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Journal articles on the topic 'Tetrahydropyridine derivatives'

Author: Grafiati

Published: 5 June 2025

Last updated: 1 August 2025

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1

W. Ardley, Tiffany. "The Chemistry and Pharmacology of Tetrahydropyridines: Part 2." Clinical Medical Reviews and Reports 5, no. 01 (2023): 01–16. https://doi.org/10.31579/2690-8794/135.

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Tetrahydropyridines (THPs) have sparked notable interest as an auspicious heterocyclic moiety. Existing in distinct structural isomers including 1,2,3,4-tetrahydropyridine, 1,2,3,6-tetrahydropyridine, 2,3,4,5-tetrahydropyridine, its presence has been identified in both natural products and synthetic pharmaceutical agents. Many THP-containing compounds have been synthesized by the inspiration of known bioactive natural products and have been found to possess biologically active properties. For this reason, more innovative methods have been developed for the synthesis of substituted-tetrahydropy

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2

Šilhánková, Alexandra, Dagmar Davidová, Michaela Šputová, et al. "Photoaddition of alcohols to some 1,2,3,6-tetrahydropyridines." Collection of Czechoslovak Chemical Communications 52, no. 5 (1987): 1298–304. http://dx.doi.org/10.1135/cccc19871298.

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Photochemical addition of methanol to 1,2,3,6-tetrahydropyridine derivatives Ia, Ib, Id-Ii and III afforded methoxypiperidines IIa-IIg and IV as Markovnikov type addition products. Reduction of 4-methyl-1-(2-propenyl)pyridinium bromide with sodium borohydride yielded 4-methyl-1-(2-propenyl)-1,2,3,6-tetrahydropyridine (Ig).

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3

Li, Jun, Xiaochen Chi, Long Meng, et al. "Palladium-catalyzed heck-type cascade cyclization of (Z)-1-iodo-1,6-dienes with N-tosyl hydrazones." Organic & Biomolecular Chemistry 16, no. 40 (2018): 7356–60. http://dx.doi.org/10.1039/c8ob01821a.

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4

Berti, Francesco, Federico Malossi, Fabio Marchetti, and Mauro Pineschi. "A highly enantioselective Mannich reaction of aldehydes with cyclic N-acyliminium ions by synergistic catalysis." Chemical Communications 51, no. 71 (2015): 13694–97. http://dx.doi.org/10.1039/c5cc04416b.

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A novel enantioselective synthesis of carbamoyl isoquinoline and tetrahydropyridine derivatives is accomplished using matched combinations of Lewis or Brønsted acids and secondary amine organocatalysts.

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5

Jahanshahi, R., and B. Akhlaghinia. "Cu(ii)-grafted SBA-15 functionalized S-methylisothiourea aminated epibromohydrin (SBA-15/E-SMTU-CuII): a novel and efficient heterogeneous mesoporous catalyst." New Journal of Chemistry 41, no. 15 (2017): 7203–19. http://dx.doi.org/10.1039/c7nj00849j.

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6

Jiang, Yu, Xiang-Ying Tang, and Min Shi. "A Rh-catalyzed 1,2-sulfur migration/aza-Diels–Alder cascade initiated by aza-vinyl carbenoids from sulfur-tethered N-sulfonyl-1,2,3-triazoles." Chemical Communications 51, no. 11 (2015): 2122–25. http://dx.doi.org/10.1039/c4cc08829h.

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A novel Rh(ii) catalyzed intramolecular 1,2-sulfur migration/intermolecular aza-Diels–Alder cascade of sulfur-tethered N-sulfonyl-1,2,3-triazoles has been developed, efficiently affording sulfur-containing tetrahydropyridine derivatives.

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7

Zhu, Yu-Jie, Xiao-Feng Guo, Zhi-Jin Fan, et al. "Approach to thiazole-containing tetrahydropyridines via Aza–Rauhut–Currier reaction and their potent fungicidal and insecticidal activity." RSC Advances 6, no. 113 (2016): 112704–11. http://dx.doi.org/10.1039/c6ra24342h.

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Insecticidal and fungicidal active thiazole-containing tetrahydropyridine derivatives with accurately predicted 3D QSAR model againstAphis LaburniKaltenbach and predicted potential anti-fungus target of fumarate reductase without cross resistance were synthesized.

