of heterocyclic systems in which 4-thiazolidinone nucleus

APA, Harvard, Vancouver, ISO, and other styles

3

Abu-Hashem, Ameen Ali, Khadiga Mohamed Abu-Zied, Magdi Elsayed AbdelSalam Zaki, Mohamed Fathy El-Shehry, Hanem Mohamed Awad, and Mohammed Abdou Khedr. "Design, Synthesis, and Anticancer Potential of the Enzyme (PARP-1) Inhibitor with Computational Studies of New Triazole, Thiazolidinone, - Thieno [2, 3-d] Pyrimidinones." Letters in Drug Design & Discovery 17, no. 6 (2020): 799–817. http://dx.doi.org/10.2174/1570180817666200117114716.

Full text

Abstract:

Background: Thienopyrimidine, triazole and thiazolidinone derivatives have recently gained attention due to their effective pharmacological activities. They show antioxidant, antitumor, antimicrobial, antiviral, anti-inflammatory and analgesic properties. Objective: Synthesis of new ethyl 2-amino-4-isopropyl-5-methylthiophene-3-carboxylate (2) was used as a starting material to produce 2-mercapto-methylthienopyrimidinone (3), (4) and 2- hydrazinyl-methylthienopyrimidinone (5), through high yields and evaluating anticancer activities. Method: A series of novel Schiff's bases (6-9) were produced

APA, Harvard, Vancouver, ISO, and other styles

4

C., Mallikarjunaswamy*1 V. Lakshmi Ranganatha2 L. Mallesha1 D.G. Bhadregowda3. "NOVEL PYRIMIDINE SCHIFF BASES: SYNTHESIS AND PHARMACOLOGICAL SCREENING." INDO AMERICAN JOURNAL OF PHARMACEUTICAL RESEARCH 07, no. 01 (2017): 7329–39. https://doi.org/10.5281/zenodo.1005166.

Full text

Abstract:

Schiff bases are aldehydelike compounds in which an imine group replaces the carbonyl group. They are widely used for industrial purposes and also exhibit a broad range of biological activities. This study represents the synthesis of a new series of (E) -N-benzylidene-5-bromo-2-chloropyrimidin-4-amine derivatives (6a-l). The newly synthesized compounds were characterized by different spectral studies. All these new compounds screened for their anti-inflammatory, antimicrobial and in vitro antioxidant activities. Structure–activity relationship analysis demonstrates that hydroxyl groups on the

APA, Harvard, Vancouver, ISO, and other styles

5

Amić, Ana, and Elena Gotal. "Selected Thermodynamic Parameters of Antioxidant Activity of Coumarin Based Heterocyclic Compounds." Chemistry Proceedings 3, no. 1 (2020): 109. http://dx.doi.org/10.3390/ecsoc-24-08385.

Full text

Abstract:

Coumarin and coumarin derivatives are bioactive compounds that have an important role in medicinal chemistry, for example in the development of anti-inflammatory, anticancer and antiviral drugs. These compounds are also very powerful antioxidants that successfully scavenge free radicals and prevent or alleviate oxidative stress. The antioxidant potential of selected heterocyclic compounds containing coumarin core was investigated theoretically, the focus of this study was on hydrogen atom transfer mechanism (HAT) and single electron transfer followed by a proton transfer mechanism (SET-PT). Us

APA, Harvard, Vancouver, ISO, and other styles

6

Premlata, Gupta, Jat Kamal, Singh Solanki Vijendra, and Shrivastava Ruchi. "An efficient synthesis, characterization and biological activity of novel Schiff bases of 2-aryl-1H-benzo[d]imidazole-4-carbohydrazide derivatives." Journal of India Chemical Society Vol. 95, Feb 2018 (2018): 173–79. https://doi.org/10.5281/zenodo.5638706.

Full text

Abstract:

Department of Chemistry IPS Academy, Indore-452 012, Madhya Pradesh, India E-mail : drpremlataguptachem@gmail.com <em>Manuscript received 20 December 2017, revised 31 January 2018, accepted 19 February 2018</em> A series of <em>N'</em>-aryllidene-2-aryl-1<em>H</em>-benzo[<em>d</em>]imidazole-4-carbohydrazide (Schiff bases) 3a<sub>1</sub>-3d<sub>4</sub> were synthesized by condensation reaction of 2-aryl-1<em>H</em>-benzo[<em>d</em>]imidazole-4-carbohydrazide (2a-2d) with substituted aromatic aldehyde. The characterization of all these novel synthesized compounds 3a<sub>1</sub>-3d<sub>4</su

APA, Harvard, Vancouver, ISO, and other styles

7

Rani, U. Usha, and A. Sreedevi. "Synthesis and Biological Evaluation of 3-(2-Benzoyl-4-chlorophenyl)-4H-spiro [indole-3,2-[1,3]thiazolidine]-2,4(1H)- dione Derivatives for Anti-tubercular and Antimicrobial Activities." Indian Journal Of Science And Technology 17, no. 20 (2024): 2101–9. http://dx.doi.org/10.17485/ijst/v17i20.1434.

