Academic literature on the topic 'Inhibitors compounds'

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Journal articles on the topic "Inhibitors compounds"

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Flores-Garcia, N. S., C. D. Arrieta-Gonzalez, J. J. Ramos-Hernandez, et al. "Rare Earth-Based Compounds as Inhibitors of Hot-Corrosion Induced by Vanadium Salts." Materials 12, no. 22 (2019): 3796. http://dx.doi.org/10.3390/ma12223796.

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In this study, the performance evaluation of lanthanum compounds as corrosion inhibitors of vanadium salts was performed. The inhibitors tested were lanthanum acetate and La2O3. The performance of the inhibitors was tested using sodium metavanadate (NaVO3) as a corrosive medium at 700, 800, and 900 °C. The corrosion inhibitory effect was evaluated on the corrosion process of 304H stainless steel. The corrosion rate of the steel was determined by the mass loss technique after 100 h of immersion in the corrosive salt with and without the addition of the corrosion inhibitor. The results show that
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Edmonds, S., A. Gibb, and E. Sim. "Effect of thiol compounds on human complement component C4." Biochemical Journal 289, no. 3 (1993): 801–5. http://dx.doi.org/10.1042/bj2890801.

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Thiol compounds have been investigated as inhibitors of the covalent binding reaction of human complement protein C4 using Sepharose-C1s as a combined activating and binding surface. o- and p-substituted aminothiophenols are equally effective inhibitors, whereas the m-substituted compound is a less potent inhibitor. The anti-hypertensive drug captopril is also shown to inhibit the covalent binding reaction. A comparison of the effects of these compounds on the covalent binding reaction of isolated C4A and C4B has been made. Results suggest that a Pro-to-Leu substitution in C4B is likely to acc
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Honma, Masaru, Mark Stubbs, Ian Collins, Paul Workman, Wynne Aherne, and Fiona M. Watt. "Identification of Novel Keratinocyte Differentiation Modulating Compounds by High-Throughput Screening." Journal of Biomolecular Screening 11, no. 8 (2006): 977–84. http://dx.doi.org/10.1177/1087057106292556.

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The authors have designed high-throughput screens to identify compounds that promote or inhibit terminal differentiation of primary human epidermal keratinocytes. Eleven known inhibitors of signaling pathways and approximately 4000 compounds of diverse structure were screened using an In-Cell Western system based on immunofluorescent staining of the terminal differentiation marker, involucrin. Staurosporine, a nonspecific protein kinase C inhibitor, and H89, a protein kinase A inhibitor, promoted expression of involucrin. Conversely, U0126, a MEK inhibitor, and SAHA or SBHA, 2 histone deacetyl
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Adachi, Ryutaro, Tsuyoshi Ishii, Shinichi Matsumoto, Takuya Satou, Junichi Sakamoto, and Tomohiro Kawamoto. "Discovery of Human Intestinal MGAT Inhibitors Using High-Throughput Mass Spectrometry." SLAS DISCOVERY: Advancing the Science of Drug Discovery 22, no. 4 (2016): 360–65. http://dx.doi.org/10.1177/1087057116673181.

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Monoacylglycerol acyltransferase (MGAT) activity catalyzes the synthesis of diacylglycerol (DAG) from fatty acyl-CoA and monoacylglycerol as substrates. It is important for the resynthesis of triacylglycerol (TAG) in the intestine. In the present study, we developed a MGAT enzymatic assay of human intestinal microsomes using a high-throughput mass spectrometry (MS)–based detection system. After screening with small-molecular-weight libraries for compounds exhibiting inhibitions against DAG and the consequent TAG syntheses, we identified multiple compounds that specifically inhibit intestinal M
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Sharma, Rajesh, Jitendra Sainy, and Subhash Chaturvedi. "2-Amino-5-sulfanyl-1,3,4-thiadiazoles: A new series of selective cyclooxygenase-2 inhibitors." Acta Pharmaceutica 58, no. 3 (2008): 317–26. http://dx.doi.org/10.2478/v10007-008-0011-6.