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8

Shakurova, Elvira R., and Lyudmila V. Parfenova. "Synthesis of N-Heterocyclic Analogues of 28-O-Methyl Betulinate, and Their Antibacterial and Antifungal Properties." Molbank 2020, no. 1 (2019): M1100. http://dx.doi.org/10.3390/m1100.

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The paper presents the results on the one-pot pyridine quaternization using betulinic 28-O-methyl ester (1) and Tempo+Br3− cation followed by reduction of the resulting salt (2) to 1,2,5,6-tetrahydropyridine derivative (3). The structures of new compounds are confirmed by means of 1D and 2D-NMR spectroscopy, as well as MALDI TOF/TOF spectrometry. The derivatives 2 and 3 are active against S. aureus at the minimum inhibitory concentration (MIC) of 4 μg/mL and 16 μg/mL, correspondingly.

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9

Ivanova, Evgeniya V., Nikolay N. Zhukov, Irina I. Surova, Maria B. Nikishina, Loik G. Mukhtorov, and Yuri M. Atroshchenko. "STUDY OF THE EFFECT OF NEW 6-R-3,5-DINITRO-1,2,3,4-TETRAHYDROPYRIDINES ON THE ACCUMULATION OF PHOTOSYNTHETIC PIGMENTS AND ASCORBIC ACID IN PLANT TISSUES." Siberian Journal of Life Sciences and Agriculture 14, no. 6 (2022): 372–87. http://dx.doi.org/10.12731/2658-6649-2022-14-6-372-387.

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Background. The problem of finding new effective plant protection products remains an urgent task of modern agrochemistry. It is known that tetrahydropyridine derivatives exhibit a broad spectrum of biological activity, including fungicidal activity. However, compounds with potential biological activity can also be highly toxic to humans, cultivated crops, and the environment as a whole, so it is necessary to study their environmental safety. The content of photosynthetic pigments and ascorbic acid are one of the most important biochemical indicators of plant response to environmental stress f

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10

Gizur, T., B. Kiss, K. Harsányi, et al. "Novel 1,2,3,6-tetrahydropyridine derivatives with potent antihypoxic activity." European Journal of Medicinal Chemistry 29, no. 5 (1994): 349–55. http://dx.doi.org/10.1016/0223-5234(94)90059-0.

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11

Braña, Miguel F., Marina Morán, María Jesús Pérez de Vega, and Isabel Pita-Romero. "Enediynes as Antitumor Compounds: Synthesis of Tetrahydropyridine Derivatives." Journal of Organic Chemistry 61, no. 4 (1996): 1369–74. http://dx.doi.org/10.1021/jo951188l.

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12

Csekö, József, H. Olga Hankovszky, and Kálmán Hideg. "Synthesis of novel, highly reactive 1-oxyl-2,2,6,6-tetramethyl-1,2,5,6-tetrahydropyridine derivatives." Canadian Journal of Chemistry 63, no. 4 (1985): 940–43. http://dx.doi.org/10.1139/v85-156.

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New multipurpose spin labels and synthons can be synthesized from 1-oxyl-2,2,6,6-tetramethyl-1,2,5,6-tetrahydropyridine-4-carboxylic acid (1). Either 1, its pentafluorophenylester (2), or acylcarbonate (3) (prepared from 1 with ethyl chloroformate) can be reduced to 1-oxyl-2,2,6,6-tetramethyl-4-hydroxymethyl-1,2,5,6-tetrahydropyridine (4). The methanesulfonate (6) and the bromo compound (7) are highly reactive alkylating reagents due, in large part, to the allylic linkage in the nitroxide ring. The latter can be reacted with KSSO2CH3 to give methanethiolsulfonate (9). A novel side chain spin-l

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13

Bogdanowicz-Szwed, Krystyna, та Małgorzata Krasodomska. "Efficient Synthesis of Polyfunctionalised Pyridines by Conjugate Addition of 2-Thienylcarbonyl (Thioacetanilides) to αβ-Unsaturated Nitriles". Journal of Chemical Research 2002, № 4 (2002): 149–50. http://dx.doi.org/10.3184/030823402103171645.

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Conjugate addition of 2-thienylcarbonyl(thioacetanilides) (1) to arylmethylenemalononitriles (2) yielded 2-amino-1,4-diaryl-5-(2-thienylcarbonyl)-6-thioxo-1,4,5,6-tetrahydropyridine-3-carbonitriles (4), which when oxidised with HgO gave functionalised 2,6-dioxopiperidines (6), whereas with MCPBA they afforded pyrido[2,1-b]benzothiazole-2-carbonitrile derivatives (7).

