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Relevant bibliographies by topics / Thiazolidine Derivative

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Academic literature on the topic 'Thiazolidine Derivative'

Author: Grafiati

Published: 4 June 2021

Last updated: 2 February 2022

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Journal articles on the topic "Thiazolidine Derivative"

1

Fawzi, Mourad, Aziz Auhmani, Moulay Youssef Ait Itto, Abdelkhalek Riahi, Sylviane Chevreux, and El Mostafa Ketatni. "Crystal structure of methyl (Z)-2-[(Z)-3-methyl-2-({(E)-1-[(R*)-4-methylcyclohex-3-en-1-yl]ethylidene}hydrazinylidene)-4-oxothiazolidin-5-ylidene]acetate." Acta Crystallographica Section E Crystallographic Communications 73, no. 11 (2017): 1626–29. http://dx.doi.org/10.1107/s2056989017014311.

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The new title 4-thiazolidinone derivative, C16H21N3O3S, was obtained from the cyclization reaction of 4-methyl-3-thiosemicarbazone and dimethyl acetylenedicarboxylate (DMAD). The cyclohexylidene ring has an envelope conformation with the stereogenic centre C atom as the flap. Its mean plane makes a dihedral angle of 56.23 (9)° with the thiazolidine ring mean plane. In the crystal, molecules are linked by C—H...O hydrogen bonds forming chains propagating in the [001] direction. Within the chains there are offset π–π interactions between the thiazolidine rings of inversion-related molecules [cen

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Almeida, Marcel L., Douglas C. F. Viana, Valécia C. M. da Costa, et al. "Synthesis, Antitumor Activity and Molecular Docking Studies on Seven Novel Thiazacridine Derivatives." Combinatorial Chemistry & High Throughput Screening 23, no. 5 (2020): 359–68. http://dx.doi.org/10.2174/1386207323666200319105239.

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Aim and Objective: In the last decades, cancer has become a major problem in public health all around the globe. Chimeric chemical structures have been established as an important trend on medicinal chemistry in the last years. Thiazacridines are hybrid molecules composed of a thiazolidine and acridine nucleus, both pharmacophores that act on important biological targets for cancer. By the fact it is a serious disease, seven new 3-acridin-9-ylmethyl-thiazolidine-2,4-dione derivatives were synthesized, characterized, analyzed by computer simulation and tested in tumor cells. In order to find ou

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PAYNE, David J., John H. BATESON, David TOLSON та ін. "Phosphonamidate analogues of dipeptides with carboxypeptidase A and β-lactamase-inhibitory activity: elucidation of the mechanism of β-lactamase inhibition by electrospray mass spectrometry". Biochemical Journal 314, № 2 (1996): 457–61. http://dx.doi.org/10.1042/bj3140457.

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A series of phosphonamidate compounds with different P1´ amino acid residues have been shown to be irreversible inactivators of the serine β-lactamase from Enterobacter cloacae P99. The efficiency of inhibition (based on k2/K values) of P99 by these derivatives, ordered in decreasing potency, is: β-phenyl-β-Ala> L-Phe> β-Ala> Gly>D-Phe>D-Pro> D-thiazolidine. The D- and L-Phe compounds also inhibit carboxypeptidase A. The proline and thiazolidine derivatives were phosphonamidate methyl esters, whereas the others were salts of diacids. Electrospray mass spectrometry showed that

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Moreno-Fuquen, Rodolfo, Juan C. Castillo, Rodrigo Abonia, Javier Ellena, and Carlos A. De Simone. "Crystal structure of (±)-3-[(benzo[d][1,3]dioxol-5-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-1,3-thiazolidin-4-one." Acta Crystallographica Section E Structure Reports Online 70, no. 12 (2014): o1235—o1236. http://dx.doi.org/10.1107/s160053681402340x.

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In the title thiazolidine-4-one derivative, C20H21NO6S, the central thiazolidine ring is essentially planar (r.m.s. deviation for all non-H atoms = 0.0287 Å) and forms a dihedral angle of 88.25 (5)° with the methoxy-substituted benzene ring and 74.21 (4)° with the 1,3-benzodioxole ring. The heterocyclic ring (with two O atoms) fused to benzene ring adopts an envelope conformation with the non-ring-junction C atom as the flap. In the crystal, the molecules are linked into chains along [001] through weak C—H...O interactions, formingR44(28) edge-fused rings.

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Cambie, RC, GR Clark, TC Jones, PS Rutledge, GA Strange та PD Woodgate. "vic-Iodo Thiocyanates and Iodo Isothiocyanates. IX. A Synthesis of Penam and Other Polycyclic Β-Lactams". Australian Journal of Chemistry 38, № 5 (1985): 745. http://dx.doi.org/10.1071/ch9850745.

