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Journal articles on the topic '-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl]propyl)-2'

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Published: 4 June 2025
Last updated: 1 August 2025

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1

Drapak, Іryna, Borys Zimenkovsky, Lina Perekhoda, et al. "Qsar-analysis of 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl]propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one’s derivatives as potential antioxidants." Pharmacia 66, no. 1 (2019): 33–40. http://dx.doi.org/10.3897/pharmacia.66.e35083.

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Aim. The aim of study was to determine of the parameters of the molecular structure of new 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl]propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one derivatives and QSAR-analysis. The latter can be considered as the theoretical basis for de novo design of new potential antioxidants. Materials and methods. 14 new derivatives of 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl] propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one were involved in the study and their antioxidant activities were evaluated. Hyper-Chem 7.59 and BuildQSAR software were used
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2

Drapak, Іryna, Borys Zimenkovsky, Lina Perekhoda, et al. "QSAR-analysis of 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl]propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one's derivatives as potential antioxidants." Pharmacia 66, no. (1) (2019): 33–40. https://doi.org/10.3897/pharmacia.66.e35083.

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Aim. The aim of study was to determine of the parameters of the molecular structure of new 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl]propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one derivatives and QSAR-analysis. The latter can be considered as the theoretical basis for de novo design of new potential antioxidants. Materials and methods. 14 new derivatives of 1-[2-(R-phenylimino)-4-methyl-3-(3-[morpholine-4-yl] propyl)-2,3-dihydro-1,3-thiazol-5-yl]ethane-1-one were involved in the study and their antioxidant activities were evaluated. Hyper-Chem 7.59 and BuildQSAR software were used
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3

Desai, S. N. Mamle, Rudrax N. S. Priolkar, Harshank A. Naik Karmali, Prabhav D. Ambe, and B. S. Biradar. "SYNTHESIS, CHARACTERIZATION AND EVALUATION OF 4-HYDROXY-1-PHENYL/METHYL-3-(3-SUBSTITUTED-1-(SUBSTITUTEDIMINO) PROPYL) QUINOLINE-2(1H)-ONE DERIVATIVES AND 4-HYDROXY-1-PHENYL/METHYL-3-(1-(SUBSTITUEDIMINO) ETHYL) QUINOLINE-2(1H)-ONE DERIVATIVES AS POSSIBLE ANTICANCER AGENTS." International Journal of Pharmacy and Pharmaceutical Sciences 9, no. 10 (2017): 240. http://dx.doi.org/10.22159/ijpps.2017v9i10.20184.

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Objective: Synthesis, characterization and evaluation of quinolin-2-one derivatives as possible anticancer agents.Methods: A series of novel 4-hydroxy-1-phenyl/methyl-3-(3-substituted-1-(substitutedimino)propyl)quinolin-2(1H)-one derivatives IIa(1-5)/IIb(1-5) and 4-hydroxy-1-phenyl/methyl-3-(1-(substituedimino)ethyl)quinolin-2(1H)-one derivatives IIIa(1-3)/IIIb(1-3) were synthesised by nucleophilic addition of substituted anilines on 3-acetyl-4-hydroxy-1-phenyl/methylquinolin-2(1H)-one (a/b) and 4-hydroxy-3-(3-substitutedpropanoyl)-1-phenyl/methyl quinolin-2(1H)-one (Ia/Ib); respectively. The
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4

Pranay, Shah, I. Patel R., and J. Vyas P. "Preparation and Biological Screening of Novel Heterocyclic Compounds." International Journal of Trend in Scientific Research and Development 3, no. 3 (2019): 632–36. https://doi.org/10.31142/ijtsrd22815.

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The Pyrimidone derivatives say, N arylidine 6 methyl 2 oxo 4 phenyl 1,2,3, 4 tetrahydropyrimidonecarbohydrazides 2a e were synthesized by condensation of Benzaldehyde derivatives with 6 Methyl 2 oxo 4 phenyl 1,2,3,4 tetrahydro pyrimidone carbohydrazides 1 in good yield. The so called hydrazone were cyclocondensed with succinic anhydride to afford 1 6 methyl 2 oxo 4 phenyl 1,2,3, 4 tetrahydropyrimidone 5 carboxamido 5 oxo 2 aryl pyrrolidine 3 carboxylic acid 3a e . These 3a e on Mannich reaction with formaldehyde and morpholine offered 2 aryl 1 6 methyl 2 oxo 4 phenyl 1, 2, 3, 4 tetrahydropyrim
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5

Mali, Suraj N., Sudhir Sawant, Hemchandra K. Chaudhari, and Mustapha C. Mandewale. "In Silico Appraisal, Synthesis, Antibacterial Screening and DNA Cleavage for 1,2,5-thiadiazole Derivative." Current Computer-Aided Drug Design 15, no. 5 (2019): 445–55. http://dx.doi.org/10.2174/1573409915666190206142756.

