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Relevant bibliographies by topics / Thiazolidone compound

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Academic literature on the topic 'Thiazolidone compound'

Author: Grafiati

Published: 5 June 2025

Last updated: 15 July 2025

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Journal articles on the topic "Thiazolidone compound"

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Varenichenko, S. A., A. V. Kharchenko, and O. K. Farat. "Synthesis and in silico ADMET profiling of novel 5-arylidene-2-(2,3,5,6,7,8-hexahydroacridin-4(1H)-ylidene)-1,3-thiazolidin-4-ones." Voprosy Khimii i Khimicheskoi Tekhnologii, no. 6 (December 2023): 37–43. http://dx.doi.org/10.32434/0321-4095-2023-151-6-37-43.

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The corresponding thiazolidone derivative was synthesized with a good yield by the reaction of 1,2,3,4,5,6,7,8-octahydroacridine-4-carbonitrile with thioglycolic acid. It was found that this compound is present in DMSO in the form of two isomers, (2E)-2-(2,3,5,6,7,8-hexahydroacridin-4(1H)-ylidene)-1,3-thiazolidin-4-one and (2Z)-2-(2,3,5,6,7,8-hexahydroacridin-4(1H)-ylidene)-1,3-thiazolidin-4-one in a ratio of 9:1, respectively, whereas it is present only in the form of the E-isomer in chloroform. The corresponding 5-arylidene-2-(2,3,5,6,7,8-hexahydroacridin-4(1H)-ylidene)-1,3-thiazolidin-4-one

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Al-Abboodi1, Doaa Hashim, and Naeemah Al-lami. "NEW METHDOLOGY OF SYNTHESIS PYRAZOLO- THIAZOLO DERIVATIVES WITH STUDY ANTIMICROBAL ACTIVITIES." iraqi journal of market research and consumer protection 16, no. 1 (2024): 1–12. http://dx.doi.org/10.28936/jmracpc16.1.2024.(1).

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In this contribution, new derivatives of thiosemicarbazon, cyclic thiazolidinone, yilidine thiazolidinone, and parazolo-thiazole were synthesized, starting from the reaction of 2 -aminobenzothiazole with p-bromo phenacyl bromide to give the first step of 2(4-bromo phenyl) imidazole (2,1 -b) benzo thiazole (1). Compound (1) then was subjected under Viels Myer Haack to yield 3-carbaldehyde linking with imidazo-benzothiazol (2). Compound (2) condensed with thiosemicarbazide togivenewsynthesis of thiosemicarbazon derivative (3). Compound 4-Oxo-1,3-thiazolidine (4) was constituted from reacting com

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Allahyani, Mamdouh, Mazen Almehmadi, Osama Abdulaziz, et al. "Synthesis and in vitro antimicrobial screening of some 5-methyl-2-substituted phenyl-3- (phenylsulfonyl)thiazolidin-4-ones." INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY 34, no. 04 (2024): 499. https://doi.org/10.59467/ijhc.2024.34.499.

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The synthesis of some new thiazolidine-sulfonamide derivatives was achieved in two steps. In the first step, appropriate aryl aldehyde reacted with benzene sulfonamide to yield N-arylidene benzene sulfonamide derivatives (1a-h). In the second step, compounds (1a-h) reacted with thiolactic acid to give the 5-methyl-2-substituted phenyl-3-(phenylsulfonyl) thiazolidin-4-one derivatives (2a-h). The compounds 2a-h were screened for their in vitro antimicrobial activity by agar disc diffusion method. The results showed that compounds 2b, 2c, and 2d exhibited anti-microbial activity against the teste

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Amit Kumar, Nitin Mittal, Mukesh Gupta, and Shikha Sharma. "Synthesis and Antibacterial Activity of Some Newer Thiazolidine-2,4-Dione Derivatives." Journal of Biomedical and Pharmaceutical Research 12, no. 4 (2023): 11–21. http://dx.doi.org/10.32553/jbpr.v12i4.1008.