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2-Amino-5-sulfanyl-1,3,4-thiadiazoles: A new series of selective cyclooxygenase-2 inhibitorsA new series of cyclooxygenase-2 inhibitors with 2-amino--5-sulfanyl-1,3,4-thiadiazole as the central scaffold unit has been synthesized. The newly synthesized compounds were characterized by analytical and spectral methods. Compounds were screened for cyclooxygenase inhibitory activity by the colorimetric COX (ovine) inhibitor screening assay, anti-inflammatory activity by the carrageenean induced rat paw oedema test and analgesic activity by the tail flick method. Some compounds exhibited significant
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Suwanhom, Paptawan, Jirakrit Saetang, Pasarat Khongkow, Teerapat Nualnoi, Varomyalin Tipmanee, and Luelak Lomlim. "Synthesis, Biological Evaluation, and In Silico Studies of New Acetylcholinesterase Inhibitors Based on Quinoxaline Scaffold." Molecules 26, no. 16 (2021): 4895. http://dx.doi.org/10.3390/molecules26164895.

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A quinoxaline scaffold exhibits various bioactivities in pharmacotherapeutic interests. In this research, twelve quinoxaline derivatives were synthesized and evaluated as new acetylcholinesterase inhibitors. We found all compounds showed potent inhibitory activity against acetylcholinesterase (AChE) with IC50 values of 0.077 to 50.080 µM, along with promising predicted drug-likeness and blood–brain barrier (BBB) permeation. In addition, potent butyrylcholinesterase (BChE) inhibitory activity with IC50 values of 14.91 to 60.95 µM was observed in some compounds. Enzyme kinetic study revealed the
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Dong, Hang, Hao Yin, Chunlong Zhao, Jiangying Cao, Wenfang Xu, and Yingjie Zhang. "Design, Synthesis and Biological Evaluation of Novel Osimertinib-Based HDAC and EGFR Dual Inhibitors." Molecules 24, no. 13 (2019): 2407. http://dx.doi.org/10.3390/molecules24132407.

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Herein a novel series of histone deacetylases (HDACs) and epidermal growth factor receptor (EGFR) dual inhibitors were designed and synthesized based on the structure of the approved EGFR inhibitor osimertinib (AZD9291). Among them, four compounds 5D, 5E, 9D and 9E exhibited more potent total HDAC inhibition than the approved HDAC inhibitor SAHA. However, these compounds only showed moderate to low inhibitory potency towards EGFR with compounds 5E and 9E possessing IC50 values against EGFRWT and EGFRT790M in the micromolar range. 3-[4,5-dimethyl-2-thiazolyl]-2,5-diphenyl-2H-tetrazolium bromide
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da Silva, Edson Roberto, Júlio Abel Alfredo dos Santos Simone Come, Simone Brogi, et al. "Cinnamides Target Leishmania amazonensis Arginase Selectively." Molecules 25, no. 22 (2020): 5271. http://dx.doi.org/10.3390/molecules25225271.

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Caffeic acid and related natural compounds were previously described as Leishmania amazonensis arginase (L-ARG) inhibitors, and against the whole parasite in vitro. In this study, we tested cinnamides that were previously synthesized to target human arginase. The compound caffeic acid phenethyl amide (CAPA), a weak inhibitor of human arginase (IC50 = 60.3 ± 7.8 μM) was found to have 9-fold more potency against L-ARG (IC50 = 6.9 ± 0.7 μM). The other compounds that did not inhibit human arginase were characterized as L-ARG, showing an IC50 between 1.3–17.8 μM, and where the most active was compo
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Ommeh, Sheila, Eunice Nduati, Eddy Mberu, et al. "In Vitro Activities of 2,4-Diaminoquinazoline and 2,4-Diaminopteridine Derivatives against Plasmodium falciparum." Antimicrobial Agents and Chemotherapy 48, no. 10 (2004): 3711–14. http://dx.doi.org/10.1128/aac.48.10.3711-3714.2004.

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ABSTRACT The activities of 28 6-substituted 2,4-diaminoquinazolines, 2,4-diamino-5,6,7,8-tetrahydroquinazolines, and 2,4-diaminopteridines against Plasmodium falciparum were tested. The 50% inhibitory concentrations (IC50s) of six compounds were <50 nM, and the most potent compound was 2,4-diamino-5-chloro-6-[N-(2,5-dimethoxybenzyl)amino]quinazoline (compound 1), with an IC50 of 9 nM. The activity of compound 1 was potentiated by the dihydropteroate synthase inhibitor dapsone, an indication that these compounds are inhibitors of dihydrofolate reductase. Further studies are warranted to asse
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Bule, Mohammed Hussen, Roghaieh Esfandyari, Tadesse Bekele Tafesse, Mohsen Amini, Mohammad Ali Faramarzi та Mohammad Abdollahi. "Synthesis, Molecular Docking and α-Glucosidase Inhibitory Activity Study of 2,4,6-triaryl Pyrimidine Derivatives". Letters in Drug Design & Discovery 17, № 10 (2020): 1216–26. http://dx.doi.org/10.2174/1570180817666200103130536.

