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Dissertations / Theses on the topic 'Synthesis of oxazolidinones'

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Published: 5 June 2025

Last updated: 1 August 2025

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1

Phung, Chau V. "The Synthesis of Oxazolidinones from Aziridines and Carbon Dioxide." University of Cincinnati / OhioLINK, 2016. http://rave.ohiolink.edu/etdc/view?acc_num=ucin1470741529.

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2

Ho, Hoi Tong Lawrence. "New methods in chiral synthesis." Thesis, University of Bath, 1999. https://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.301557.

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3

Zheng, Zilong. "Synthesis of Oxazolidinone Derivatives and Anti-Influenza Agents." Ohio University / OhioLINK, 2016. http://rave.ohiolink.edu/etdc/view?acc_num=ohiou1470739369.

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4

Orac, Crina M. "Stereochemical Synthesis of Ring E Analogs of Methyllycaconitine and 4,5-Disubstituted Oxazolidinones." Ohio University / OhioLINK, 2009. http://rave.ohiolink.edu/etdc/view?acc_num=ohiou1258046479.

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5

Ella-Menye, Jean-Rene. "Synthesis of Novel Chiral Heterocyclic Compounds for Antibacterial Agents and Peptidomimetics." ScholarWorks@UNO, 2007. http://scholarworks.uno.edu/td/611.

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Small chiral molecules are very important building blocks in the synthesis of biologically active compounds. These building blocks include nitrogen and oxygen-containing heterocycles such as 2-oxazolidinones, 1,3-oxazinan-2-ones, 2-oxazolines, oxazines, morpholine and morpholinones. Because of their interesting properties, chiral heterocycles have stirred great interest in the synthetic chemist community to develop useful and efficient strategies to these molecules. In this dissertation, the design and syntheses of various heterocyclic building blocks are presented, as well as the testing of t

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6

Revell, Kevin David. "Mode of action and structure-activity studies of N-alkylthio beta-lactams and N-alkylthio-2-oxazolidinones, and synthesis of second-generation disulfide Inhibitors of beta-Ketoacyl-Acyl Carrer Protein Synthase III (FabH) as potent antibacterial agents." [Tampa, Fla] : University of South Florida, 2006. http://purl.fcla.edu/usf/dc/et/SFE0001453.

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7

Fang, Fang. "Synthesis of Bicyclic and Tricyclic Analogues of Oxazolidinone." Ohio University / OhioLINK, 2013. http://rave.ohiolink.edu/etdc/view?acc_num=ohiou1357312054.

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8

Karmakar, S. "Synthetic studies towards pseudotheonamides, herbarium III, bicyclic thiohydantoins and oxazolidinone -5- one." Thesis(Ph.D.), CSIR-National Chemical Laboratory, Pune, 2006. http://dspace.ncl.res.in:8080/xmlui/handle/20.500.12252/2479.

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9

Bhandare, Richie R. "Investigation into the bioisosteric approach in the design, synthesis and evaluation of muscarinic receptor ligands." Diss., Temple University Libraries, 2013. http://cdm16002.contentdm.oclc.org/cdm/ref/collection/p245801coll10/id/214985.

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Pharmaceutical Sciences<br>Ph.D.<br>The acetylcholine (ACh) receptor system belongs to rhodopsin GPCR family and is an integral membrane protein divided into two types: muscarinic and nicotinic. The naturally occurring neurotransmitter acetylcholine binds to these two receptor systems non- selectively. The regulatory effects of the neurotransmitter acetylcholine are diverse ranging from autonomic nervous system and the central nervous system through different types of neurons innervated by cholinergic inputs. Muscarinic acetylcholine receptors (mAChRs) are divided into five receptor subtypes (

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10

Zhang, Jianjun. "Library Synthesis of Anticancer and Antibacterial Agents via Azide Chemistry." DigitalCommons@USU, 2010. https://digitalcommons.usu.edu/etd/711.

