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Journal articles on the topic 'Synthesis of oxazolidinones'

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Published: 5 June 2025

Last updated: 1 August 2025

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1

Aoki, Hiroyuki, Lizhu Ke, Susan M. Poppe, et al. "Oxazolidinone Antibiotics Target the P Site on Escherichiacoli Ribosomes." Antimicrobial Agents and Chemotherapy 46, no. 4 (2002): 1080–85. http://dx.doi.org/10.1128/aac.46.4.1080-1085.2002.

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ABSTRACT The oxazolidinones are a novel class of antimicrobial agents that target protein synthesis in a wide spectrum of gram-positive and anaerobic bacteria. The oxazolidinone PNU-100766 (linezolid) inhibits the binding of fMet-tRNA to 70S ribosomes. Mutations to oxazolidinone resistance in Halobacterium halobium, Staphylococcus aureus, and Escherichia coli map at or near domain V of the 23S rRNA, suggesting that the oxazolidinones may target the peptidyl transferase region responsible for binding fMet-tRNA. This study demonstrates that the potency of oxazolidinones corresponds to increased

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2

McKee, E. E., M. Ferguson, A. T. Bentley, and T. A. Marks. "Inhibition of Mammalian Mitochondrial Protein Synthesis by Oxazolidinones." Antimicrobial Agents and Chemotherapy 50, no. 6 (2006): 2042–49. http://dx.doi.org/10.1128/aac.01411-05.

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ABSTRACT The effects of a variety of oxazolidinones, with different antibacterial potencies, including linezolid, on mitochondrial protein synthesis were determined in intact mitochondria isolated from rat heart and liver and rabbit heart and bone marrow. The results demonstrate that a general feature of the oxazolidinone class of antibiotics is the inhibition of mammalian mitochondrial protein synthesis. Inhibition was similar in mitochondria from all tissues studied. Further, oxazolidinones that were very potent as antibiotics were uniformly potent in inhibiting mitochondrial protein synthes

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3

Sangita, Km, Geeta Gupta, Anita Pandey, and Peetam Singh. "Oxazolidinones: Mechanism of action and molecular characterization of resistance mechanisms in staphylococci." Journal of Medical Society 39, no. 1 (2025): 15–21. https://doi.org/10.4103/jms.jms_156_24.

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ABSTRACT Oxazolidinones are a new class of antibiotics effective in treating infections caused by various Gram-positive bacteria including methicillin-resistant staphylococci and vancomycin-resistant enterococci. Linezolid, the first oxazolidinone available, has become a valuable clinical option for treating infections due to multidrug-resistant Gram-positive bacteria. It has been used for patients with bacteremia, osteomyelitis, endocarditis, and skin and soft tissue infections, particularly when other therapies failed. Oxazolidinones inhibit the initiation of protein synthesis by specificall

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4

Nagiec, Eva E., Luping Wu, Steve M. Swaney, et al. "Oxazolidinones Inhibit Cellular Proliferation via Inhibition of Mitochondrial Protein Synthesis." Antimicrobial Agents and Chemotherapy 49, no. 9 (2005): 3896–902. http://dx.doi.org/10.1128/aac.49.9.3896-3902.2005.

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ABSTRACT The oxazolidinones are a relatively new structural class of antibacterial agents that act by inhibiting bacterial protein synthesis. The oxazolidinones inhibit mitochondrial protein synthesis, as shown by [35S]methionine incorporation into intact rat heart mitochondria. Treatment of K562 human erythroleukemia cells with the oxazolidinone eperezolid resulted in a time- and concentration-dependent inhibition of cell proliferation. The cells remained viable, but an increase in doubling time was observed with eperezolid treatment. Inhibition was reversible, since washing and refeeding of

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5

Foti, Claudia, Anna Piperno, Angela Scala, and Ottavia Giuffrè. "Oxazolidinone Antibiotics: Chemical, Biological and Analytical Aspects." Molecules 26, no. 14 (2021): 4280. http://dx.doi.org/10.3390/molecules26144280.