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Background: α-Glucosidase inhibitors hinder the carbohydrate digestion and play an important role in the treatment of diabetes mellitus. α-glucosidase inhibitors available on the market are acarbose, miglitol, and voglibose. However, the use of acarbose is diminishing due to related side effects like diarrhea, bloating and abdominal distension. Objectives: This study aimed to synthesize 2,4,6-triaryl pyrimidines derivatives, screen their α- glucosidase inhibitory activity, perform kinetic and molecular docking studies. Methods: A series of 2,4,6-triaryl pyrimidine derivatives were synthesized
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Dissertations / Theses on the topic "Inhibitors compounds"

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Tan, Swee Hain. "Organic corrosion inhibitors." Murdoch University, 1991. http://wwwlib.murdoch.edu.au/adt/browse/view/adt-MU20060818.150145.

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The overall aims of this thesis were to conduct a broad survey of possible organic corrosion inhibitors in near-neutral chloride solutions and to elucidate the mechanisms of such action. Altogether, 130 organic compounds were studied as possible corrosion inhibitors for pure iron, mild steel, copper and aluminium in aerated near-neutral (pH = 8.4) solutions containing 500 ppm NaCl and 100 ppm NaHCO,, conditions often encountered in water-based automotive engine coolants. Inhibitor behaviour was investigated using steady-state electrochemical techniques including polarisation curves, Stern-Gear
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Geraets, Liesbeth. "Dietary PARP-1 inhibitors as anti-inflammatory compounds." Maastricht : Maastricht : Universitaire Pers ; University Library, Universiteit Maastricht [host], 2008. http://arno.unimaas.nl/show.cgi?fid=14252.

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McNab, Donald. "Boron-containing compounds as inhibitors of HIV proteinase." Thesis, University of St Andrews, 1997. http://hdl.handle.net/10023/14305.

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HIV Proteinase (HIV PR) has proved to be an excellent target for the development of anti-AIDS drugs. Four inhibitors of this enzyme are now approved for clinical use but they, like others, suffer from shortcomings associated with their size and the fact they are peptides. In this thesis the development of small non-peptidic cyclic compounds is described. They were designed to inhibit HIV PR principally by targeting its unique structural features rather than by mimicking its natural substrates. The designed compounds all contained the borinic acid functional group which it was anticipated would
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Corredor, Sánchez Miriam. "Chemical Modulation of Identified Hit Compounds as Apoptosis Inhibitors." Doctoral thesis, Universitat Ramon Llull, 2013. http://hdl.handle.net/10803/117361.

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L’apoptosi és un procés biològic rellevant en moltes malalties. Un punt de regulació d’aquest procés és la formació d’un complex multiproteic anomenat apoptosoma; per tant, aquest complex té un gran interès per al desenvolupament de moduladors apoptòtics. El nostre grup ha descrit prèviament una piperazina-2,5-diona substituïda en posició 3 com a potent modulador apoptòtic. Estudis estructurals d’aquest compost han permès veure la presència dels isòmers cis / trans de l’enllaç de l’amida terciària exocíclica en un procés d’intercanvi lent, fet que pot ser important per a la interacció amb la d
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Ryle, Peter Robert. "Ethanol-induced fatty liver : protective action of (+)-catechin compounds." Thesis, University of Surrey, 1986. http://epubs.surrey.ac.uk/847975/.

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The aim of the work presented in this thesis was to assess the protective properties of the bioflavanoid drug, (+)-catechin, and its palmityl ester, 3-palmitoyl-(+)-catechin, against ethanol hepato-toxicity (ie: fatty liver) in the rat. In initial experiments, both (+)-catechin compounds were found to protect against the hepatic lipid accumulation (mainly triglyceride) after acute ethanol dosing, and after long-term feeding of ethanol in a liquid diet. In the latter situation, 3-palmitoyl-(+)-catechin was significantly more effective than (+)-catechin itself at preventing fatty liver, probably
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Abner, Erik 1986. "Identification of HIV-1 reactivating quinoline compounds as bromodomain inhibitors." Doctoral thesis, Universitat Pompeu Fabra, 2016. http://hdl.handle.net/10803/565528.