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Background: : Thiadiazole not only acts as “hydrogen binding domain” and “two-electron donor system” but also as constrained pharmacophore. Methods:: The maleate salt of 2-((2-hydroxy-3-((4-morpholino-1, 2,5-thiadiazol-3-yl) oxy) propyl) amino)- 2-methylpropan-1-ol (TML-Hydroxy)(4) has been synthesized. This methodology involves preparation of 4-morpholino-1, 2,5-thiadiazol-3-ol by hydroxylation of 4-(4-chloro-1, 2,5-thiadiazol-3-yl) morpholine followed by condensation with 2-(chloromethyl) oxirane to afford 4-(4-(oxiran-2-ylmethoxy)-1,2,5-thiadiazol- 3-yl) morpholine. Oxirane ring of this com
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6

Perekhoda, L. O., H. O. Yeromina, I. V. Drapak, I. A. Sych, A. M. Demchenko та S. O. Komykhov. "The synthesis of N-[4-methyl(41-chlorophenyl)-2-R-phenylіmіnothіazol-3-yl]-morpholine derivatives by Hantzsch reaction". Journal of Organic and Pharmaceutical Chemistry 14, № 3(55) (2016): 52–57. http://dx.doi.org/10.24959/ophcj.16.890.

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7

Suhak, O. A., О. I. Panasenko, and Ye G. Knysh. "Synthesis, physic and chemical properties of 2-(4-R-5-(thiophene-2-ylmethyl)-4h-1,2,4-triazole-3-ylthio)acetate acids and their salts." Farmatsevtychnyi zhurnal, no. 2 (August 14, 2018): 48–54. http://dx.doi.org/10.32352/0367-3057.2.17.06.

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Derivatives of 1,2,4-triazole are inherent in various types of biological activity. They can be used as pesticide and medicinal drugs (anticonvulsants, analgetics, antitumor and antibacterial). In this regard the search of new methods of synthesis and investigation of biological activity of 2-(4-R-5-(thiophene-2-ylmethyl)-4H-1,2,4-triazole-3-ylthio)acetate acids and their salts is relevant nowadays.
 With the aim of finding the new biologically active compounds 2-(4-R-5-(thiophene-2-ylmethyl)-4H-1,2,4-triazole-3-ylthio)acetate acids and their salts are synthesized, where R is methyl, ethy
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8

Kumar Reddy, G. Mahesh, Raghu Babu Korupolu, B. Kishore Babu, et al. "Hydrolytic Degradation Study of Rivaroxaban: Degradant Products Identification by LC-MS Isolation by Prep-HPLC and Characterization by HRMS, NMR and FT-IR." Asian Journal of Chemistry 32, no. 12 (2020): 3035–42. http://dx.doi.org/10.14233/ajchem.2020.22888.

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Present work illustrates the stress degradation behaviour of rivaroxaban under hydrolytic, oxidative, thermal and photolytic conditions as per ICH guidelines. Under thermal and photolytic conditions drug had a fair stability where as in other stress conditions degradation products were observed. Initial identification of the degradation products was performed by hyphenated mass spectrometry coupled to ultra-performance liquid chromatography (UPLC-MS) and mass directed auto purification (MDAP) was used for isolation. Various 1D and 2D nuclear magnetic resonance (NMR) were performed to character
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9

Anwar, Sh, F. Mahmood, N. A. Tahir, and G. F. Salih. "SECONDARY COMPOUNDS RELEASED BY RHIZOSPHERIC BACTERIA EXHIBIT FUNGISTATIC EFFECTS AGAINST PHYTOPATHOGENIC FUNGUS." IRAQI JOURNAL OF AGRICULTURAL SCIENCES 53, no. 5 (2022): 1174–83. http://dx.doi.org/10.36103/ijas.v53i5.1631.

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The aim of conducted research was to devalute the inhibition effect of metabolites secreted by some Rhizospheric bacteria on the growth of two pathogenic fungi: Rhizoctonia solani and Fussarium solani, 330 bacteria isolates were obtained from the rhizosphere of the wheat, tomato, cowpea and Mt. Atlas mastic tree grown in the Sulaimani. Thirty-five isolates were screened for suppression of phytopathogeneic fungus. Results showed that most of these rhizospheric bacteria were have fungistatic potential in different degrees. The highest inhibition of the linear growth of fungi was noted for R. sol
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10

Fawcett, James A., and Robert G. Harvey. "Proso Millet (Panicum miliaceum) Control in Corn (Zea mays) by Postemergence-Directed Herbicides." Weed Science 36, no. 2 (1988): 215–20. http://dx.doi.org/10.1017/s0043174500074737.