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Thiazolidin-2,4-diones were intensively studied for its antidiabetic property in 1982. Thiazolidin-2,4-diones have also been demonstrated to possess different biological activity like anticancer, anti-HIV, antitumor, antimicrobial, antiviral and antiproliferative activity. 3-Benzoyl-5-(substituted benzylidine)-thiazolidin-2,4-diones and 3-p-Tolyl-5-(substituted benzylidine)-thiazolidin-2,4-diones have evaluated as structurally novel antimicrobials. A series of 5-[(SubstitutedPhenylamino)benzylidine]thiazolidine-2,4-dione derivatives 17(a-j) were synthesized by nucleophilic substitution reactio

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Kumar, Shiv, Nitin Kumar, Sushma Drabu, et al. "Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide Based Thiazolidinone Derivatives as Potent Antibacterial and Antifungal Agents." E-Journal of Chemistry 9, no. 4 (2012): 2155–65. http://dx.doi.org/10.1155/2012/857514.

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Twelve compounds belonging to series 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)-N-[4-oxo-2-(substituted)phenyl-1,3-thiazolidin-3-yl]acetamide (5a-l) were synthesized. These compounds were evaluated for theirin-vitroantibacterial againstE. coli, S. aureus, K. pneumoniae, P. aeruginosa & antifungalactivity againstC. albicans, A. niger & A. flavusby cup-plate method. Structures of all the newly synthesized compounds were confirmed by elemental analysis,1H-NMR & FT-IR spectral data interpretation. Compounds 5d & 5h having p-nitrophenyl &p-trifluoromethylphenyl group respectively on

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Rosy P., Jacquline, Jebastin Sonia Jas M., Santhanalakshmi K, Venkat Kumar Shanmugam, and Prabhakaran A. "Identification of Potential Inhibitor Targeting InhA, Molecular Docking, ADMET, Molecular Dynamic Simulation and Antibacterial Activity of Thiazolidinone Derivatives: A Computational Approach." International Journal of Zoological Investigations 08, special issue (2022): 191–202. http://dx.doi.org/10.33745/ijzi.2022.v08i0s.024.

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This study was performed to examine molecular docking of newly synthesised thiazolidinone compounds and discover potential InhA inhibitors. MIC screening produced thiazolidinone derivatives for Staphylococcus aureus illness. KBr pellet FT-IR spectra were collected on a Thermo Nicolet AVATAR-330 spectrometer. Bruker obtained 400 MHz 1H spectra of all chemicals in DMSO-d6. Five 4 thiazolidinone derivatives:4-(4-oxo-2-phenylthiazolidin-3yl)amino)benzyl)oxazolidin-2-one(8), ((2-(4 chlorophenyl)-4oxothiazolidin-3yl)amino)benzyl)- oxazolidin-2-one(9), ((2-(4-fluorophenyl)-4-oxothiazolidin-3 yl)amino

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Perepelytsya, O. O., I. M. Yaremiy, K. P. Kupchanko, N. V. Panasenko, M. K. Bratenko, and M. V. Vovk. "Synthesis and hypoglycemic activity of derivatives of 4-((1,3-thiazolydine-5-yliden)methy)pyrazole-3-carbonic acid and its esters." Chernivtsi University Scientific Herald. Chemistry, no. 819 (2019): 37–44. http://dx.doi.org/10.31861/chem-2019-819-06.

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An effective preparative method of synthesis of a series of new (pyrazole-4-il)methylenethiazolidine structures has been elaborated. The structures are functionalized in the 3rd position by the carboxylate or carboxyle group and in the 3rd and 5th positions of the thiazolidine cycle – by the oxo-, thio- or iminogroups. The method involves condensation of 4-formylpyrazole-3-carbonic acids and their ethyl esters with a series of the substituted thiazolidines: 1,3-thiazolidine-2,4-dione, 4-thioxo-1,3-thiazolidine-2-one, 2-thioxo-1,3-thiazolidine-4-one and 2-imino-1,3-thiazolidine-4-one. A group o

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Kumar, Nitin, and Sanjay Sharma. "SYNTHESIS AND ANTICANCER ACTIVITY OF N-SUBSTITUTED INDOLE DERIVATIVES." INDIAN DRUGS 58, no. 12 (2022): 16–21. http://dx.doi.org/10.53879/id.58.12.12496.

