Log in

Relevant bibliographies by topics / Substituted acetamides

Contents

Journal articles
Dissertations / Theses
Book chapters
Conference papers

Academic literature on the topic 'Substituted acetamides'

Author: Grafiati

Published: 4 June 2021

Last updated: 3 February 2022

Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles

Select a source type:

Consult the lists of relevant articles, books, theses, conference reports, and other scholarly sources on the topic 'Substituted acetamides.'

Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.

You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.

Journal articles on the topic "Substituted acetamides"

1

Gowda, Basavalinganadoddy Thimme, Jozef Kožíšek, Ingrid Svoboda, and Hartmut Fuess. "Effect of Meta-Substitution on Solid State Geometry of N-(Aryl)-2,2,2-trichloro-acetamides, 3-XC6H4NH-CO-CCl3 and 3,5-X2C6H3NH-CO-CCl3 (X = Cl, CH3)." Zeitschrift für Naturforschung A 62, no. 1-2 (2007): 91–100. http://dx.doi.org/10.1515/zna-2007-1-213.

Full text

Abstract:

The crystal structures of N-(meta-substituted phenyl)-2,2,2-trichloro-acetamides such as N- (3-methylphenyl)-2,2,2-trichloro-acetamide, 3-CH3C6H4NH-CO-CCl3 (3MPTCA); N-(3-chlorophenyl)- 2,2,2-trichloro-acetamide, 3-ClC6H4NH-CO-CCl3 (3CPTCA); N-(3,5-dimethylphenyl)- 2,2,2-trichloro-acetamide, 3,5-(CH3)2C6H3NH-CO-CCl3 (35DMPTCA) and N-(3,5-dichlorophenyl)- 2,2,2-trichloro-acetamide, 3,5-Cl2C6H3NH-CO-CCl3 (35DCPTCA) have been determined at room temperature. The crystal system, space group, formula units and lattice constants (Å ) of the new structures are: 3MPTCA: orthorhombic, Pbca, Z = 8, a = 1

APA, Harvard, Vancouver, ISO, and other styles

2

Angel, April J., Anne E. Finefrock, Kristen L. French, et al. "Preparation of N-aryl-4-oxo-4H-1-benzothiopyran-2-acetamides from trilithiated acetoacetanilides and lithiated methyl thiosalicylate." Canadian Journal of Chemistry 77, no. 1 (1999): 94–97. http://dx.doi.org/10.1139/v98-216.

Full text

Abstract:

Acetoacetanilide and substituted acetoacetanilides were trilithiated in excess lithium diisopropylamide, and the polylithiated intermediates were regioselectively condensed with lithiated methyl thiosalicylate, followed by acid cyclization to afford substituted N-aryl-4-oxo-4H-1-benzothiopyran-2-acetamides (thiochromone-2-acetamides).Key words: thiochromones, strong-base multiple anion synthesis, Claisen-type condensation.

APA, Harvard, Vancouver, ISO, and other styles

3

Alagarsamy, Veerachamy, Viswas Raja Solomon, Mohaideen Thasthagir Sulthana, Meduri Satyasai Vijay, and Bandi Narendhar. "Design and synthesis of quinazolinyl acetamides for their analgesic and anti-inflammatory activities." Zeitschrift für Naturforschung B 70, no. 8 (2015): 597–604. http://dx.doi.org/10.1515/znb-2015-0035.

Full text

Abstract:

AbstractA variety of novel 2-(substituted)-N-(4-oxo-2-phenylquinazolin-3(3H)-yl)acetamides were synthesized by the reaction of 2-chloro-N-(4-oxo-2-phenylquinazolin-3(3H)-yl)acetamide with various amines. The starting material, 2-chloro-N-(4-oxo-2-phenylquinazolin-3(3H)-yl)acetamide, was synthesized from anthranilic acid by the multistep process. The title compounds were investigated for analgesic, anti-inflammatory, and ulcerogenic index activities. Among those, the compound 2-(ethylamino)-N-(4-oxo-2-phenylquinazolin-3(3H)-yl)acetamide (V9) showed most potent analgesic and anti-inflammatory ac

APA, Harvard, Vancouver, ISO, and other styles

4

Krivoshein, Arcadius V. "α-Substituted Lactams and Acetamides: Ion Channel Modulators that Show Promise in Treating Drug-resistant Epilepsy". Central Nervous System Agents in Medicinal Chemistry 20, № 2 (2020): 79–87. http://dx.doi.org/10.2174/1871524920666200510005458.