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14

Uhrín, Dušan, та Bohumil Proksa. "Study of conformation of α-narcotine N-oxide and related compounds". Collection of Czechoslovak Chemical Communications 54, № 2 (1989): 498–505. http://dx.doi.org/10.1135/cccc19890498.

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Conformation of quaternary derivatives of (-)-α-narcotine (I) in solution was investigated using α-narcotine N-oxide hydrochloride (IV) as the model compound. In solution, compound IV exists predominantly in the form with torsion angle H-C(1)-C(9)-H of about 270° and with half-chair conformation of the isoquinoline tetrahydropyridine ring.

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15

O'Callaghan, Conor N., and T. Brian H. McMurry. "Conversion by Hydrazinolysis of Tetrahydropyridine Ester Derivatives into 1-Ammoniotetrahydropyridine 6-oxide Derivatives." Journal of Chemical Research, no. 9 (1998): 491. http://dx.doi.org/10.1039/a801665h.

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16

Horáčková, Jaroslava, and Vojeslav Štěrba. "Coupling Kinetics of Benzenediazonium Ions with 2,6-Dioxo-3-(p-substituted phenylhydrazono)-1,2,3,6-tetrahydropyridine-4-carboxylic Acid." Collection of Czechoslovak Chemical Communications 57, no. 9 (1992): 1915–27. http://dx.doi.org/10.1135/cccc19921915.

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The kinetics have been measured of the reactions of 4-nitro-, 4-chloro-, and 4-methoxybenzenediazonium ions with substituted phenylazo derivatives of citrazinic acid in buffer solutions, and the pKa values of the corresponding monoazo and bisazo compounds have been estimated. The reactions of 4-nitrobenzenediazonium ion with 4-chloro- and 4-methoxyphenylazo derivatives and of 4-chlorobenzenediazonium ion with 4-methoxyphenylazo derivative were accompanied by a partial replacement of the substituted phenylazo group by the 4-nitro- and 4-chlorophenylazo groups, respectively. The reactions of 4-c

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17

Hall, Larry, Sam Murray, Kay Castagnoli, and Neal Castagnoli. "Studies on 1,2,3,6-tetrahydropyridine derivatives as potential monoamine oxidase inactivators." Chemical Research in Toxicology 5, no. 5 (1992): 625–33. http://dx.doi.org/10.1021/tx00029a006.

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18

Gwaltney, Stephen L., Stephen J. O'Connor, Lissa T. J. Nelson, et al. "Aryl tetrahydropyridine inhibitors of farnesyltransferase: glycine, phenylalanine and histidine derivatives." Bioorganic & Medicinal Chemistry Letters 13, no. 7 (2003): 1359–62. http://dx.doi.org/10.1016/s0960-894x(03)00095-7.

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19

Plate, Ralf, Marc J. M. Plaum, Thijs de Boer, John S. Andrews, Duncan R. Rae, and Sam Gibson. "Synthesis and muscarinic activities of 3-(pyrazolyl)-1,2,5,6-tetrahydropyridine derivatives." Bioorganic & Medicinal Chemistry 4, no. 2 (1996): 227–37. http://dx.doi.org/10.1016/0968-0896(96)00001-6.

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20

BRANA, M. F., M. MORAN, M. J. PEREZ DE VEGA, and I. PITA-ROMERO. "ChemInform Abstract: Enediynes as Antitumor Compounds: Synthesis of Tetrahydropyridine Derivatives." ChemInform 27, no. 30 (2010): no. http://dx.doi.org/10.1002/chin.199630303.

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21

GIZUR, T., B. KISS, K. HARSANYI, et al. "ChemInform Abstract: Novel 1,2,3,6-Tetrahydropyridine Derivatives with Potent Antihypoxic Activity." ChemInform 25, no. 43 (2010): no. http://dx.doi.org/10.1002/chin.199443163.

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22

Maret, Gérard, Bernard Testa, Peter Jenner, Nabil El Tayar, and Pierre-Alain Carrupt. "The MPTP Story: Mao Activates Tetrahydropyridine Derivatives to Toxins Causing Parkinsonism." Drug Metabolism Reviews 22, no. 4 (1990): 291–332. http://dx.doi.org/10.3109/03602539009041087.

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23

Shvekhgeimer, Mai-Genrikh A. "2,3,4,5-Tetrahydropyridine (Δ1-piperideine) and its derivatives. Synthesis and chemical properties". Russian Chemical Reviews 67, № 12 (1998): 1031–60. http://dx.doi.org/10.1070/rc1998v067n12abeh000434.