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Tras la infección por VIH-1, el establecimiento de un depósito de células T en reposo infectadas latentemente con VIH impide la erradicación del virus en pacientes. Para lograr la erradicación, la terapia retroviral existente debe combinarse con medicamentos que reactiven los virus latentes. Previamente, nuestro grupo describió un nuevo compuesto químico, MMQO (8-metoxi-6-metilquinolin-4-ol) que es capaz de reactivar la transcripción viral a través de un mecanismo desconocido. El objetivo de este proyecto fue identificar los proteínas que interaccionan con MMQO e investigar su papel en la reac
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Cunningham, Bernadette D. M. "Flavones and related compounds as inhibitors of protein tyrosine kinases." Thesis, Aston University, 1987. http://publications.aston.ac.uk/12513/.

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Aberrant tyrosine protein kinase activity has been implicated in the formation and maintenance of malignancy and so presents a potential target for cancer chemotherapy. Quercetin, a naturally occuring flavonoid, inhibits the tyrosine protein kinase encoded by the Rous sarcoma virus but also exhibits many other effects. Analogues of this compound were synthesised by the acylation of suitable 2-hydroxyacetophenones with appropriately substituted aromatic (or alicyclic) acid chlorides, followed by base catalysed rearrangement to the 1-(2-hydroxyphenyl)-3-phenylpropan-1,3-diones. Acid catalysed ri
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García, Reyes Balbina [Verfasser]. "Validation of new Casein Kinase 1 (CK1) small molecule inhibitor compounds and characterization of Inhibitors of Wnt Production (IWPs) as inhibitors of CK1δ / Balbina García Reyes". Ulm : Universität Ulm, 2018. http://d-nb.info/1151938424/34.

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Byrom, Daniel. "Synthesis of TGF-Beta inhibitors and compounds for spatiotemporal drug release." Doctoral thesis, Universitat de Barcelona, 2018. http://hdl.handle.net/10803/665149.

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During this doctoral thesis, we have synthesised hundreds of grams of the TGF-β inhibitor LY2157299 (Galunisertib). This product was used by the group of Eduard Batlle in their investigations into the roles that TGF-β plays in colorectal cancer. During the initial synthesis and subsequent scale up, we overcame hurdles including optimisation of the penultimate step of the reaction - giving reproducible results - as well as optimising conditions of the final solid form to provide a product which is suitable for formulation for the in vivo experiments. After discovering some of the drawback of LY
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Omune, Duncan Otieno. "Synthetic analogs of equisetin as potential HIV-1 integrase inhibitors." Diss., Online access via UMI:, 2004. http://wwwlib.umi.com/dissertations/fullcit/3150487.

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Books on the topic "Inhibitors compounds"

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Kato, T., W. Krämer, K. H. Kuck, D. M. Norris, and H. Scheinpflug, eds. Sterol Biosynthesis Inhibitors and Anti-Feeding Compounds. Springer Berlin Heidelberg, 1986. http://dx.doi.org/10.1007/978-3-642-69790-6.

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Kuznetsov, Yurii I. Organic inhibitors of corrosion of metals. Edited by Thomas J. G. N. Plenum Press, 1996.

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Cunningham, Bernadette Deirdre Mary. Flavones and related compounds as inhibitors of protein tyrosine kinases. Aston University. Department of Pharmaceutical Sciences, 1987.

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Handbook of compounds with anti-inflammatory and anti-platelet aggregation activities isolated from plants. Nova Science Publishers, 2008.

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1946-, Kato T., ed. Sterol biosynthesis inhibitors and anti-feeding compounds. Springer-Verlag, 1986.

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E, Stütz Arnold, ed. Iminosugars as glycosidase inhibitors: Nojirimycin and beyond. Wiley-VCH, 1999.

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Stu, Arnold E. Iminosugars As Glycosidase Inhibitors: Nojirimycin and Beyond. John Wiley & Sons, 1999.

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Ramesh C. Gupta, PhD, DABT, FACT, FATS. Toxicology of Organophosphate & Carbamate Compounds. Academic Press, 2005.

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Toxicology of Organophosphate & Carbamate Compounds. Academic Press, 2005.

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Böldicke, Thomas. Protein Targeting Compounds: Prediction, Selection and Activity of Specific Inhibitors. Springer, 2018.

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Book chapters on the topic "Inhibitors compounds"

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Büning, H., and U. T. Hacker. "Inhibitors of Angiogenesis." In Protein Targeting Compounds. Springer International Publishing, 2015. http://dx.doi.org/10.1007/978-3-319-22473-2_12.