Full text

Abstract:

The two main problems in the pharmacotherapy of epilepsy are resistance to currently available first-line medications (which occurs in about one third of patients) and the high incidence of side effects. To address these two challenges, extensive efforts are being undertaken to design new, structurally distinct antiepileptic drugs with a broad spectrum of anticonvulsant activity. Tests in animal models of epilepsy indicate that α-substituted lactams and acetamides show a broad spectrum of anticonvulsant activity (including very promising activity in drug-resistant models) as well as an excelle

APA, Harvard, Vancouver, ISO, and other styles

5

Yadav, Smriti, Bharath Kumar Inturi, Shrinidhi B.R, Pooja H.J, Neenu Ganesh, and Gurubasavaraj V. Pujar. "Design, Synthesis and Antitubercular Evaluation of New Benzimidazole Scaffolds." Anti-Infective Agents 18, no. 4 (2021): 375–83. http://dx.doi.org/10.2174/2211352518666200108091454.

Full text

Abstract:

Background: To overcome one of the resistance mechanisms of Isoniazid (INH), there is a need for an antitubercular agent that can inhibit InhA enzyme by circumventing the formation of INH-NAD+ adduct. Objective: The objective of the study is the development of novel antitubercular agents that target Mycobacterium tuberculosis InhA (Enoyl Acyl Carrier Protein Reductase). Methods: A small-molecule chemical library was used for the identification of the novel InhA inhibitors using primary screening and molecular docking studies followed by the scaffold hopping approach. The designed molecules, 2-

APA, Harvard, Vancouver, ISO, and other styles

6

Gowda, Basavalinganadoddy Thimme, Shilpa Lakshmipathy, and Jayalakshmi K. Lakshmipathy. "Synthetic and 1H and 13C NMRSpectral Studies on N-(Mono-substitutedphenyl)- acetamides and Substituted Acetamides, 2/3/4-YC6H4NH-COCH3–iXi (Y = CH3, F, Cl, Br, NO2; X = Cl, CH3; i = 0, 1, 2, 3)." Zeitschrift für Naturforschung A 61, no. 10-11 (2006): 595–99. http://dx.doi.org/10.1515/zna-2006-10-1113.

Full text

Abstract:

Nineteen N-(2/3/4-methyl/halo/nitro-phenyl)-acetamides and substituted acetamides, 2/3/4- YC6H4NH-CO-CH3−iXi (Y = CH3, F, Cl, Br or NO2; X = Cl or CH3 and i = 0, 1, 2 or 3), have been prepared, characterized, and their 1H and 13C NMR spectra in solution measured and correlated. 1H and 13C NMR chemical shifts were assigned to the protons and carbon atoms, respectively, in line with those for similar compounds. Since the chemical shifts are dependent on the electron density around the nucleus or associated with the atom to which it is bound, the incremental shifts of the aromatic protons or carb

APA, Harvard, Vancouver, ISO, and other styles

7

Raghavendra, N. M., P. P. Thampi, and P. M. Gurubasavarajaswamy. "Synthesis and Antimicrobial Activity of Some Novel Substituted Piperazinyl-quinazolin-3(4H)-ones." E-Journal of Chemistry 5, no. 1 (2008): 23–33. http://dx.doi.org/10.1155/2008/410157.

Full text

Abstract:

Several substituted-quinazolin-3(4H)-ones were synthesized by condensation of 2-chloro-N-(4-oxo-substituted-quinazolin-3(4H)-yl)-acetamides with various substituted piperazines through single step reaction. Elemental analysis, IR,1HNMR and mass spectral data confirmed the structure of the newly synthesized compounds. Synthesized quinazolin-4-one derivatives were investigated for their antibacterial and antifungal activities.

APA, Harvard, Vancouver, ISO, and other styles

8

Su, Weike, Bibo Yang, and Yongshu Li. "A Novel Synthesis of N-substituted 2-(benzotriazol-1-yl) Acetamides Promoted by Samarium Diiodide." Journal of Chemical Research 2002, no. 11 (2002): 542–43. http://dx.doi.org/10.3184/030823402103170934.

Full text

APA, Harvard, Vancouver, ISO, and other styles

9

Xu, Di, Lena Frank, Tina Nguyen, et al. "Magnesium-Catalyzed N2-Regioselective Alkylation of 3-Substituted Pyrazoles." Synlett 31, no. 06 (2019): 595–99. http://dx.doi.org/10.1055/s-0039-1690160.

Full text

Abstract:

A highly regioselective Mg-catalyzed alkylation of 3-substituted pyrazoles has been developed to provide N2-alkylated regioisomers. Using α-bromoacetates and acetamides as alkylating agents, this new method was applied to a variety of 3-substituted and 3,4-disubstituted pyrazoles to produce the N2-alkylated products with high regioselectivities ranging from 76:24 to 99:1 and 44–90% yields.