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This review covers the main aspects concerning the chemistry, the biological activity and the analytical determination of oxazolidinones, the only new class of synthetic antibiotics advanced in clinical use over the past 50 years. They are characterized by a chemical structure including the oxazolidone ring with the S configuration of substituent at C5, the acylaminomethyl group linked to C5 and the N-aryl substituent. The synthesis of oxazolidinones has gained increasing interest due to their unique mechanism of action that assures high antibiotic efficiency and low susceptibility to resistan

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6

Swaney, Steve M., Hiroyuki Aoki, M. Clelia Ganoza, and Dean L. Shinabarger. "The Oxazolidinone Linezolid Inhibits Initiation of Protein Synthesis in Bacteria." Antimicrobial Agents and Chemotherapy 42, no. 12 (1998): 3251–55. http://dx.doi.org/10.1128/aac.42.12.3251.

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ABSTRACT The oxazolidinones represent a new class of antimicrobial agents which are active against multidrug-resistant staphylococci, streptococci, and enterococci. Previous studies have demonstrated that oxazolidinones inhibit bacterial translation in vitro at a step preceding elongation but after the charging ofN-formylmethionine to the initiator tRNA molecule. The event that occurs between these two steps is termed initiation. Initiation of protein synthesis requires the simultaneous presence of N-formylmethionine-tRNA, the 30S ribosomal subunit, mRNA, GTP, and the initiation factors IF1, I

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7

Siddaraj, Ranjith, Shivaraja Govindaiah, Raghu Ningegowda, Nanjunda Swamy Shivananju, and Babu Shubha Priya. "A novel and expeditious synthesis of oxazolidinone drugs linezolid and eperezolid." European Journal of Chemistry 9, no. 4 (2018): 353–59. http://dx.doi.org/10.5155/eurjchem.9.4.353-359.1783.

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A concise and efficient synthesis of linezolid and eperezolid were accomplished through a convergent scheme utilizing diverse reaction conditions. The synthesis demonstrates utility of a new approach to facilitate the expeditious construction of 3-aryl-5-(substituted methyl)-2-oxazolidinones and easier insertion of N-acetyl group. This new approach offers the possibility of accessing related 2-oxazolidinone members easily as well as making additional analogues of Linezolid. The adopted method afforded high purity and excellent yield compared to other existing synthetic methods. The compounds w

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8

Zadsirjan, Vahideh, and Majid M. Heravi. "Oxazolidinones as Chiral Auxiliaries in the Asymmetric 1,4-Conjugate Addition Reaction Applied to the Total Synthesis of Natural Products: A Supplemental Mini-Review." Current Organic Synthesis 15, no. 1 (2018): 3–20. http://dx.doi.org/10.2174/1570179414666170601115831.

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Background: The most frequently used chiral auxiliaries, oxazolidinones (Evans' oxazolidinones) have been employed in 1,4-congugate addition reactions to α,β-unsaturated carbonyl compounds. Supplementary to our previous reports in this mini-review, we attempted to underscore the applications of this strategy in a step (steps) in the total synthesis of some naturally occurring compounds exhibiting diverse biological activities. Objective: In this mini-review, we try to underscore the applications of oxazolidinones (Evans’ oxazolidinones) in 1,4-congugate addition reactions to α,β-unsaturated ca

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9

Pi, Shao-Feng, Yue-Meng Guo, Zheng-Rui Zhou, Han-zhou Sun, and Bing Yi. "Synthesis of N-substituted-4-methylene-oxazolidinones via base-catalyzed cyclization of propargylic alcohols with p-toluenesulfonyl isocyanate." Journal of Chemical Research 44, no. 9-10 (2020): 521–23. http://dx.doi.org/10.1177/1747519820907304.

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A practical method is developed for the synthesis of oxazolidinone derivatives, an important class of heterocyclic compounds. The effect of bases and solvents on this cyclization reaction is discussed and a simple new base–solvent system (triethylamine in toluene) is found to be the most effective. The reaction conditions developed here are mild and no by-products are observed. Moreover, using optimized conditions, a number of differently substituted propargylic alcohols are cyclized to the corresponding N-substituted-4-methylene-oxazolidinones in yields of up to 99%.

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10

Schwarz, Jacob, and Kaitlyn Weeber. "Synthesis of Cyanoacetyl Oxazolidinones." Synthesis 44, no. 13 (2012): 1993–96. http://dx.doi.org/10.1055/s-0031-1291123.

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11

Davies, H., and R. Reddy. "Enantioselective Synthesis of Oxazolidinones." Synfacts 2007, no. 1 (2007): 0020. http://dx.doi.org/10.1055/s-2006-955744.