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Kuck, Karl-Heinz, Klaus Stenzel, and Jean-Pierre Vors. "Sterol Biosynthesis Inhibitors." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2012. http://dx.doi.org/10.1002/9783527644179.ch19.

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Stenzel, Klaus, and Jean-Pierre Vors. "Sterol Biosynthesis Inhibitors*." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2019. http://dx.doi.org/10.1002/9783527699261.ch19.

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Lickfeldt, Darin W., Denise P. Cudworth, Daniel D. Loughner, and Lowell D. Markley. "Microtubulin Assembly Inhibitors (Pyridines)." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2012. http://dx.doi.org/10.1002/9783527644179.ch10.

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Wenger, Jean, Thierry Niderman, and Chris Mathews. "Acetyl-CoA Carboxylase Inhibitors." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2012. http://dx.doi.org/10.1002/9783527644179.ch11.

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Theodoridis, George, Rex Liebl, and Cyrill Zagar. "Protoporphyrinogen IX Oxidase Inhibitors." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2012. http://dx.doi.org/10.1002/9783527644179.ch3.

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Dietrich, Hansjörg, and Bernd Laber. "Inhibitors of Cellulose Biosynthesis." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2012. http://dx.doi.org/10.1002/9783527644179.ch7.

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Lickfeldt, Darin W., Denise P. Cudworth, Daniel D. Loughner, and Lowell D. Markley. "Microtubulin Assembly Inhibitors (Pyridines)." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2019. http://dx.doi.org/10.1002/9783527699261.ch10.

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Wenger, Jean, Thierry Niderman, Chris Mathews, and Steve Wailes. "Acetyl-CoA Carboxylase Inhibitors." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2019. http://dx.doi.org/10.1002/9783527699261.ch11.

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Zagar, Cyrill, Rex Liebl, George Theodoridis, and Matthias Witschel. "Protoporphyrinogen IX Oxidase Inhibitors." In Modern Crop Protection Compounds. Wiley-VCH Verlag GmbH & Co. KGaA, 2019. http://dx.doi.org/10.1002/9783527699261.ch3.

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Conference papers on the topic "Inhibitors compounds"

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Jansen, J. W. C. M. "EFFECTS OF INHIBITORS ON COLLAGEN INDUCED PLATELET AGGREGATION IN SIX DIFFERENT SPECIES." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643445.

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One approach to the development of antithrombotics is inhibition of platelet aggregation. The pharmacological approach often used is to test compounds on collagen induced platelet aggregation measured in platelet rich plasma. Therefore we have compared inhibitors with different mechanism of action on aggregation of platelets from six different species commonly used in pharmacological studies. Aggregation was induced with submaximal amounts of collagen (Hormone Chemie).Inhibitors of the cyclooxygenase system, aspirin and indomethacin, were very potent in inhibiting aggregation of platelets from
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Beretz, A., F. Lanza, A. Stierlé, and J.-P. Cazenave. "CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITORS PREVENT AGGREGATION AND SECRETION OF HUMAN PLATELETS BY RAISING CYCLIC AMP AND REDUCING CYTOPLASMIC FREE CALCIUM MOBILIZATION." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643586.

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Drugs that raise platelet cyclic AMP (cAMP) are potent inhibitors of platelet activation. We have studied the effects of 5 inhibitors of cyclic nucleotide phosphodiesterase (PDE) of different chemical structures (quercetin, Ro 15-2041, HL-725, cilostamide and MY-5445), which are all potent inhibitors of platelet function. The concentrations that inhibit by 50 % crude cAMP-PDE activity (IC50) from human platelets are: 0.06 μM(HL-725), 0.15 μM(Ro 15-2041 ), 0.23 μM(cilostamide), 6.9 μM(MY-5445) and 44.4 μM(quercetin). We measured on the same preparation of washed human platelets loaded with quin
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Ng, Jun Hong Clarence, Tariq Almubarak, and Hisham A. Nasr-El-Din. "Seed Extracts as Natural, Green, Non-Toxic Corrosion Inhibitors." In SPE Trinidad and Tobago Section Energy Resources Conference. SPE, 2021. http://dx.doi.org/10.2118/200935-ms.