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Penam (4-thia-1-azabicyclo[3.2.0]heptan-7-one) and 2,3-disubstituted penams are prepared conveniently from vic-iodo isothiocyanates beginning with the facile cyclization of the latter with di -t-butyl sodiomalonates. Treatment of the resulting di -t-butyl 2-(thiazolidin-2- ylene ) malonates with trifluoroacetic acid gives t-butyl 2-thiazolin-2- ylacetate derivatives which are reduced to the corresponding thiazolidines with aluminium amalgam. Cleavage of these t-butyl esters with hydrogen chloride affords β-amino acid hydrochlorides, which are cyclized to penam and its derivatives with 1-[3-( d

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Hayashi, Tateki, Clayton A. Reece, and Takayuki Shibamoto. "Gas Chromatographic Determination of Formaldehyde in Coffee Via Thiazolidine Derivative." Journal of AOAC INTERNATIONAL 69, no. 1 (1986): 101–5. http://dx.doi.org/10.1093/jaoac/69.1.101.

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Abstract Thiazolidine formed from trace quantities of formaldehyde in an aqueous solution containing cysteamine at pH 8 was extracted with chloroform and subsequently analyzed by a gas chromatograph equipped with a fused silica capillary column and a thermionic nitrogen-phosphorus specific detector. Recoveries of formaldehyde from the aqueous solutions at levels lower than 1 ppm were slightly over 100%. Quantitative analysis of formaldehyde in commercial brewed and instant coffees showed 3.4-4.5 ppm in the brewed and 10-16.3 ppm in the instant coffee.

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Chande, Madhukar S., and Vijay Suryanarayan. "Synthesis of Spirocyclohexanone Ring Containing Thiazolidine Nucleus: A Regioselective Approach." Journal of Chemical Research 2005, no. 6 (2005): 345–47. http://dx.doi.org/10.3184/0308234054506749.

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The paper highlights the Michael addition reactions of 2-arylimino-3-aryl-thiazolidin-4-one 1 with acceptors like methyl acrylate and acrylonitrile to furnish the diadducts 5 and 8. Dieckmann condensation of 5 affords the spirocyclohexanone derivative. Also discussed is the interaction of 1 with 1,5-diarylpenta-1,4-dien-3-ones 9.

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Gyertyán, István, Lujza Petöcz, István Gacsályi, Márton I. K. Fekete, Kornélia Tekes, and László Kápolnai. "Psychopharmacological effects of an imino-thiazolidine derivative antidepressant candidate, EGYT-4201." Drug Development Research 22, no. 4 (1991): 385–99. http://dx.doi.org/10.1002/ddr.430220410.

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Norisada, Nobuyoshi, Hiroaki Masuzaki, Muneya Fujimoto, et al. "Antidiabetic and adipogenic properties in a newly synthesized thiazolidine derivative, FPFS-410." Metabolism 53, no. 12 (2004): 1532–37. http://dx.doi.org/10.1016/j.metabol.2004.06.020.

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Journal, Baghdad Science. "Synthesis of Some Heterocyclic Compounds derived from 2-mercapto pyrimidine." Baghdad Science Journal 7, no. 2 (2010): 1014–22. http://dx.doi.org/10.21123/bsj.7.2.1014-1022.

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In this work 2-hydrazino pyrimidine (1) was prepared from 2-mercapto pyrimidine with hydrazine hydrate. Treatment of (1) with active methylene compounds gave 2-(3,5-dimethyl -1 H – Pyrazole-1-yl) pyrimidine , whereas the reaction of (1) with carboxylic anhydride namely maleic anhydride or 1,2,3,6-tetra hydro phthalic anhydride yielded 1-Pyrimidine-2-yl-1,2-dihydro pyridazine-3,6-dione (3) and 2 – Pyrimidin -2-yl -2,3,4 a ,5,8 a – hexahydro phthalazine 1,4 – dione (4) . Reaction of (1) with phenyl isothiocyanate and ethyl chloro acetate afforded 3-Phenyl-1,3-thiazolidine-2,4-dione-2( pyrimidine

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Dissertations / Theses on the topic "Thiazolidine Derivative"

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Norisada, Nobuyoshi. "Antidiabetic and adipogenic properties in a newly-synthesized thiazolidine derivative, FPFS-410." Kyoto University, 2007. http://hdl.handle.net/2433/135906.

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Novo, Fernández Olalla. "New contributions to the preparation of compounds derived from L-cysteine with biological activity." Doctoral thesis, Universitat de Lleida, 2017. http://hdl.handle.net/10803/440527.