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Various anticancer and antibacterial agents have been synthesized via azide chemistry by taking advantage of carbohydrate. Starting from the synthesis of 14 glycosyl azides, a library of carbohydrate-oxazolidinone conjugates and a library of carbohydrate-cyclopamine conjugates with biological interests were synthesized based on a highly efficient "click reaction" assisted by sonication. Some of the conjugates have improved solubility and enhanced anticancer activity. A library of neomycin B derivatives with various modifications at the 5" position has been synthesized. Two leads exhibit

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11

Murray, Adrian James. "The use of a bicyclic -oxazolidinone as a key precursor towards the total synthesis of (-)- kainic acid and (-)-swainsonine." Thesis, University of Sussex, 2007. http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.487581.

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12

Bhetuwal, Bishwa Raj. "Stereoselective Synthesis of β-Mannosides and β-Mannosamines via Cs₂CO₃-Mediated Anomeric O-Alkylation". University of Toledo / OhioLINK, 2020. http://rave.ohiolink.edu/etdc/view?acc_num=toledo1606049621805782.

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13

DELAUNAY, DOMINIQUE. "Contribution a l'etude des 2-oxazolidinones, 2-oxazolidinethiones et 2-thiazolidinethiones. Preparation de beta-aminothiols et utilisation en synthese asymetrique." Rennes 1, 1995. http://www.theses.fr/1995REN10055.

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Le travail presente dans ce memoire apporte une contribution a l'etude de la synthese des beta-aminothiols et de leur utilisation en catalyse asymetrique. L'elaboration de ces composes a partir des beta-aminoalcools nous a conduits a mettre au point les conditions d'acces a plusieurs heterocycles: oxazolidinones, oxazolidinethiones et thiazolidinethiones. Dans la premiere partie, nous avons mis en evidence deux voies d'acces aux oxazolidinones a partir des alpha-aminoesters. La premiere, tres directe, consiste, a condenser un organomagnesien sur des carbamates esters, mais ce procede conduit a

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14

Zhang, Yang. "Dynamic Systems : Enzymatic Synthesis, Exchange Reactions and Applications in Materials Science." Doctoral thesis, KTH, Organisk kemi, 2015. http://urn.kb.se/resolve?urn=urn:nbn:se:kth:diva-173480.

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This thesis is divided into three parts, revolving around the developments of dynamic systems utilized in dynamic kinetic resolution (DKR) and constitutional dynamic chemistry (CDC). The first section gives an introduction to constitutional dynamics, the core concept of this thesis. Constitutional dynamics can be tuned through reversible interactions. Then, the basic principles of constitutional dynamics in DKR and CDC are discussed, along with their applications. The second section explores the asymmetric synthesis of oxazolidinone derivatives using lipase catalysis through kinetic resolution

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15

Denis, Alexis. "Fonctionnalisations selectives a l'aide des complexes du palladium : synthese de composes d'interet biologiques, cyclopropanes vinyliques, aryl-3 oxazolidinones-2 (inhibiteurs potentiels de la monoamine oxydase)." Paris 6, 1987. http://www.theses.fr/1987PA066335.

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Ce travail porte sur l'utilisation du palladium (o) pour la synthese de molecules d'interet biologique. En premier lieu, on decrit la synthese stereoselective de cyclopropanes vinyliques et de pyrethrinoides. Dans un second temps, on etudie l'echange acetate phenol et l'amination de derives allyliques fibonctionnels. Enfin, on presente la synthese d'aryl-3 dihydroxy-5,5 oxazolidones-2 erythro et threo et etudie leur utilisation en tant qu'inhibiteur d'enzyme monoamine oxidase

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16

Tang, Ya-Ping, and 湯雅評. "Synthesis and Structure-Activity Relationships of Oxazolidines and Oxazolidinones." Thesis, 2005. http://ndltd.ncl.edu.tw/handle/20323261878776123488.

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碩士<br>大仁科技大學<br>製藥科技研究所<br>93<br>Many previous reports mainly concentrated on chemical synthesis and reactivity of this class of oxazolidines, so far few investigations have been reported on the anticancer activity of these compounds against tumor cell lines in vitro. Especially the lack of any information concerning the influence on the biological activity of an aromatic substitution attached to the 2 position of oxazolidine prompted us to attempt the preparation of these compounds. 2-aryl-1,3-oxazolidines were formed from ?aminoalcohol with various aromatic aldehyde. On the other hand, we

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17

Hein, Jason Ellis. "Tools for efficient asymmetric synthesis: design, synthesis and application of fluorous oxazolidinone chiral auxiliaries." Thesis, 2006. http://hdl.handle.net/1993/187.