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12

Shinabarger, D. L., K. R. Marotti, R. W. Murray, et al. "Mechanism of action of oxazolidinones: effects of linezolid and eperezolid on translation reactions." Antimicrobial Agents and Chemotherapy 41, no. 10 (1997): 2132–36. http://dx.doi.org/10.1128/aac.41.10.2132.

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The oxazolidinones are a new class of synthetic antibiotics with good activity against gram-positive pathogenic bacteria. Experiments with a susceptible Escherichia coli strain, UC6782, demonstrated that in vivo protein synthesis was inhibited by both eperezolid (formerly U-100592) and linezolid (formerly U-100766). Both linezolid and eperezolid were potent inhibitors of cell-free transcription-translation in E. coli, exhibiting 50% inhibitory concentrations (IC50s) of 1.8 and 2.5 microM, respectively. The ability to demonstrate inhibition of in vitro translation directed by phage MS2 RNA was

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13

M, Heravi; Majid, and V. Zadsirjan. "Oxazolidinones as chiral auxiliaries in the asymmetric 1,4-conjugate addition reaction applied to the total synthesis of natural products: A supplemental mini-review." Current Organic Synthesis 15, no. 1 (2018): 3–20. https://doi.org/10.2174/1570179414666170601115831.

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Background: The most frequently used chiral auxiliaries, oxazolidinones (Evans’ oxazolidinones) have been employed in 1,4-congugate addition reactions to α,β-unsaturated carbonyl compounds. Supplementary to our previous reports in this mini-review, we attempted to underscore the applications of this strategy in a step (steps) in the total synthesis of some naturally occurring compounds exhibiting diverse biological activities. Objective: In this mini-review, we try to underscore the applications of oxazolidinones (Evans’ oxazolidi-nones) in 1,4-congugate addition reactio

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14

Brickner, Steven J. "Oxazolidinone Antibacterial Agents." Current Pharmaceutical Design 2, no. 2 (1996): 175–94. http://dx.doi.org/10.2174/1381612802666220921173820.

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The oxazolidinones are a new class of synthetic antibacterial agents. These compounds demonstrate potent in vitro and in vivo activity against important human pathogens, including multiple antibiotic-resistant strains of gram positive organisms including the staphylococci, streptococci, and enterococci. The oxazolidinones have a novel mechanism of action, inhibiting bacterial protein synthesis at a very early step prior to initiation. Literature disclosures have described the inability to detect in vitro bacterial resistance development to the oxazolidinones. Only the (S)-enantiomer is active;

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15

Demir, Esra, Ozlem Sari, Yasin Çetinkaya, Ufuk Atmaca, Safiye Sağ Erdem, and Murat Çelik. "One-pot synthesis of oxazolidinones and five-membered cyclic carbonates from epoxides and chlorosulfonyl isocyanate: theoretical evidence for an asynchronous concerted pathway." Beilstein Journal of Organic Chemistry 16 (July 21, 2020): 1805–19. http://dx.doi.org/10.3762/bjoc.16.148.

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The one-pot reaction of chlorosulfonyl isocyanate (CSI) with epoxides having phenyl, benzyl and fused cyclic alkyl groups in different solvents under mild reaction conditions without additives and catalysts was studied. Oxazolidinones and five-membered cyclic carbonates were obtained in ratios close to 1:1 in the cyclization reactions. The best yields of these compounds were obtained in dichloromethane (DCM). Together with 16 known compounds, two novel oxazolidinone derivatives and two novel cyclic carbonates were synthesized with an efficient and straightforward method. Compared to the existi

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16

Aurelio, Luigi, Robert T. C. Brownlee, Andrew B. Hughes, and Brad E. Sleebs. "The Facile Production of N-Methyl Amino Acids via Oxazolidinones." Australian Journal of Chemistry 53, no. 5 (2000): 425. http://dx.doi.org/10.1071/ch99082.

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A range of oxazolidinones derived from N-carbamoyl α-amino acids were prepared by an efficient method as key intermediates in the synthesis of N-methyl amino acids and peptides. The method was readily applied to most α-amino acids except those with basic side chains. The oxazolidinones were converted by reductive cleavage into N-methyl α-amino acids.

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17

Lin, A. H., R. W. Murray, T. J. Vidmar, and K. R. Marotti. "The oxazolidinone eperezolid binds to the 50S ribosomal subunit and competes with binding of chloramphenicol and lincomycin." Antimicrobial Agents and Chemotherapy 41, no. 10 (1997): 2127–31. http://dx.doi.org/10.1128/aac.41.10.2127.