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Thizolidine-2,4-dione (1), on reaction with p-fluorobenzaldehyde in the presence of piperidine and toluene, gives (Z)-5-(2-fluororobenzylidin)-thiazolidin-2,4-dione (2), which on reaction with indole and o-chlorobenzaldehyde in the presence of ethanol yielded final derivatives i.e (Z)-5-(4-fluororobenzylidene)-3-[(1H-indol-1-yl) (substituted phenyl) methyl] thiazolidine-2,4-dione (3a-3e). All the synthesized compounds were characterized by UV, FTIR, 1 H NMR, MASS spectroscopy and elemental analysis. These compounds were screened for their anticancer activity against MCF-7 human breast cancer c

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Nuriye, Ahmed, Hemant Yennawar, Kevin Cannon, and John Tierney. "Crystal structures of two thiazolidinone derivatives bearing a trichloromethyl substituent at the 2-position." Acta Crystallographica Section E Crystallographic Communications 74, no. 10 (2018): 1509–12. http://dx.doi.org/10.1107/s2056989018013257.

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The title compounds 2-trichloromethyl-3-phenyl-1,3-thiazolidin-4-one (C10H8Cl3NOS),1and 3-(4-chlorophenyl)-2-trichloromethyl-1,3-thiazolidin-4-one (C10H7Cl4NOS)2, are structurally related with one atom substitution difference in theparaposition of the benzene ring. In both structures, the thiazolidinone ring adopts an envelope conformation with the S atom as the flap. The dihedral angles between the rings [48.72 (11) in1and 48.42 (9)° in2] are very similar and the molecules are almost superimposable. In both crystal structures, C—H...O `head-to-tail' interactions between the chiral carbon atom

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da Silva Santos, Jonas, Joel Jones Junior, and Flavia M. da Silva. "1,3-Thiazolidin-4-ones: Biological Potential, History, Synthetic Development and Green Methodologies." Current Organic Synthesis 15, no. 8 (2018): 1109–23. http://dx.doi.org/10.2174/1570179415666180919125625.

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Background: We present here the synthesis of 1,3-thiazolidin-4-one (1) and its functionalised analogues, such as the classical isosteres, glitazone (1,3-thiazolidine-2,4-dione) (2), rhodanine (2-thioxo-1,3- thiazolidin-4-one) (3) and pseudothiohydantoin (2-imino-1,3-thiazolidin-4-one) (4) started in the midnineteenth century to the present day (1865-2018). Objective: The review focuses on the differences in the representation of the molecular structures discussed here over time since the first discussions about the structural theory by Kekulé, Couper and Butlerov. Moreover, advanced synthesis

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Dissertations / Theses on the topic "Thiazolidone compound"

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Laduranty, Joëlle. "Mise au point de la préparation de molécules polyfonctionnelles comportant l'unité structurale SCCN de la cystéamine : applications en radioprotection et synthèse organique." Poitiers, 1988. http://www.theses.fr/1988POIT2013.

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CAVALCANTE, SILVA JACQUELINE. "Effects of a new thiazolidine compound (GQ-11) on tissue repair process in models of insulin resistance and ischemia/reperfusion." Doctoral thesis, Università degli studi di Genova, 2019. http://hdl.handle.net/11567/982439.

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The thiazolidinediones (TZDs) class comprises drugs with hypoglycemic effects, reducing insulin resistance in peripheral tissues. Our group has demonstrated in preliminary in vivo data that a new TZD, GQ-11, improves insulin resistance as well as modulates cytokines involved in inflammatory process, suggesting an interesting approach for therapeutic alternatives in tissue repair, especially in metabolic decompensation cases, as insulin resistance and ischemia-reperfusion. In this context, the aim of this study was to investigate GQ-11 effects in tissue repair in three different models: insulin

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Novo, Fernández Olalla. "New contributions to the preparation of compounds derived from L-cysteine with biological activity." Doctoral thesis, Universitat de Lleida, 2017. http://hdl.handle.net/10803/440527.