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A new class of oxazolidinone chiral auxiliary has been synthesized from various α-amino acids, incorporating a perfluoroalkyl functional chain as a soluble support. This feature allows the chiral auxiliaries to be employed under standard solution-phase reaction conditions, and rapidly purified from crude mixtures using fluorous solid phase extraction (FSPE). Our investigation of these new materials has been divided into two main sections. To obtain the chiral auxiliaries in multi-gram quantities a synthetic protocol was designed, where efficiency and reproducibility were the primary obje

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18

Siuts, Antje. "Synthese von neuen 3-Aryl-2-oxazolidinonen als antibakterielle Wirkstoffe /." 1994. http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&doc_number=006651747&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA.

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19

Lin, Shih-Che, and 林士哲. "Joined Use of Oxazolidinone and Desymmetric Amino Protection in Application of Oligosaccharide Synthesis." Thesis, 2010. http://ndltd.ncl.edu.tw/handle/87344166396453512090.

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碩士<br>國立交通大學<br>應用化學研究所<br>98<br>Joined use of N-benzyl oxazolidinone and N-benzyl-N-benzyloxycarbonyl (N-BnCbz) desymmetric amino-protecting function is reported. The new synthetic approach enables the facile preparation of type 1 and type 2 LacNAc disaccharide in satisfactory yield. One-pot deprotection of N-BnCbz and O-benzyl ether is achieved by hydrogenolysis under mild conditions. Further application of this protection strategy realizes the synthesis of trisaccharide H blood group substrate.

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20

(6859052), Jacqueline N. Williams. "DESIGN, SYNTHESIS, AND BIOLOGICAL EVALUATION OF POTENT HIV-1 PROTEASE INHIBITORS WITH NOVEL BICYCLIC OXAZOLIDINONE AND BIS SQUARAMIDE SCAFFOLDS." Thesis, 2019.

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<p>In 2018, the World Health Organization (WHO) reported approximately 37 million people are living with the Human Immunodeficiency Virus (HIV). Suppressing replication of the virus down to undetectable levels was achieved by combination antiretroviral therapy (cART) which effectively reduced the mortality and morbidity rates of HIV positive individuals. Despite the improvements towards combatting HIV/AIDS, no successful treatment exists to eradicate the virus from an infected individual. Treatment regimens are lifelong and prompt less than desirable side effects including but not limited to;

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21

Mathre, David John. "I. The Disastereoselective Alkylation of Chiral 2-Oxazolidinone Imide Enolates. II. Efforts Directed Toward the Enantioselective Total Synthesis of Ferensimycin B." Thesis, 1985. https://thesis.library.caltech.edu/11401/1/Mathre_DJ_1985.pdf.

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<p>The diastereoselective alkylation of chiral 2-oxazolidinone imide enolates is described. The requisite chiral N-acyl 2-oxazolididones are prepared from readily available amino acid and amino alcohol precursors. The lithium and sodium enolates, derived from these chiral imides, react in a highly diastereoselective manner with a variety of electrophiles. Furthermore, the diasteromers are often separable by liquid chromateography affording products with a diastereomeric purity ≥ 99:1. Several methods are described for the non–destructive removal of the chiral auxiliary to afford enantiomerical

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22

Hsu, Mei-Yuan, and 許媄媛. "Synthesis of di- and tri-substituted imidazoles mediated by tributylphosphine via [3+2] cyclization of in situ generated oxazolidinone and ethyl cyanoformate." Thesis, 2010. http://ndltd.ncl.edu.tw/handle/21540813001552023488.

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碩士<br>淡江大學<br>化學學系碩士班<br>98<br>In the current study, we take advantage of oxazolidinone and ethyl formate to carry out [3+2] cycloaddition aimed at synthesizing a series of di- and tri-substituted imidazoles. Regarding the synthesis of di-substituted imidazoles, glycine was taken to couple with benzoyl chloride, followed by the dehydration mediated by 1-ethyl-3-(3-dimethyl- aminopropyl)carbodiimide hydrochloride(EDCI) in DCM to generate oxazolidinone 68 in 30 mins. Without purification, ethyl formate and tributylphosphine (PBu3, 0.6 eq) were further added in the solution and the mixture was st

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