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The oxazolidinones are a novel class of antibiotics that act by inhibiting protein synthesis. It as been reported that the drug exerts its primary activity on the initiation phase of translation. In order to study the possibility of direct interaction between the drug and the ribosome, we have developed a binding assay using 14C-labelled eperezolid (PNU-100592; formerly U-100592). Eperezolid binds specifically to the 50S ribosomal subunit of Escherichia coli. The specific binding of eperezolid is dose dependent and is proportional to the ribosome concentrations. Scatchard analysis of the bindi

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18

Weeber, Kaitlyn M., and Jacob B. Schwarz. "ChemInform Abstract: Synthesis of Cyanoacetyl Oxazolidinones." ChemInform 43, no. 42 (2012): no. http://dx.doi.org/10.1002/chin.201242133.

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19

Shang, Jianpeng, Zuopeng Li, Caina Su, Yong Guo, and Youquan Deng. "Efficient synthesis of 2-oxazolidinones from epoxides and carbamates catalyzed by amine-functionalized ionic liquids." RSC Advances 5, no. 88 (2015): 71765–69. http://dx.doi.org/10.1039/c5ra09838f.

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20

Wang, Peixue, Qinghe Li, Shimin Liu, and Youquan Deng. "Converting urea into high value-added 2-oxazolidinones under solvent-free conditions." RSC Advances 6, no. 97 (2016): 94382–86. http://dx.doi.org/10.1039/c6ra21809a.

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21

Zurenko, G. E., B. H. Yagi, R. D. Schaadt, et al. "In vitro activities of U-100592 and U-100766, novel oxazolidinone antibacterial agents." Antimicrobial Agents and Chemotherapy 40, no. 4 (1996): 839–45. http://dx.doi.org/10.1128/aac.40.4.839.

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Oxazolidinones make up a relatively new class of antimicrobial agents which possess a unique mechanism of bacterial protein synthesis inhibition. U-100592 (S)-N-[[3-[3-fluoro-4-[4-(hydroxyacetyl)-1-piperazinyl]- phenyl]-2-oxo-5-oxazolidinyl]methyl]-acetamide and U-100766 (S)-N-[[3-[3-fluoro-4-(4-morpholinyl)phenyl]- 2-oxo-5-oxazolidinyl]methyl]-acetamide are novel oxazolidinone analogs from a directed chemical modification program. MICs were determined for a variety of bacterial clinical isolates; the respective MICs of U-100592 and U-100766 at which 90% of isolates are inhibited were as follo

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22

Xiong, Liqun, Patricia Kloss, Stephen Douthwaite, et al. "Oxazolidinone Resistance Mutations in 23S rRNA ofEscherichia coli Reveal the Central Region of Domain V as the Primary Site of Drug Action." Journal of Bacteriology 182, no. 19 (2000): 5325–31. http://dx.doi.org/10.1128/jb.182.19.5325-5331.2000.

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ABSTRACT Oxazolidinone antibiotics inhibit bacterial protein synthesis by interacting with the large ribosomal subunit. The structure and exact location of the oxazolidinone binding site remain obscure, as does the manner in which these drugs inhibit translation. To investigate the drug-ribosome interaction, we selected Escherichia colioxazolidinone-resistant mutants, which contained a randomly mutagenized plasmid-borne rRNA operon. The same mutation, G2032 to A, was identified in the 23S rRNA genes of several independent resistant isolates. Engineering of this mutation by site-directed mutage

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23

Heravi, Majid M., Vahideh Zadsirjan, and Behnaz Farajpour. "Applications of oxazolidinones as chiral auxiliaries in the asymmetric alkylation reaction applied to total synthesis." RSC Advances 6, no. 36 (2016): 30498–551. http://dx.doi.org/10.1039/c6ra00653a.

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24

Gu, Zheng-Yang, and Ji-Bao Xia. "[3 + 1 + 1] cyclization of vinyl oxiranes with azides and CO by tandem palladium catalysis: efficient synthesis of oxazolidinones." Organic Chemistry Frontiers 8, no. 15 (2021): 4112–17. http://dx.doi.org/10.1039/d1qo00591j.