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Abstract Acid treatments are commonly used in the oilfield to remove inorganic scale or to stimulate formatio ns. These treatments typically consist of using hydrochloric acid (HCl), acetic acid, formic acid, or chelating agents. At elevated temperatures, these acids are highly corrosive and can cause severe damage to tubulars as well as downhole equipment. To reduce damage from these acids, corrosion inhibitors are added to the treatment solution. Corrosion inhibitors used in the oil and gas industry are typically quaternary amines or sulfur-containing compounds. These compounds adsorb to the
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Mathew, Shilu M., Fatiha Benslimane, Asmaa A. Althani, and Hadi M. Yassine. "Virtual Screening of Anti-Viral Drugs and Natural Compounds for Potential Inhibition of the Novel SARS-Cov-2 Spike Receptor-Binding Domain." In Qatar University Annual Research Forum & Exhibition. Qatar University Press, 2020. http://dx.doi.org/10.29117/quarfe.2020.0281.

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Background: The spike (S) protein of SARS-CoV-2 harbors the receptor-binding domain (RBD) that mediates the virus's entry to host cells. The aim of this study was to identify novel inhibitors that target the RBD domain of S-protein through computational screening of chemical and natural compounds. Method: The S protein was modelled from the recently resolved and the previously described SARS-CoV protein structures. CLC Drug Discovery was used to computationally screen for potential inhibitory effects of currently prescribed drugs (n= 22) anti-viral natural drugs (n=100), natural compounds (n=
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Kumar, T., S. Vishwanatham, _. Emranuzzaman, and B. N. Talukdar. "Nitrogen Containing Organic Compounds as Corrosion Inhibitors of Mild Steel." In SPE India Oil and Gas Conference and Exhibition. Society of Petroleum Engineers, 1998. http://dx.doi.org/10.2118/39534-ms.

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Hannon, C. L., J. Gerstmann, F. B. Mansfeld, and Z. Sun. "Development of Corrosion Inhibitors for Absorption Heat Pumps." In ASME 2002 International Mechanical Engineering Congress and Exposition. ASMEDC, 2002. http://dx.doi.org/10.1115/imece2002-33411.

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This paper describes the results of a research project to develop a non-toxic corrosion in hibitor for the protection of carbon steel surfaces of ammonia-water absorption heat pumps through the use of rare earth metal salt (REMS) compounds. Chromate compounds are currently used as corrosion inhibitors in these systems, but are toxic, environmentally harmful, and their use is being phased out. Corrosion concerns in ammonia-water absorption systems are primarily those of non-condensable (NC) gases generated by corrosion reactions impeding the heat and mass transfer processes in the system. The r
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Tiwari, Laxmikant. "Design & Development of Quaternary Amine Compounds: Corrosion Inhibitors with Improved Environmental Profiles." In SPE International Symposium on Oilfield Corrosion. Society of Petroleum Engineers, 2005. http://dx.doi.org/10.2118/95081-ms.

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Lindamulage, Indeewari K., Hai-Yen Vu, Dr Piyush Trivedi, and Dr Hoyun Lee. "Abstract 3100: Characterisation of novel chalcone derivatives, CTR compounds as tubulin polymerisation inhibitors." In Proceedings: AACR 106th Annual Meeting 2015; April 18-22, 2015; Philadelphia, PA. American Association for Cancer Research, 2015. http://dx.doi.org/10.1158/1538-7445.am2015-3100.

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Saeh, Jamal C., Bin Yang, Bo Peng, et al. "Abstract 2916: Discovery of pyrazolimidazopyridine compounds as potentin vitroandin vivoanaplastic lymphoma kinase inhibitors." In Proceedings: AACR 103rd Annual Meeting 2012‐‐ Mar 31‐Apr 4, 2012; Chicago, IL. American Association for Cancer Research, 2012. http://dx.doi.org/10.1158/1538-7445.am2012-2916.

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Korolev, Vjacheslav, Аlexej Alekseev, Natalia Merkulova, et al. "INHIBITORS OF ADP-INDUCED PLATELET AGGREGATION BASED ON IMIDAZO [4,5-E] BENZO [1,2-C; 3,4-C ’] DIFUROXAN." In Chemistry of nitro compounds and related nitrogen-oxygen systems. LLC MAKS Press, 2019. http://dx.doi.org/10.29003/m793.aks-2019/361-365.

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Reports on the topic "Inhibitors compounds"

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Perez-Acle, Tomas. Development of Lead Compounds as Fusion Inhibitors for Dengue Virus. Defense Technical Information Center, 2009. http://dx.doi.org/10.21236/ada604418.

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2

Klipp, Robert. Novel Compound, 84F2, Inhibits Calmodulin Deficient RyR2. Portland State University Library, 2000. http://dx.doi.org/10.15760/etd.5368.

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