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Proso millet (Panicum miliaceumL. # PANMI) was controlled in corn (Zea maysL. ‘Pioneer 3747’) with postemergence-directed herbicides applied following a standard preplant-incorporated application of butylate[S-ethylbis(2-methylpropyl)carbamothioate] plus dichlormid (2,2-dichloro-N,N-di-2-propenylacetamide) plus cyanazine {2-[[4-chloro-6-(ethylamino)-1,3,5-triazin-2-yl]amino]-2-methylpropanenitrile}. Postemergence-directed applications of ametryn [N-ethyl-N′-(1-methylethyl)-6-(methylthio)-1,3,5-triazine-2,4-diamine], cloproxydim {(E,E)-2-[1-[[(3-chloro-2-propenyl)oxy]imino]butyl]-5-[2-(ethylthi
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11

Pedder, Simon C. J., Robert I. Wilcox, John M. Tuchek, Dennis D. Johnson, and R. D. Crawford. "Attenuation of febrile seizures in epileptic chicks by N-methyl-D-aspartate receptor antagonists." Canadian Journal of Physiology and Pharmacology 68, no. 1 (1990): 84–88. http://dx.doi.org/10.1139/y90-012.

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Experimental febrile seizures can be evoked in epileptic chicks by elevation of their body temperature. Both competitive N-methyl-D-aspartate (NMDA) receptor antagonists [(3-(±)2-carboxypiperazin-4-yl)-propyl-1-phosphonic acid (CPP), DL-2-amino-7-phosphosphonoheptanoic acid (APH), DL-2-amino-5-phosphonovaleric acid (APV), D-α-aminoadipic acid (AAA), and DL-α,ε-diaminopimelic acid (DAP)] and the noncompetitive NMDA antagonist (+)-5-methyl-10,11-dihydro-5H-dibenzo [a,d] cyclohepten-5,10-imine maleate (MK-801) produced dose-dependent increases in latency to the onset of seizures. Of the drugs tes
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12

Kaminski, John E., Peter H. Dernoeden, and Cale A. Bigelow. "Creeping Bentgrass Seedling Tolerance to Herbicides and Paclobutrazol." HortScience 39, no. 5 (2004): 1126–29. http://dx.doi.org/10.21273/hortsci.39.5.1126.

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The tolerance of creeping bentgrass (Agrostis stolonifera L.) seedlings to many herbicides has not been evaluated. Three field studies were conducted between fall and spring from 1998 to 2002 to assess creeping bentgrass seedling tolerance to five herbicides and paclobutrazol. The primary objectives of this investigation were to assess bentgrass tolerance to these chemicals when applied at various timings following seedling emergence, and establishment of new seedlings as influenced by potential soil residues in the spring following a fall application of the chemicals. Treatments were applied
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13

Courteix, Christine, Anne-Marie Privat, Teresa Pélissier, Alejandro Hernandez, Alain Eschalier, and Joseph Fialip. "Agmatine Induces Antihyperalgesic Effects in Diabetic Rats and a Superadditive Interaction with R(–)-3-(2-Carboxypiperazine-4-yl)-propyl-1-phosphonic Acid, a N-Methyl-d-aspartate-Receptor Antagonist." Journal of Pharmacology and Experimental Therapeutics 322, no. 3 (2007): 1237–45. http://dx.doi.org/10.1124/jpet.107.123018.

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14

Thompson, Kenira J., Mario L. Mata, James E. Orfila, Edwin J. Barea-Rodriguez, and Joe L. Martinez. "Metabotropic Glutamate Receptor Antagonist AIDA Blocks Induction of Mossy Fiber-CA3 LTP In Vivo." Journal of Neurophysiology 93, no. 5 (2005): 2668–73. http://dx.doi.org/10.1152/jn.00901.2004.

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Metabotropic glutamate receptors (mGluR) are implicated in long-term memory storage. mGluR-I and mGluR-II antagonists impede various forms of learning and long-term potentiation (LTP) in animals. Despite the evidence linking mGluR to learning mechanisms, their role in mossy fiber-CA3 long-term potentiation (LTP) is not yet clear. To explain the involvement of mGluR-I in memory mechanisms, we examined the function of the mGluR-I antagonist 1-aminoindan-1, 5-dicarboxylic acid (AIDA) on the induction of mossy fiber-CA3 LTP in vivo in male Sprague Dawley and Fischer 344 (F344) rats. Acute extracel
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15

Ahn, Seongmo, Jin Hyeok Jang, Jung Min Joo, and Hye Ryung Byon. "Dicationic Heteroaryl Pyridinium As a Highly Stable, Soluble, and Crossover-Resistant Anolyte for Nonaqueous Redox Flow Batteries." ECS Meeting Abstracts MA2022-01, no. 48 (2022): 2031. http://dx.doi.org/10.1149/ma2022-01482031mtgabs.