Full text

Abstract:

Objectives: To synthesize a new scaff fold of 3'-(2-Benzoyl-4-chlorophenyl)-4'H-spiro [indole-3,2'-[1,3] thiazolidine]-2,4'(1H)-dione derivatives and to assess the compounds for anti-tubercular and antimicrobial activities. Methods : A new series of 3'-(2-Benzoyl-4-chlorophenyl)-4'H-spiro [indole-3,2'- [1,3] thiazolidine]-2,4'(1H)-dione derivatives were prepared by synthesizing schiff’s bases followed by condensing schiff base with 2-mercaptopropanoic acid in the presence of zinc chloride. Synthesized compounds were characterized by IR, NMR and Mass spectral data. Their antimicrobial, antitube

APA, Harvard, Vancouver, ISO, and other styles

8

Somani, R., P. Dubey, and S. Zine. "MICROWAVE ASSISTED SYNTHESIS OF BIPHENYL BASED SCHIFF’S BASES AND THEIR ANTIMICROBIAL EVALUATION." INDIAN DRUGS 55, no. 03 (2018): 13–18. http://dx.doi.org/10.53879/id.55.03.11218.

Full text

Abstract:

Schiff’s base constitutes a significant class of compounds for new drug development. They are widely used for industrial purposes and also exhibit a broad range of biological activities. The search for Schiff’s base containing compounds with more selective activity and lower side effects continues to be an active area of argument examination in medicinal chemistry. The biphenyl molecule consists of two connected phenyl rings. Biphenyl ring scaffolds are fairly non-reactive in nature. They enhance the log-P values; increase the tropical polar surface area (TPSA) of the molecule, act as hydropho

APA, Harvard, Vancouver, ISO, and other styles

9

Sumathy, A., R. Suresh, and N. L. Gowrishankar. "In-silico DESIGN SCREENING OF SOME PYRAZOLONE FUSED HETEROCYCLIC ANALOGUES AS HER2 INHIBITORS TARGETING BREAST CANCER." Rasayan Journal of Chemistry 15, no. 01 (2022): 497–503. http://dx.doi.org/10.31788/rjc.2022.1516738.

Full text

Abstract:

In human breast cancers, the human epidermal development factor receptor-2 is a membrane tyrosine kinase that is overexpressed, and gene amplified. Pyrazolone fused heterocyclic moieties- thiazolidinone, carboxymethyl thiazolidinone, azetidinone are significant DNA-intercalating agents here human epidermal development factor receptor-2 amplification and over expression are linked to tumour cell proliferation and the pathway of instances in breast cancer. Few novel pyrazolone fused heterocyclic analogues are designed by in-silico-technique for their human epidermal development factor receptor-2

APA, Harvard, Vancouver, ISO, and other styles

10

Padmaja, Devi M. S* Dr. Prasobh G.R. Dr. Sandhya S.M Visal C. S. Reena Athira. "SYNTHESIS AND SCREENING OF ANALGESIC AND ANTI-INFLAMMATORY ACTIVITY OF NOVEL BENZTRIAZOLE DERIVATIVES." INDO AMERICAN JOURNAL OF PHARMACEUTICAL SCIENCES o6, no. 07 (2019): 13632–48. https://doi.org/10.5281/zenodo.3345871.

Full text

Abstract:

<em>Benzotriazole is a  lead molecule for designing potential bioactive molecule. Benzotriazole and its derivatives exhibits anti inflammatory, analgesic, antimicrobial and anticonvulsant activities. 1,2,4 triazole is one of the most biologically active classes of compounds possessing wide spectrum of activities including anti-inflammatory, analgesic, CNS stimulants, sedatives, antianxiety, antimicrobial agents and antimycotic agents. In this study, we planned to synthesize various Schiff’s bases of 5 [1H,1,2,3 benzotriazol 1yl methyl] 4 [substituted amino]4H-1,2,4 triazole-3 &ndash

APA, Harvard, Vancouver, ISO, and other styles

More sources

We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!