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25

Baruah, Shyamal, Amrit Puzari, Farhana Sultana, and Jayanta Barman. "Synthesis, Characterization and Evaluation of Antimicrobial Properties of (R)-(-)-4-Phenyl-2 Oxazolidinone Based Azetidinones." Anti-Infective Agents 16, no. 2 (2018): 104–13. http://dx.doi.org/10.2174/2211352516666180619153317.

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Introduction: A series of (R)-(-)-4-Phenyl-2 oxazolidinone based azetidinones (4a-i) were synthesized from the reaction of (2-Oxo-4-phenyl-oxazolidin-3-yl) acetic acid with aromatic imines (3a-i) in the presence of Thionyl chloride and Triethylamine as a base. Methods: The transformation proceeds through the formation of acid chloride to ketene which finally forms the azetidinones through [2+2] cycloaddition with aromatic imines. Products obtained were screened to evaluate their antibacterial activity with respect to known bacteria like Escherichia Coli (E. Coli) and Bacillus subtilis. Results

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26

Kalia, Vandana, Rajni Miglani, Kedar P. Purnapatre, et al. "Mode of Action of Ranbezolid against Staphylococci and Structural Modeling Studies of Its Interaction with Ribosomes." Antimicrobial Agents and Chemotherapy 53, no. 4 (2008): 1427–33. http://dx.doi.org/10.1128/aac.00887-08.

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ABSTRACT Oxazolidinones are known to inhibit protein biosynthesis and act against a wide spectrum of gram-positive bacteria. A new investigational oxazolidinone, ranbezolid, inhibited bacterial protein synthesis in Staphylococcus aureus and Staphylococcus epidermidis. In S. epidermidis, ranbezolid showed inhibition of cell wall and lipid synthesis and a dose-dependent effect on membrane integrity. A kill-kinetics study showed that ranbezolid was bactericidal against S. epidermidis. In vitro translation of the luciferase gene done using bacterial and mammalian ribosomes indicated that ranbezoli

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27

Ghosh, Arun K., Alessandro Grillo, Satish Kovela, and Margherita Brindisi. "Asymmetric Diels–Alder reaction of 3-(acyloxy)acryloyl oxazolidinones: optically active synthesis of a high-affinity ligand for potent HIV-1 protease inhibitors." RSC Advances 9, no. 71 (2019): 41755–63. http://dx.doi.org/10.1039/c9ra10178k.

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28

Xia, Shumei, Yu Song, Xuedong Li, Hongru Li, and Liang-Nian He. "Ionic Liquid-Promoted Three-Component Domino Reaction of Propargyl Alcohols, Carbon Dioxide and 2-Aminoethanols: A Thermodynamically Favorable Synthesis of 2-Oxazolidinones." Molecules 23, no. 11 (2018): 3033. http://dx.doi.org/10.3390/molecules23113033.

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To circumvent the thermodynamic limitation of the synthesis of oxazolidinones starting from 2-aminoethanols and CO2 and realize incorporation CO2 under atmospheric pressure, a protic ionic liquid-facilitated three-component reaction of propargyl alcohols, CO2 and 2-aminoethanols was developed to produce 2-oxazolidinones along with equal amount of α-hydroxyl ketones. The ionic liquid structure, reaction temperature and reaction time were in detail investigated. And 15 mol% 1,5,7-triazabicylo[4.4.0]dec-5-ene ([TBDH][TFE]) trifluoroethanol was found to be able to synergistically activate the subs

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29

Li, Wei, Marco Wollenburg, and Frank Glorius. "Enantioselective synthesis of 2-oxazolidinones by ruthenium(ii)–NHC-catalysed asymmetric hydrogenation of 2-oxazolones." Chemical Science 9, no. 29 (2018): 6260–63. http://dx.doi.org/10.1039/c8sc01869c.

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30

Logan, Matthew W., Yuen A. Lau, Yongsheng Zheng, et al. "Heterogeneous photoredox synthesis of N-hydroxy-oxazolidinones catalysed by metal–organic frameworks." Catalysis Science & Technology 6, no. 14 (2016): 5647–55. http://dx.doi.org/10.1039/c6cy00054a.

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31

Arshadi, Sattar, Alireza Banaei, Saeideh Ebrahimiasl, Aazam Monfared, and Esmail Vessally. "Solvent-free incorporation of CO2 into 2-oxazolidinones: a review." RSC Advances 9, no. 34 (2019): 19465–82. http://dx.doi.org/10.1039/c9ra00551j.