APA, Harvard, Vancouver, ISO, and other styles

10

Chordia, Mahendra D., Sanjay N. Karmarkar, Shriniwas L. Kelkar, and Murzban S. Wadia. "Use of Substituted Acetamides for the Synthesis of 3-Substituted 2-Aminoquinolines." Synthesis 1987, no. 09 (1987): 810–11. http://dx.doi.org/10.1055/s-1987-28080.

Full text

APA, Harvard, Vancouver, ISO, and other styles

Dissertations / Theses on the topic "Substituted acetamides"

1

Zink, Landon. "Synthesis of N-(substituted phenyl) acetamides." Digital Commons @ East Tennessee State University, 2011. https://dc.etsu.edu/honors/131.

Full text

APA, Harvard, Vancouver, ISO, and other styles

2

Flanigan, David L. "Studies in rhodium catalyzed intramolecular C-H insertion of amino acid derived [alpha]-diazo-[alpha]-(substituted)acetamides and its application to the total synthesis of clasto-lactacystin [beta]-lactone." [Tampa, Fla.] : University of South Florida, 2004. http://purl.fcla.edu/fcla/etd/SFE0000418.

Full text

APA, Harvard, Vancouver, ISO, and other styles

3

Flanigan, David L. Jr. "Studies in Rhodium Catalyzed Intramolecular C-H Insertion of Amino Acid Derived α-Diazo-α-(substituted)acetamides and its Application to the Total Synthesis of clasto-Lactacystin β-Lactone". Scholar Commons, 2004. https://scholarcommons.usf.edu/etd/1037.

Full text

Abstract:

Lactacystin is a microbial metabolite isolated by Omura that exhibits neurotrophic activity in neuroblastoma cell lines. Lactacystin and especially its β-lactone analog are the first examples of non-polypeptide small molecules capable of specifically inhibiting the 20S proteasome. Various asymmetric total syntheses of lactacystin and its analogs have been reported. The total synthesis of clasto -lactacystin β-lactone is achieved using L-serine methyl ester as the starting material and the sole source of stereochemical induction. The success of this synthesis hinges on two featured transformati

APA, Harvard, Vancouver, ISO, and other styles

4

Peixoto, Isabelle Nogueira. "Estudos químicos de derivados mesoiônicos do sistema 1,3- Tiazólio-5-tiolato com acetamidas substituídas e suas Potencialidades antifúngicas contra cepas de candida Albicans." Universidade Federal da Paraíba, 2016. http://tede.biblioteca.ufpb.br:8080/handle/tede/9002.

Full text

Abstract:

Submitted by Maike Costa (maiksebas@gmail.com) on 2017-06-20T11:50:06Z No. of bitstreams: 1 arquivototal.pdf: 10487656 bytes, checksum: 9f874336a1873756d7bc4d26e57ee76d (MD5)<br>Made available in DSpace on 2017-06-20T11:50:06Z (GMT). No. of bitstreams: 1 arquivototal.pdf: 10487656 bytes, checksum: 9f874336a1873756d7bc4d26e57ee76d (MD5) Previous issue date: 2016-05-13<br>This work describes the synthesis, characterization and antifungal potential of twelve mesoionic derivatives from the 1,3-thiazolium-5-thiolate system. The compounds, totally unprecedented, were divided in two classes:

APA, Harvard, Vancouver, ISO, and other styles

5

Gomes, Roberto da Silva. "Análise conformacional e das interações eletrônicas de algumas N-metóxi-N-metil-acetamidas-α-heterossubstituídas." Universidade de São Paulo, 2011. http://www.teses.usp.br/teses/disponiveis/46/46136/tde-31082011-144942/.

Full text

Abstract:

A presente tese trata da síntese e a análise conformacional de algumas N-metóxi-N-metil-amidas α-heterossubstituídas (amidas de Weinreb) Z-C(O)-N(OMe)Me (Z= CH2F (1), CH2OMe (2), CH2OPh (3), CH2Cl (4), CH2Br (5), CH2SEt (6) e Me2CSEt (7). A análise da banda da carbonila no infravermelho apoiada por cálculos teóricos B3LYP/6311++G(3df, 3pd), juntamente com a análise de NBO indicou a existência de um equilíbrio conformacional cis/gauche, isto é, (c) e (g) para (1) e (3), (c1, c2) e (g1, g2) para (2), (c) e (g1, g2) para (4-6) e (g1, g2) para (7). Em fase gasosa a população do confôrmero gau

APA, Harvard, Vancouver, ISO, and other styles

6

Yan-JhuChen and 陳彥竹. "Synthesis of Highly Substituted 2-Quinolinones via Intramolecular Cyclization of Acetamide Derivatives." Thesis, 2016. http://ndltd.ncl.edu.tw/handle/44316335157697510707.