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Una gran varietat de productes naturals i fàrmacs que inclouen sofre en les seves estructures presenten diverses activitats biològiques i aplicacions. Un exemple és la L-cisteïna, un aminoàcid essencial necessari en processos bioquímics dels éssers vius. D’una banda, aquest treball es centra en l’obtenció de tiazolidines a partir de la L-cisteïna amb un grau de qualitat alimentària. La metodologia es basa en un procés de síntesi en continu i en un sistema d’assecatge d’atomització. A més, es va realitzar un estudi per investigar el rol de la tiazolidina derivada de la D-ribosa com a agent quim

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Chiu, Hsiao-shan, and 邱筱珊. "Synthesis, Characterization and Crystal Engineering Structural Transformation of L-Thiazolidine-4-carboxylate-containing Homochiral Coordination Compounds." Thesis, 2013. http://ndltd.ncl.edu.tw/handle/28282970174106855902.

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碩士<br>國立中央大學<br>化學學系<br>101<br>This thesis focuses on the preparation of a series of metal complexes via the use of a combination of metal (Zn(II), Co(II), Ni(II), Cd(II) salts with a LTP (L-thiazolidine-4-carboxylate)) ligand under mild reaction conditions. Their structures were characterized by single-crystal X-ray diffraction analyses. The structures of the first series [M(LTP)2(H2O)2] (M = Zn(II) 1, Co(II) 2, Ni(II) 3) show that the metal ion is six-coordinated in a distorted octahedral geometry and bonded to two N and two O atoms from two LTP ligands with bis-chelating coordination mode a

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Book chapters on the topic "Thiazolidone compound"

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Pardasani, R. T., and P. Pardasani. "Magnetic properties of nickel(II) complex with 1,3-thiazolidine-2-thionate." In Magnetic Properties of Paramagnetic Compounds. Springer Berlin Heidelberg, 2017. http://dx.doi.org/10.1007/978-3-662-54234-7_364.

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Pardasani, R. T., and P. Pardasani. "Molar magnetic moment of dichloro[2-(2-pyridyl)imino-kN-N-(2-thiazolin-kN-2-yl)thiazolidine]." In Magnetic Properties of Paramagnetic Compounds, Magnetic Susceptibility Data, Volume 2. Springer Berlin Heidelberg, 2021. http://dx.doi.org/10.1007/978-3-662-62466-1_226.

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Pardasani, R. T., and P. Pardasani. "Magnetic properties of copper(II) complex with 2-(2-pyridyl)imino-N-(2-thiazolin-2-yl)-thiazolidine." In Magnetic Properties of Paramagnetic Compounds, Magnetic Susceptibility Data, Volume 4. Springer Berlin Heidelberg, 2021. http://dx.doi.org/10.1007/978-3-662-62474-6_12.

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Pardasani, R. T., and P. Pardasani. "Magnetic properties of binuclear copper(II) complex with 2-(2-pyridyl)imino-N-(2-thiazolin-2-yl)thiazolidine." In Magnetic Properties of Paramagnetic Compounds, Magnetic Susceptibility Data, Volume 4. Springer Berlin Heidelberg, 2021. http://dx.doi.org/10.1007/978-3-662-62474-6_168.

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Cha, J. K. "Acylation of Thiazolidines." In Three Carbon-Heteroatom Bonds: Esters and Lactones; Peroxy Acids and R(CO)OX Compounds; R(CO)X, X=S, Se, Te. Georg Thieme Verlag KG, 2005. http://dx.doi.org/10.1055/sos-sd-021-00303.

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Kryshchyshyn, Anna, Danylo Kaminskyy, Philippe Grellier, and Roman Lesyk. "Thiazolidinone-Related Heterocyclic Compounds as Potential Antitrypanosomal Agents." In Azoles - Synthesis, Properties, Applications and Perspectives [Working Title]. IntechOpen, 2020. http://dx.doi.org/10.5772/intechopen.91861.

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Conference papers on the topic "Thiazolidone compound"

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Cozar, I. B., A. Pı̂rnău, N. Vedeanu, and C. Nastasă. "Structural investigation of a new antimicrobial thiazolidine compound." In PROCESSES IN ISOTOPES AND MOLECULES (PIM 2013). AIP, 2013. http://dx.doi.org/10.1063/1.4833691.