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32

Renslo, Adam R., Priyadarshini Jaishankar, Revathy Venkatachalam, et al. "Conformational Constraint in Oxazolidinone Antibacterials. Synthesis and Structure−Activity Studies of (Azabicyclo[3.1.0]hexylphenyl)oxazolidinones." Journal of Medicinal Chemistry 48, no. 15 (2005): 5009–24. http://dx.doi.org/10.1021/jm058204j.

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33

Das, Biswajit, A. V. S. Rajarao, Sonali Rudra, et al. "Synthesis and biological activity of novel oxazolidinones." Bioorganic & Medicinal Chemistry Letters 19, no. 22 (2009): 6424–28. http://dx.doi.org/10.1016/j.bmcl.2009.09.054.

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34

Baldwin, Jack E., та E. Lee. "Synthesis of bicyclic γ-lactams via oxazolidinones". Tetrahedron 42, № 23 (1986): 6551–54. http://dx.doi.org/10.1016/s0040-4020(01)88118-7.

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35

Lebel, Hélène, Laura Mamani Laparra, Maroua Khalifa, et al. "Synthesis of oxazolidinones: rhodium-catalyzed C–H amination of N-mesyloxycarbamates." Organic & Biomolecular Chemistry 15, no. 19 (2017): 4144–58. http://dx.doi.org/10.1039/c7ob00378a.

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36

Toda, Yasunori, Shoya Tanaka, Shuto Gomyou, Ayaka Kikuchi, and Hiroyuki Suga. "4-Hydroxymethyl-substituted oxazolidinone synthesis by tetraarylphosphonium salt-catalyzed reactions of glycidols with isocyanates." Chemical Communications 55, no. 41 (2019): 5761–64. http://dx.doi.org/10.1039/c9cc01983a.

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37

Casado-Sánchez, Antonio, Pablo Domingo-Legarda, Silvia Cabrera, and José Alemán. "Visible light photocatalytic asymmetric synthesis of pyrrolo[1,2-a]indoles via intermolecular [3+2] cycloaddition." Chemical Communications 55, no. 75 (2019): 11303–6. http://dx.doi.org/10.1039/c9cc05838a.

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The asymmetric synthesis of pyrrolo[1,2-a]indoles is developed through a [3+2] cycloaddition between silyl-indole derivatives and α,β-unsaturated N-acyl oxazolidinones by merging photocatalysis and Lewis acid catalysis.

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38

Galetto, Fábio Z., Cleiton da Silva, Ricardo I. M. Beche та ін. "Decarboxylative ring-opening of 2-oxazolidinones: a facile and modular synthesis of β-chalcogen amines". RSC Advances 12, № 53 (2022): 34496–502. http://dx.doi.org/10.1039/d2ra06070a.

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This study includes a new protocol for the synthesis of primary and secondary β-chalcogen amines (Se, Te and S) from the ring-opening reaction of non-activated 2-oxazolidinones with chalcogenolate anions.

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39

Hu, Yulin, Zongyan Tang, and Xiaobing Liu. "Novel and Highly Efficient Carboxylative Cyclization of CO2 to 2-Oxazolidinones Using Nano-SiO2-Supported Ionic Liquid Sustainable Catalysts." Molecules 30, no. 3 (2025): 633. https://doi.org/10.3390/molecules30030633.

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The conversion of CO2 into 2-oxazolidinones through carboxylative cyclization with propargylic amines is considered an effective method for utilizing waste gas as a sustainable C1 resource and mitigating the greenhouse effect. In this context, a series of nano-SiO2-supported ionic liquids have been prepared and developed as multifunctional heterogeneous catalysts in the carboxylative cyclization of propargylic amines with CO2. The catalyst IL-SbF6@nano-SiO2 demonstrated a high compatibility with various propargylic amines, achieving excellent yields (90~98%) for the desired 2-oxazolidinones un

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40

Scrimin, Paolo, Giorgio Cavicchioni, Ferruccio D'Angeli, Amiram Goldblum, and Flavio Maran. "Chemistry of 2-bromo-2-methylpropanamides. Synthesis and solvolytic behaviour of oxazolidinones and spiro-oxazolidinones." Journal of the Chemical Society, Perkin Transactions 1, no. 1 (1988): 43. http://dx.doi.org/10.1039/p19880000043.