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24

Yankin, Andrei N., and Maksim V. Dmitriev. "Nickel complexes as efficient catalysts in multicomponent synthesis of tetrahydropyridine derivatives." Synthetic Communications 50, no. 22 (2020): 3481–89. http://dx.doi.org/10.1080/00397911.2020.1803357.

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25

Kita, Yoshio, Hirofumi Maekawa, Yasuhiro Yamasaki, and Ikuzo Nishiguchi. "Selective and facile electroreductive synthesis of dihydro- and tetrahydropyridine dicarboxylic acid derivatives." Tetrahedron Letters 40, no. 49 (1999): 8587–90. http://dx.doi.org/10.1016/s0040-4039(99)01789-x.

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26

Wang, Jiao-dan, Qiao-li Lin, Jun Qiu, et al. "NO2-Fe(III)PcCl@C -catalyzed one-pot synthesis of tetrahydropyridine derivatives." Russian Journal of General Chemistry 87, no. 4 (2017): 821–28. http://dx.doi.org/10.1134/s1070363217040259.

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27

Eda, Masahiro, and Mark J. Kurth. "Solid-phase Zincke route to pyridinium, tetrahydropyridine, and piperidine derivatives: vesamicol analogs." Tetrahedron Letters 42, no. 11 (2001): 2063–68. http://dx.doi.org/10.1016/s0040-4039(00)02351-0.

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28

Zuo, Zeping, Miaomiao Chen, Xiaoni Shao, et al. "Design and biological evaluation of tetrahydropyridine derivatives as novel human GPR119 agonists." Bioorganic & Medicinal Chemistry Letters 30, no. 4 (2020): 126855. http://dx.doi.org/10.1016/j.bmcl.2019.126855.

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29

Mochona, Bereket, and Kinfe K. Redda. "Synthesis of N-benzoylamino-1,2,3,6-tetrahydropyridine derivatives as potential anti-inflammatory agents." Journal of Heterocyclic Chemistry 44, no. 6 (2007): 1383–87. http://dx.doi.org/10.1002/jhet.5570440622.

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30

Araldi, Gian Luca, and Yu-Wen Hwang. "Development of Novel Fluorinated Polyphenols as Selective Inhibitors of DYRK1A/B Kinase for Treatment of Neuroinflammatory Diseases including Parkinson’s Disease." Pharmaceuticals 16, no. 3 (2023): 443. http://dx.doi.org/10.3390/ph16030443.

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Natural polyphenol derivatives such as those found in green tea have been known for a long time for their useful therapeutic activity. Starting from EGCG, we have discovered a new fluorinated polyphenol derivative (1c) characterized by improved inhibitory activity against DYRK1A/B enzymes and by considerably improved bioavailability and selectivity. DYRK1A is an enzyme that has been implicated as an important drug target in various therapeutic areas, including neurological disorders (Down syndrome and Alzheimer’s disease), oncology, and type 2 diabetes (pancreatic β-cell expansion). Systematic

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31

Jílek, Jiří, Miroslav Rajšner, Vladimír Valenta, et al. "Synthesis of piperidine derivatives as potential analgetic agents." Collection of Czechoslovak Chemical Communications 55, no. 7 (1990): 1828–53. http://dx.doi.org/10.1135/cccc19901828.

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Reaction of N-(1-(2-phenylethyl)-4-piperidinyl)propionanilide (I) with phosphorus pentasulfide gave the thioamide VI. Acylation of N-(1-(2-phenylethyl)-4-piperidinyl)aniline with 2-(methoxy)acetic and 2-(methylthio)acetic anhydrides afforded the amides II and III. Treatment of 4-anilino-1-benzylpiperidine-4-methanol with thionyl chloride gave the spirocyclic sulfurous acid ester amide XIV. Reduction of the hydrochloride of ethyl 3-(1-ethoxycarbonyl-4-phenylimino-3-piperidinyl)propionate (XXII) with sodium cyanoborohydride gave the perhydro-1,6-naphthyridine derivative XIX, a model compound in

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32

Nakao, Akira, Nobuyuki Ohkawa, Takayoshi Nagasaki, et al. "Tetrahydropyridine derivatives with inhibitory activity on the production of proinflammatory cytokines: Part 1." Bioorganic & Medicinal Chemistry Letters 19, no. 16 (2009): 4607–10. http://dx.doi.org/10.1016/j.bmcl.2009.06.094.