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Živković, Marijana, Stepan Stepanović, and Dušan Sladić. "STEROIDAL THIAZOLIDIN-4-ONES: IN SILICO PREDICTION OF TOXICITY." In 3rd International Symposium on Biotechnology. University of Kragujevac, Faculty of Agronomy in Čačak, 2025. https://doi.org/10.46793/sbt30.67mz.

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Cancer remains a leading cause of death worldwide, and as a result, scientists are focused on discovering new drugs to combat this disease. To save both time and money, it is desirable to predict the drug-likeness and toxicity of new compounds. According to RDKit library, previosly synthesized, highly cytotoxic and selective steroidal thazolidin-4-ones (TZDs) were drug-like. Based on in vitro cytotoxicity results in HeLa cells for 12 TZDs, a reliable in silico toxicity model was developed for other similar compounds. The polar surface area and number of H-bond acceptors of the tested TZDs were

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Rašović, Aleksandar, and Vladimir A. Blagojević. "THE C(2)C(2′) SINGLE BOND LENGTHS OF THE TRANSITION STATES IN THE CONFIGURATIONAL ISOMERIZATION OF 2-ALKYLIDENE-4-OXOTHIAZOLIDINES BY THE MEANES TO QUANTIFY THEIR PUSH-PULL EFFECT UNDER SOLVENT CONDITIONS." In 17th International Conference on Fundamental and Applied Aspects of Physical Chemistry. Society of Physical Chemists of Serbia, 2024. https://doi.org/10.46793/phys.chem24i.261r.

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We reported previously that the barriers to rotation (DG‡) around the C(2)C(2′) double of the selected thiazolidine derivatives 1-2 proved to be an efficient parameter to quantify the push–pull effect of these compounds both under the same and different solvent conditions. As a continuation of the research of potential parameters that could be applied for this purpose, this work explored calculated C(2)C(2′) single bonds of their transition states (TS). Regarding this, they showed to be of great interest.

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Živković, Marijana B., Srđan J. Tufegdžić, Sandra B. Šegan, Neda O. Đorđević, and Dušan Sladić. "IN SILICO DRUG-LIKENESS OF STEROIDAL THIAZOLIDIN-4-ONES." In 8th Workshop Food and Drug Safety and Qualit. Vinča Institute of Nuclear Sciences - National Institute of the Republic of Serbia, 2024. http://dx.doi.org/10.46793/8fdsq.pc7mz.

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In silico assessment of drug-likeness of 15 steroidal mono- and bis-thiazolidinones was performed. Androstrane (1−5) and progesterone types (6) mono-derivatives had no violations of Lipinski’s rule of five, while bis-derivatives had slightly higher molecular masses than 500 Da, and cholestane derivatives (8−9) showed high lipophilicity and Caco-2 permeability. All examined compounds showed great intestinal absorption potential.

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Rašović, Aleksandar, and Vladimir A. Blagojević. "AN EXTENDED STUDY OF THE APPLICATION OF THE BARRIERS TO ROTATION AROUND THE C=C BOND OF 2-ALKYLIDENE-4-OXOTHIAZOLIDINES TO QUANTIFY THEIR PUSH-PULL EFFECT UNDER SOLVENT CONDITIONS." In 17th International Conference on Fundamental and Applied Aspects of Physical Chemistry. Society of Physical Chemists of Serbia, 2024. https://doi.org/10.46793/phys.chem24i.257r.

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As we reported previously, the barriers to rotation (DG‡) around the C(2)C(2′) double of the selected thiazolidine derivatives 1-2 showed to be an efficient parameter to quantify their push–pull effect both under the same and different solvent conditions (at least three solvents studied: chloroform, dimethyl sulfoxide, and water). This work reports an extended study regarding solvent conditions. Additionally, this research has involved model compound 3, which does not possess a push–pull effect. The archived excellent linear correlations between the barriers to rotation (DG‡) around the C(2)C(

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Azeez, Hashim, and Bana Abdulrahman. "Synthesis and Spectroscopic Characterization of a New Series of Thiazolidin-4-One Compounds from Heterocyclic Schiff Bases." In 2018 International Conference on Pure and Applied Science. Koya University, 2018. http://dx.doi.org/10.14500/icpas2018.ach77.

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