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41

Diaz, Gaspar, Michelle de Freitas, Maria Ricci-Silva, and Marisa Diaz. "Easy Access to Evans’ Oxazolidinones. Stereoselective Synthesis and Antibacterial Activity of a New 2-Oxazolidinone Derivative." Molecules 19, no. 6 (2014): 7429–39. http://dx.doi.org/10.3390/molecules19067429.

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42

Hua-Yue, Wu, Ding Jin-Chang, and Liu Yun-Kui. "Samarium triiodide catalyzed cycloaddition of epoxides with isocyanates : a facile synthesis of oxazolidinones." Journal of Indian Chemical Society Vol. 80, Jan 2003 (2003): 36–37. https://doi.org/10.5281/zenodo.5835576.

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Department of Chemistry. Wenzhou Normal College, Wenzhou 325027, P. R. China <em>E-mail :</em> hywu3@ 163.com Fax : 86-577-88339081 Department of Chemistry, Zhejiang University (Campus Xixi), Hangzhou 310028, P.R. China <em>Manuscript received 6 May 2002.accepted 6 September 2002</em> Oxazolidinones were synthesized in high yields via cycloaddition of epoxides with isocyanates catalyzed by samarium triiodide.

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43

Beattie, Christopher, and Michael North. "VanadiumV(salen) catalysed synthesis of oxazolidinones from epoxides and isocyanates." RSC Adv. 4, no. 59 (2014): 31345–52. http://dx.doi.org/10.1039/c4ra04427d.

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The combination of a vanadium<sup>V</sup>(salen) complex V<sup>+</sup>O(salen) EtOSO<sub>3</sub><sup>−</sup> and tetrabutylammonium bromide forms a highly active catalyst system for the reaction between epoxides and isocyanates leading to oxazolidinones.

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44

Hughes, Andrew B., та Brad E. Sleebs. "Synthesis of New β-Amino Acids via 5-Oxazolidinones and the Arndt - Eistert Procedure". Australian Journal of Chemistry 58, № 11 (2005): 778. http://dx.doi.org/10.1071/ch05199.

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N-Methyl β-amino acids are potentially useful amino acid derivatives for incorporation in lead peptide therapeutics. The syntheses of five such compounds are presented. Their synthesis via 6-oxazinanones was low yielding. Alternatively, reductive cleavage of a 5-oxazolidinone gave the N-methyl α-amino acid, which was then homologated via an Arndt–Eistert procedure in high yield to give the N-methyl β-amino acid.

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45

Wang, Guijun. "Synthesis and Antibacterial Properties of Oxazolidinones and Oxazinanones." Anti-Infective Agents in Medicinal Chemistry 7, no. 1 (2008): 32–49. http://dx.doi.org/10.2174/187152108783329771.

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Song, Qing-Wen, Ya-Nan Zhao, Liang-Nian He, Jian Gao, and Zhen-Zhen Yang. "Synthesis of Oxazolidinones/Polyurethanes from Aziridines and CO2." Current Catalysise 1, no. 2 (2012): 107–24. http://dx.doi.org/10.2174/2211544711201020107.

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Kumar, Pankaj, Jennifer Fernandes, and Abhishek Kumar. "Synthesis and Antimicrobial Evaluation of Substituted Oxazolidinones Moieties." Research Journal of Pharmacy and Technology 10, no. 1 (2017): 98. http://dx.doi.org/10.5958/0974-360x.2017.00023.3.

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Liu, Jidong, Baoyuan He, Aizhen Yu, and Weicheng Zhou. "Synthesis and Antibacterial Activity of Substituted Oxotriazolylphenyl Oxazolidinones." Chemical Biology & Drug Design 70, no. 1 (2007): 65–69. http://dx.doi.org/10.1111/j.1747-0285.2007.00531.x.

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Rmedi, Hamdi. "Design and synthesis of fused cyclic sulfamides-oxazolidinones." Tetrahedron 75, no. 10 (2019): 1337–42. http://dx.doi.org/10.1016/j.tet.2019.01.046.

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50

Phillips, O. A., E. E. Udo, A. A. M. Ali, and N. Al-Hassawi. "Synthesis and antibacterial activity of 5-substituted oxazolidinones." Bioorganic & Medicinal Chemistry 11, no. 1 (2003): 35–41. http://dx.doi.org/10.1016/s0968-0896(02)00423-6.

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