Full text

Abstract:

碩士<br>國立成功大學<br>化學系<br>104<br>Three effective methods for the synthesis of 2-quinolinones were reported. We use α-substituted N-[2-(phenylethynyl)phenyl]acetamides as substrates, undergoes a 6-exo-dig cyclization and consequently produce 3,4-disubstituted 2-quinolinones. Surprisingly, heterocyclic substrates could also be used to generate the corresponding 2-quinolinones. To our delight, a variety of functional groups, including benzoyl, methoxycarbonyl and cyano groups, were used in these reaction conditions.

APA, Harvard, Vancouver, ISO, and other styles

7

Lo, Pei-Ching, and 羅珮菁. "Gold-Catalyzed Cyclization of N-(2-ethynylphenyl)-N-((methylthio)methyl)acetamide Derivatives with 1,3-Migration to Substituted indoles." Thesis, 2018. http://ndltd.ncl.edu.tw/handle/csu36q.

Full text

Abstract:

碩士<br>國立中山大學<br>生物科學系研究所<br>106<br>Molecules that contain the indole substructure exhibit a broad spectrum of biological activities, such as anti-cancer, anti-oxidant, anti-rheumatoidal, anti-HIV, anti-microbial, anti-inflamatory, analgesic, antipyretic, anti-convulsant and anthelmintic activities. Treatment of N-(2-ethynylphenyl)-N-((methylthio)methyl)acetamide as precursor with 0.1 equivalent of (furyl)3PAuCl and 0.1 equivalent of AgSbF6 in refluxing acetonitrile for 24 hours afforded cyclized and hydrolyzed indole derivatives. Preliminary results showed precursor bearing electron donating g

APA, Harvard, Vancouver, ISO, and other styles

Book chapters on the topic "Substituted acetamides"

1

Kikelj, D., and U. Urleb. "From N-Substituted 2-[(Thioacyl)sulfanyl]acetamides." In Five-Membered Hetarenes with One Chalcogen and One Additional Heteroatom. Georg Thieme Verlag KG, 2002. http://dx.doi.org/10.1055/sos-sd-011-00908.

Full text

APA, Harvard, Vancouver, ISO, and other styles

2

"DFT Study on Some Synthetic Compounds: (2,6), (2,4) and (3,4) Dichloro Substituted Phenyl-N-(1- 3-thiazol-2-yl) Acetamides." In DFT Based Studies on Bioactive Molecules, edited by Ambrish Kumar Srivastava and Neeraj Misra. BENTHAM SCIENCE PUBLISHERS, 2021. http://dx.doi.org/10.2174/9789814998369121010005.

Full text

APA, Harvard, Vancouver, ISO, and other styles

3

Schmued, Larry. "Fluoro-Gold and 4-Acetamido-4′-isothiocyanostilbene-2,2′-disulfonic Acid: Use of Substituted Stilbenes in Neuroanatomical Studies." In Quantitative and Qualitative Microscopy. Elsevier, 1990. http://dx.doi.org/10.1016/b978-0-12-185255-9.50022-5.

Full text

APA, Harvard, Vancouver, ISO, and other styles

Conference papers on the topic "Substituted acetamides"

1

Nikalje, Anna Pratima, Mangesh Ghodke, Shailee Tiwari, Julio Seijas Vázquez, and M. Pilar Vazquez-Tato. "Microwave-Assisted Facile Synthesis and anticonvulsant evaluation of Novel N-(3-chloro-2-oxo-4-substituted phenyl azetidin-1-yl)-2-(1, 3-dioxoisoindolin-2-yl) acetamides." In The 21st International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2017. http://dx.doi.org/10.3390/ecsoc-21-04810.

Full text

APA, Harvard, Vancouver, ISO, and other styles

2

Nikalje, Anna Pratima. "Synthesis and Anti-Inflammatory Evaluation of 2-(3-(2-(1,3-Dioxoisoindolun-2-YL) Acetamido)-4-OXO-2-Substituted Thiazolidin-5-YL) Acetic Acid Derivatives." In The 18th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2014. http://dx.doi.org/10.3390/ecsoc-18-c010.

Full text

APA, Harvard, Vancouver, ISO, and other styles

We offer discounts on all premium plans for authors whose works are included in thematic literature selections. Contact us to get a unique promo code!