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Una gran varietat de productes naturals i fàrmacs que inclouen sofre en les seves estructures presenten diverses activitats biològiques i aplicacions. Un exemple és la L-cisteïna, un aminoàcid essencial necessari en processos bioquímics dels éssers vius. D’una banda, aquest treball es centra en l’obtenció de tiazolidines a partir de la L-cisteïna amb un grau de qualitat alimentària. La metodologia es basa en un procés de síntesi en continu i en un sistema d’assecatge d’atomització. A més, es va realitzar un estudi per investigar el rol de la tiazolidina derivada de la D-ribosa com a agent quim

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Huber-Villaume, Sophie. "Impact des ligands de PPARs, et leurs dérivés, sur les cellules cancéreuses coliques humaines : modifications des statuts redox et glycolytique." Thesis, Université de Lorraine, 2014. http://www.theses.fr/2014LORR0217/document.

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La Pioglitazone appartient à la famille des thiazolidinédiones et le Fénofibrate à la famille des fibrates. Ces molécules sont, respectivement, des agonistes synthétiques du récepteur activable par les proliférateurs de peroxysomes γ (PPARγ) et PPARα, membres de la famille des récepteurs nucléaires aux hormones. Le traitement de cellules cancéreuses humaines par ces molécules limite la croissance et peut induire leur apoptose. Cependant, l’impact de ces traitements sur les cellules cancéreuses est en partie dû à une action indépendante de l’activation du récepteur et met en cause la génération

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Wang, Hui-Min, and 王惠民. "Utilization of derivatives of thiazolidine-2-thione." Thesis, 1988. http://ndltd.ncl.edu.tw/handle/57766773753850809928.

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Lu, Hsueh-Yuan, and 呂學遠. "(I) Multicomponent Reaction Synthesis of Thiazolidine-Linked Benzimidazole Derivatives (II) Synthesis of Tetrahydroisoquinoline Heterocyclic Small Molecule Derivatives via Radical Pictet-Spengler Reaction." Thesis, 2019. http://ndltd.ncl.edu.tw/handle/feduqz.

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Book chapters on the topic "Thiazolidine Derivative"

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Cordero, F. M., and S. Cicchi. "Reaction of Thiazolidin-4-ones with Nitrosobenzene." In Three Carbon-Heteroatom Bonds: Amides and Derivatives; Peptides; Lactams. Georg Thieme Verlag KG, 2005. http://dx.doi.org/10.1055/sos-sd-022-00380.

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Conference papers on the topic "Thiazolidine Derivative"

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Sankar, P. Siva, K. Divya, G. Dinneswara Reddy, V. Padmavathi, and Grigory V. Zyryanov. "Synthesis, characterization and antimicrobial activity of azetidinone and thiazolidinone derivatives." In PROCEEDINGS OF THE 3RD INTERNATIONAL CONFERENCE ON AUTOMOTIVE INNOVATION GREEN ENERGY VEHICLE: AIGEV 2018. Author(s), 2019. http://dx.doi.org/10.1063/1.5087379.

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2

Szymanowski, Wojciech, Kamila Buzun, Anna Szymanowska, et al. "The cytotoxic potential of a novel 2-thioxo-4-thiazolidinone derivative used with anti-HER2 antibodies in AGS gastric cancer cells." In RAD Conference. RAD Centre, 2021. http://dx.doi.org/10.21175/rad.abstr.book.2021.8.2.

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Buzun, Kamila, Agnieszka Gornowicz, Robert Czarnomysy, Roman Lesyk, Krzysztof Bielawski, and Anna Bielawska. "The pro-apoptotic effect of new 2-thioxo-4-thiazolidinone derivative Les-3331 on MCF-7 and MDA-MB-231 cell lines." In RAD Conference. RAD Centre, 2021. http://dx.doi.org/10.21175/rad.abstr.book.2021.8.4.

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4

Kobylinska, L., B. Zimenkovsky, R. Panchuk, et al. "Complex of synthetic 4-thiazolidinone derivatives with PEG-containing polymeric nanocarrier improve of biocompatibility and protects against toxicity in laboratory rats." In 2017 IEEE 7th International Conference "Nanomaterials: Application & Properties" (NAP). IEEE, 2017. http://dx.doi.org/10.1109/nap.2017.8190321.

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Nikalje, Anna Pratima. "Synthesis and Anti-Inflammatory Evaluation of 2-(3-(2-(1,3-Dioxoisoindolun-2-YL) Acetamido)-4-OXO-2-Substituted Thiazolidin-5-YL) Acetic Acid Derivatives." In The 18th International Electronic Conference on Synthetic Organic Chemistry. MDPI, 2014. http://dx.doi.org/10.3390/ecsoc-18-c010.

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