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33

Nakao, Akira, Nobuyuki Ohkawa, Takayoshi Nagasaki, et al. "Tetrahydropyridine derivatives with inhibitory activity on the production of proinflammatory cytokines: Part 2." Bioorganic & Medicinal Chemistry Letters 20, no. 8 (2010): 2435–37. http://dx.doi.org/10.1016/j.bmcl.2010.03.022.

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34

Shakurova, Elvira R., Elena V. Salimova, Ekaterina S. Mescheryakova, and Lyudmila V. Parfenova. "One-pot synthesis of quaternary pyridinium salts and tetrahydropyridine derivatives of fusidane triterpenoids." Chemistry of Heterocyclic Compounds 55, no. 12 (2019): 1204–10. http://dx.doi.org/10.1007/s10593-019-02602-6.

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35

Nakao, Akira, Nobuyuki Ohkawa, Takayoshi Nagasaki, et al. "Tetrahydropyridine derivatives with inhibitory activity on the production of proinflammatory cytokines: Part 3." Bioorganic & Medicinal Chemistry Letters 20, no. 16 (2010): 4774–78. http://dx.doi.org/10.1016/j.bmcl.2010.06.122.

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36

Shvekhgeimer, M. G. A. "ChemInform Abstract: 2,3,4,5-Tetrahydropyridine (Δ1-Piperideine) and Its Derivatives. Synthesis and Chemical Properties". ChemInform 30, № 24 (2010): no. http://dx.doi.org/10.1002/chin.199924291.

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37

Wu, Yen-Ku, and Viresh H. Rawal. "Rapid construction of tetrahydropyridine scaffolds via formal imino Diels–Alder reactions of Schiff bases and Nazarov reagents." Organic & Biomolecular Chemistry 17, no. 39 (2019): 8827–31. http://dx.doi.org/10.1039/c9ob01880h.

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38

Sharma, Ganesh, and C. S. Sharma. "Tetrahydropyridine appended 8-aminoquinoline derivatives: Design, synthesis, in silico, and in vitro antimalarial studies." Bioorganic Chemistry 151 (October 2024): 107674. http://dx.doi.org/10.1016/j.bioorg.2024.107674.

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39

Shishkin, O. V. "Conformational analysis of 2-oxo-1,2,3,4,-tetrahydropyridine and its alkyl- and phenyl-substituted derivatives." Russian Chemical Bulletin 46, no. 9 (1997): 1510–12. http://dx.doi.org/10.1007/bf02502929.

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40

Aiello, Daniele, Hendrik Jonas, Anna Carbone, et al. "Synthesis and Antioxidative Properties of 1,2,3,4-Tetrahydropyridine Derivatives with Different Substituents in 4-Position." Molecules 27, no. 21 (2022): 7423. http://dx.doi.org/10.3390/molecules27217423.

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Natural products are an excellent source of inspiration for the development of new drugs. Among them, betalains have been extensively studied for their antioxidant properties and potential application as natural food dyes. Herein, we describe the seven-step synthesis of new betalamic acid analogs without carboxy groups in the 2- and 6-position with an overall yield of ~70%. The Folin–Ciocalteu assay was used to determine the antioxidant properties of protected intermediate 21. Additionally, the five-step synthesis of betalamic acid analog 35 with three ester moieties was performed. Using NMR t

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41

Aeluri, Raghunath, Manjula Alla, Vittal Rao Bommena, Ramalinga Murthy, and Nishant Jain. "Synthesis and Antiproliferative Activity of Polysubstituted Tetrahydropyridine and Piperidin-4-one-3-carboxylate Derivatives." Asian Journal of Organic Chemistry 1, no. 1 (2012): 71–79. http://dx.doi.org/10.1002/ajoc.201200010.

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42

Kita, Yoshio, Hirofumi Maekawa, Yasuhiro Yamasaki, and Ikuzo Nishiguchi. "ChemInform Abstract: Selective and Facile Electroreductive Synthesis of Dihydro- and Tetrahydropyridine Dicarboxylic Acid Derivatives." ChemInform 31, no. 9 (2010): no. http://dx.doi.org/10.1002/chin.200009142.

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43

Melikyan, G. G., K. A. Atanesyan, G. Kh Aslanyan, M. R. Tirakyan, L. A. Khachatryan, and Sh O. Badanyan. "Synthesis of 1,4,5,6-tetrahydropyridine derivatives starting from trans-3-chloro-1,3-alkadien-5-ones." Chemistry of Heterocyclic Compounds 23, no. 4 (1987): 414–17. http://dx.doi.org/10.1007/bf00546737.