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Recently, redox flow batteries (RFBs) have emerged as one of the promising candidates for safe and economical grid-scale energy storage system (ESS) that store the intermittent energies such as wind or solar energy. Unlike the conventional aqueous vanadium RFBs, the design of new molecules in nonaqueous RFB (NRFB) has been in the spotlight for the high energy density, cycling stability, and low cost. Among the redox active materials, in particular, organic molecule has various structures through functionalization, and thus its redox potential, solubility, and chemical stability can be controll
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16

Bracci, E., L. Ballerini, and A. Nistri. "Spontaneous rhythmic bursts induced by pharmacological block of inhibition in lumbar motoneurons of the neonatal rat spinal cord." Journal of Neurophysiology 75, no. 2 (1996): 640–47. http://dx.doi.org/10.1152/jn.1996.75.2.640.

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1. The effects of blocking gamma-aminobutyric acid- and glycine-mediated synaptic transmission by bicuculline and strychnine on the neonatal rat isolated spinal cord were investigated by intracellular recording from motoneurons with the use of current-clamp and voltage-clamp techniques and by extracellular recording from homologous ventral roots of the L5 segment. 2. Bicuculline per se evoked irregular bursts of motoneuron membrane potential, often comprising individual events fused together. Strychnine alone did not elicit spontaneous bursting in the large majority of preparations. Simultaneo
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17

O'Boyle, Michael P., Viet Do, Brian E. Derrick, and Brenda J. Claiborne. "In Vivo Recordings of Long-Term Potentiation and Long-Term Depression in the Dentate Gyrus of the Neonatal Rat." Journal of Neurophysiology 91, no. 2 (2004): 613–22. http://dx.doi.org/10.1152/jn.00307.2003.

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Previous in vitro studies demonstrated that long-term potentiation (LTP) could be elicited at medial perforant path (MPP) synapses onto hippocampal granule cells in slices from 7-day-old rats. In contrast, in vivo studies suggested that LTP at perforant path synapses could not be induced until at least days 9 or 10 and then in only a small percentage of animals. Because several characteristics of the oldest granule cells are adult-like on day 7, we re-examined the possibility of eliciting LTP in 7-day-old rats in vivo. We also recorded from 8- and 9-day-old rats to further elucidate the occurr
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18

Gunduz, Mithat, Upendra A. Argikar, Amanda L. Cirell, Alan P. Brown, Simone Bonazzi, and Markus Walles. "Species-specific Bioactivation of Morpholines as a Causative of DrugInduced Liver Injury Observed in Monkeys." Drug Metabolism and Bioanalysis Letters 16 (December 1, 2023). http://dx.doi.org/10.2174/0118723128260455231104180653.

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Background: Everolimus, an allosteric mechanistic target of rapamycin (mTOR) inhibitor, recently demonstrated the therapeutic value of mTOR inhibitors for Central Nervous System (CNS) indications driven by hyperactivation of mTOR. A newer, potent brain-penetrant analog of everolimus, referred to as (1) in this manuscript [(S)-3-methyl-4-(7-((R)-3-methylmorpholino)-2- (thiazol-4-yl)-3H-imidazo[4,5-b]pyridin-5-yl)morpholine,(1)] catalytically inhibits mTOR function in the brain and increases the lifespan of mice with neuronal mTOR hyperactivation Introduction: Early evaluation of the safety of 1
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19

Cao, Meng-meng, Xin-ling Wang, Wen-ke Yang, Jing Yang та Xia Wang. "Crystal structure of diiodo-bis(1-((2-propyl-1H-benzo[d]imidazol-1-yl)methyl)-1H-benzo[d][1,2,3]triazole-κ1 N)cadmium(II), C34H34CdI2N10". Zeitschrift für Kristallographie - New Crystal Structures, 15 липня 2025. https://doi.org/10.1515/ncrs-2025-0231.

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Abstract C34H34CdI2N10, monoclinic, C2/c (no. 15), a = 17.1805(4) Å, b = 12.8107(2) Å, c = 17.6543(4) Å, β = 113.821(3)°, Z = 4, V = 3554.59(15) Å3, R gt(F) = 0.0447, wR ref(F 2) = 0.1192, T = 293(2)K.
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20

Cheng, Ling-He, Meng-meng Cao, Hai-Long Zhang, Xiao Wang та Yang-Yu Liu. "Crystal structure of poly[(μ2-nitrato-κ3 O,O′:O′′)(μ2-1-[(2-propyl-1H-benzimidazole-1-yl)methyl]-1H-benzotriazole-k2 N:N′)silver(I)], C17H17AgN6O3". Zeitschrift für Kristallographie - New Crystal Structures, 23 травня 2025. https://doi.org/10.1515/ncrs-2025-0114.

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