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44

Tu, Shujiang, Fang Fang, Songlei Zhu, et al. "Microwave-assisted synthesis of phenylenedi(4′,4“-tetrahydroquinoline) and di(4′,4”-tetrahydropyridine) derivatives." Journal of Heterocyclic Chemistry 42, no. 1 (2005): 29–32. http://dx.doi.org/10.1002/jhet.5570420105.

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45

Tong, Shuo, and Mei-Xiang Wang. "Catalytic Enantioselective Synthesis of 4-Amino-1,2,3,4-tetrahydropyridine Derivatives from Intramolecular Nucleophilic Addition Reaction of Tertiary Enamides." Synlett 30, no. 04 (2018): 483–87. http://dx.doi.org/10.1055/s-0037-1610384.

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A general and efficient method for the synthesis of highly enantiopure 4-amino-1,2,3,4-tetradydropyridine derivatives based on chiral phosphoric acid catalyzed intramolecular nucleophilic addition of tertiary enamides to imines has been developed. We have also demonstrated a substrate engineering strategy to significantly improve the enantioselectivity of asymmetric catalysis

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46

Bibik, E. Yu, L. I. Kurbanov, S. A. Grygoryan, et al. "The analgesic activity of new sulfur-containing di- and tetrahydropyridine derivatives in the hot plate test." JOURNAL of SIBERIAN MEDICAL SCIENCES, no. 3 (2021): 45–55. http://dx.doi.org/10.31549/2542-1174-2021-3-45-55.

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Nowadays the search of new high-efficiency and safe drugs for the pharmacotherapy of diseases accompanied by pain syndrome is an active area of modern pharmacological research. 170 new derivatives of di- and tetrahydropyridines synthesized on the basis of the Chemex Research Laboratory, Vladimir Dahl Lugansk State University were exposed to the virtual bioscreening using the Swiss Target Prediction software. The paper describes screening studies in vivo of 5 samples of sulfur-containing di- and tetrahydropyridines (laboratory codes d02-138, as-262, f02-079, cv-074, cv-143) in the standard hot

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47

Redda, Kinfe Ken, Madhavi Gangapuram, Absera W. Haile, and Suresh Eyunni. "Abstract 5742: Synthesis of substituted benzimidazole tetrahydropyridines as anti-breast cancer agents." Cancer Research 85, no. 8_Supplement_1 (2025): 5742. https://doi.org/10.1158/1538-7445.am2025-5742.

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Abstract Breast cancer is the most common type of cancer worldwide. In 2023, the World Health Organization (WHO) reported that 2.3 million women were diagnosed with breast cancer, leading to 670, 000 deaths. Furthermore, the incidence rates of breast cancer have been rising at 3% each year. Overexpression of COX-2 in breast cancer tissues is associated with poor prognosis, including higher tumor grade, increased metastatic potential, and resistance to therapy. Selective COX-2 inhibitors have demonstrated potential in reducing tumor growth in preclinical and some clinical studies. These inhibit

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48

Khasanova, A. A., D. R. Kireeva, N. N. Gibadullina, Z. N. Fazletdinova, A. R. Sakhabutdinova, and R. R. Garafutdinov. "The influence of hexahydropyrimidine, bis(1,2,3,4-tetrahydropyridine) derivatives and tetrahydropyrimidinium salt on polymerase chain reaction." Biomics 11, no. 1 (2019): 14–22. http://dx.doi.org/10.31301/2221-6197.bmcs.2019-03.

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49

Nimkar, Sandeep K., Andrea H. Anderson, John M. Rimoldi, et al. "Synthesis and Monoamine Oxidase B Catalyzed Oxidation of C-4 Heteroaromatic Substituted 1,2,3,6-Tetrahydropyridine Derivatives." Chemical Research in Toxicology 9, no. 6 (1996): 1013–22. http://dx.doi.org/10.1021/tx960063o.

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50

Dong, Xu, Ying Han, Fachao Yan, et al. "Palladium-Catalyzed 6-Endo Selective Alkyl-Heck Reactions: Access to 5-Phenyl-1,2,3,6-tetrahydropyridine Derivatives." Organic Letters 18, no. 15 (2016): 3774–77. http://dx.doi.org/10.1021/acs.orglett.6b01787.

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